Compile Data Set for Download or QSAR
Report error Found 5126 of affinity data for UniProtKB/TrEMBL: Q01959
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50067772(Rhenium complex of 3-(2-Bromo-2,2,2-triformyl-3-me...)
Affinity DataIC50: 0.146nMAssay Description:The compound was tested in vitro for high binding affinity for the Dopamine transporter (DAT) using competitive binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50101075((2S,3S)-methyl 3-(3,4-dichlorophenyl)-8-methyl-8-a...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]CFT from human DAT expressed in COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50004167((2R,3S)-3-(4-Chloro-phenyl)-2-((E)-2-chloro-vinyl)...)
Affinity DataKi:  0.220nMAssay Description:Binding constant for the ability to displace [3H]mazindol to dopamine receptor was calculated from the Cheng-Prusoff relationshipMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50067771(3-(2-Methylsulfanyl-ethylsulfanyl)-propionic acid ...)
Affinity DataIC50: 0.227nMAssay Description:The compound was tested in vitro for high binding affinity for the Dopamine transporter (DAT) using competitive binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50260904((1R,2R,3S,5S)-2-(2,2-dibromovinyl)-8-methyl-3-p-to...)
Affinity DataIC50: 0.230nMAssay Description:Displacement of [3H]WIN-35428 from dopamine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50102589(3-(3,4-Dichloro-phenyl)-7-hydroxy-8-methyl-8-aza-b...)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of [3H]WIN-35428 binding to Dopamine transporter in rhesus (Macaca mulatta) or cynomolgus monkey (Macaca fascicularis) caudate-putamenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50260905((1R,2R,3S,5S)-3-(4-chlorophenyl)-2-(2,2-dibromovin...)
Affinity DataIC50: 0.320nMAssay Description:Displacement of [3H]WIN-35428 from dopamine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50085072(GBR-12909 | 1-{2-[(3-Fluoro-phenyl)-(4-fluoro-phen...)
Affinity DataKi:  0.360nMAssay Description:Competitive binding versus [N-methyl-3H]WIN-35428 in murine kidney cells transfected with human dopamine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50004167((2R,3S)-3-(4-Chloro-phenyl)-2-((E)-2-chloro-vinyl)...)
Affinity DataIC50: 0.360nMAssay Description:Displacement of [3H]mazindol from dopamine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50004167((2R,3S)-3-(4-Chloro-phenyl)-2-((E)-2-chloro-vinyl)...)
Affinity DataIC50: 0.360nMAssay Description:Displacement of [3H]mazindol from dopamine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50334460(RTI-229 | CHEMBL1643896 | ((1R,2S,3S,5S)-3-(4-iodo...)
Affinity DataIC50: 0.370nMAssay Description:Inhibition of DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50323773(N-((E)-4-Fluorobut-2-en-1-yl)-2beta-carbomethoxy-3...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [125I]RTI55 from human DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50183549((S)-(+)-4-[2-[bis-(4-fluorophenyl)methoxy]ethyl]-1...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50035730(3-(3,4-Dichloro-phenyl)-8-methyl-8-aza-bicyclo[3.2...)
Affinity DataIC50: 0.400nMAssay Description:inhibition of [3H]WIN-35428 binding to the dopamine transporter (DAT) in monkey caudate-putamen.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM81946(CAS_96850-13-4 | LU 19-005 | LU 19,005)
Affinity DataKi:  0.410nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2012
Entry Details
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50118598(4-{2-[Bis-(4-fluoro-phenyl)-methoxy]-ethyl}-1-(3-p...)
Affinity DataKi:  0.450nMAssay Description:Binding affinity towards dopamine transporter (DAT) by using [125I]RTI-55 radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50006774(CHEMBL311347 | (2S,3S)-methyl 3-(4-iodophenyl)-8-m...)
Affinity DataKi:  0.480nMAssay Description:Binding affinity to dopamine transporter in membranes of cells selectively expressing the human genes for DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50085071(3-(4-Iodo-phenyl)-6-methyl-6-aza-bicyclo[3.2.2]non...)
