BDBM25761 Anapriline::Avlocardyl::CHEMBL27::PROPANOLOL(-)::PROPRANOLOL, d::PROPRANOLOL, l-::PROPRANOLOL,(+)::PROPRANOLOL,(-)::Propanolol::Propanolol,(+/-)::Propranolol::[2-hydroxy-3-(naphthalen-1-yloxy)propyl](propan-2-yl)amine
SMILES CC(C)NCC(O)COc1cccc2ccccc12
InChI Key InChIKey=AQHHHDLHHXJYJD-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 21 hits for monomerid = 25761
Affinity DataKi: 6.5nMAssay Description:Evaluated for beta-receptor affinity determined in rat brain membrane fraction with [3H]- dihydroalprenololMore data for this Ligand-Target Pair
Affinity DataKd: 2.40nMAssay Description:Antagonism of the isoprenaline-induced positive chronotropic effect on the atria of guinea pigMore data for this Ligand-Target Pair
Affinity DataKd: 8.70nMAssay Description:Antagonist activity of compound against Beta-1 adrenergic receptor in isolated guinea pig left atriaMore data for this Ligand-Target Pair
Affinity DataKd: 2nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparationMore data for this Ligand-Target Pair
Affinity DataKd: 1.70nMAssay Description:In vitro beta-1 adrenergic receptor activity was determined via inhibition of the positive chronotropic actions of isoproterenol in isolated guinea p...More data for this Ligand-Target Pair
Affinity DataKd: 2.40nMAssay Description:Beta-1 adrenergic receptor blocking activity in atria of guinea pig.More data for this Ligand-Target Pair
Affinity DataKd: 3.10nMAssay Description:Compound was evaluated for competitive antagonism of beta-1 adrenergic receptor in guinea pig atria measured as pA2 (-log KB)More data for this Ligand-Target Pair
Affinity DataKd: 3.39nMAssay Description:The apparent pA2 value was measured for beta-2 adrenergic blocking activity on the trachea of guinea pigMore data for this Ligand-Target Pair
Affinity DataKd: 43.6nMAssay Description:Antagonist activity of compound against Beta-2 adrenergic receptor in isolated guinea pig tracheaMore data for this Ligand-Target Pair
Affinity DataKd: 1.26nMAssay Description:Ability to block Beta-2 adrenergic receptor in guinea pig trachea preparationMore data for this Ligand-Target Pair
Affinity DataKd: 3.02nMAssay Description:In vitro beta-2 adrenergic receptor activity was determined by measuring inhibition of the isoproterenol induced relaxation in isolated guinea pig tr...More data for this Ligand-Target Pair
Affinity DataKd: 3.39nMAssay Description:Beta-2 adrenergic receptor blocking activity in trachea of guinea pig.More data for this Ligand-Target Pair
Affinity DataKd: 1.78nMAssay Description:Compound was evaluated for competitive antagonism of beta-2 adrenergic receptor in rat uterus measured as pA2 (-log KB)More data for this Ligand-Target Pair