Compile Data Set for Download or QSAR
maximum 50k data
Found 31 Enz. Inhib. hit(s) with all data for entry = 50043076
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435635(CHEMBL2391601)
Affinity DataEC50:  24nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435665(CHEMBL2391602)
Affinity DataEC50:  310nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435637(CHEMBL2391599)
Affinity DataEC50:  300nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435638(CHEMBL2391598)
Affinity DataEC50:  89nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435639(CHEMBL2391597)
Affinity DataEC50:  68nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435640(CHEMBL2391596)
Affinity DataEC50:  91nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435641(CHEMBL2391595)
Affinity DataEC50:  450nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435642(CHEMBL2391594)
Affinity DataEC50:  160nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435643(CHEMBL2391593)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435644(CHEMBL2391592)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435645(CHEMBL2391436)
Affinity DataEC50:  610nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435646(CHEMBL2391435)
Affinity DataEC50:  2.95E+3nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435647(CHEMBL2391434)
Affinity DataEC50:  350nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435648(CHEMBL2391433)
Affinity DataEC50:  31nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435649(CHEMBL2391432)
Affinity DataEC50:  2.74E+3nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435650(CHEMBL2391431)
Affinity DataEC50:  4.00E+3nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435651(CHEMBL2391430)
Affinity DataEC50:  130nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435652(CHEMBL2391429)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435653(CHEMBL2391614)
Affinity DataEC50:  2.06E+3nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435654(CHEMBL2391613)
Affinity DataEC50:  2.12E+3nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435655(CHEMBL2391612)
Affinity DataEC50:  1.71E+3nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435656(CHEMBL2391611)
Affinity DataEC50:  440nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435657(CHEMBL2391610)
Affinity DataEC50:  380nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435658(CHEMBL2391609)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435659(CHEMBL2391608)
Affinity DataEC50:  960nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435660(CHEMBL2391607)
Affinity DataEC50:  380nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435661(CHEMBL2391606)
Affinity DataEC50:  270nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435662(CHEMBL2391605)
Affinity DataEC50:  810nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435663(CHEMBL2391604)
Affinity DataEC50:  660nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435664(CHEMBL2391603)
Affinity DataEC50:  8.40E+3nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435636(CHEMBL2391600)
Affinity DataEC50:  1.06E+3nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed