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Found 55 with Last Name = 'azim' and Initial = 'mk'
TargetCarbonic anhydrase 2(Bos taurus)
University of Karachi

LigandPNGBDBM222435(N'',N'''-Bis[(E)-(2,6-dichlorophenyl)methylide...)
Affinity DataKi:  1.78E+3nMpH: 7.4Assay Description:Kinetic studies were performed by using different concentration of inhibitors over different concentrations of substrate (4-NPA) such as 0.175, 0.35,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Bos taurus)
University of Karachi

LigandPNGBDBM222429(N'',N'''-Bis[(E)-(2-nitrophenyl)methylidene]ca...)
Affinity DataKi:  1.81E+3nMpH: 7.4Assay Description:Kinetic studies were performed by using different concentration of inhibitors over different concentrations of substrate (4-NPA) such as 0.175, 0.35,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Bos taurus)
University of Karachi

LigandPNGBDBM222428(N'',N'''-Bis[(E)-(4-nitrophenyl)methylidene]ca...)
Affinity DataKi:  2.35E+3nMpH: 7.4Assay Description:Kinetic studies were performed by using different concentration of inhibitors over different concentrations of substrate (4-NPA) such as 0.175, 0.35,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Bos taurus)
University of Karachi

LigandPNGBDBM222431(N'',N'''-Bis[(E)-(4-bromophenyl)methylidene]ca...)
Affinity DataKi:  2.52E+3nMpH: 7.4Assay Description:Kinetic studies were performed by using different concentration of inhibitors over different concentrations of substrate (4-NPA) such as 0.175, 0.35,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Bos taurus)
University of Karachi

LigandPNGBDBM222430(N'',N'''-Bis[(E)-(2-chloro-5-nitrophenyl)methy...)
Affinity DataKi:  3.58E+3nMpH: 7.4Assay Description:Kinetic studies were performed by using different concentration of inhibitors over different concentrations of substrate (4-NPA) such as 0.175, 0.35,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Bos taurus)
University of Karachi

LigandPNGBDBM222433(N'',N'''-Bis[(E)-(2-chlorophenyl)methylidene]c...)
Affinity DataKi:  4.12E+3nMpH: 7.4Assay Description:Kinetic studies were performed by using different concentration of inhibitors over different concentrations of substrate (4-NPA) such as 0.175, 0.35,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50377588(CHEMBL257594)
Affinity DataIC50:  0.130nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin-2 by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50377588(CHEMBL257594)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of human cathepsin D by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM912((3S,4S)-3-hydroxy-4-[(2S)-2-[(3S,4S)-3-hydroxy-6-m...)
Affinity DataIC50:  0.550nMAssay Description:Inhibition of human cathepsin D by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetPlasmepsin II(Plasmodium falciparum)
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM912((3S,4S)-3-hydroxy-4-[(2S)-2-[(3S,4S)-3-hydroxy-6-m...)
Affinity DataIC50:  0.680nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin-2 by FRET assayMore data for this Ligand-Target Pair
TargetPlasmepsin II(Plasmodium falciparum)
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50377587(CHEMBL404394)
Affinity DataIC50:  4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin-2 by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50377587(CHEMBL404394)
Affinity DataIC50:  9nMAssay Description:Inhibition of human cathepsin D by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM233139(2-Nitrobenzohydrazide | Mr-I-53b)
Affinity DataIC50:  1.00E+3nMpH: 5.0Assay Description:The assay was performed with plasmepsin-II/cathepsin D (1.2 nM) and substrate (malaria FRET-1; 1.0 μM) in 0.1 M sodium acetate buffer pH 5, contai...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM233141(1,2-Diphenylhydrazine | Mr-II-10)
Affinity DataIC50:  1.05E+3nMpH: 5.0Assay Description:The assay was performed with plasmepsin-II/cathepsin D (1.2 nM) and substrate (malaria FRET-1; 1.0 μM) in 0.1 M sodium acetate buffer pH 5, contai...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM233138(Butanohydrazide | Mr-I-33)
Affinity DataIC50:  1.25E+3nMpH: 5.0Assay Description:The assay was performed with plasmepsin-II/cathepsin D (1.2 nM) and substrate (malaria FRET-1; 1.0 μM) in 0.1 M sodium acetate buffer pH 5, contai...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM233139(2-Nitrobenzohydrazide | Mr-I-53b)
Affinity DataIC50:  1.30E+3nMpH: 5.0Assay Description:The assay was performed with plasmepsin-II/cathepsin D (1.2 nM) and substrate (malaria FRET-1; 1.0 μM) in 0.1 M sodium acetate buffer pH 5, contai...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Bos taurus)
University of Karachi

