Compile Data Set for Download or QSAR
Report error Found 56 of affinity data for UniProtKB/TrEMBL: P29410
LigandChemical structure of BindingDB Monomer ID 50367049BDBM50367049(CHEMBL604399)
Affinity DataKi:  60nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of ATP, non competitive inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50367049BDBM50367049(CHEMBL604399)
Affinity DataKi:  60nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of AMP, competitive inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50367044BDBM50367044(CHEMBL605639)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of AMP, competitive inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50367044BDBM50367044(CHEMBL605639)
Affinity DataKi:  2.80E+3nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of AMP, non competitive inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50367040BDBM50367040(CHEMBL606017)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of ATP, non competitive inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50367040BDBM50367040(CHEMBL606017)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of AMP, competitive inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50367048BDBM50367048(CHEMBL605430)
Affinity DataKi:  5.20E+4nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of AMP, competitive inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50010310BDBM50010310(CHEMBL3251359)
Affinity DataKi:  5.50E+4nMAssay Description:Competitive inhibition of Sprague-Dawley rat liver adenylate kinase 2 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50010310BDBM50010310(CHEMBL3251359)
Affinity DataKi:  6.00E+4nMAssay Description:Competitive binding inhibition constant(Ki) of rat adenylate kinase (AK II) isozymes was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50367048BDBM50367048(CHEMBL605430)
Affinity DataKi:  6.30E+4nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of AMP, competitive and non competitive inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50010311BDBM50010311(CHEMBL2364580)
Affinity DataKi:  7.50E+4nMAssay Description:Competitive inhibition of Sprague-Dawley rat liver adenylate kinase 2 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50010309BDBM50010309(CHEMBL3251358)
Affinity DataKi:  8.00E+4nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50010309BDBM50010309(CHEMBL3251358)
Affinity DataKi:  8.00E+4nMAssay Description:Competitive inhibition of Sprague-Dawley rat liver adenylate kinase 2 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 18137BDBM18137(adenosine 5 -monophosphate | CHEMBL752 | [(2R,3S,4...)
Affinity DataKi:  8.00E+4nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of AMPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50010312BDBM50010312(CHEMBL3251360)
Affinity DataKi:  8.00E+4nMAssay Description:Competitive inhibition of Sprague-Dawley rat liver adenylate kinase 2 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50366480BDBM50366480(ATP | ADENOSINE TRIPHOSPHATE)
Affinity DataKi:  9.00E+4nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of ATP, non competitive inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50010314BDBM50010314(CHEMBL3251362)
Affinity DataKi:  1.45E+5nMAssay Description:Competitive inhibition of Sprague-Dawley rat liver adenylate kinase 2 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50010313BDBM50010313(CHEMBL3251361)
Affinity DataKi:  2.50E+5nMAssay Description:Competitive inhibition of Sprague-Dawley rat liver adenylate kinase 2 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50367068BDBM50367068(CHEMBL609795 | CHEMBL3350524)
Affinity DataKi:  3.00E+5nMAssay Description:Ability to inhibit rat adenylate kinase II, activity expressed as Inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50010308BDBM50010308(CHEMBL3251357)
Affinity DataKi:  3.20E+5nMAssay Description:Competitive inhibition of Sprague-Dawley rat liver adenylate kinase 2 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50010315BDBM50010315(CHEMBL3251363)
Affinity DataKi:  3.20E+5nMAssay Description:Competitive inhibition of Sprague-Dawley rat liver adenylate kinase 2 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50010315BDBM50010315(CHEMBL3251363)
Affinity DataKi:  3.20E+5nMAssay Description:Competitive binding inhibition constant (Ki) of rat adenylate kinase (AK II) isozymes was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50367104BDBM50367104(CHEMBL607646)
Affinity DataKi:  3.80E+5nMAssay Description:Competitive inhibitory constant with Rat adenylate kinase II isozymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50367038BDBM50367038(CHEMBL604815)
Affinity DataKi:  4.50E+5nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of ATP, competitive inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50367046BDBM50367046(CHEMBL604395)
Affinity DataKi:  4.50E+5nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of ATP, non competitive inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50367042BDBM50367042(CHEMBL606221)
Affinity DataKi:  5.40E+5nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of ATP, non competitive inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50027451BDBM50027451(Phosphoric acid mono-[5-(6-amino-purin-9-yl)-4-hyd...)
Affinity DataKi:  9.40E+5nMAssay Description:Competitive inhibitory constant with Rat adenylate kinase II isozymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50027422BDBM50027422(1N-{4-[9-(3,4-dihydroxy-5-hydroxymethyltetrahydro-...)