Affinity DataKi:  0.480nMAssay Description:In vitro affinity determined using [3H]WIN-35428 in murine kidney cells transfected with human dopamine transporter (DAT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50006774(CHEMBL311347 | (2S,3S)-methyl 3-(4-iodophenyl)-8-m...)
Affinity DataKi:  0.480nMAssay Description:In vitro competitive binding versus [N-methyl-3H]WIN-35428 in murine kidney cells transfected with cDNA for human dopamine transporter (DAT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50063324(8-Methyl-3-naphthalen-2-yl-8-aza-bicyclo[3.2.1]oct...)
Affinity DataIC50: 0.490nMAssay Description:Inhibition of [3H]WIN-35428 binding to the dopamine transporter in cynomolgus (macaca fascicularis) monkey caudate putamen.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50183539(CHEMBL381256 | CHEMBL429492 | trans-(R,R)-4-[2-[bi...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50323774(N-((E)-4-Fluorobut-2-en-1-yl)-2beta-carbomethoxy-3...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [125I]RTI55 from human DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50090975(8-Methyl-3-naphthalen-2-yl-8-aza-bicyclo[3.2.1]oct...)
Affinity DataIC50: 0.570nMAssay Description:Inhibition of [3H]WIN-35428 binding to the dopamine transporter in cynomolgus (macaca fascicularis) monkey caudate putamen.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50063324(8-Methyl-3-naphthalen-2-yl-8-aza-bicyclo[3.2.1]oct...)
Affinity DataIC50: 0.570nMAssay Description:Inhibition of [3H]WIN-35428 binding to Dopamine transporter in rhesus (Macaca mulatta) or cynomolgus monkey (Macaca fascicularis) caudate-putamenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50063324(8-Methyl-3-naphthalen-2-yl-8-aza-bicyclo[3.2.1]oct...)
Affinity DataIC50: 0.570nMAssay Description:Inhibition of [3H]WIN-35428 binding to Dopamine transporter in rhesus (Macaca mulatta) or cynomolgus monkey (Macaca fascicularis) caudate-putamenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50323772(N-((E)-4-Fluorobut-2-en-1-yl)-2beta-carbomethoxy-3...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [125I]RTI55 from human DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50127392(3-(4-Chloro-3-methyl-phenyl)-8-methyl-8-aza-bicycl...)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of dopamine (DA) reuptake using cloned human dopamine transporter was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50046734(3-(3,4-Dichloro-phenyl)-8-aza-bicyclo[3.2.1]octane...)
Affinity DataIC50: 0.660nMAssay Description:Inhibition of [3H]3-beta-(4-fluorophenyl)tropane-2beta-carboxylic acid methyl ester binding to dopamine transporter of cynomolgus monkey striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50106857(3-(4-Iodo-phenyl)-8-aza-bicyclo[3.2.1]octane-2-car...)
Affinity DataKi:  0.690nMAssay Description:In vitro binding affinity against human dopamine transporter in dog kidney cell line by using [125I]RTI-55 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM160629(US9045468, 45)
Affinity DataIC50: 0.700nMpH: 7.9 T: 2°CAssay Description:Compounds were dissolved in 100% DMSO at a concentration 100 times the desired highest assay concentration, serially diluted 1:3 in 100% DMSO, and 0....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2015
Entry Details
US Patent

TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM22165(Vanoxerine | CHEMBL542933 | GBR-12909 | CHEMBL5438...)
Affinity DataIC50: 0.710nMAssay Description:Displacement of [125I]RTI-55 from recombinant human DAT expressed in CHOK1 cells after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/25/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50118599(4-(2-(bis(4-fluorophenyl)methoxy)ethyl)-1-(naphtha...)
Affinity DataKi:  0.710nMAssay Description:Binding affinity towards dopamine transporter (DAT) by using [125I]RTI-55 radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50118600(2-((4-(2-(bis(4-fluorophenyl)methoxy)ethyl)piperid...)
