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Found 75 with Last Name = 'martin' and Initial = 'ac'
TargetPlatelet-activating factor acetylhydrolase(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50125265(CHEMBL204021 | N-(2-Diethylamino-ethyl)-2-[2-(4-fl...)
Affinity DataIC50:  0.0490nMAssay Description:Inhibition of human recombinant Lp-PLA2 using 2-thio-PAF as substrate after 20 mins by CPM-based fluorescence assayMore data for this Ligand-Target Pair
TargetPlatelet-activating factor acetylhydrolase(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182422(CHEMBL3818650)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of human recombinant Lp-PLA2 using 2-thio-PAF as substrate after 20 mins by CPM-based fluorescence assayMore data for this Ligand-Target Pair
TargetPlatelet-activating factor acetylhydrolase(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182421(CHEMBL3817896)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of human recombinant Lp-PLA2 using 2-thio-PAF as substrate after 20 mins by CPM-based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor acetylhydrolase(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182420(CHEMBL3819600)
Affinity DataIC50:  3.60nMAssay Description:Inhibition of human recombinant Lp-PLA2 using 2-thio-PAF as substrate after 20 mins by CPM-based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor acetylhydrolase(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182419(CHEMBL3819444)
Affinity DataIC50:  9.5nMAssay Description:Inhibition of human recombinant Lp-PLA2 using 2-thio-PAF as substrate after 20 mins by CPM-based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA ligase(Staphylococcus aureus)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444582(CHEMBL3099715)
Affinity DataIC50:  15nMAssay Description:Inhibition of C-terminal 6xHis-tagged full length recombinant Staphylococcus aureus DNA ligase (1 to 312) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor acetylhydrolase(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182422(CHEMBL3818650)
Affinity DataIC50:  18nMAssay Description:Inhibition of Lp-PLA2 in human whole plasma using 2-thio-PAF as substrate preincubated for 15 mins followed by substrate addition measured after 3 mi...More data for this Ligand-Target Pair
TargetPlatelet-activating factor acetylhydrolase(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182421(CHEMBL3817896)
Affinity DataIC50:  28nMAssay Description:Inhibition of Lp-PLA2 in human whole plasma using 2-thio-PAF as substrate preincubated for 15 mins followed by substrate addition measured after 3 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor acetylhydrolase(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50125265(CHEMBL204021 | N-(2-Diethylamino-ethyl)-2-[2-(4-fl...)
Affinity DataIC50:  35nMAssay Description:Inhibition of Lp-PLA2 in human whole plasma using 2-thio-PAF as substrate preincubated for 15 mins followed by substrate addition measured after 3 mi...More data for this Ligand-Target Pair
TargetPlatelet-activating factor acetylhydrolase(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182428(CHEMBL3819632)
Affinity DataIC50:  180nMAssay Description:Inhibition of human recombinant Lp-PLA2 using 2-thio-PAF as substrate after 20 mins by CPM-based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA ligase(Staphylococcus aureus)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444581(CHEMBL3099713)
Affinity DataIC50:  220nMAssay Description:Inhibition of C-terminal 6xHis-tagged full length recombinant Staphylococcus aureus DNA ligase (1 to 312) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor acetylhydrolase(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182429(CHEMBL3818759)
Affinity DataIC50:  230nMAssay Description:Inhibition of human recombinant Lp-PLA2 using 2-thio-PAF as substrate after 20 mins by CPM-based fluorescence assayMore data for this Ligand-Target Pair
TargetDNA ligase(Staphylococcus aureus)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444580(CHEMBL3099714)
Affinity DataIC50:  230nMAssay Description:Inhibition of C-terminal 6xHis-tagged full length recombinant Staphylococcus aureus DNA ligase (1 to 312) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
TargetPlatelet-activating factor acetylhydrolase(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182423(CHEMBL3819367)
Affinity DataIC50:  230nMAssay Description:Inhibition of human recombinant Lp-PLA2 using 2-thio-PAF as substrate after 20 mins by CPM-based fluorescence assayMore data for this Ligand-Target Pair
TargetPlatelet-activating factor acetylhydrolase(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182420(CHEMBL3819600)
Affinity DataIC50:  320nMAssay Description:Inhibition of Lp-PLA2 in human whole plasma using 2-thio-PAF as substrate preincubated for 15 mins followed by substrate addition measured after 3 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor acetylhydrolase(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182419(CHEMBL3819444)
Affinity DataIC50:  560nMAssay Description:Inhibition of Lp-PLA2 in human whole plasma using 2-thio-PAF as substrate preincubated for 15 mins followed by substrate addition measured after 3 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor acetylhydrolase(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182432(CHEMBL3818591)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of human recombinant Lp-PLA2 using 2-thio-PAF as substrate after 20 mins by CPM-based fluorescence assayMore data for this Ligand-Target Pair
TargetPlatelet-activating factor acetylhydrolase(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182431(CHEMBL3819446)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human recombinant Lp-PLA2 using 2-thio-PAF as substrate after 20 mins by CPM-based fluorescence assayMore data for this Ligand-Target Pair
TargetPlatelet-activating factor acetylhydrolase(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182423(CHEMBL3819367)
Affinity DataIC50:  7.10E+3nMAssay Description:Inhibition of Lp-PLA2 in human whole plasma using 2-thio-PAF as substrate preincubated for 15 mins followed by substrate addition measured after 3 mi...More data for this Ligand-Target Pair
TargetDNA ligase(Staphylococcus aureus)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444579(CHEMBL3099712)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of C-terminal 6xHis-tagged full length recombinant Staphylococcus aureus DNA ligase (1 to 312) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA ligase(Staphylococcus aureus)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444578(CHEMBL3099706)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of C-terminal 6xHis-tagged full length recombinant Staphylococcus aureus DNA ligase (1 to 312) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA ligase(Staphylococcus aureus)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444577(CHEMBL3099711)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of C-terminal 6xHis-tagged full length recombinant Staphylococcus aureus DNA ligase (1 to 312) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor acetylhydrolase(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182430(CHEMBL3819099)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of human recombinant Lp-PLA2 using 2-thio-PAF as substrate after 20 mins by CPM-based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA ligase(Staphylococcus aureus)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444575(CHEMBL3099710)
Affinity DataIC50:  5.30E+4nMAssay Description:Inhibition of C-terminal 6xHis-tagged full length recombinant Staphylococcus aureus DNA ligase (1 to 312) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor acetylhydrolase(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182425(CHEMBL3819345)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of human recombinant Lp-PLA2 using 2-thio-PAF as substrate after 20 mins by CPM-based fluorescence assayMore data for this Ligand-Target Pair
TargetPlatelet-activating factor acetylhydrolase(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182425(CHEMBL3819345)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of human recombinant Lp-PLA2 using PED6 as substrate preincubated for 30 mins followed by substrate addition measured for 20 mins by fluor...More data for this Ligand-Target Pair
TargetDNA ligase(Staphylococcus aureus)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444574(CHEMBL3099708)
Affinity DataIC50:  1.30E+5nMAssay Description:Inhibition of C-terminal 6xHis-tagged full length recombinant Staphylococcus aureus DNA ligase (1 to 312) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA ligase(Staphylococcus aureus)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444573(CHEMBL3099709)
Affinity DataIC50:  1.40E+5nMAssay Description:Inhibition of C-terminal 6xHis-tagged full length recombinant Staphylococcus aureus DNA ligase (1 to 312) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA ligase(Staphylococcus aureus)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444572(CHEMBL3099707)
Affinity DataIC50:  3.00E+5nMAssay Description:Inhibition of C-terminal 6xHis-tagged full length recombinant Staphylococcus aureus DNA ligase (1 to 312) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor acetylhydrolase(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182424(CHEMBL3818090)
Affinity DataIC50:  5.00E+5nMAssay Description:Inhibition of human recombinant Lp-PLA2 using PED6 as substrate preincubated for 30 mins followed by substrate addition measured for 20 mins by fluor...More data for this Ligand-Target Pair
TargetPlatelet-activating factor acetylhydrolase(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM12414(CHEMBL27601 | benzenesulfonamide | hCA inhibitor, ...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of human recombinant Lp-PLA2 using PED6 as substrate preincubated for 30 mins followed by substrate addition measured for 20 mins by fluor...More data for this Ligand-Target Pair
TargetPlatelet-activating factor acetylhydrolase(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182426(CHEMBL3819543)
Affinity DataIC50:  1.00E+6nMAssay Description:Inhibition of human recombinant Lp-PLA2 using PED6 as substrate preincubated for 30 mins followed by substrate addition measured for 20 mins by fluor...More data for this Ligand-Target Pair
TargetPlatelet-activating factor acetylhydrolase(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182427(CHEMBL3181806)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of human recombinant Lp-PLA2 using PED6 as substrate preincubated for 30 mins followed by substrate addition measured for 20 mins by fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor acetylhydrolase(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM12414(CHEMBL27601 | benzenesulfonamide | hCA inhibitor, ...)
Affinity DataKd:  3.40E+6nMAssay Description:Binding affinity to N-terminal His6-tagged Lp-PLA2 (47 to 429 residues) (unknown origin) expressed in sf21 insect cells by ITC assayMore data for this Ligand-Target Pair
TargetPlatelet-activating factor acetylhydrolase(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182424(CHEMBL3818090)
Affinity DataKd:  9.80E+5nMAssay Description:Binding affinity to N-terminal His6-tagged Lp-PLA2 (47 to 429 residues) (unknown origin) expressed in sf21 insect cells by ITC assayMore data for this Ligand-Target Pair
TargetDNA ligase(Staphylococcus aureus)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444576(CHEMBL3099705)
Affinity DataKd:  3.80E+4nMAssay Description:Binding affinity to C-terminal 6xHis-tagged Staphylococcus aureus DNA ligase (1 to 312) expressed in Escherichia coli BL21 (DE3) by ITC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA ligase(Staphylococcus aureus)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444578(CHEMBL3099706)
Affinity DataKd:  1.00E+4nMAssay Description:Binding affinity to C-terminal 6xHis-tagged Staphylococcus aureus DNA ligase (1 to 312) expressed in Escherichia coli BL21 (DE3) by ITC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA ligase(Staphylococcus aureus)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444582(CHEMBL3099715)
Affinity DataKd:  25nMAssay Description:Binding affinity to C-terminal 6xHis-tagged Staphylococcus aureus DNA ligase (1 to 312) expressed in Escherichia coli BL21 (DE3) by ITC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukocyte surface antigen CD47(Homo sapiens (Human))
Sorbonne University

