Compile Data Set for Download or QSAR
Report error Found 1052 Enz. Inhib. hit(s) with Target = 'B2 bradykinin receptor'
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074991((E)-Penta-2,4-dienoic acid ({[2,4-dichloro-3-(2-me...)
Affinity DataEC50:  260nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074994(5-[({[4-Methoxy-3-(2-methyl-quinolin-8-yloxymethyl...)
Affinity DataEC50:  480nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074992((E)-N-({[4-Chloro-2-methoxy-3-(2-methyl-quinolin-8...)
Affinity DataEC50:  55nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074997((E)-3-(6-Acetylamino-pyridin-3-yl)-N-({[4-methoxy-...)
Affinity DataEC50:  59nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074983((E)-N-({[2-Chloro-4-methoxy-3-(2-methyl-quinolin-8...)
Affinity DataEC50:  130nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074990(4-[3-({[4-Chloro-2-cyano-3-(2-methyl-quinolin-8-yl...)
Affinity DataEC50:  400nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074982((E)-N-({[2,4-Dichloro-3-(2-methyl-benzothiazol-4-y...)
Affinity DataEC50:  54nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074995((E)-N-({[2-Methoxy-3-(2-methyl-quinolin-8-yloxymet...)
Affinity DataEC50:  1.10E+3nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074979((E)-3-(4-Methoxy-phenyl)-N-({methyl-[3-(2-methyl-q...)
Affinity DataEC50:  660nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074998((E)-N-({[4-Methoxy-3-(2-methyl-quinolin-8-yloxymet...)
Affinity DataEC50:  220nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50075000((E)-N-({[4-Chloro-2-cyano-3-(2-methyl-quinolin-8-y...)
Affinity DataEC50:  4.10nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074978(2-[3-(4-Amino-butyl)-ureido]-N-[4-chloro-2-cyano-3...)
Affinity DataEC50:  350nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074986(N-(2-((4-chloro-2-cyano-3-((2-methylquinolin-8-ylo...)
Affinity DataEC50:  56nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074980((E)-N-({[2,4-Dichloro-3-(2-methyl-benzothiazol-4-y...)
Affinity DataEC50:  100nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074999(N-[4-Chloro-2-cyano-3-(2-methyl-quinolin-8-yloxyme...)
Affinity DataEC50:  290nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074984((E)-N-({[2,4-Dichloro-3-(2-methyl-benzothiazol-4-y...)
Affinity DataEC50:  23nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074989((E)-N-({[2,4-Dichloro-3-(2-phenyl-benzothiazol-4-y...)
Affinity DataEC50:  2.00E+4nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074987(N-[2-Cyano-4-methoxy-3-(2-methyl-quinolin-8-yloxym...)
Affinity DataEC50:  450nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074988((E)-N-({[3-(Benzothiazol-4-yloxymethyl)-2,4-dichlo...)
Affinity DataEC50:  1.30E+3nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093761(1-[(R)-5-Amino-1-(4-aminomethyl-benzylcarbamoyl)-p...)
Affinity DataKd:  2.80E+4nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093760(4-Aminomethyl-N-(3-amino-propyl)-N-(2,2-dibutyl-be...)
Affinity DataKd:  1.40E+4nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093759((R)-3-Amino-N-(4-aminomethyl-benzyl)-2-{2-[(2-cycl...)
Affinity DataKd:  1.70E+4nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093762(3-Aminomethyl-1-(3-amino-propyl)-7-dibenzylamino-5...)
Affinity DataKd:  4.30E+3nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093763(N-{3-[7-Dibenzylamino-3-(2-guanidino-ethyl)-2-oxo-...)
Affinity DataKd:  4.50E+3nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093764(cyclic nonapeptide analogue | CHEMBL2369879)
Affinity DataKd:  200nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cells; 0.2-16More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093765((R)-3-Amino-N-(4-aminomethyl-benzyl)-2-{2-[(2-cycl...)
Affinity DataKd:  1.01E+5nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093767(1-(3-Aminomethyl-benzyl)-6,6-dibenzyl-1,4,5,6-tetr...)
