Affinity DataEC50: >5.00E+5nMAssay Description:In vitro evaluation for inhibitor of human topoisomerase II from HeLa cells.More data for this Ligand-Target Pair
Affinity DataEC50: >2.50E+5nMAssay Description:In vitro evaluation for inhibitor of human topoisomerase II from HeLa cells.More data for this Ligand-Target Pair
Affinity DataEC50: >2.10E+5nMAssay Description:In vitro evaluation for inhibitor of human topoisomerase II from HeLa cells.More data for this Ligand-Target Pair
Affinity DataEC50: 2.00E+4nMAssay Description:In vitro evaluation for inhibitor of human topoisomerase II from HeLa cells.More data for this Ligand-Target Pair
Affinity DataEC50: >2.20E+5nMAssay Description:In vitro evaluation for inhibitor of human topoisomerase II from HeLa cells.More data for this Ligand-Target Pair
Affinity DataEC50: 550nMAssay Description:In vitro evaluation for inhibitor of human topoisomerase II from HeLa cells.More data for this Ligand-Target Pair
Affinity DataEC50: 9.00E+4nMAssay Description:In vitro evaluation for inhibitor of human topoisomerase II from HeLa cells.More data for this Ligand-Target Pair
Affinity DataEC50: >2.20E+5nMAssay Description:In vitro evaluation for inhibitor of human topoisomerase II from HeLa cells.More data for this Ligand-Target Pair
Affinity DataEC50: 1.60E+3nMAssay Description:In vitro evaluation for inhibitor of human topoisomerase II from HeLa cells.More data for this Ligand-Target Pair
Affinity DataEC50: 5.10E+5nMAssay Description:In vitro evaluation for inhibitor of human topoisomerase II from HeLa cells.More data for this Ligand-Target Pair
Affinity DataEC50: 500nMAssay Description:In vitro evaluation for inhibitor of human topoisomerase II from HeLa cells.More data for this Ligand-Target Pair
Affinity DataEC50: 330nMAssay Description:In vitro evaluation for inhibitor of human topoisomerase II from HeLa cells.More data for this Ligand-Target Pair
Affinity DataEC50: >2.40E+5nMAssay Description:In vitro evaluation for inhibitor of human topoisomerase II from HeLa cells.More data for this Ligand-Target Pair
Affinity DataEC50: >2.30E+5nMAssay Description:In vitro evaluation for inhibitor of human topoisomerase II from HeLa cells.More data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+4nMAssay Description:In vitro evaluation for inhibitor of human topoisomerase II from HeLa cells.More data for this Ligand-Target Pair
Affinity DataEC50: >2.60E+5nMAssay Description:In vitro evaluation for inhibitor of human topoisomerase II from HeLa cells.More data for this Ligand-Target Pair
Affinity DataEC50: >2.20E+5nMAssay Description:In vitro evaluation for inhibitor of human topoisomerase II from HeLa cells.More data for this Ligand-Target Pair
Affinity DataEC50: >4.80E+5nMAssay Description:In vitro evaluation for inhibitor of human topoisomerase II from HeLa cells.More data for this Ligand-Target Pair
Affinity DataEC50: >2.70E+5nMAssay Description:In vitro evaluation for inhibitor of human topoisomerase II from HeLa cells.More data for this Ligand-Target Pair
Affinity DataEC50: 720nMAssay Description:In vitro inhibitior of human DNA topoisomerase II from HeLa cells.More data for this Ligand-Target Pair
Affinity DataEC50: >2.60E+5nMAssay Description:In vitro evaluation for inhibitor of human topoisomerase II from HeLa cells.More data for this Ligand-Target Pair
Affinity DataEC50: >2.10E+5nMAssay Description:In vitro evaluation for inhibitor of human topoisomerase II from HeLa cells.More data for this Ligand-Target Pair
Affinity DataEC50: >2.40E+5nMAssay Description:In vitro evaluation for inhibitor of human topoisomerase II from HeLa cells.More data for this Ligand-Target Pair
Affinity DataEC50: 3.00E+3nMAssay Description:In vitro evaluation for inhibitor of human topoisomerase II from HeLa cells.More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Concentration of compound at which inhibitory activity detected against DNA topoisomerase IIMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Concentration of compound at which inhibitory activity detected against DNA topoisomerase IIMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Concentration of compound at which inhibitory activity detected against DNA topoisomerase IIMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Concentration of compound at which inhibitory activity detected against DNA topoisomerase IIMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+3nMAssay Description:Concentration of compound at which inhibitory activity detected against DNA topoisomerase IIMore data for this Ligand-Target Pair
Affinity DataEC50: 5.60E+3nMAssay Description:Concentration of compound at which inhibitory activity detected against DNA topoisomerase IIMore data for this Ligand-Target Pair
Affinity DataEC50: 5.60E+4nMAssay Description:In vitro inhibitory activity against DNA topoisomerase IIMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Concentration of compound at which inhibitory activity detected against DNA topoisomerase IIMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Concentration of compound at which inhibitory activity detected against DNA topoisomerase IIMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+3nMAssay Description:Concentration of compound at which inhibitory activity detected against DNA topoisomerase IIMore data for this Ligand-Target Pair
Affinity DataEC50: 5.60E+4nMAssay Description:Concentration of compound at which inhibitory activity detected against DNA topoisomerase IIMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Concentration of compound at which inhibitory activity detected against DNA topoisomerase IIMore data for this Ligand-Target Pair
Affinity DataEC50: 7.60E+3nMAssay Description:Inhibitory activity in a DNA cleavage assay using HeLa DNA topoisomerase II yielding its effective concentrationMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+4nMAssay Description:In vitro activity against topoisomerase-2 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+4nMAssay Description:In vitro activity against topoisomerase-2 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+4nMAssay Description:In vitro activity against topoisomerase-2 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+4nMAssay Description:In vitro activity against topoisomerase-2 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+4nMAssay Description:In vitro activity against topoisomerase-2 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+4nMAssay Description:In vitro activity against topoisomerase-2 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+4nMAssay Description:In vitro activity against topoisomerase-2 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+4nMAssay Description:In vitro activity against topoisomerase-2 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+4nMAssay Description:In vitro activity against topoisomerase-2 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+4nMAssay Description:In vitro activity against topoisomerase-2 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+4nMAssay Description:In vitro activity against topoisomerase-2 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+4nMAssay Description:In vitro activity against topoisomerase-2 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+4nMAssay Description:In vitro activity against topoisomerase-2 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair




















3D Structure (crystal)


























