BDBM50005410 CHEMBL139197::CHEMBL2137199
SMILES OC(c1ccc(c(F)c1)-c1ccc(CN2CCN(Cc3ccncc3)CC2)cc1)(C(F)(F)F)C(F)(F)F
InChI Key InChIKey=KVHKWAZUPPBMLL-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50005410
Affinity DataKi: 105nMAssay Description:Binding affinity to RORc (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Displacement of [3H]T0901317 from human RoRc expressed in HepG2 cells by scintillation proximity binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 320nMAssay Description:Agonist activity at RoRc-LBD (unknown origin) expressed in HEK293 cells assessed as transcriptional activity by GAL4 reporter assayMore data for this Ligand-Target Pair