Compile Data Set for Download or QSAR
Report error Found 282 Enz. Inhib. hit(s) with Target = 'Beta-1/Beta-2/Beta-3 adrenergic receptor'
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50007477(CHEMBL10453 | 4-(3-tert-Butylamino-2-hydroxy-propo...)
Affinity DataEC50:  9.20nMAssay Description:Beta adrenergic receptor agonistic activity for the stimulation of accumulation of cyclic AMP in cultured C6 glioma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50007476(CHEMBL266619 | 4-(3-tert-Butylamino-2-hydroxy-prop...)
Affinity DataEC50:  8.20nMAssay Description:Beta adrenergic receptor agonistic activity for the stimulation of accumulation of cyclic AMP in cultured C6 glioma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataEC50:  7nMAssay Description:Beta adrenergic receptor agonistic activity for the stimulation of accumulation of cyclic AMP in cultured C6 glioma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50019060(CHEMBL287587 | 4-(2-Amino-1-hydroxy-ethyl)-3-fluor...)
Affinity DataEC50:  2.00E+3nMAssay Description:Displacement of [3H]dihydroalprenolol from beta-adrenergic receptor in Sprague-Dawley rat cerebral cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM35234(Noradrenaline,(+) | NOREPINEPHRINE | DL-[7-3H]nore...)
Affinity DataEC50:  5.00E+3nMAssay Description:Agonist activity at beta-adrenergic receptor in Sprague-Dawley rat cerebral cortex assessed as [3H]cAMP accumulation by liquid scintillation spectros...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50042998(5-(2-Amino-1-hydroxy-ethyl)-3-fluoro-benzene-1,2-d...)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at beta-adrenergic receptor in Sprague-Dawley rat cerebral cortex assessed as [3H]cAMP accumulation by liquid scintillation spectros...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50019061(CHEMBL281232 | 4-(2-Amino-1-hydroxy-ethyl)-5-fluor...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at beta-adrenergic receptor in Sprague-Dawley rat cerebral cortex assessed as [3H]cAMP accumulation by liquid scintillation spectros...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50019061(CHEMBL281232 | 4-(2-Amino-1-hydroxy-ethyl)-5-fluor...)
Affinity DataEC50: >1.00E+5nMAssay Description:Displacement of [3H]dihydroalprenolol from beta-adrenergic receptor in Sprague-Dawley rat cerebral cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM35234(Noradrenaline,(+) | NOREPINEPHRINE | DL-[7-3H]nore...)
Affinity DataEC50:  800nMAssay Description:Displacement of [3H]dihydroalprenolol from beta-adrenergic receptor in Sprague-Dawley rat cerebral cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50019060(CHEMBL287587 | 4-(2-Amino-1-hydroxy-ethyl)-3-fluor...)
Affinity DataEC50:  5.00E+3nMAssay Description:Agonist activity at beta-adrenergic receptor in Sprague-Dawley rat cerebral cortex assessed as [3H]cAMP accumulation by liquid scintillation spectros...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50042998(5-(2-Amino-1-hydroxy-ethyl)-3-fluoro-benzene-1,2-d...)
Affinity DataEC50:  4.00E+3nMAssay Description:Displacement of [3H]dihydroalprenolol from beta-adrenergic receptor in Sprague-Dawley rat cerebral cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50106979(4-(4-{2-[(R)-2-Hydroxy-2-(4-hydroxy-3-methanesulfo...)
Affinity DataEC50:  10nMAssay Description:In vitro agonistic activity against cAMP accumulation level in CHO cells expressing human beta-AR receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50106973(4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-propy...)
Affinity DataEC50:  77nMAssay Description:In vitro agonistic activity against cAMP accumulation level in CHO cells expressing human beta-AR receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50029050(4-[(1R)-1-hydroxy-2-(methylamino)ethyl]benzene-1,2...)
Affinity DataEC50:  230nMAssay Description:Agonistic potency at beta adrenergic receptor for the stimulation of accumulation of cyclic AMP in cultured C6 glioma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50019057((+/-)4-Fluoro-5-(1-hydroxy-2-methylamino-ethyl)-be...)
Affinity DataEC50: >1.50E+3nMAssay Description:Agonistic potency at beta adrenergic receptor for the stimulation of accumulation of cyclic AMP in cultured C6 glioma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50019059(3-Fluoro-4-(1-hydroxy-2-methylamino-ethyl)-benzene...)
Affinity DataEC50:  40nMAssay Description:Agonistic potency at beta adrenergic receptor for the stimulation of accumulation of cyclic AMP in cultured C6 glioma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50019057((+/-)4-Fluoro-5-(1-hydroxy-2-methylamino-ethyl)-be...)
Affinity DataEC50: >1.50E+3nMAssay Description:Stimulation of cyclic AMP accumulation in C6 glioma cells expressing adrenergic beta receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50019060(CHEMBL287587 | 4-(2-Amino-1-hydroxy-ethyl)-3-fluor...)
Affinity DataEC50:  63nMAssay Description:Stimulation of cyclic AMP accumulation in C6 glioma cells expressing adrenergic beta receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50019059(3-Fluoro-4-(1-hydroxy-2-methylamino-ethyl)-benzene...)
Affinity DataEC50:  40nMAssay Description:Stimulation of cyclic AMP accumulation in C6 glioma cells expressing adrenergic beta receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50042997(4-(2-Amino-1-hydroxy-ethyl)-3,5-difluoro-benzene-1...)
Affinity DataEC50: >1.00E+5nMAssay Description:Stimulation of cyclic AMP accumulation in C6 glioma cells expressing adrenergic beta receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50019061(CHEMBL281232 | 4-(2-Amino-1-hydroxy-ethyl)-5-fluor...)
Affinity DataEC50: >1.00E+4nMAssay Description:Stimulation of cyclic AMP accumulation in C6 glioma cells expressing adrenergic beta receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50029050(4-[(1R)-1-hydroxy-2-(methylamino)ethyl]benzene-1,2...)
Affinity DataEC50:  230nMAssay Description:Stimulation of cyclic AMP accumulation in C6 glioma cells expressing adrenergic beta receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50029051(4-[(1R)-2-amino-1-hydroxyethyl]benzene-1,2-diol | ...)
Affinity DataEC50:  52nMAssay Description:Stimulation of cyclic AMP accumulation in C6 glioma cells expressing adrenergic beta receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50212978(CHEMBL541542)
Affinity DataEC50: >3.00E+4nMAssay Description:Beta-adrenergic agonistic activity in guinea-pig atrium preincubated with phenoxybenzamine (12 uM) for 30 minMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2018
Entry Details

TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50212979(CHEMBL543333)
Affinity DataEC50: >3.00E+4nMAssay Description:Beta-adrenergic agonistic activity in guinea-pig atrium preincubated with phenoxybenzamine (12 uM) for 30 minMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2018
Entry Details

TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50212980(CHEMBL553039 | SR-58997A)
Affinity DataEC50: >3.00E+4nMAssay Description:Beta-adrenergic agonistic activity in guinea-pig atrium preincubated with phenoxybenzamine (12 uM) for 30 minMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2018
Entry Details

TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50212977(AMIBEGRON HYDROCHLORIDE | Amibegron HCl | SR-58611...)
Affinity DataEC50: >3.00E+4nMAssay Description:Beta-adrenergic agonistic activity in guinea-pig atrium preincubated with phenoxybenzamine (12 uM) for 30 minMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2018
Entry Details

TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50212981(CHEMBL543099 | SR-59062A)
Affinity DataEC50: >3.00E+4nMAssay Description:Beta-adrenergic agonistic activity in guinea-pig atrium preincubated with phenoxybenzamine (12 uM) for 30 minMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2018
Entry Details

TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50212977(AMIBEGRON HYDROCHLORIDE | Amibegron HCl | SR-58611...)
Affinity DataEC50: >3.00E+4nMAssay Description:Beta-adrenergic agonistic activity in guinea-pig atrium preincubated with phenoxybenzamine (12 uM) for 30 minMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2018
Entry Details

TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50222540(CHEMBL19679)
Affinity DataKd:  200nMAssay Description:Binding affinity against Beta adrenergic receptor in C6-2B astrocytoma cells, using [125I]-iodohydroxybenzylpindolol-benzylpindolol([125I]-HYP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2018
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50222722(CHEMBL20234)
Affinity DataKd:  40nMAssay Description:Binding affinity against Beta adrenergic receptor in C6-2B astrocytoma cells, using [125I]-iodohydroxybenzylpindolol-benzylpindolol([125I]-HYP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2018
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50222723(CHEMBL19422)
Affinity DataKd:  15nMAssay Description:Binding affinity against Beta adrenergic receptor in C6-2B astrocytoma cells, using [125I]-iodohydroxybenzylpindolol-benzylpindolol([125I]-HYP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2018
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50222724(CHEMBL19669)
Affinity DataKd:  2.00E+3nMAssay Description:Binding affinity against Beta adrenergic receptor in C6-2B astrocytoma cells, using [125I]-iodohydroxybenzylpindolol-benzylpindolol([125I]-HYP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2018
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50222773(CHEMBL20909)
Affinity DataKd:  50nMAssay Description:Binding affinity against Beta adrenergic receptor in C6-2B astrocytoma cells, using [125I]-iodohydroxybenzylpindolol-benzylpindolol([125I]-HYP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2018
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50246936(S-(-)-propanolol | (-)-(S)-Propranolol | [2-Hydrox...)
Affinity DataKd:  0.700nMAssay Description:Binding affinity against Beta adrenergic receptor in C6-2B astrocytoma cells, using [125I]-iodohydroxybenzylpindolol-benzylpindolol([125I]-HYP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2018
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50222776(CHEMBL19770)
Affinity DataKd:  5nMAssay Description:Binding affinity against Beta adrenergic receptor in C6-2B astrocytoma cells, using [125I]-iodohydroxybenzylpindolol-benzylpindolol([125I]-HYP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2018
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50222775(CHEMBL19591)
Affinity DataKd:  500nMAssay Description:Binding affinity against Beta adrenergic receptor in C6-2B astrocytoma cells, using [125I]-iodohydroxybenzylpindolol-benzylpindolol([125I]-HYP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2018
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50222770(CHEMBL19593)
Affinity DataKd:  200nMAssay Description:Binding affinity against Beta adrenergic receptor in C6-2B astrocytoma cells, using [125I]-iodohydroxybenzylpindolol-benzylpindolol([125I]-HYP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2018
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50222768(CHEMBL19680)
Affinity DataKd:  2.00E+3nMAssay Description:Binding affinity against Beta adrenergic receptor in C6-2B astrocytoma cells, using [125I]-iodohydroxybenzylpindolol-benzylpindolol([125I]-HYP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2018
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50222769(CHEMBL19809)
Affinity DataKd:  300nMAssay Description:Binding affinity against Beta adrenergic receptor in C6-2B astrocytoma cells, using [125I]-iodohydroxybenzylpindolol-benzylpindolol([125I]-HYP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2018
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50029051(4-[(1R)-2-amino-1-hydroxyethyl]benzene-1,2-diol | ...)
Affinity DataEC50:  2.60E+3nMAssay Description:Evaluated for Beta adrenergic receptor agonistic property in isolated guinea pig atriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2018
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50224296(CHEMBL161974)
Affinity DataEC50:  10nMAssay Description:Evaluated for Beta adrenergic receptor agonistic property in isolated guinea pig atriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2018
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50067212(CHEBI:8093 | Cyclomydril | Duo-Medihaler | Phenyle...)
Affinity DataEC50:  6.00E+3nMAssay Description:Evaluated for Beta adrenergic receptor agonistic property in isolated guinea pig atriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2018
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50224297(CHEMBL158865)
Affinity DataEC50:  20nMAssay Description:Evaluated for Beta adrenergic receptor agonistic property in isolated guinea pig atriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2018
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataEC50:  30nMAssay Description:Evaluated for Beta adrenergic receptor agonistic property in isolated guinea pig atriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2018
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50224298(CHEMBL159016)
Affinity DataEC50:  3.00E+4nMAssay Description:Evaluated for Beta adrenergic receptor agonistic property in isolated guinea pig atriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2018
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50225367(Bromoacetyl Alprenolol Menthane)
Affinity DataKd:  19.8nMAssay Description:Equilibrium dissociation constant (KD) against beta adrenergic receptor of rat lung tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2018
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50225368(CHEMBL47370)
Affinity DataKd:  391nMAssay Description:Equilibrium dissociation constant (KD) against beta adrenergic receptor of rat heart tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2018
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50225367(Bromoacetyl Alprenolol Menthane)
Affinity DataKd:  42.4nMAssay Description:Equilibrium dissociation constant (KD) against beta adrenergic receptor of rat heart tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2018
Entry Details Article
PubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50225368(CHEMBL47370)
Affinity DataKd:  2.80nMAssay Description:Dissociation constant against beta adrenergic receptor using [3H]dihydroalprenolol in rat lung tissue at 1*10e-6 concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2018
Entry Details Article
PubMed
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