LigandPNGBDBM222428(N'',N'''-Bis[(E)-(4-nitrophenyl)methylidene]ca...)
Affinity DataIC50:  1.33E+3nMpH: 7.4 T: 2°CAssay Description:In this assay, 4-nitrophenyl acetate (4-NPA), a colorless compound, was hydrolyzed to 4-nitrophenol and CO2. The reaction was followed by measuring t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM233140(2-Nitrobenzohydrazide | Mr-I-179)
Affinity DataIC50:  1.35E+3nMpH: 5.0Assay Description:The assay was performed with plasmepsin-II/cathepsin D (1.2 nM) and substrate (malaria FRET-1; 1.0 μM) in 0.1 M sodium acetate buffer pH 5, contai...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Bos taurus)
University of Karachi

LigandPNGBDBM222430(N'',N'''-Bis[(E)-(2-chloro-5-nitrophenyl)methy...)
Affinity DataIC50:  1.37E+3nMpH: 7.4 T: 2°CAssay Description:In this assay, 4-nitrophenyl acetate (4-NPA), a colorless compound, was hydrolyzed to 4-nitrophenol and CO2. The reaction was followed by measuring t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM233138(Butanohydrazide | Mr-I-33)
Affinity DataIC50:  1.40E+3nMpH: 5.0Assay Description:The assay was performed with plasmepsin-II/cathepsin D (1.2 nM) and substrate (malaria FRET-1; 1.0 μM) in 0.1 M sodium acetate buffer pH 5, contai...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM233142(1,2-Dipyridinylhydrazine | Mr-II-80)
Affinity DataIC50:  1.45E+3nMpH: 5.0Assay Description:The assay was performed with plasmepsin-II/cathepsin D (1.2 nM) and substrate (malaria FRET-1; 1.0 μM) in 0.1 M sodium acetate buffer pH 5, contai...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Bos taurus)
University of Karachi

LigandPNGBDBM222435(N'',N'''-Bis[(E)-(2,6-dichlorophenyl)methylide...)
Affinity DataIC50:  1.46E+3nMpH: 7.4 T: 2°CAssay Description:In this assay, 4-nitrophenyl acetate (4-NPA), a colorless compound, was hydrolyzed to 4-nitrophenol and CO2. The reaction was followed by measuring t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50001676(CHEMBL3237776 | Mr-I-27)
Affinity DataIC50:  1.50E+3nMpH: 5.0Assay Description:The assay was performed with plasmepsin-II/cathepsin D (1.2 nM) and substrate (malaria FRET-1; 1.0 μM) in 0.1 M sodium acetate buffer pH 5, contai...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM233140(2-Nitrobenzohydrazide | Mr-I-179)
Affinity DataIC50:  1.60E+3nMpH: 5.0Assay Description:The assay was performed with plasmepsin-II/cathepsin D (1.2 nM) and substrate (malaria FRET-1; 1.0 μM) in 0.1 M sodium acetate buffer pH 5, contai...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50001676(CHEMBL3237776 | Mr-I-27)
Affinity DataIC50:  1.65E+3nMpH: 5.0Assay Description:The assay was performed with plasmepsin-II/cathepsin D (1.2 nM) and substrate (malaria FRET-1; 1.0 μM) in 0.1 M sodium acetate buffer pH 5, contai...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Bos taurus)
University of Karachi

LigandPNGBDBM222429(N'',N'''-Bis[(E)-(2-nitrophenyl)methylidene]ca...)
Affinity DataIC50:  1.85E+3nMpH: 7.4 T: 2°CAssay Description:In this assay, 4-nitrophenyl acetate (4-NPA), a colorless compound, was hydrolyzed to 4-nitrophenol and CO2. The reaction was followed by measuring t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Bos taurus)
University of Karachi

