Compile Data Set for Download or QSAR
Report error Found 149 Enz. Inhib. hit(s) with all data for entry = 11288
TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605125BDBM605125((2S,5S)-5-{(2S,3S)-3-Methyl-2- [(pyridine-4-carbon...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605124BDBM605124((2S,5S)-5-{(2S,3S)-3-Methyl-2- [(pyridine-3-carbon...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605123BDBM605123((2S,5S)-5-{(2S,3S)-3-Methyl-2- [(pyridine-2-carbon...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605122BDBM605122((2S,5S)-5-[(S)-2-(4-Methoxy- benzoylamino)-3-methy...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605128BDBM605128((2S,5S)-5-{(S)-3-Methyl-2-[(pyridine-4- carbonyl)-...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605127BDBM605127((2S,5S)-5-{(S)-3-Methyl-2-[(pyridine-3- carbonyl)-...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605126BDBM605126((2S,5S)-5-{(S)-3-Methyl-2-[(pyridine-2- carbonyl)-...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605133BDBM605133((2S,5S)-5-((S)-2-Benzoylamino-2- cyclopentyl-acety...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605132BDBM605132((2S,5S)-5-[(S)-2-(2-Benzo[b]thiophen-3- yl-acetyla...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605131BDBM605131((2S,5S)-5-((S)-2-Acetylamino-3-ethyl- pentanoylami...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605134BDBM605134((2S,5S)-5-((S)-2-Acetylamino-2- cyclopentyl-acetyl...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605109BDBM605109((2S,5S)-5-[(S)-3-Methyl-2-(4-methyl- benzoylamino)...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605108BDBM605108((2S,5S)-5-[(S)-3-Methyl-2-(3-methyl- benzoylamino)...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605107BDBM605107((2S,5S)-5-[(S)-3-Methyl-2-(2-methyl- benzoylamino)...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605113BDBM605113((2S,5S)-5-{(S)-2-[2-(2-Fluoro-ethoxy)- acetylamino...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605112BDBM605112((2S,5S)-5-((S)-2-Benzoylamino-4,4,4- trifluoro-3-m...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605111BDBM605111((2S,5S)-5-[(2S,3R)-2-(2- Benzo[b]thiophen-3-yl-ace...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605110BDBM605110((2S,5S)-5-((2S,3R)-2-Benzoylamino-3- methyl-pentan...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605117BDBM605117((2S,5S)-5-[(2S,3S)-2-(2-Methoxy- benzoylamino)-3-m...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605116BDBM605116((2S,5S)-5-[(2S,3S)-2-(2-Fluoro- acetylamino)-3-met...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605115BDBM605115(US11667645, Compound C058 | (2S,5S)-5-{(2S,3S)-2-[...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605114BDBM605114((2S,5S)-5-[(S)-2-(2-Fluoro-acetylamino)- 3-methyl-...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605121BDBM605121((2S,SS)-5-[(S)-2-(3-Methoxy- benzoylamino)-3-methy...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605120BDBM605120((2S,5S)-5-[(S)-2-(2-Methoxy- benzoylamino)-3-methy...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605119BDBM605119((2S,5S)-5-[(2S,3S)-2-(4-Methoxy- benzoylamino)-3-m...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605118BDBM605118((2S,5S)-5-[(2S,3S)-2-(3-Methoxy- benzoylamino)-3-m...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605157BDBM605157((1S,8S)-8-((S)-2-Benzoylamino-3- methyl-butyrylami...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605156BDBM605156((1S,8S)-8-{(2S,3S)-2-[2-(2-Fluoro- ethoxy)-acetyla...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605155BDBM605155((1S,8S)-8-[(2S,3S)-2-(2-Fluoro- acetylamino)-3-met...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605154BDBM605154((1S,8S)-8-((2S,3S)-2-Acetylamino-3- methyl-pentano...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605160BDBM605160((1S,8S)-8-{(S)-2-[2-(2-Fluoro-ethoxy)- acetylamino...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605159BDBM605159((1S,8S)-8-[(S)-2-(2-Fluoro-acetylamino)- 3-methyl-...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605158BDBM605158((1S,8S)-8-((S)-2-Acetylamino-3-methyl- butyrylamin...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605141BDBM605141((2S,5S)-5-((S)-2-Benzoylamino-2- cyclobutyl-acetyl...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605140BDBM605140((2S,5S)-5-((S)-2-Acetylamino-2- cyclobutyl-acetyla...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605153BDBM605153((1S,8S)-8-((2S,3S)-2-Benzoylamino-3- methyl-pentan...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605189BDBM605189((3S,6S)-3-{(2S,3S)-2-[2-(2-Fluoro- ethoxy)-acetyla...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605188BDBM605188((2S,5S)-5-{(2S,3S)-2-[(2-Fluoro-pyridine- 4-carbon...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605187BDBM605187((2S,5S)-5-{(2S,3S)-2-[(6-Fluoro-pyridine- 3-carbon...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605192BDBM605192((1S,8S)-8-[(2S,3S)-2-(2- Benzo[b]thiophen-3-yl-ace...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605115BDBM605115(US11667645, Compound C058 | (2S,5S)-5-{(2S,3S)-2-[...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605063BDBM605063((2S,5S)-5-[(2S,3S)-2-(2- Benzo[b]thiophen-3-yl-ace...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605190BDBM605190((3S,6S)-3-{(2S,3S)-2-[2-(2-Fluoro- ethoxy)-acetyla...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605197BDBM605197((2S,5S)-5-[(2S,3S)-2-(2-Benzofuran-2-yl- acetylami...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605196BDBM605196((2S,5S)-5-[(2S,3S)-2-(2- Benzo[b]thiophen-2-yl-ace...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605200BDBM605200((2S,5S)-5-[(2S,3S)-2-(2-1H- Benzoimidazol-2-yl-ace...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605199BDBM605199((2S,5S)-5-[(2S,3S)-2-(2-1H-Indol-2-yl- acetylamino...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605071BDBM605071((2S,5S)-5-((S)-3-Methyl-2- phenylacetylamino-butyr...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605198BDBM605198((2S,5S)-5-[(2S,3S)-2-(2-Benzooxazol-2- yl-acetylam...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

TargetGranzyme B(Human)
Cytosite Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 605175BDBM605175((2S,5S)-5-{(2S,3S)-2-[2-(2-Fluoro- ethoxy)-acetyla...)
Affinity DataIC50: 150nMAssay Description:Buffer pH7.4: Prepare 1 (M) KH2PO4 and 1 (M) K2HPO4. Titrate 1(M) K2HPO4 with 1 (M) KH2PO4 to obtain pH 7.40. Dilute this buffer 10 fold in Water (30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
US Patent

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