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Found 783 with Last Name = 'parker' and Initial = 'j'
Targetneuronal acetylcholine receptor subunit alpha-2(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86041(NFEP)
Affinity DataKi:  0.00240nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM86042(NEP)
Affinity DataKi:  0.00310nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM86041(NFEP)
Affinity DataKi:  0.00380nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM86040(NBEP)
Affinity DataKi:  0.00400nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-4(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86042(NEP)
Affinity DataKi:  0.00850nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-4(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86041(NFEP)
Affinity DataKi:  0.00920nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-4(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86040(NBEP)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-2(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86040(NBEP)
Affinity DataKi:  0.0130nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-2(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86042(NEP)
Affinity DataKi:  0.0280nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinergic receptor, nicotinic alpha 1(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86040(NBEP)
Affinity DataKi:  0.0440nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-2(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86040(NBEP)
Affinity DataKi:  0.0550nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-2(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86045(NNEP)
Affinity DataKi:  0.0620nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM86045(NNEP)
Affinity DataKi:  0.0770nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinergic receptor nicotinic alpha 5 subunit(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86040(NBEP)
Affinity DataKi:  0.220nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-4(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86045(NNEP)
Affinity DataKi:  0.350nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinergic receptor, nicotinic alpha 1(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86041(NFEP)
Affinity DataKi:  0.480nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-2(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86041(NFEP)
Affinity DataKi:  1.20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50338518(1-((3S,4S)-4-amino-1-(4-(3,3-difluoropyrrolidin-1-...)
Affinity DataKi:  2.10nMAssay Description:Inhibition of DPP4 in rat plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinergic receptor nicotinic alpha 5 subunit(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86041(NFEP)
Affinity DataKi:  2.10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinergic receptor, nicotinic alpha 1(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86042(NEP)
Affinity DataKi:  3.20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-2(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86042(NEP)
Affinity DataKi:  3.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-2(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86045(NNEP)
Affinity DataKi:  3.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinergic receptor, nicotinic alpha 1(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86045(NNEP)
Affinity DataKi:  4.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50152799((R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic a...)
Affinity DataKi:  6.40nMAssay Description:Displacement of [125I]NDP-MSH from HEK293 cells expressing human melanocortin-4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinergic receptor nicotinic alpha 5 subunit(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86045(NNEP)
Affinity DataKi:  7.20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-2(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86044(NTEP)
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50152800(1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid ...)
Affinity DataKi:  11nMAssay Description:Displacement of [125I]NDP-MSH from HEK293 cells expressing human melanocortin-4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinergic receptor nicotinic alpha 5 subunit(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86042(NEP)
Affinity DataKi:  11nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50152808((R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic a...)
Affinity DataKi:  11nMAssay Description:Displacement of [125I]NDP-MSH from HEK293 cells expressing human melanocortin-4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50152808((R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic a...)
Affinity DataKi:  12nMAssay Description:Tested for inhibition of binding to MC4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50152807((R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic a...)
Affinity DataKi:  12nMAssay Description:Displacement of [125I]NDP-MSH from HEK293 cells expressing human melanocortin-4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50152802((R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic a...)
Affinity DataKi:  13nMAssay Description:Displacement of [125I]NDP-MSH from HEK293 cells expressing human melanocortin-4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50152795(1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid ...)
Affinity DataKi:  13nMAssay Description:Displacement of [125I]NDP-MSH from HEK293 cells expressing human melanocortin-4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50155393(4-Amino-N-[(R)-1-(4-chloro-benzyl)-2-oxo-2-(4-{2-[...)
Affinity DataKi:  14nMAssay Description:Tested for inhibition of binding to MC4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50152816((R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic a...)
Affinity DataKi:  14nMAssay Description:Displacement of [125I]NDP-MSH from HEK293 cells expressing human melanocortin-4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50338518(1-((3S,4S)-4-amino-1-(4-(3,3-difluoropyrrolidin-1-...)
Affinity DataKi:  14nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50063218((R)-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]...)
Affinity DataKi:  14nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50155370(CHEMBL186074 | Piperidine-3-carboxylic acid [(R)-1...)
Affinity DataKi:  15nMAssay Description:Tested for inhibition of binding to MC4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50152813(1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid ...)
Affinity DataKi:  19nMAssay Description:Displacement of [125I]NDP-MSH from HEK293 cells expressing human melanocortin-4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50155390(3-Amino-N-[(R)-1-(4-chloro-benzyl)-2-oxo-2-(4-{2-[...)
Affinity DataKi:  21nMAssay Description:Tested for inhibition of binding to MC4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50152817((R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic a...)
Affinity DataKi:  23nMAssay Description:Displacement of [125I]NDP-MSH from HEK293 cells expressing human melanocortin-4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50134486((R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic a...)
Affinity DataKi:  24nMAssay Description:Displacement of [125I]-NDP-MSH from HEK293 cells expressing human melanocortin-3 receptor at 10 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50152810(1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid ...)
Affinity DataKi:  24nMAssay Description:Displacement of [125I]NDP-MSH from HEK293 cells expressing human melanocortin-4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50152797((R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic a...)
Affinity DataKi:  24nMAssay Description:Displacement of [125I]NDP-MSH from HEK293 cells expressing human melanocortin-4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50152796(1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid ...)
Affinity DataKi:  25nMAssay Description:Displacement of [125I]NDP-MSH from HEK293 cells expressing human melanocortin-4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50155401(CHEMBL363122 | Piperidine-4-carboxylic acid [(R)-1...)
Affinity DataKi:  26nMAssay Description:Tested for inhibition of binding to MC4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50152818(1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid ...)
Affinity DataKi:  27nMAssay Description:Displacement of [125I]NDP-MSH from HEK293 cells expressing human melanocortin-4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50152806((R)-N-((R)-1-(4-(2-(aminomethyl)phenyl)piperazin-1...)
Affinity DataKi:  27nMAssay Description:Displacement of [125I]NDP-MSH from HEK293 cells expressing human melanocortin-1 receptor at 10 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50140541((S)-2-Amino-2-cyclohexyl-1-(3,3-difluoro-pyrrolidi...)
Affinity DataKi:  28nMAssay Description:Inhibitory constant against Dipeptidylpeptidase IV activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50155374(2-Amino-4-methyl-pentanoic acid [(R)-1-(4-chloro-b...)
Affinity DataKi:  30nMAssay Description:Tested for inhibition of binding to MC4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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