Compile Data Set for Download or QSAR
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Found 55 Enz. Inhib. hit(s) with all data for entry = 50015054
TargetMelanocortin receptor 5(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150842(4-[((R)-N-Cyclohexyl-3-methyl-piperazine-1-carboxi...)
Affinity DataKi:  2.10nMAssay Description:Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150835(4-[N''-(2-Amino-2-methyl-propyl)-N''''-cyclohexyl-...)
Affinity DataKi:  5.30nMAssay Description:Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150837(4-[((S)-N-(R)-Cyclohexyl-2,5-dimethyl-piperazine-1...)
Affinity DataKi:  5.90nMAssay Description:Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150829(4-[(N-Cyclohexyl-3,5-dimethyl-piperazine-1-carboxi...)
Affinity DataKi:  11nMAssay Description:Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150830(4-[(N-Cyclohexyl-piperazine-1-carboximidoyl)-amino...)
Affinity DataKi:  18nMAssay Description:Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150833(4-[((S)-N-Cyclohexyl-3-methyl-piperazine-1-carboxi...)
Affinity DataKi:  21nMAssay Description:Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150836(4-(N''-Cyclohexyl-N''''-pyrrolidin-3-yl-guanidino)...)
Affinity DataKi:  26nMAssay Description:Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150831(4-[(N-Cyclohexyl-3-methylamino-pyrrolidine-1-carbo...)
Affinity DataKi:  36nMAssay Description:Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150840(4-[(4-Benzyl-N-cyclohexyl-piperazine-1-carboximido...)
Affinity DataKi:  44nMAssay Description:Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150834(4-[(N-Cyclohexyl-4-methyl-piperazine-1-carboximido...)
Affinity DataKi:  50nMAssay Description:Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150849(4-[N''-Cyclohexyl-N''''-(3,5-difluoro-benzyl)-guan...)
Affinity DataKi:  70nMAssay Description:Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150845(4-[(N-Cyclohexyl-4-pyrrolidin-1-yl-piperidine-1-ca...)
Affinity DataKi:  77nMAssay Description:Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150847(CHEMBL184612 | N-[2-(2,4-Dichloro-phenyl)-ethyl]-4...)
Affinity DataKi:  91nMAssay Description:Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150839(4-[(N-Cyclohexyl-3,5-dimethyl-piperidine-1-carboxi...)
Affinity DataKi:  144nMAssay Description:Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150832(4-[(4-Amino-N-cyclohexyl-piperidine-1-carboximidoy...)
Affinity DataKi:  230nMAssay Description:Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150838(4-[(N-Cyclohexyl-4-phenyl-piperazine-1-carboximido...)
Affinity DataKi:  290nMAssay Description:Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150844(4-[(N-Cyclohexyl-4-pyrimidin-2-yl-piperazine-1-car...)
Affinity DataKi:  305nMAssay Description:Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150850(4-[(N-Cyclohexyl-2,6-dimethyl-morpholine-4-carboxi...)
Affinity DataKi:  350nMAssay Description:Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150843(4-(N''''-Cyclohexyl-N'',N''-dipropyl-guanidino)-N-...)
Affinity DataKi:  360nMAssay Description:Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150837(4-[((S)-N-(R)-Cyclohexyl-2,5-dimethyl-piperazine-1...)
Affinity DataKi:  360nMAssay Description:Binding affinity for human melanocortin 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150830(4-[(N-Cyclohexyl-piperazine-1-carboximidoyl)-amino...)
Affinity DataKi:  400nMAssay Description:Binding affinity for human melanocortin 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150848(4-[(N-Cyclohexyl-3-oxo-piperazine-1-carboximidoyl)...)
Affinity DataKi:  560nMAssay Description:Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150833(4-[((S)-N-Cyclohexyl-3-methyl-piperazine-1-carboxi...)
Affinity DataKi:  580nMAssay Description:Binding affinity for human melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150829(4-[(N-Cyclohexyl-3,5-dimethyl-piperazine-1-carboxi...)
Affinity DataKi:  590nMAssay Description:Binding affinity for human melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150830(4-[(N-Cyclohexyl-piperazine-1-carboximidoyl)-amino...)
Affinity DataKi:  650nMAssay Description:Binding affinity for human melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150842(4-[((R)-N-Cyclohexyl-3-methyl-piperazine-1-carboxi...)
Affinity DataKi:  840nMAssay Description:Binding affinity for human melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150837(4-[((S)-N-(R)-Cyclohexyl-2,5-dimethyl-piperazine-1...)
