Compile Data Set for Download or QSAR
maximum 50k data
Found 243 with Last Name = 'giridhar' and Initial = 'r'
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50131385((2R,3R,4R,5S)-3,4,5-Trihydroxy-1-(4-phenoxy-benzen...)
Affinity DataKi:  0.0610nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50004154(2-Butyl-4-chloro-6-methyl-1-[2'-(1H-tetrazol-5-yl)...)
Affinity DataKi:  1nMAssay Description:Binding affinity to angiotensin AT1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50030727(4''-[3-Butyl-5-oxo-1-(2-trifluoromethyl-phenyl)-1,...)
Affinity DataKi:  1.70nMAssay Description:Binding affinity to angiotensin AT1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50131385((2R,3R,4R,5S)-3,4,5-Trihydroxy-1-(4-phenoxy-benzen...)
Affinity DataKi:  2.30nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM11548(CHEMBL100570 | N-hydroxy-2-[(4-methoxy-1,1-bipheny...)
Affinity DataKi:  3.80nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50044739(3-Butyl-2-[2'-(1H-tetrazol-5-yl)-biphenyl-4-yloxy]...)
Affinity DataKi:  4.5nMAssay Description:Binding affinity to angiotensin AT2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50247674(2-[7-(3,5-Dimethoxy-benzyloxy)-1,1-dioxo-1,3,4,5-t...)
Affinity DataKi:  5nMAssay Description:Inhibition of pig TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50335930(CHEMBL1668000 | N-(4'-((3-butyl-6,9-dioxo-2,3-diaz...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-angiotensin 2 from angiotensin AT1 receptor in human PLC-PRF5 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50039342(5-Methyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataKi:  24nMAssay Description:Binding affinity to angiotensin AT1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50335929(2-((2'-(1H-tetrazol-5-yl)biphenyl-4-yl)methyl)-3-b...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]-angiotensin 2 from angiotensin AT1 receptor in human PLC-PRF5 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50335923(1-(2'-(1H-tetrazol-5-yl)biphenyl-4-yl)-2,2-difluor...)
Affinity DataKi:  29nMAssay Description:Binding affinity to angiotensin AT1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM11548(CHEMBL100570 | N-hydroxy-2-[(4-methoxy-1,1-bipheny...)
Affinity DataKi:  46.7nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM11548(CHEMBL100570 | N-hydroxy-2-[(4-methoxy-1,1-bipheny...)
Affinity DataKi:  55nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50335923(1-(2'-(1H-tetrazol-5-yl)biphenyl-4-yl)-2,2-difluor...)
Affinity DataKi:  480nMAssay Description:Binding affinity to angiotensin AT2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
The M. S. University of Baroda

LigandPNGBDBM86095(2-Cyanopyrrolidine Derivative, 24)
Affinity DataKi:  5.30E+3nM ΔG°:  -29.9kJ/molepH: 6.0 T: 2°CAssay Description:The fluorescence for the assay was monitored on a Varian Gemini spectrofluorometer with the excitation and emission wavelengths at 380 and 440nm. Th...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
The M. S. University of Baroda

LigandPNGBDBM86096(2-Cyanopyrrolidine Derivative, 25)
Affinity DataKi:  8.60E+3nM ΔG°:  -28.7kJ/molepH: 6.0 T: 2°CAssay Description:The fluorescence for the assay was monitored on a Varian Gemini spectrofluorometer with the excitation and emission wavelengths at 380 and 440nm. Th...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
The M. S. University of Baroda

LigandPNGBDBM86094(2-Cyanopyrrolidine Derivative, 23)
Affinity DataKi:  6.70E+4nM ΔG°:  -23.7kJ/molepH: 6.0 T: 2°CAssay Description:The fluorescence for the assay was monitored on a Varian Gemini spectrofluorometer with the excitation and emission wavelengths at 380 and 440nm. Th...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
The M. S. University of Baroda

LigandPNGBDBM86099(2-Cyanopyrrolidine Derivative, 28)
Affinity DataKi:  7.50E+4nM ΔG°:  -23.4kJ/molepH: 6.0 T: 2°CAssay Description:The fluorescence for the assay was monitored on a Varian Gemini spectrofluorometer with the excitation and emission wavelengths at 380 and 440nm. Th...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
The M. S. University of Baroda

