Compile Data Set for Download or QSAR
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Found 24 Enz. Inhib. hit(s) with all data for entry = 50013856
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135494(4-(5-Fluoro-3-methyl-benzo[b]thiophene-2-sulfonyla...)
Affinity DataIC50:  56nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135493(5-Fluoro-3-methyl-benzo[b]thiophene-2-sulfonic aci...)
Affinity DataIC50:  82nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135496(CHEMBL130156 | [4-(5-Fluoro-3-methyl-benzo[b]thiop...)
Affinity DataIC50:  154nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135499(2-[4-(5-Fluoro-3-methyl-benzo[b]thiophene-2-sulfon...)
Affinity DataIC50:  159nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135509(5-Fluoro-3-methyl-benzo[b]thiophene-2-sulfonic aci...)
Affinity DataIC50:  192nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135495(4-(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonyla...)
Affinity DataIC50:  203nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135502(3-Methanesulfonyl-4-(3-methyl-benzo[b]thiophene-2-...)
Affinity DataIC50:  305nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135497(4-(3,5-Dimethyl-benzo[b]thiophene-2-sulfonylamino)...)
Affinity DataIC50:  325nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135506(5-Fluoro-3-methyl-benzo[b]thiophene-2-sulfonic aci...)
Affinity DataIC50:  337nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135501(4-(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonyla...)
Affinity DataIC50:  594nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135505(4-(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonyla...)
Affinity DataIC50:  663nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135507(4-(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonyla...)
Affinity DataIC50:  880nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135498(4-(5-Fluoro-3-methyl-benzo[b]thiophene-2-sulfonyla...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135508(4-(5-Fluoro-3-methyl-benzo[b]thiophene-2-sulfonyla...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135495(4-(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonyla...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity of the compound against bovin chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135494(4-(5-Fluoro-3-methyl-benzo[b]thiophene-2-sulfonyla...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity of the compound against human cathepsin GMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135495(4-(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonyla...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity of the compound against human cathepsin GMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135494(4-(5-Fluoro-3-methyl-benzo[b]thiophene-2-sulfonyla...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity of the compound against bovin chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135493(5-Fluoro-3-methyl-benzo[b]thiophene-2-sulfonic aci...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity of the compound against bovin chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135493(5-Fluoro-3-methyl-benzo[b]thiophene-2-sulfonic aci...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity of the compound against human cathepsin GMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135503(5-Fluoro-3-methyl-benzo[b]thiophene-2-sulfonic aci...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135504(4-(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonyla...)
Affinity DataIC50:  1.65E+3nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50135500(4-(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonyla...)
Affinity DataIC50:  4.21E+3nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Toa Eiyo

Curated by ChEMBL
LigandPNGBDBM50121657(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonic aci...)
Affinity DataIC50:  1.06E+4nMAssay Description:In vitro inhibitory activity against human chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed