Compile Data Set for Download or QSAR
maximum 50k data
Found 51 Enz. Inhib. hit(s) with all data for entry = 50005010
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537670(CHEMBL4641380)
Affinity DataIC50:  20nMAssay Description:Tested for inhibition of cGMP-dependent protein kinase from bovine lungMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537669(CHEMBL4643608)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at CB1 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537671(CHEMBL4633843)
Affinity DataIC50:  30nMAssay Description:Tested for inhibition of cGMP-dependent protein kinase from bovine lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537648(CHEMBL4640596)
Affinity DataIC50:  40nMAssay Description:Inhibitory potency against isolated epidermal growth factor receptor (EGFR) from human A431 carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537661(CHEMBL4648946)
Affinity DataIC50:  40nMAssay Description:Antagonist activity at CB1 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537646(CHEMBL512270)
Affinity DataIC50:  40nMAssay Description:Inhibitory potency against isolated epidermal growth factor receptor (EGFR) from human A431 carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537649(CHEMBL1723285)
Affinity DataIC50:  50nMAssay Description:Inhibition of Epidermal growth factor receptor autophosphorylation in A431 human epidermoid carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537665(CHEMBL4648066)
Affinity DataIC50:  50nMAssay Description:Antagonist activity at CB1 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537662(CHEMBL4647748)
Affinity DataIC50:  50nMAssay Description:Antagonist activity at CB1 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537643(CHEMBL1506565)
Affinity DataIC50:  50nMAssay Description:Inhibitory potency against isolated epidermal growth factor receptor (EGFR) from human A431 carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537629(CHEMBL4635339)
Affinity DataIC50:  58nMAssay Description:Inhibitory potency against isolated epidermal growth factor receptor (EGFR) from human A431 carcinoma cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537628(CHEMBL4643853)
Affinity DataIC50:  66nMAssay Description:Inhibitory potency against isolated epidermal growth factor receptor (EGFR) from human A431 carcinoma cellsMore data for this Ligand-Target Pair
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537628(CHEMBL4643853)
Affinity DataIC50:  66.1nMAssay Description:Tested for inhibition of cGMP-dependent protein kinase from bovine lungMore data for this Ligand-Target Pair
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537659(CHEMBL4646298)
Affinity DataIC50:  80nMAssay Description:Antagonist activity at CB1 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537647(CHEMBL1403506)
Affinity DataIC50:  80nMAssay Description:Inhibitory potency against isolated epidermal growth factor receptor (EGFR) from human A431 carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537667(CHEMBL4639207)
Affinity DataIC50:  140nMAssay Description:Antagonist activity at CB1 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537668(CHEMBL4647815)
Affinity DataIC50:  140nMAssay Description:Antagonist activity at CB1 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537652(CHEMBL4640293)
Affinity DataIC50:  180nMAssay Description:Antagonist activity at CB1 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537639(CHEMBL4639296)
Affinity DataIC50:  324nMAssay Description:Inhibitory potency against isolated epidermal growth factor receptor (EGFR) from human A431 carcinoma cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537641(CHEMBL4647303)
Affinity DataIC50:  575nMAssay Description:Inhibitory potency against isolated epidermal growth factor receptor (EGFR) from human A431 carcinoma cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537626(CHEMBL4645869)
Affinity DataIC50:  603nMAssay Description:Inhibition of Epidermal growth factor receptor autophosphorylation in A431 human epidermoid carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537664(CHEMBL4637016)
Affinity DataIC50:  820nMAssay Description:Antagonist activity at CB1 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537653(CHEMBL4643582)
Affinity DataIC50:  860nMAssay Description:Antagonist activity at CB1 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537645(CHEMBL467988)
Affinity DataIC50:  970nMAssay Description:Inhibitory potency against isolated epidermal growth factor receptor (EGFR) from human A431 carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537637(CHEMBL4644624)
Affinity DataIC50:  1.29E+3nMAssay Description:Inhibition of Epidermal growth factor receptor autophosphorylation in A431 human epidermoid carcinoma cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537655(CHEMBL4649728)
Affinity DataIC50:  1.36E+3nMAssay Description:Antagonist activity at CB1 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537660(CHEMBL4634222)
