BindingDB PrimarySearch

BDBM17657 (2S)-2-aminopentanedioic acid::(S)-Glu::D-Glutamate::Glutamate::L-Glu::L-Glutamate::L-Glutamic acid::L-[14C(U)]glutamate::L-gluatmate

SMILES: C(CC(=O)O)[C@@H](C(=O)O)N

InChI Key: InChIKey=WHUUTDBJXJRKMK-UHFFFAOYSA-N

Data: 92 KI 23 IC50 121 EC50

PDB links: 31 PDB IDs match this monomer.

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 236 hits for monomerid = 17657
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Glutamate carboxypeptidase 2 [44-750] (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	4.28E+5	n/a	n/a	n/a	n/a	7.4	37
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Excitatory amino acid transporter 4 (Rat)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	1.30E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Excitatory amino acid transporter 4 (Rat)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	1.32E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Excitatory amino acid transporter 2 (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	5.25E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Excitatory amino acid transporter 3 (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	3.24E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Excitatory amino acid transporter 1 (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	1.10E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Excitatory amino acid transporter 3 (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	3.20E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Excitatory amino acid transporter 2 (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	5.20E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Excitatory amino acid transporter 1 (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	1.15E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Prolyl 4-hydroxylase (PBCV-1)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	>1.00E+6	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Glutamate receptor 3 (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	2.34E+4	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Glutamate receptor 4 (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	4.80E+3	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Glutamate receptor 3 (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	2.40E+4	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Glutamate receptor 2 (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	5.62E+4	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Glutamate receptor 2 (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	5.70E+4	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Glutamate receptor 4 (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	4.90E+3	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Glutamate receptor 1 (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	3.30E+4	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Glutamate receptor 1 (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	3.31E+4	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Metabotropic glutamate receptor 5 (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	1.60E+4	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Excitatory amino acid transporter 4 (Rat)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	1.20E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Excitatory amino acid transporter 4 (Rat)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	1.26E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Excitatory amino acid transporter 1 (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	1.12E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Excitatory amino acid transporter 1 (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	1.10E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Excitatory amino acid transporter 2 (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	8.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Excitatory amino acid transporter 2 (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	7.94E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Excitatory amino acid transporter 3 (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	5.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Excitatory amino acid transporter 3 (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	5.01E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Glutamate receptor ionotropic, NMDA 2A (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	70	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Glutamate receptor 1 (Rat)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	6.40E+3	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Glutamate receptor 3 (Rat)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	1.30E+3	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Glutamate receptor 1 (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	2.20E+4	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Glutamate receptor 2 (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	6.20E+3	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Glutamate receptor 3 (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	3.50E+4	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Glutamate receptor 1 (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	2.26E+3	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Glutamate receptor 2 (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	2.19E+3	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Glutamate receptor 3 (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	3.66E+3	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Glutamate receptor 1 (Rat)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	5.10E+4	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Glutamate receptor 2 (Rat)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	1.90E+5	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Glutamate receptor 3 (Rat)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	5.20E+4	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Glutamate receptor 4 (Rat)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	2.00E+4	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Metabotropic glutamate receptor 2 (Rat)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	610	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Metabotropic glutamate receptor 3 (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	2.50E+3	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Glutamate receptor ionotropic, kainate 1 (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	7.50E+4	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Glutamate receptor ionotropic, kainate 2 (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	2.50E+4	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Glutamate receptor ionotropic, kainate 1 (Rat)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	3.52E+4	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Metabotropic glutamate receptor 1 (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	1.05E+3	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Metabotropic glutamate receptor 8 (Rat)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	8.00E+3	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Metabotropic glutamate receptor 1 (Rat)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	3.00E+3	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Metabotropic glutamate receptor 2 (Rat)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	1.60E+4	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Metabotropic glutamate receptor 2 (Human)	BDBM17657 (L-Glutamic acid \| L-Glu \| (2S)-2-aminopentanedioic...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	7.40E+3	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair

Displayed 1 to 50 (of 236 total ) | Next | Last >>