Compile Data Set for Download or QSAR
Report error Found 45 Enz. Inhib. hit(s) with all data for entry = 50048457
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216719BDBM50216719(CHEMBL348433)
Affinity DataKi:  330nMpH: 7.1Assay Description:Binding affinity was evaluated towards 3-phosphoglycerate kinase at 37 degrees Celsius in 0.1 m NaCl pH 7.1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216635BDBM50216635(CHEMBL356436)
Affinity DataKi:  690nMpH: 7.1Assay Description:Binding affinity was evaluated towards 3-phosphoglycerate kinase at 37 degrees Celsius in 0.1 m NaCl pH 7.1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216704BDBM50216704(CHEMBL150751)
Affinity DataIC50: 840nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216708BDBM50216708(CHEMBL151887)
Affinity DataIC50: 880nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216723BDBM50216723(CHEMBL150369)
Affinity DataIC50: 960nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216696BDBM50216696(CHEMBL357952)
Affinity DataIC50: 980nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216716BDBM50216716(CHEMBL348186)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216634BDBM50216634(CHEMBL356655)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216714BDBM50216714(CHEMBL149734)
Affinity DataIC50: 1.08E+3nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216726BDBM50216726(CHEMBL149786)
Affinity DataIC50: 1.15E+3nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216701BDBM50216701(CHEMBL148974)
Affinity DataIC50: 1.17E+3nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216635BDBM50216635(CHEMBL356436)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216719BDBM50216719(CHEMBL348433)
Affinity DataIC50: 1.34E+3nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216707BDBM50216707(CHEMBL422133)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216636BDBM50216636(CHEMBL347337)
Affinity DataIC50: 1.98E+3nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216700BDBM50216700(CHEMBL149264)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216722BDBM50216722(CHEMBL149115)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216695BDBM50216695(CHEMBL149058)
Affinity DataIC50: 8.35E+3nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216679BDBM50216679(CHEMBL149129)
Affinity DataIC50: 9.40E+3nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216710BDBM50216710(CHEMBL345538)
Affinity DataIC50: 1.07E+4nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216720BDBM50216720(CHEMBL149998)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216705BDBM50216705(CHEMBL149943)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216724BDBM50216724(CHEMBL356430)
Affinity DataKi:  6.10E+4nMpH: 7.1Assay Description:Binding affinity was evaluated towards 3-phosphoglycerate kinase at 37 degrees Celsius in 0.1 m NaCl pH 7.1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216699BDBM50216699(CHEMBL147415)
Affinity DataKi:  6.10E+4nMpH: 7.1Assay Description:Binding affinity was evaluated towards 3-phosphoglycerate kinase at 37 degrees Celsius in 0.1 m NaCl pH 7.1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216709BDBM50216709(CHEMBL148780)
Affinity DataIC50: 6.88E+4nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216702BDBM50216702(CHEMBL148792)
Affinity DataIC50: 7.30E+4nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216698BDBM50216698(CHEMBL341829)
Affinity DataKi:  7.50E+4nMpH: 7.1Assay Description:Binding affinity was evaluated towards 3-phosphoglycerate kinase at 37 degrees Celsius in 0.1 m NaCl pH 7.1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216717BDBM50216717(CHEMBL149729)
Affinity DataIC50: 7.80E+4nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216703BDBM50216703(CHEMBL148705)
Affinity DataKi:  8.00E+4nMpH: 7.1Assay Description:Binding affinity was evaluated towards 3-phosphoglycerate kinase at 37 degrees Celsius in 0.1 m NaCl pH 7.1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216724BDBM50216724(CHEMBL356430)
Affinity DataIC50: 8.70E+4nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216699BDBM50216699(CHEMBL147415)
Affinity DataIC50: 8.70E+4nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216713BDBM50216713(CHEMBL345282)
Affinity DataIC50: 8.90E+4nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216715BDBM50216715(CHEMBL151547)
Affinity DataIC50: 9.90E+4nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216694BDBM50216694(CHEMBL150532)
Affinity DataIC50: 1.02E+5nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216712BDBM50216712(CHEMBL149219)
Affinity DataIC50: 1.07E+5nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216711BDBM50216711(CHEMBL147362)
Affinity DataKi:  1.20E+5nMpH: 7.1Assay Description:Binding affinity was evaluated towards 3-phosphoglycerate kinase at 37 degrees Celsius in 0.1 m NaCl pH 7.1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216725BDBM50216725(CHEMBL149333)
Affinity DataIC50: 1.38E+5nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216721BDBM50216721(CHEMBL149259)
Affinity DataIC50: 1.47E+5nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216698BDBM50216698(CHEMBL341829)
Affinity DataIC50: 1.50E+5nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216697BDBM50216697(CHEMBL357982)
Affinity DataKi:  1.56E+5nMpH: 7.1Assay Description:Binding affinity was evaluated towards 3-phosphoglycerate kinase at 37 degrees Celsius in 0.1 m NaCl pH 7.1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216697BDBM50216697(CHEMBL357982)
Affinity DataIC50: 1.63E+5nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216706BDBM50216706(CHEMBL148654)
Affinity DataIC50: 1.81E+5nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216703BDBM50216703(CHEMBL148705)
Affinity DataIC50: 1.82E+5nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216718BDBM50216718(CHEMBL358865)
Affinity DataIC50: 1.93E+5nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed
TargetPhosphoglycerate kinase 1(Human)
Sheffield University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216711BDBM50216711(CHEMBL147362)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibitory activity against 3-phosphoglycerate kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2018
Entry Details Article
PubMed