Affinity DataKi:  840nMAssay Description:Binding affinity for human melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150841(4-[(N-Cyclohexyl-2-methyl-3-oxo-piperazine-1-carbo...)
Affinity DataKi:  1.05E+3nMAssay Description:Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150835(4-[N''-(2-Amino-2-methyl-propyl)-N''''-cyclohexyl-...)
Affinity DataKi:  1.30E+3nMAssay Description:Binding affinity for human melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150831(4-[(N-Cyclohexyl-3-methylamino-pyrrolidine-1-carbo...)
Affinity DataKi:  1.40E+3nMAssay Description:Binding affinity for human melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150836(4-(N''-Cyclohexyl-N''''-pyrrolidin-3-yl-guanidino)...)
Affinity DataKi:  1.50E+3nMAssay Description:Binding affinity for human melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150846(4-{[N-Cyclohexyl-4-(2,5-dimethyl-phenyl)-piperazin...)
Affinity DataKi:  1.76E+3nMAssay Description:Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150836(4-(N''-Cyclohexyl-N''''-pyrrolidin-3-yl-guanidino)...)
Affinity DataKi:  1.90E+3nMAssay Description:Binding affinity for human melanocortin 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150830(4-[(N-Cyclohexyl-piperazine-1-carboximidoyl)-amino...)
Affinity DataKi:  2.20E+3nMAssay Description:Binding affinity for human melanocortin 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150831(4-[(N-Cyclohexyl-3-methylamino-pyrrolidine-1-carbo...)
Affinity DataKi:  2.30E+3nMAssay Description:Binding affinity for human melanocortin 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150835(4-[N''-(2-Amino-2-methyl-propyl)-N''''-cyclohexyl-...)
Affinity DataKi:  2.40E+3nMAssay Description:Binding affinity for human melanocortin 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150836(4-(N''-Cyclohexyl-N''''-pyrrolidin-3-yl-guanidino)...)
Affinity DataKi:  2.50E+3nMAssay Description:Binding affinity for human melanocortin 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150833(4-[((S)-N-Cyclohexyl-3-methyl-piperazine-1-carboxi...)
Affinity DataKi:  2.80E+3nMAssay Description:Binding affinity for human melanocortin 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150837(4-[((S)-N-(R)-Cyclohexyl-2,5-dimethyl-piperazine-1...)
Affinity DataKi:  2.80E+3nMAssay Description:Binding affinity for human melanocortin 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150842(4-[((R)-N-Cyclohexyl-3-methyl-piperazine-1-carboxi...)
Affinity DataKi:  3.50E+3nMAssay Description:Binding affinity for human melanocortin 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150829(4-[(N-Cyclohexyl-3,5-dimethyl-piperazine-1-carboxi...)
Affinity DataKi:  3.90E+3nMAssay Description:Binding affinity for human melanocortin 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150842(4-[((R)-N-Cyclohexyl-3-methyl-piperazine-1-carboxi...)
Affinity DataIC50:  70nMAssay Description:Inhibition of human Melanocortin 5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150829(4-[(N-Cyclohexyl-3,5-dimethyl-piperazine-1-carboxi...)
Affinity DataIC50:  80nMAssay Description:Inhibition of [125I]NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150837(4-[((S)-N-(R)-Cyclohexyl-2,5-dimethyl-piperazine-1...)
Affinity DataIC50:  380nMAssay Description:Inhibition of human Melanocortin 5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150833(4-[((S)-N-Cyclohexyl-3-methyl-piperazine-1-carboxi...)
Affinity DataIC50:  380nMAssay Description:Inhibition of [125I]NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150830(4-[(N-Cyclohexyl-piperazine-1-carboximidoyl)-amino...)
Affinity DataIC50:  460nMAssay Description:Inhibition of [125I]NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150835(4-[N''-(2-Amino-2-methyl-propyl)-N''''-cyclohexyl-...)
Affinity DataIC50:  530nMAssay Description:Inhibition of [125I]NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150836(4-(N''-Cyclohexyl-N''''-pyrrolidin-3-yl-guanidino)...)
Affinity DataIC50:  530nMAssay Description:Inhibition of [125I]NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150831(4-[(N-Cyclohexyl-3-methylamino-pyrrolidine-1-carbo...)
Affinity DataIC50:  630nMAssay Description:Inhibition of human Melanocortin 5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50150835(4-[N''-(2-Amino-2-methyl-propyl)-N''''-cyclohexyl-...)
Affinity DataEC50:  2.90E+3nMAssay Description:Binding affinity for human melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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