Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50036296
TargetD(2) dopamine receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50038287(N-{4-[2-(4-Pyridin-2-yl-piperazin-1-yl)-ethyl]-cyc...)
Affinity DataEC50:  4.90nMAssay Description:In vitro inhibition of forskolin-stimulated cAMP accumulation in GH4C1 cells transfected with the human Dopamine D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM84637(NSC_54562 | CHEMBL240773 | QUINPIROLE | CAS_85760-...)
Affinity DataEC50:  7.60nMAssay Description:In vitro inhibition of forskolin-stimulated cAMP accumulation in GH4C1 cells transfected with the human Dopamine D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50038284(N-[(2R,4aS,6S,8aR)-6-(4-Pyridin-2-yl-piperazin-1-y...)
Affinity DataEC50:  10nMAssay Description:In vitro inhibition of forskolin-stimulated cAMP accumulation in GH4C1 cells transfected with the human Dopamine D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50038284(N-[(2R,4aS,6S,8aR)-6-(4-Pyridin-2-yl-piperazin-1-y...)
Affinity DataIC50: 73nMAssay Description:Binding affinity towards Dopamine D2 receptor from rat striatal membranes, using [3H]- spiperone as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50453480(CHEMBL2112745)
Affinity DataEC50:  240nMAssay Description:In vitro inhibition of forskolin-stimulated cAMP accumulation in GH4C1 cells transfected with the human Dopamine D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50038287(N-{4-[2-(4-Pyridin-2-yl-piperazin-1-yl)-ethyl]-cyc...)
Affinity DataIC50: 443nMAssay Description:Binding affinity towards Dopamine D2 receptor from rat striatal membranes, using [3H]- spiperone as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50038282(N-[(2R,4aS,6R,8aR)-6-(4-Pyridin-2-yl-piperazin-1-y...)
Affinity DataEC50: >1.00E+3nMAssay Description:In vitro inhibition of forskolin-stimulated cAMP accumulation in GH4C1 cells transfected with the human Dopamine D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50038283(N-[(2S,4aS,6R,8aR)-6-(4-Pyridin-2-yl-piperazin-1-y...)
Affinity DataEC50: >1.00E+3nMAssay Description:In vitro inhibition of forskolin-stimulated cAMP accumulation in GH4C1 cells transfected with the human Dopamine D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50453480(CHEMBL2112745)
Affinity DataIC50: 1.10E+3nMAssay Description:Binding affinity towards Dopamine D2 receptor from rat striatal membranes, using [3H]- spiperone as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50038282(N-[(2R,4aS,6R,8aR)-6-(4-Pyridin-2-yl-piperazin-1-y...)
Affinity DataIC50: 5.80E+3nMAssay Description:Binding affinity towards Dopamine D2 receptor from rat striatal membranes, using [3H]- spiperone as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50038283(N-[(2S,4aS,6R,8aR)-6-(4-Pyridin-2-yl-piperazin-1-y...)
Affinity DataIC50: 7.10E+3nMAssay Description:Binding affinity towards Dopamine D2 receptor from rat striatal membranes, using [3H]- spiperone as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed