TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of soluble epoxide hydrolase (unknown origin)More data for this Ligand-Target Pair
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of soluble epoxide hydrolase (unknown origin)More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of AT1 receptor (unknown origin)More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant N-terminal His-tagged human iNOS expressed in Escherichia coli using L-arginine as substrate preincubated for 15 mins follo...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
Affinity DataIC50: 58nMAssay Description:Inhibition of recombinant mouse iNOS using [3H]L-arginine as substrate preincubated for 15 mins followed by NADPH addition measured after 20 mins in ...More data for this Ligand-Target Pair
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
Affinity DataIC50: 69nMAssay Description:Inhibition of soluble epoxide hydrolase (unknown origin)More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Inhibition of recombinant N-terminal His-tagged human iNOS expressed in Escherichia coli using L-arginine as substrate preincubated for 15 mins follo...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
Affinity DataIC50: 101nMAssay Description:Inhibition of recombinant mouse iNOS using [3H]L-arginine as substrate preincubated for 15 mins followed by NADPH addition measured after 20 mins in ...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Inhibition of recombinant mouse iNOS using [3H]L-arginine as substrate preincubated for 15 mins followed by NADPH addition measured after 20 mins in ...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
Affinity DataIC50: 253nMAssay Description:Inhibition of recombinant mouse iNOS using [3H]L-arginine as substrate preincubated for 15 mins followed by NADPH addition measured after 20 mins in ...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
Affinity DataIC50: 276nMAssay Description:Inhibition of recombinant mouse iNOS using [3H]L-arginine as substrate preincubated for 15 mins followed by NADPH addition measured after 20 mins in ...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: 428nMAssay Description:Inhibition of recombinant N-terminal His-tagged human iNOS expressed in Escherichia coli using L-arginine as substrate preincubated for 15 mins follo...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
Affinity DataIC50: 446nMAssay Description:Inhibition of recombinant mouse iNOS using [3H]L-arginine as substrate preincubated for 15 mins followed by NADPH addition measured after 20 mins in ...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
Affinity DataIC50: 450nMAssay Description:Inhibition of recombinant mouse iNOS using [3H]L-arginine as substrate preincubated for 15 mins followed by NADPH addition measured after 20 mins in ...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
Affinity DataIC50: 534nMAssay Description:Inhibition of recombinant mouse iNOS using [3H]L-arginine as substrate preincubated for 15 mins followed by NADPH addition measured after 20 mins in ...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: 681nMAssay Description:Inhibition of recombinant N-terminal His-tagged human iNOS expressed in Escherichia coli using L-arginine as substrate preincubated for 15 mins follo...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
Affinity DataIC50: 1.03E+3nMAssay Description:Inhibition of recombinant mouse iNOS using [3H]L-arginine as substrate preincubated for 15 mins followed by NADPH addition measured after 20 mins in ...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
Affinity DataIC50: 1.23E+3nMAssay Description:Inhibition of recombinant mouse iNOS using [3H]L-arginine as substrate preincubated for 15 mins followed by NADPH addition measured after 20 mins in ...More data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of recombinant human nNOS expressed in Escherichia coli using L-arginine as substrate preincubated for 15 mins followed by NADPH addition ...More data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of recombinant rat nNOS using [3H]L-arginine as substrate preincubated for 15 mins followed by NADPH addition measured after 20 mins in pr...More data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of recombinant human nNOS expressed in Escherichia coli using L-arginine as substrate preincubated for 15 mins followed by NADPH addition ...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant mouse iNOS using [3H]L-arginine as substrate preincubated for 15 mins followed by NADPH addition measured after 20 mins in ...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant mouse iNOS using [3H]L-arginine as substrate preincubated for 15 mins followed by NADPH addition measured after 20 mins in ...More data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant rat nNOS using [3H]L-arginine as substrate preincubated for 15 mins followed by NADPH addition measured after 20 mins in pr...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant mouse iNOS using [3H]L-arginine as substrate preincubated for 15 mins followed by NADPH addition measured after 20 mins in ...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant mouse iNOS using [3H]L-arginine as substrate preincubated for 15 mins followed by NADPH addition measured after 20 mins in ...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant mouse iNOS using [3H]L-arginine as substrate preincubated for 15 mins followed by NADPH addition measured after 20 mins in ...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant mouse iNOS using [3H]L-arginine as substrate preincubated for 15 mins followed by NADPH addition measured after 20 mins in ...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant mouse iNOS using [3H]L-arginine as substrate preincubated for 15 mins followed by NADPH addition measured after 20 mins in ...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant mouse iNOS using [3H]L-arginine as substrate preincubated for 15 mins followed by NADPH addition measured after 20 mins in ...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant mouse iNOS using [3H]L-arginine as substrate preincubated for 15 mins followed by NADPH addition measured after 20 mins in ...More data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human eNOS using L-argininge as substrate preincubated for 15 mins followed by NADPH addition and measured after 20 mins by OPA/NAC rea...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant mouse iNOS using [3H]L-arginine as substrate preincubated for 15 mins followed by NADPH addition measured after 20 mins in ...More data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant bovine eNOS using [3H]L-arginine as substrate preincubated for 15 mins followed by NADPH addition measured after 20 mins in...More data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
Affinity DataIC50: 2.11E+5nMAssay Description:Inhibition of recombinant bovine eNOS using [3H]L-arginine as substrate preincubated for 15 mins followed by NADPH addition measured after 20 mins in...More data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
Affinity DataIC50: 2.65E+5nMAssay Description:Inhibition of recombinant bovine eNOS using [3H]L-arginine as substrate preincubated for 15 mins followed by NADPH addition measured after 20 mins in...More data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of recombinant bovine eNOS using [3H]L-arginine as substrate preincubated for 15 mins followed by NADPH addition measured after 20 mins in...More data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: 3.04E+5nMAssay Description:Inhibition of human eNOS using L-argininge as substrate preincubated for 15 mins followed by NADPH addition and measured after 20 mins by OPA/NAC rea...More data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
Affinity DataIC50: 3.31E+5nMAssay Description:Inhibition of recombinant bovine eNOS using [3H]L-arginine as substrate preincubated for 15 mins followed by NADPH addition measured after 20 mins in...More data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
Affinity DataIC50: 3.84E+5nMAssay Description:Inhibition of recombinant bovine eNOS using [3H]L-arginine as substrate preincubated for 15 mins followed by NADPH addition measured after 20 mins in...More data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of recombinant bovine eNOS using [3H]L-arginine as substrate preincubated for 15 mins followed by NADPH addition measured after 20 mins in...More data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of recombinant bovine eNOS using [3H]L-arginine as substrate preincubated for 15 mins followed by NADPH addition measured after 20 mins in...More data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of recombinant bovine eNOS using [3H]L-arginine as substrate preincubated for 15 mins followed by NADPH addition measured after 20 mins in...More data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
University Of Chieti "G. D'Annunzio
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of recombinant bovine eNOS using [3H]L-arginine as substrate preincubated for 15 mins followed by NADPH addition measured after 20 mins in...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
Affinity DataEC50: 2.02E+3nMAssay Description:Transactivation of GAL4-tagged human PPARgamma expressed in African green monkey COS7 cells after 36 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair