Affinity DataKi: 11nMAssay Description:Antagonist activity at LPAR1/LPAR3 in rat glioma C62B cells assessed as inhibition of LPA-induced reduction in isoproterenol-stimulated [3H]cAMP accu...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Rattus norvegicus)
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 497nMAssay Description:Activity at LPA1 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Rattus norvegicus)
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 652nMAssay Description:Activity at LPA1 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Rattus norvegicus)
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 1.93E+3nMAssay Description:Activity at LPA1 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Rattus norvegicus)
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Antagonist activity at LPA1 receptor in rat hepatic stellate cells assessed as inhibition of lysophosphatidic acid-induced intracellular calcium infl...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Rattus norvegicus)
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of LPA in rat plasma after 18 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Rattus norvegicus)
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 48nMAssay Description:Antagonist activity at LPA1 receptor in rat hepatic stellate cells assessed as inhibition of lysophosphatidic acid-induced intracellular calcium infl...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Rattus norvegicus)
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 56nMAssay Description:Antagonist activity at LPA1 receptor in rat hepatic stellate cells assessed as inhibition of lysophosphatidic acid-induced intracellular calcium infl...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Rattus norvegicus)
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 72nMAssay Description:Antagonist activity at LPA1 receptor in rat hepatic stellate cells assessed as inhibition of lysophosphatidic acid-induced intracellular calcium infl...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Rattus norvegicus)
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 73nMAssay Description:Antagonist activity at LPA1 receptor in rat hepatic stellate cells assessed as inhibition of lysophosphatidic acid-induced intracellular calcium infl...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Rattus norvegicus)
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 74nMAssay Description:Antagonist activity at LPA1 receptor in rat hepatic stellate cells assessed as inhibition of lysophosphatidic acid-induced intracellular calcium infl...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Rattus norvegicus)
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 81nMAssay Description:Antagonist activity at LPA1 receptor in rat hepatic stellate cells assessed as inhibition of lysophosphatidic acid-induced intracellular calcium infl...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Rattus norvegicus)
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Antagonist activity at LPA1 receptor in rat hepatic stellate cells assessed as inhibition of lysophosphatidic acid-induced intracellular calcium infl...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Rattus norvegicus)
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Antagonist activity at LPA1 receptor in rat hepatic stellate cells assessed as inhibition of lysophosphatidic acid-induced intracellular calcium infl...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Rattus norvegicus)
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Antagonist activity at LPA1 receptor in rat hepatic stellate cells assessed as inhibition of lysophosphatidic acid-induced intracellular calcium infl...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Rattus norvegicus)
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Antagonist activity at LPA1 receptor in rat hepatic stellate cells assessed as inhibition of lysophosphatidic acid-induced intracellular calcium infl...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Rattus norvegicus)
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 915nMAssay Description:Activity at LPA1 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Rattus norvegicus)
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 1.11E+3nMAssay Description:Activity at LPA1 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Rattus norvegicus)
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 4.66E+3nMAssay Description:Activity at LPA1 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Rattus norvegicus)
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: >2.00E+4nMAssay Description:Antagonist activity at LPA1 receptor in rat hepatic stellate cells assessed as inhibition of lysophosphatidic acid-induced intracellular calcium infl...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Rattus norvegicus)
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 981nMAssay Description:Activity at LPA1 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Rattus norvegicus)
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 1.41E+3nMAssay Description:Activity at LPA1 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Rattus norvegicus)
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 1.58E+3nMAssay Description:Activity at LPA1 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Rattus norvegicus)
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 3.60E+3nMAssay Description:Activity at LPA1 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Rattus norvegicus)
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Activity at LPA1 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Rattus norvegicus)
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 1.56E+3nMAssay Description:Activity at LPA1 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Rattus norvegicus)
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 2.26E+3nMAssay Description:Activity at LPA1 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair