Compile Data Set for Download or QSAR
Report error Found 87 Enz. Inhib. hit(s) with all data for entry = 412
LigandPNGBDBM267062(Butyl 4-{[(4,5-dichloro-2-thienyl)sulfonyl]amino}-...)
Affinity DataIC50: 200nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267057(2-Hydroxyethyl 4-{[(5'-fluoro-2'-hydroxybiphenyl-3...)
Affinity DataIC50: 200nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267074(3-Morpholin-4-ylpropyl 4-({[5-chloro-4-(5-fluoro-2...)
Affinity DataIC50: 600nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267054(2-(1H-Pyrrol-1-yl)ethyl 4-{[(4,5-dichlorothiophen-...)
Affinity DataIC50: 600nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267055(2-Methoxyethyl 4-({[3-(2,3-dihydro-1-benzofuran-5-...)
Affinity DataIC50: 700nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267031(4-{[(5-Chloro-4-phenyl-2-thienyl)sulfonyl]amino}-2...)
Affinity DataIC50: 800nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267082(3-[(5-Methylisoxazol-3-yl)amino]propyl 4-{[(5'-flu...)
Affinity DataIC50: 800nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267065(2-Methoxy-1-methylethyl 4-{[(4,5-dichlorothiophen-...)
Affinity DataIC50: 800nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267064(Benzyl 4-{[(4,5-dichloro-2-thienyl)sulfonyl]amino}...)
Affinity DataIC50: 800nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267066(2-Methoxyethyl 4-({[5-chloro-4-(2,3-dihydro-1-benz...)
Affinity DataIC50: 900nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267031(4-{[(5-Chloro-4-phenyl-2-thienyl)sulfonyl]amino}-2...)
Affinity DataIC50: 900nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267068(General Procedure 9 | US9718809, 82)
Affinity DataIC50: 1.08E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267035(2-Methoxyethyl 4-({[5-chloro-4-(2-hydroxyphenyl)-2...)
Affinity DataIC50: 1.20E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267063(1-Methyl-3-morpholin-4-ylpropyl 4-{[(4,5-dichlorot...)
Affinity DataIC50: 1.20E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267030(Methyl 2-hydroxy-4-({[(2'-hydroxybiphenyl-4-yl)met...)
Affinity DataIC50: 1.40E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267061(2-Methoxy-1-(methoxymethyl)ethyl 4-{[(3,5-dichloro...)
Affinity DataIC50: 1.40E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267076(2-Hydroxyethyl 4-{[(5-chloro-4-phenyl-2-thienyl)su...)
Affinity DataIC50: 1.40E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267039(Methyl 2-hydroxy-4-({[3-(piperidin-1-yl)phenyl]sul...)
Affinity DataIC50: 1.50E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267033(Methyl 2-(acetyloxy)-4-{[(4,5-dichlorothiophen-2-y...)
Affinity DataIC50: 1.50E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267071(Methyl 4-[(biphenyl-3-ylsulfonyl)amino]-2-hydroxyb...)
Affinity DataIC50: 1.60E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267077(Methyl 4-({[3-(5-acetyl-2-thienyl)phenyl]sulfonyl}...)
Affinity DataIC50: 1.70E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267025(4-{[(4-Bromo-2,5-dichlorothiophen-3-yl)sulfonyl]am...)
Affinity DataIC50: 1.70E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267024(Methyl 4-({[3-(2,3-dihydro-1-benzofuran-5-yl)-5-(t...)
Affinity DataIC50: 1.70E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267070(1-Benzylpyrrolidin-3-yl 2-hydroxy-4-{[(2,4,5-trich...)
Affinity DataIC50: 1.80E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267021(Methyl 4-[(tert-butoxycarbonyl)amino]-2-hydroxyben...)
Affinity DataIC50: 1.90E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267080(General Procedure 14 | US9718809, 230)
Affinity DataIC50: 1.90E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267026(Methyl 4-({[5-(2,5-difluorophenyl)thiophen-2-yl]su...)
Affinity DataIC50: 2.00E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267049(Methyl 4-({[5-chloro-4-(5-fluoro-2-hydroxyphenyl)-...)
Affinity DataIC50: 2.00E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267078(2-Methoxy-1-(methoxymethyl)ethyl 4-({[5-chloro-4-(...)
Affinity DataIC50: 2.00E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267038(Methyl 4-({[5-(dimethylamino)naphthalen-1-yl]sulfo...)
Affinity DataIC50: 2.10E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267029(Methyl 4-{[(2,5-dichloro-3-thienyl)sulfonyl]amino}...)
Affinity DataIC50: 2.30E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267041(Methyl 4-[({5-chloro-4-[3-(dimethylcarbamoyl)pheny...)
Affinity DataIC50: 2.40E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267079(Methyl 2-hydroxy-4-({[4'-(trifluoromethoxy)bipheny...)
Affinity DataIC50: 2.40E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267057(2-Hydroxyethyl 4-{[(5'-fluoro-2'-hydroxybiphenyl-3...)
Affinity DataIC50: 2.60E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267051(3-Morpholin-4-ylpropyl 4-({[4-(1,3-benzodioxol-5-y...)
Affinity DataIC50: 2.80E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267016(Methyl 4-({[4-(3-aminophenyl)-5-chlorothiophen-2-y...)
Affinity DataIC50: 2.80E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267047(General Procedure 10 | US9718809, 156)
Affinity DataIC50: 2.80E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267048(General Procedure 5 | US9718809, 53)
Affinity DataIC50: 3.10E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267067(2-Methoxyethyl 4-{[(4-bromo-2,5-dichlorothiophen-3...)
Affinity DataIC50: 3.50E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267036(Methyl 4-{[(4-fluoro-1-naphthyl)sulfonyl]amino}-2-...)
Affinity DataIC50: 3.60E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267094(3-Morpholin-4-ylpropyl 4-{[(5'-fluoro-2'-hydroxybi...)
Affinity DataIC50: 3.60E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267056(3-Morpholin-4-ylpropyl 4-{[(4,5-dichlorothiophen-2...)
Affinity DataIC50: 4.00E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267075(Methyl 2-hydroxy-4-{[(3-quinolin-6-ylphenyl)sulfon...)
Affinity DataIC50: 4.50E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267023(Methyl 2-hydroxy-4-({[4-(trifluoromethyl)phenyl]su...)
Affinity DataIC50: 4.60E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267020(Methyl 4-{[(5-chloro-4-pyridin-3-ylthiophen-2-yl)s...)
Affinity DataIC50: 4.60E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267034(Methyl 4-{[(3-chloro-4-fluorophenyl)sulfonyl]amino...)
Affinity DataIC50: 4.80E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267045(Methyl 4-({[6-chloro-5-(2,3-dihydro-1-benzofuran-5...)
Affinity DataIC50: 4.90E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267043(Methyl 4-{[(2',5'-difluorobiphenyl-3-yl)sulfonyl]a...)
Affinity DataIC50: 5.10E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267060(Tetrahydrofuran-3-yl 4-{[(2,5-dichloro-3-thienyl)s...)
Affinity DataIC50: 5.20E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

LigandPNGBDBM267022(Methyl 4-{[(3'-carbamoylbiphenyl-3-yl)sulfonyl]ami...)
Affinity DataIC50: 5.40E+3nMAssay Description:6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFK-2/BPase-2) is a bi-functional enzyme that catalyses the formation and degradation of fructo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
US Patent

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