Affinity DataKi:  1.10E+6nMAssay Description:Competitive inhibition of adenylate kinase III in rat liver with respect to ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50367067BDBM50367067(CHEMBL612174 | CHEMBL3350514)
Affinity DataKi:  1.60E+6nMAssay Description:Ability to inhibit rat adenylate kinase II, activity expressed as Inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50367066BDBM50367066(CHEMBL610373 | CHEMBL3350509)
Affinity DataKi:  1.80E+6nMAssay Description:Ability to inhibit rat adenylate kinase II, activity expressed as Inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50367073BDBM50367073(CHEMBL609819 | CHEMBL3350528)
Affinity DataKi:  1.90E+6nMAssay Description:Ability to inhibit rat adenylate kinase II, activity expressed as Inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50367037BDBM50367037(CHEMBL606008)
Affinity DataKi:  2.00E+6nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of ATP, competitive inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50367098BDBM50367098(CHEMBL607630)
Affinity DataKi:  2.10E+6nMAssay Description:Competitive inhibitory constant with Rat adenylate kinase II isozymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50027448BDBM50027448(Phosphoric acid mono-[6-(6-amino-purin-9-yl)-2,2-d...)
Affinity DataKi:  2.10E+6nMAssay Description:Competitive inhibitory constant with Rat adenylate kinase II isozymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50367039BDBM50367039(CHEMBL604398)
Affinity DataKi:  2.20E+6nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50367103BDBM50367103(CHEMBL608483)
Affinity DataKi:  2.40E+6nMAssay Description:Non-competitive/Competitive inhibitory constant of compound with Rat adenylate kinase II isozymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50027455BDBM50027455(Phosphoric acid mono-[6-(6-amino-purin-9-yl)-2-eth...)
Affinity DataKi:  2.70E+6nMAssay Description:Competitive inhibitory constant with Rat adenylate kinase II isozymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50027446BDBM50027446(Phosphoric acid mono-[6-(6-amino-purin-9-yl)-2-met...)
Affinity DataKi:  2.70E+6nMAssay Description:Competitive inhibitory constant with Rat adenylate kinase II isozymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50367045BDBM50367045(CHEMBL605010)
Affinity DataKi:  3.20E+6nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of AMP, non competitive inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50367045BDBM50367045(CHEMBL605010)
Affinity DataKi:  3.20E+6nMAssay Description:Competitive inhibitory constant with Rat adenylate kinase II isozymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50027447BDBM50027447(Phosphoric acid mono-[5-(6-amino-purin-9-yl)-3-hyd...)
Affinity DataKi:  3.60E+6nMAssay Description:Competitive inhibitory constant with Rat adenylate kinase II isozymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50367106BDBM50367106(CHEMBL609083 | CHEMBL1230507)
Affinity DataKi:  4.20E+6nMAssay Description:Competitive inhibitory constant with Rat adenylate kinase II isozymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50367100BDBM50367100(CHEMBL607942)
Affinity DataKi:  5.40E+6nMAssay Description:Competitive inhibitory constant with Rat adenylate kinase II isozymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50367110BDBM50367110(CHEMBL609073)
Affinity DataKi:  5.80E+6nMAssay Description:Competitive inhibitory constant with Rat adenylate kinase II isozymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50367069BDBM50367069(CHEMBL609792 | CHEMBL3350522)
Affinity DataKi:  7.30E+6nMAssay Description:Ability to inhibit rat adenylate kinase II, activity expressed as Inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50367041BDBM50367041(CHEMBL603556)
Affinity DataKi:  9.80E+6nMAssay Description:Competitive inhibitory constant with Rat adenylate kinase II isozymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50367041BDBM50367041(CHEMBL603556)
Affinity DataKi:  9.80E+6nMAssay Description:Inhibitory activity against rat adenylate kinase II was determined in the presence of AMP, non competitive inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50367102BDBM50367102(CHEMBL608353)
Affinity DataKi:  1.14E+7nMAssay Description:Competitive inhibitory constant with Rat adenylate kinase II isozymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50367089BDBM50367089(CHEMBL1788163)
Affinity DataKi:  1.14E+7nMAssay Description:Non competitive binding inhibition constant (Ki) of rat adenylate kinase (AK II) isozymes was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50367088BDBM50367088(CHEMBL1788161)
Affinity DataKi:  1.26E+7nMAssay Description:Non competitive binding inhibition constant (Ki) of rat adenylate kinase (AK II) isozymes was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
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