Compile Data Set for Download or QSAR
Report error Found 76 Enz. Inhib. hit(s) with all data for entry = 50048109
LigandChemical structure of BindingDB Monomer ID 100152BDBM100152(cid_5359389 | SMR001233259 | HARMINE | 7-methoxy-1...)
Affinity DataIC50: 29nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 100152BDBM100152(cid_5359389 | SMR001233259 | HARMINE | 7-methoxy-1...)
Affinity DataIC50: 72nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204658BDBM50204658(CHEMBL3908596)
Affinity DataIC50: 700nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204646BDBM50204646(CHEMBL3962894)
Affinity DataIC50: 890nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204644BDBM50204644(CHEMBL3935442)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204647BDBM50204647(CHEMBL3917542)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204653BDBM50204653(CHEMBL3945429)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetCasein kinase I delta/epsilon(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 100152BDBM100152(cid_5359389 | SMR001233259 | HARMINE | 7-methoxy-1...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of CK1 delta/epsilon (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204659BDBM50204659(CHEMBL3923825)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50204658BDBM50204658(CHEMBL3908596)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50204646BDBM50204646(CHEMBL3962894)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50204644BDBM50204644(CHEMBL3935442)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50204653BDBM50204653(CHEMBL3945429)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50204659BDBM50204659(CHEMBL3923825)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50204647BDBM50204647(CHEMBL3917542)
Affinity DataIC50: 8.90E+3nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50204660BDBM50204660(CHEMBL3939584)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50204657BDBM50204657(CHEMBL3930589)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetCasein kinase I delta/epsilon(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204652BDBM50204652(CHEMBL3974565)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CK1 delta/epsilon (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetCasein kinase I delta/epsilon(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204645BDBM50204645(CHEMBL3957926)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CK1 delta/epsilon (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetCasein kinase I delta/epsilon(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204643BDBM50204643(CHEMBL3921647)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CK1 delta/epsilon (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204645BDBM50204645(CHEMBL3957926)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204656BDBM50204656(CHEMBL3903644)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50204652BDBM50204652(CHEMBL3974565)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50204655BDBM50204655(CHEMBL3902603)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetCasein kinase I delta/epsilon(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204657BDBM50204657(CHEMBL3930589)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CK1 delta/epsilon (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204652BDBM50204652(CHEMBL3974565)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GSK-3 alpha/beta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204644BDBM50204644(CHEMBL3935442)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GSK-3 alpha/beta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204649BDBM50204649(CHEMBL3936539)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetCasein kinase I delta/epsilon(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204658BDBM50204658(CHEMBL3908596)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CK1 delta/epsilon (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204655BDBM50204655(CHEMBL3902603)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GSK-3 alpha/beta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204651BDBM50204651(CHEMBL3911609)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GSK-3 alpha/beta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50204645BDBM50204645(CHEMBL3957926)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetCasein kinase I delta/epsilon(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204649BDBM50204649(CHEMBL3936539)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CK1 delta/epsilon (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetCasein kinase I delta/epsilon(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204647BDBM50204647(CHEMBL3917542)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CK1 delta/epsilon (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204656BDBM50204656(CHEMBL3903644)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GSK-3 alpha/beta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204653BDBM50204653(CHEMBL3945429)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GSK-3 alpha/beta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204650BDBM50204650(CHEMBL3912662)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204657BDBM50204657(CHEMBL3930589)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GSK-3 alpha/beta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204647BDBM50204647(CHEMBL3917542)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GSK-3 alpha/beta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204649BDBM50204649(CHEMBL3936539)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GSK-3 alpha/beta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetCasein kinase I delta/epsilon(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204653BDBM50204653(CHEMBL3945429)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CK1 delta/epsilon (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204652BDBM50204652(CHEMBL3974565)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50204643BDBM50204643(CHEMBL3921647)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204650BDBM50204650(CHEMBL3912662)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GSK-3 alpha/beta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetCasein kinase I delta/epsilon(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204656BDBM50204656(CHEMBL3903644)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CK1 delta/epsilon (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetCasein kinase I delta/epsilon(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204651BDBM50204651(CHEMBL3911609)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CK1 delta/epsilon (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204658BDBM50204658(CHEMBL3908596)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GSK-3 alpha/beta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetCasein kinase I delta/epsilon(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204642BDBM50204642(CHEMBL3985735)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CK1 delta/epsilon (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetCasein kinase I delta/epsilon(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204646BDBM50204646(CHEMBL3962894)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CK1 delta/epsilon (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
TargetCasein kinase I delta/epsilon(Human)
Paris-Sud University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50204659BDBM50204659(CHEMBL3923825)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CK1 delta/epsilon (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details Article
PubMed
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