Affinity DataKd:  7.60E+3nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093766(((2R,4R)-2-Aminomethyl-4-benzyloxy-pyrrolidin-1-yl...)
Affinity DataKd:  6.60E+4nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093768(5-Dibutylamino-pentanoic acid [(S)-1-(4-butyl-pyri...)
Affinity DataKd:  2.30E+4nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50218386(CHEMBL3142416)
Affinity DataKd:  200nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cells; 0.2-16More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093770(4-Aminomethyl-N-[(S)-1-(4-butyl-pyridin-2-yl)-2-cy...)
Affinity DataKd:  7.40E+3nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093771(N-[(S)-1-(4-Butyl-pyridin-2-yl)-2-cyclohexyl-ethyl...)
Affinity DataKd:  5.00E+3nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093772(N-[3-(7-Dibenzylamino-3-guanidinomethyl-2-oxo-5-ph...)
Affinity DataKd:  1.20E+4nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093773(3-(2-Amino-ethyl)-1-(3-amino-propyl)-7-dibenzylami...)
Affinity DataKd:  1.50E+4nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093774(N-[(2R,4R)-4-Benzyloxy-1-(naphthalene-2-carbonyl)-...)
Affinity DataKd:  1.50E+4nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093775(5-Amino-pentanoic acid [(S)-1-(4-butyl-pyridin-2-y...)
Affinity DataKd:  6.20E+4nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50093776(4-Aminomethyl-N-(2,2-dibutyl-benzo[1,3]dioxol-4-yl...)
Affinity DataKd:  1.30E+4nMAssay Description:Compound was assayed for binding against the human Bradykinin receptor B2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rabbit)
Institute De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50407804(CHEMBL406472)
Affinity DataKd:  3.39E+3nMAssay Description:In vitro antagonistic activity against kinin-induced rabbit jugular vein contraction.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rabbit)
Institute De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50407806(CHEMBL304374)
Affinity DataKd:  468nMAssay Description:In vitro antagonistic activity against kinin-induced rabbit jugular vein contraction.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rabbit)
Institute De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50407815(CHEMBL65100)
Affinity DataKd:  363nMAssay Description:In vitro antagonistic activity against kinin-induced rabbit jugular vein contraction.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rabbit)
Institute De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50407816(CHEMBL63532)
Affinity DataKd:  3.02E+3nMAssay Description:In vitro antagonistic activity against kinin-induced rabbit jugular vein contraction.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rabbit)
Institute De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50407817(CHEMBL294278)
Affinity DataKd:  251nMAssay Description:In vitro antagonistic activity against kinin-induced rabbit jugular vein contraction.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50408044(CHEMBL3038104)
Affinity DataKd:  174nMAssay Description:In vitro Bradykinin receptor B2 antagonist activity by using rat uterus functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50408045(CHEMBL2372278)
Affinity DataKd:  0.490nMAssay Description:In vitro Bradykinin receptor B2 antagonist activity by using rat uterus functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50408047(CHEMBL3038096)
Affinity DataKd:  18.6nMAssay Description:In vitro Bradykinin receptor B2 antagonist activity by using rat uterus functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50408053(CHEMBL3038094)
Affinity DataKd:  3.16nMAssay Description:In vitro Bradykinin receptor B2 antagonist activity by using rat uterus functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50408055(CHEMBL3038102)
Affinity DataKd:  50.1nMAssay Description:In vitro Bradykinin receptor B2 antagonist activity by using rat uterus functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50408815(B-9430 | CHEMBL384857)
Affinity DataKd:  6.31nMAssay Description:Antagonistic activity against Bradykinin receptor B2 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50408806(B-9858 | CHEMBL410358)
Affinity DataKd:  3.16E+3nMAssay Description:Antagonistic activity against Bradykinin receptor B2 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50413782(CHEMBL1627325)
Affinity DataEC50:  0.0339nMAssay Description:Antagonist activity at human recombinant bradykinin 2 receptor expressed in CHO cells assessed as inhibition of bradykinin-induced intracellular calc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
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