Affinity DataIC50:  1.72E+3nMAssay Description:Antagonist activity at CB1 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM154387(US9012443, 427)
Affinity DataIC50:  1.78E+3nMAssay Description:Inhibitory potency against isolated epidermal growth factor receptor (EGFR) from human A431 carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM154206(US9012443, 219)
Affinity DataIC50:  1.78E+3nMAssay Description:Inhibitory potency against isolated epidermal growth factor receptor (EGFR) from human A431 carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537644(CHEMBL1582054)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibitory potency against isolated epidermal growth factor receptor (EGFR) from human A431 carcinoma cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537638(CHEMBL4648561)
Affinity DataIC50:  2.95E+3nMAssay Description:Inhibitory potency against isolated epidermal growth factor receptor (EGFR) from human A431 carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537635(CHEMBL4634771)
Affinity DataIC50:  3.02E+3nMAssay Description:Inhibitory potency against isolated epidermal growth factor receptor (EGFR) from human A431 carcinoma cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537633(CHEMBL4635573)
Affinity DataIC50:  3.24E+3nMAssay Description:Inhibition of Epidermal growth factor receptor autophosphorylation in A431 human epidermoid carcinoma cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537630(CHEMBL4633966)
Affinity DataIC50:  4.07E+3nMAssay Description:Inhibitory potency against isolated epidermal growth factor receptor (EGFR) from human A431 carcinoma cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537642(CHEMBL4638594)
Affinity DataIC50:  4.37E+3nMAssay Description:Inhibitory potency against isolated epidermal growth factor receptor (EGFR) from human A431 carcinoma cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537632(CHEMBL4594142)
Affinity DataIC50:  6.17E+3nMAssay Description:Inhibitory potency against isolated epidermal growth factor receptor (EGFR) from human A431 carcinoma cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537627(CHEMBL4641013)
Affinity DataIC50:  6.76E+3nMAssay Description:Inhibitory potency against isolated epidermal growth factor receptor (EGFR) from human A431 carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537634(CHEMBL4639502)
Affinity DataIC50:  7.59E+3nMAssay Description:Inhibitory potency against isolated epidermal growth factor receptor (EGFR) from human A431 carcinoma cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537625(CHEMBL4648044)
Affinity DataIC50:  7.94E+3nMAssay Description:Inhibitory potency against isolated epidermal growth factor receptor (EGFR) from human A431 carcinoma cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537624(CHEMBL4635045)
Affinity DataIC50:  8.13E+3nMAssay Description:Inhibitory potency against isolated epidermal growth factor receptor (EGFR) from human A431 carcinoma cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537640(CHEMBL4637484)
Affinity DataIC50:  9.12E+3nMAssay Description:Inhibitory potency against isolated epidermal growth factor receptor (EGFR) from human A431 carcinoma cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537631(CHEMBL4636699)
Affinity DataIC50:  9.55E+3nMAssay Description:Inhibitory potency against isolated epidermal growth factor receptor (EGFR) from human A431 carcinoma cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537636(CHEMBL4648024)
Affinity DataIC50:  9.55E+3nMAssay Description:Inhibition of Epidermal growth factor receptor autophosphorylation in A431 human epidermoid carcinoma cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537650(CHEMBL4635913)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibitory potency against isolated epidermal growth factor receptor (EGFR) from human A431 carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537656(CHEMBL4635842)
Affinity DataIC50: >1.90E+4nMAssay Description:Antagonist activity at CB1 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537658(CHEMBL4634336)
Affinity DataIC50: >1.90E+4nMAssay Description:Antagonist activity at CB1 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537654(CHEMBL4643587)
Affinity DataIC50: >1.90E+4nMAssay Description:Antagonist activity at CB1 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537663(CHEMBL4636826)
Affinity DataIC50: >1.90E+4nMAssay Description:Antagonist activity at CB1 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537666(CHEMBL4633879)
Affinity DataIC50: >1.90E+4nMAssay Description:Antagonist activity at CB1 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSepiapterin reductase(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50537657(CHEMBL4636874)
Affinity DataIC50: >1.90E+4nMAssay Description:Antagonist activity at CB1 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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