Compile Data Set for Download or QSAR
Report error Found 26 of affinity data for UniProtKB/TrEMBL: Q5U431
TargetG-protein coupled receptor 39(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50030783BDBM50030783(CHEMBL3342370)
Affinity DataEC50:  0.5nMAssay Description:Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetG-protein coupled receptor 39(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50030782BDBM50030782(CHEMBL3342371)
Affinity DataEC50:  1nMAssay Description:Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetG-protein coupled receptor 39(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50030776BDBM50030776(CHEMBL3342377)
Affinity DataEC50:  2nMAssay Description:Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetG-protein coupled receptor 39(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232391BDBM50232391(CHEMBL4100119)
Affinity DataEC50:  2.60nMAssay Description:Agonist activity at mouse GPR39 expressed in HEK293 cells co-expressing Galphaq assessed as myo-[2-3H]inositol phosphate accumulation in presence of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2019
Entry Details Article
PubMed
TargetG-protein coupled receptor 39(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50030786BDBM50030786(CHEMBL3342367)
Affinity DataEC50:  3nMAssay Description:Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetG-protein coupled receptor 39(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50030789BDBM50030789(CHEMBL3341764)
Affinity DataEC50:  3nMAssay Description:Agonist activity at mouse GPR39 by IP1 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetG-protein coupled receptor 39(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50030790BDBM50030790(CHEMBL3342357)
Affinity DataEC50:  4nMAssay Description:Agonist activity at mouse GPR39 by IP1 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetG-protein coupled receptor 39(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232401BDBM50232401(CHEMBL4077818)
Affinity DataEC50:  5nMAssay Description:Agonist activity at mouse GPR39 expressed in HEK293 cells co-expressing Galphaq assessed as myo-[2-3H]inositol phosphate accumulation in presence of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2019
Entry Details Article
PubMed
TargetG-protein coupled receptor 39(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50030779BDBM50030779(CHEMBL3342374)
Affinity DataEC50:  7nMAssay Description:Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetG-protein coupled receptor 39(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50030775BDBM50030775(CHEMBL3342378)
Affinity DataEC50:  8nMAssay Description:Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetG-protein coupled receptor 39(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50030777BDBM50030777(CHEMBL3342376)
Affinity DataEC50:  8nMAssay Description:Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetG-protein coupled receptor 39(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50030787BDBM50030787(CHEMBL3342366)
Affinity DataEC50:  10nMAssay Description:Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetG-protein coupled receptor 39(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50030781BDBM50030781(CHEMBL3342372)
Affinity DataEC50:  17nMAssay Description:Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetG-protein coupled receptor 39(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50030770BDBM50030770(CHEMBL3342362)
Affinity DataEC50:  22nMAssay Description:Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetG-protein coupled receptor 39(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50030780BDBM50030780(CHEMBL3342373)
Affinity DataEC50:  34nMAssay Description:Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetG-protein coupled receptor 39(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50030773BDBM50030773(CHEMBL3342359)
Affinity DataEC50:  115nMAssay Description:Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetG-protein coupled receptor 39(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232401BDBM50232401(CHEMBL4077818)
Affinity DataEC50:  180nMAssay Description:Agonist activity at mouse GPR39 expressed in HEK293 cells co-expressing Galphaq assessed as myo-[2-3H]inositol phosphate accumulation measured after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2019
Entry Details Article
PubMed
TargetG-protein coupled receptor 39(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50030778BDBM50030778(CHEMBL3342375)
Affinity DataEC50:  185nMAssay Description:Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetG-protein coupled receptor 39(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50030785BDBM50030785(CHEMBL3342368)
Affinity DataEC50:  304nMAssay Description:Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetG-protein coupled receptor 39(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50030767BDBM50030767(CHEMBL3342365)
Affinity DataEC50:  365nMAssay Description:Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetG-protein coupled receptor 39(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232367BDBM50232367(CHEMBL4093273)
Affinity DataEC50:  380nMAssay Description:Agonist activity at mouse GPR39 expressed in HEK293 cells co-expressing Galphaq assessed as myo-[2-3H]inositol phosphate accumulation measured after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2019
Entry Details Article
PubMed
TargetG-protein coupled receptor 39(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50030772BDBM50030772(CHEMBL3342360)
Affinity DataEC50:  1.50E+3nMAssay Description:Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetG-protein coupled receptor 39(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50030784BDBM50030784(CHEMBL3342369)
Affinity DataEC50:  2.61E+3nMAssay Description:Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetG-protein coupled receptor 39(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50030768BDBM50030768(CHEMBL3342364)
Affinity DataEC50:  6.72E+3nMAssay Description:Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetG-protein coupled receptor 39(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50030769BDBM50030769(CHEMBL3342363)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetG-protein coupled receptor 39(Mouse)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50030771BDBM50030771(CHEMBL3342361)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed