TargetGamma-aminobutyric acid receptor subunit alpha-4(Homo sapiens (Human))
Cocensys
Curated by PDSP Ki Database
Cocensys
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-4(Homo sapiens (Human))
Cocensys
Curated by PDSP Ki Database
Cocensys
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-6(Homo sapiens (Human))
Cocensys
Curated by PDSP Ki Database
Cocensys
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-4(Homo sapiens (Human))
Cocensys
Curated by PDSP Ki Database
Cocensys
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-4(Homo sapiens (Human))
Cocensys
Curated by PDSP Ki Database
Cocensys
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-6(Homo sapiens (Human))
Cocensys
Curated by PDSP Ki Database
Cocensys
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-4(Homo sapiens (Human))
Cocensys
Curated by PDSP Ki Database
Cocensys
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-6(Homo sapiens (Human))
Cocensys
Curated by PDSP Ki Database
Cocensys
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-6(Homo sapiens (Human))
Cocensys
Curated by PDSP Ki Database
Cocensys
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-4(Homo sapiens (Human))
Cocensys
Curated by PDSP Ki Database
Cocensys
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-6(Homo sapiens (Human))
Cocensys
Curated by PDSP Ki Database
Cocensys
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-6(Homo sapiens (Human))
Cocensys
Curated by PDSP Ki Database
Cocensys
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-4(Homo sapiens (Human))
Cocensys
Curated by PDSP Ki Database
Cocensys
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-4(Homo sapiens (Human))
Cocensys
Curated by PDSP Ki Database
Cocensys
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-6(Homo sapiens (Human))
Cocensys
Curated by PDSP Ki Database
Cocensys
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-6(Homo sapiens (Human))
Cocensys
Curated by PDSP Ki Database
Cocensys
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-6(Homo sapiens (Human))
Cocensys
Curated by PDSP Ki Database
Cocensys
Curated by PDSP Ki Database
Affinity DataIC50: 5nMAssay Description:Inhibitory concentration against human caspase-3More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Compound was evaluated for its inhibitory activity against the Caspase-9 enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of human caspase 9More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition concentration required against caspase-8More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibitory concentration against human caspase-3More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of human caspase 8More data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Compound was evaluated for its inhibitory activity against the Caspase-7 enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Compound was evaluated for its inhibitory activity against the Caspase-8 enzymeMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Of Oregon
Curated by ChEMBL
University Of Oregon
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Functional antagonism by electrical assays in Xenopus oocytes expressing the 1A/2B NMDA receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition concentration required against caspase-9More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition concentration required against caspase-7More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibitory concentration against Caspase-7More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of human caspase 7More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of human caspase 1More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibitory concentration against human caspase-3More data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibitory concentration against human caspase-3More data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibitory concentration against human caspase-3More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Of Oregon
Curated by ChEMBL
University Of Oregon
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Functional antagonism by electrical assays in Xenopus oocytes expressing the 1A/2B NMDA receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibitory activity against human recombinant caspase-3More data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibitory concentration against Caspase-8More data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibitory concentration against human caspase-3More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Compound was evaluated for its inhibitory activity against the Caspase-6 enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Inhibitory concentration against human caspase-3More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Compound was evaluated for its inhibitory activity against the Caspase-1 enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibitory concentration against human caspase-3More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibitory concentration against human caspase-3More data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibitory activity against human recombinant caspase-3More data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibitory activity against human recombinant caspase-3More data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibitory activity against human recombinant caspase-3More data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Inhibitory activity against human recombinant caspase-3More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibitory activity against human recombinant caspase-3More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibitory activity against human recombinant Caspase-3 enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibitory concentration against human caspase-3More data for this Ligand-Target Pair