LigandPNGBDBM86093(2-Cyanopyrrolidine Derivative, 22)
Affinity DataKi:  8.50E+4nM ΔG°:  -23.1kJ/molepH: 6.0 T: 2°CAssay Description:The fluorescence for the assay was monitored on a Varian Gemini spectrofluorometer with the excitation and emission wavelengths at 380 and 440nm. Th...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
The M. S. University of Baroda

LigandPNGBDBM86094(2-Cyanopyrrolidine Derivative, 23)
Affinity DataKi:  9.20E+4nM ΔG°:  -22.9kJ/molepH: 6.0 T: 2°CAssay Description:The fluorescence for the assay was monitored on a Varian Gemini spectrofluorometer with the excitation and emission wavelengths at 380 and 440nm. Th...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
The M. S. University of Baroda

LigandPNGBDBM86096(2-Cyanopyrrolidine Derivative, 25)
Affinity DataKi: >1.00E+5nM ΔG°: >-22.7kJ/molepH: 6.0 T: 2°CAssay Description:The fluorescence for the assay was monitored on a Varian Gemini spectrofluorometer with the excitation and emission wavelengths at 380 and 440nm. Th...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
The M. S. University of Baroda

LigandPNGBDBM86095(2-Cyanopyrrolidine Derivative, 24)
Affinity DataKi: >1.00E+5nM ΔG°: >-22.7kJ/molepH: 6.0 T: 2°CAssay Description:The fluorescence for the assay was monitored on a Varian Gemini spectrofluorometer with the excitation and emission wavelengths at 380 and 440nm. Th...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
The M. S. University of Baroda

LigandPNGBDBM86100(2-Cyanopyrrolidine Derivative, 29)
Affinity DataKi: >1.00E+5nM ΔG°: >-22.7kJ/molepH: 6.0 T: 2°CAssay Description:The fluorescence for the assay was monitored on a Varian Gemini spectrofluorometer with the excitation and emission wavelengths at 380 and 440nm. Th...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
The M. S. University of Baroda

LigandPNGBDBM86100(2-Cyanopyrrolidine Derivative, 29)
Affinity DataKi: >1.00E+5nM ΔG°: >-22.7kJ/molepH: 6.0 T: 2°CAssay Description:The fluorescence for the assay was monitored on a Varian Gemini spectrofluorometer with the excitation and emission wavelengths at 380 and 440nm. Th...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
The M. S. University of Baroda

LigandPNGBDBM86098(2-Cyanopyrrolidine Derivative, 27)
Affinity DataKi: >1.00E+5nM ΔG°: >-22.7kJ/molepH: 6.0 T: 2°CAssay Description:The fluorescence for the assay was monitored on a Varian Gemini spectrofluorometer with the excitation and emission wavelengths at 380 and 440nm. Th...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
The M. S. University of Baroda

LigandPNGBDBM86097(2-Cyanopyrrolidine Derivative, 26)
Affinity DataKi: >1.00E+5nM ΔG°: >-22.7kJ/molepH: 6.0 T: 2°CAssay Description:The fluorescence for the assay was monitored on a Varian Gemini spectrofluorometer with the excitation and emission wavelengths at 380 and 440nm. Th...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
The M. S. University of Baroda

LigandPNGBDBM86097(2-Cyanopyrrolidine Derivative, 26)
Affinity DataKi: >1.00E+5nM ΔG°: >-22.7kJ/molepH: 6.0 T: 2°CAssay Description:The fluorescence for the assay was monitored on a Varian Gemini spectrofluorometer with the excitation and emission wavelengths at 380 and 440nm. Th...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
The M. S. University of Baroda

LigandPNGBDBM86098(2-Cyanopyrrolidine Derivative, 27)
Affinity DataKi: >1.00E+5nM ΔG°: >-22.7kJ/molepH: 6.0 T: 2°CAssay Description:The fluorescence for the assay was monitored on a Varian Gemini spectrofluorometer with the excitation and emission wavelengths at 380 and 440nm. Th...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
The M. S. University of Baroda