Curated by ChEMBL
LigandPNGBDBM50192009(CHEMBL3946082)
Affinity DataKd:  1.50E+3nMAssay Description:Binding affinity to CD47 receptor in human biotinylated MEC1 cell membranes by biolayer interferometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukocyte surface antigen CD47(Homo sapiens (Human))
Sorbonne University

Curated by ChEMBL
LigandPNGBDBM50192010(CHEMBL3975422)
Affinity DataKd:  1.00E+4nMAssay Description:Binding affinity to CD47 receptor in human NT.115-labeled MEC1 cell membranes after 5 mins by MST assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukocyte surface antigen CD47(Homo sapiens (Human))
Sorbonne University

Curated by ChEMBL
LigandPNGBDBM50192009(CHEMBL3946082)
Affinity DataKd:  771nMAssay Description:Binding affinity to CD47 receptor in human NT.115-labeled MEC1 cell membranes after 5 mins by MST assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukocyte surface antigen CD47(Homo sapiens (Human))
Sorbonne University

Curated by ChEMBL
LigandPNGBDBM50192011(CHEMBL3911226)
Affinity DataKd:  1.80E+4nMAssay Description:Binding affinity to CD47 receptor in human biotinylated MEC1 cell membranes by biolayer interferometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukocyte surface antigen CD47(Homo sapiens (Human))
Sorbonne University

Curated by ChEMBL
LigandPNGBDBM50192012(CHEMBL3971661)
Affinity DataKd:  4.30E+4nMAssay Description:Binding affinity to CD47 receptor in human biotinylated MEC1 cell membranes by biolayer interferometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukocyte surface antigen CD47(Homo sapiens (Human))
Sorbonne University

Curated by ChEMBL
LigandPNGBDBM50192013(CHEMBL3974452)
Affinity DataKd:  1.90E+4nMAssay Description:Binding affinity to CD47 receptor in human biotinylated MEC1 cell membranes by biolayer interferometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukocyte surface antigen CD47(Homo sapiens (Human))
Sorbonne University

Curated by ChEMBL
LigandPNGBDBM50192014(CHEMBL3891508)
Affinity DataKd:  1.20E+3nMAssay Description:Binding affinity to CD47 receptor in human NT.115-labeled MEC1 cell membranes after 5 mins by MST assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukocyte surface antigen CD47(Homo sapiens (Human))
Sorbonne University

Curated by ChEMBL
LigandPNGBDBM50192013(CHEMBL3974452)
Affinity DataKd:  2.28E+3nMAssay Description:Binding affinity to CD47 receptor in human NT.115-labeled MEC1 cell membranes after 5 mins by MST assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukocyte surface antigen CD47(Homo sapiens (Human))
Sorbonne University

Curated by ChEMBL
LigandPNGBDBM50192015(CHEMBL3900522)
Affinity DataKd:  6.20E+3nMAssay Description:Binding affinity to CD47 receptor in human biotinylated MEC1 cell membranes by biolayer interferometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukocyte surface antigen CD47(Homo sapiens (Human))
Sorbonne University

Curated by ChEMBL
LigandPNGBDBM50192014(CHEMBL3891508)
Affinity DataKd:  4.00E+4nMAssay Description:Binding affinity to CD47 receptor in human biotinylated MEC1 cell membranes by biolayer interferometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukocyte surface antigen CD47(Homo sapiens (Human))
Sorbonne University

Curated by ChEMBL
LigandPNGBDBM50192016(CHEMBL3939184)
Affinity DataKd:  2.70E+4nMAssay Description:Binding affinity to CD47 receptor in human biotinylated MEC1 cell membranes by biolayer interferometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukocyte surface antigen CD47(Homo sapiens (Human))
Sorbonne University

Curated by ChEMBL
LigandPNGBDBM50192012(CHEMBL3971661)
Affinity DataKd:  3.04E+3nMAssay Description:Binding affinity to CD47 receptor in human NT.115-labeled MEC1 cell membranes after 5 mins by MST assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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