Affinity DataKi:  0.730nMAssay Description:Binding affinity towards dopamine transporter (DAT) by using [125I]RTI-55 radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50349803(CHEMBL1812741)
Affinity DataIC50: 0.75nMAssay Description:Inhibition of human DAT expressed in HEK293 cells assessed as inhibition of [3H]DA reuptake after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2013
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50102564(3-(3,4-Dichloro-phenyl)-7-hydroxy-8-methyl-8-aza-b...)
Affinity DataIC50: 0.760nMAssay Description:Inhibition of [3H]WIN-35428 binding to Dopamine transporter in rhesus (Macaca mulatta) or cynomolgus monkey (Macaca fascicularis) caudate-putamenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM375641(US9908897, Example 21)
Affinity DataIC50: 0.776nMAssay Description:The affinity of the compounds of the invention to the human DAT or NET or SERT transporters is assessed by using the [3H]WIN-35,428 or [3H]nisoxetine...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2020
Entry Details
US Patent

TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50260934(3beta-(4-Chlorophenyl)-2beta-(phenylethynyl)tropan...)
Affinity DataIC50: 0.800nMAssay Description:Displacement of [3H]WIN-35428 from dopamine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50260933(3beta-(4-Methylphenyl)-2beta-(phenylethynyl)tropan...)
Affinity DataIC50: 0.800nMAssay Description:Displacement of [3H]WIN-35428 from dopamine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50183535((R)-(+)-4-[2-[bis-(4-fluorophenyl)methoxy]ethyl]-1...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50199786(CHEMBL3918282)
Affinity DataKi:  0.806nMAssay Description:Inhibition of [3H]dopamine uptake from wild type human DAT expressed in COS-7 cells preincubated for 30 mins followed by [3H]dopamine addition and me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50273607((1R,2S,3S,5R)-methyl 3-(4-chloro-3-methylphenyl)-8...)
Affinity DataIC50: 0.820nMAssay Description:Displacement of [3H]WIN-35428 from DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50349805(CHEMBL1812739)
Affinity DataIC50: 0.830nMAssay Description:Inhibition of human DAT expressed in HEK293 cells assessed as inhibition of [3H]DA reuptake after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2013
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50363762(CHEMBL1947088)
Affinity DataKi:  0.870nMAssay Description:Displacement of [3H]WIN35428 from human cloned DAT receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50004167((2R,3S)-3-(4-Chloro-phenyl)-2-((E)-2-chloro-vinyl)...)
Affinity DataKi:  0.880nMAssay Description:Binding constant for [3H]dopamine uptake was calculated from the Cheng-Prusoff relationshipMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM376888(4-(aminomethyl)-1-[2,3-difluoro-5-(3-fluorophenoxy...)
Affinity DataIC50: 0.891nMAssay Description:The affinity of the compounds of the invention to the human DAT or NET or SERT transporters is assessed by using the [3H]WIN-35,428 or [3H]nisoxetine...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50085069(3-(4-Chloro-phenyl)-6-methyl-6-aza-bicyclo[3.2.2]n...)
Affinity DataKi:  0.900nMAssay Description:Inhibition constant against [N-methyl-3H]WIN-35428 in murine kidney cells transfected with human dopamine transporter.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50260935(3beta-(4-Chlorophenyl)-2beta-(4-nitrophenylethynyl...)
Affinity DataIC50: 0.900nMAssay Description:Displacement of [3H]WIN-35428 from dopamine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50177110(2-beta-(4-fluorophenyl)-3-beta-(4-methylphenyl)tro...)
Affinity DataIC50: 0.900nMAssay Description:Displacement of [3H]WIN-35428 from DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50183540((S)-(-)-4-[2-[bis-(4-fluorophenyl)methoxy]ethyl]-1...)
Affinity DataKi:  0.900nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Institut F£R Bioanorganische Und Radiopharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50183545(R-(-)-4-[2-[bis-(4-fluorophenyl)methoxy]ethyl]-1-(...)
Affinity DataKi:  0.900nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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