LigandPNGBDBM86099(2-Cyanopyrrolidine Derivative, 28)
Affinity DataKi: >1.00E+5nM ΔG°: >-22.7kJ/molepH: 6.0 T: 2°CAssay Description:The fluorescence for the assay was monitored on a Varian Gemini spectrofluorometer with the excitation and emission wavelengths at 380 and 440nm. Th...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
The M. S. University of Baroda

LigandPNGBDBM86093(2-Cyanopyrrolidine Derivative, 22)
Affinity DataKi: >1.00E+5nM ΔG°: >-22.7kJ/molepH: 6.0 T: 2°CAssay Description:The fluorescence for the assay was monitored on a Varian Gemini spectrofluorometer with the excitation and emission wavelengths at 380 and 440nm. Th...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50195927(CHEMBL391851 | N-(5-methyl-2,4,6-trioxo-hexahydrop...)
Affinity DataIC50:  0.0260nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50044402(2-Butyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataIC50:  0.0550nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortic strip assessed as inhibition of angiotensin 2-induced contractile responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50247788((2R,3S)-N1-((S)-3-(4-guanidinophenyl)-1-(methylami...)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50229322((3S,4S)-N-hydroxy-4-(4-((2-methylquinolin-4-yl)met...)
Affinity DataIC50:  0.140nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50247606((R)-2-((R)-3-amino-3-(4-((2-methylquinolin-4-yl)me...)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50041677(2-{2-Butyl-4-oxo-3-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50:  0.200nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50009718(2-Ethyl-5,7-dimethyl-3-[2'-(1H-tetrazol-5-yl)-biph...)
Affinity DataIC50:  0.200nMAssay Description:Binding affinity to angiotensin AT2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50038189(4'-(2-Ethyl-5,7-dimethyl-imidazo[4,5-b]pyridin-3-y...)
Affinity DataIC50:  0.200nMAssay Description:Binding affinity to angiotensin AT1 receptor in rabbit aortic ringsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50009718(2-Ethyl-5,7-dimethyl-3-[2'-(1H-tetrazol-5-yl)-biph...)
Affinity DataIC50:  0.300nMAssay Description:Binding affinity to angiotensin AT1 receptor in rabbit aortic ringsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50287290(CHEMBL34866 | KRH-594 | Potassium; 2-[5-ethyl-3-[2...)
Affinity DataIC50:  0.400nMAssay Description:Antagonist activity at angiotensin AT1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50042534(2-Benzyl-5-propyl-4-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataIC50:  0.420nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50042580(2-Butyl-5-(2-chloro-phenyl)-3-[2'-(1H-tetrazol-5-y...)
Affinity DataIC50:  0.550nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aorta assessed as reduction of angiotensin 2-induced contractile responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50282383(2-Ethyl-5,7-dimethyl-3-[2'-(2-oxo-2,3-dihydro-2lam...)
Affinity DataIC50:  0.700nMAssay Description:Binding affinity to angiotensin AT1 receptor in rabbit aortic ringsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50335928((R)-1-((2'-(1H-tetrazol-5-yl)biphenyl-4-yl)methyl)...)
Affinity DataIC50:  0.770nMAssay Description:Binding affinity to angiotensin AT1 receptor in rabbit aortic ringsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50043450(3,6-Dichloro-2-[5-(2-ethyl-5,7-dimethyl-3H-imidazo...)
Affinity DataIC50:  0.800nMAssay Description:Binding affinity to angiotensin AT1 receptor in rabbit aortic ringsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50043434(2-Ethyl-5,7-dimethyl-4-{1-[phenyl-(1H-tetrazol-5-y...)
Affinity DataIC50:  1nMAssay Description:Binding affinity to angiotensin AT1 receptor in rabbit aortic ringsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM26526((2R)-N-hydroxy-2-[(3S)-3-methyl-3-{4-[(2-methylqui...)
Affinity DataIC50:  1nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50247605((R)-N-hydroxy-2-(3-methyl-1-(4-((2-methylquinolin-...)
Affinity DataIC50:  1nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50152901(1-Methyl-2-[4-(2-methyl-quinolin-4-ylmethoxy)-benz...)
Affinity DataIC50:  1nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50167485(5-Methyl-5-[4-(2-methyl-quinolin-4-ylmethoxy)-phen...)
Affinity DataIC50:  1nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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