BDBM50318633 3-benzenesulfonyl-8-piperazin-1-ylquinoline::CHEMBL1083390::SB-742457
SMILES O=S(=O)(c1ccccc1)c1cnc2c(cccc2c1)N1CCNCC1
InChI Key InChIKey=JJZFWROHYSMCMU-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50318633
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]-LSD from human 5HT6R expressed in HEK293 cell membranes incubated for 1 hr by micro-beta plate reader based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5HT2A expressed in HEK293 cell membranes incubated for 1 hr by micro-beta plate reader based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 997nMAssay Description:Displacement of [3H]-raclopride from human D2L expressed in CHO-K1 cell membranes incubated for 1 hr by micro-beta plate reader based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.37E+3nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5HT1A expressed in HEK293 cell membranes incubated for 1 hr by micro-beta plate reader based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.42E+4nMAssay Description:Displacement of [3H]-5-CT from human 5HT7b expressed in HEK293 cell membranes incubated for 1 hr by micro-beta plate reader based analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMAssay Description:Inverse agonist activity at 5HT6R (unknown origin) expressed in 1321N1 cells co-expressing CAMYEL assessed as reduction in basal cAMP accumulation by...More data for this Ligand-Target Pair