Report error Found 147 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 1/2'
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity was determined in vitro against cannabinoid receptor by ability to displace [3H]CP-55940More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity was determined in vitro against cannabinoid receptor by ability to displace [3H]CP-55940More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity was determined in vitro against cannabinoid receptor by ability to displace [3H]CP-55940More data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]WIN-55,212-2 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]WIN-55,212-2 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: >2.95E+3nMAssay Description:Binding affinity for the cannabinoid receptor in the absence of phenylmethanesulfonyl fluoride (PMSF) was determined in rat fore brain membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 2.89E+3nMAssay Description:Binding affinity towards cannabinoid receptor using [3H]SR-141,716A as radioligand in rat brain membraneMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 2.79E+3nMAssay Description:Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.25E+3nMAssay Description:Binding affinity was determined in vitro against cannabinoid receptor by ability to displace [3H]CP-55940More data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 1.22E+3nMAssay Description:Displacement of [3H]WIN-55,212-2 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: >1.18E+3nMAssay Description:Binding affinity for the cannabinoid receptor in the absence of phenylmethanesulfonyl fluoride (PMSF) was determined in rat fore brain membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 1.04E+3nMAssay Description:Displacement of [3H]WIN-55,212-2 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 1.01E+3nMAssay Description:Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to Cannabinoid receptor (unknown origin)More data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 928nMAssay Description:Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 919nMAssay Description:Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 823nMAssay Description:Displacement of [3H]WIN-55,212-2 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
Affinity DataKi: 800nMAssay Description:Binding affinity for Cannabinoid receptorMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 585nMAssay Description:Binding affinity towards cannabinoid receptor using [3H]SR-141,716A as radioligand in rat brain membraneMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 466nMAssay Description:Binding affinity towards cannabinoid receptor using [3H]SR-141,716A as radioligand in rat brain membraneMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 466nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]3-(1,1-Dimethyl-heptyl)-9-hydroxymethyl-6,6-dimethyl-6a,7,8,9,10,10a-hexahydro-6H-benzo[...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 317nMAssay Description:Displacement of [3H]WIN-55,212-2 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 282nMAssay Description:Binding affinity towards cannabinoid receptor using [3H]SR-141,716A as radioligand in rat brain membraneMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 269nMAssay Description:Displacement of [3H]WIN-55,212-2 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 268nMAssay Description:Binding affinity for the cannabinoid receptor in the absence of phenylmethanesulfonyl fluoride (PMSF) was determined in rat fore brain membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 255nMAssay Description:Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 251nMAssay Description:Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 247nMAssay Description:Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 238nMAssay Description:Binding affinity towards cannabinoid receptor using [3H]SR-141,716A as radioligand in rat brain membraneMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 220nMAssay Description:Binding affinity towards cannabinoid receptor using [3H]SR-141,716A as radioligand in rat brain membraneMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 205nMAssay Description:Displacement of [3H]WIN-55,212-2 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 190nMAssay Description:Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 183nMAssay Description:Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 173nMAssay Description:Binding affinity for the cannabinoid receptor in the presence of phenylmethanesulfonyl fluoride (PMSF) was determined in rat fore brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 164nMAssay Description:Binding affinity was determined in vitro against cannabinoid receptor by ability to displace [3H]CP-55940More data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 161nMAssay Description:Binding affinity towards cannabinoid receptor using [3H]SR-141,716A as radioligand in rat brain membraneMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 158nMAssay Description:Binding affinity for the cannabinoid receptor in the absence of phenylmethanesulfonyl fluoride (PMSF) was determined in rat fore brain membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 153nMAssay Description:Binding affinity towards cannabinoid receptor using [3H]SR-141,716A as radioligand in rat brain membraneMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 149nMAssay Description:Displacement of [3H]WIN-55,212-2 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 145nMAssay Description:Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 119nMAssay Description:Binding affinity for the cannabinoid receptor in the presence of phenylmethanesulfonyl fluoride (PMSF) was determined in rat fore brain membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 82nMAssay Description:Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
Affinity DataKi: 81nMAssay Description:Binding affinity was determined in vitro against cannabinoid receptor by ability to displace [3H]CP-55940More data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 78nMAssay Description:Binding affinity for the cannabinoid receptor in the presence of phenylmethanesulfonyl fluoride (PMSF) was determined in rat fore brain membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 78nMAssay Description:Displacement of [3H]WIN-55,212-2 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
Affinity DataKi: 72nMAssay Description:Binding affinity was determined in vitro against cannabinoid receptor by ability to displace [3H]CP-55940More data for this Ligand-Target Pair


































