BDBM50005410 CHEMBL139197::CHEMBL2137199
SMILES OC(c1ccc(c(F)c1)-c1ccc(CN2CCN(Cc3ccncc3)CC2)cc1)(C(F)(F)F)C(F)(F)F
InChI Key InChIKey=KVHKWAZUPPBMLL-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50005410
Affinity DataIC50: 110nMAssay Description:Inhibition of Gal4-RORgamma-LBD (180 to 507 residues) (unknown origin) expressed in HEK293T cells after 24 hrs by dual-luciferase reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 910nMAssay Description:Displacement of N-terminal biotinylated SRC1-4 coactivator peptide from N-terminal His6-fused human RORgamma-LBD (262 to 507 residues) expressed in E...More data for this Ligand-Target Pair