LigandPNGBDBM10888(1,2-benzoxazol-3-ylmethanesulfonamide | CHEMBL750 ...)
Affinity DataIC50:  1.86E+3nMpH: 7.4 T: 2°CAssay Description:In this assay, 4-nitrophenyl acetate (4-NPA), a colorless compound, was hydrolyzed to 4-nitrophenol and CO2. The reaction was followed by measuring t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50362536(CHEMBL1941013)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human cathepsin D using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Bos taurus)
University of Karachi

LigandPNGBDBM222431(N'',N'''-Bis[(E)-(4-bromophenyl)methylidene]ca...)
Affinity DataIC50:  2.32E+3nMpH: 7.4 T: 2°CAssay Description:In this assay, 4-nitrophenyl acetate (4-NPA), a colorless compound, was hydrolyzed to 4-nitrophenol and CO2. The reaction was followed by measuring t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Bos taurus)
University of Karachi

LigandPNGBDBM222433(N'',N'''-Bis[(E)-(2-chlorophenyl)methylidene]c...)
Affinity DataIC50:  2.33E+3nMpH: 7.4 T: 2°CAssay Description:In this assay, 4-nitrophenyl acetate (4-NPA), a colorless compound, was hydrolyzed to 4-nitrophenol and CO2. The reaction was followed by measuring t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM233141(1,2-Diphenylhydrazine | Mr-II-10)
Affinity DataIC50:  2.40E+3nMpH: 5.0Assay Description:The assay was performed with plasmepsin-II/cathepsin D (1.2 nM) and substrate (malaria FRET-1; 1.0 μM) in 0.1 M sodium acetate buffer pH 5, contai...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM233142(1,2-Dipyridinylhydrazine | Mr-II-80)
Affinity DataIC50:  2.50E+3nMpH: 5.0Assay Description:The assay was performed with plasmepsin-II/cathepsin D (1.2 nM) and substrate (malaria FRET-1; 1.0 μM) in 0.1 M sodium acetate buffer pH 5, contai...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Bos taurus)
University of Karachi

LigandPNGBDBM222434(N'',N'''-Bis[(E)-(2,4-dichlorophenyl)methylide...)
Affinity DataIC50:  2.67E+3nMpH: 7.4 T: 2°CAssay Description:In this assay, 4-nitrophenyl acetate (4-NPA), a colorless compound, was hydrolyzed to 4-nitrophenol and CO2. The reaction was followed by measuring t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Bos taurus)
University of Karachi

LigandPNGBDBM222432(N'',N'''-Bis[(E)-(2-bromophenyl)methylidene]ca...)
Affinity DataIC50:  3.96E+3nMpH: 7.4 T: 2°CAssay Description:In this assay, 4-nitrophenyl acetate (4-NPA), a colorless compound, was hydrolyzed to 4-nitrophenol and CO2. The reaction was followed by measuring t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50362533(CHEMBL1941010)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin-2 using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50362535(CHEMBL1941012)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin-2 using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50362537(CHEMBL1941014)
Affinity DataIC50:  1.42E+4nMAssay Description:Inhibition of human cathepsin D using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50362536(CHEMBL1941013)
Affinity DataIC50:  1.47E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin-2 using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50362532(CHEMBL1941009)
Affinity DataIC50:  1.78E+4nMAssay Description:Inhibition of human cathepsin D using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50362529(CHEMBL1941006)
Affinity DataIC50:  1.96E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin-2 using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50362528(CHEMBL1941005)
Affinity DataIC50:  2.04E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin-2 using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50362530(CHEMBL1941007)
Affinity DataIC50:  2.12E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin-2 using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50362528(CHEMBL1941005)
Affinity DataIC50:  2.12E+4nMAssay Description:Inhibition of human cathepsin D using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50362538(CHEMBL1941015)
Affinity DataIC50:  2.12E+4nMAssay Description:Inhibition of human cathepsin D using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50362529(CHEMBL1941006)
Affinity DataIC50:  2.85E+4nMAssay Description:Inhibition of human cathepsin D using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50362532(CHEMBL1941009)
Affinity DataIC50:  3.05E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin-2 using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50362531(CHEMBL1941008)
Affinity DataIC50:  3.06E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin-2 using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50362530(CHEMBL1941007)
Affinity DataIC50:  3.19E+4nMAssay Description:Inhibition of human cathepsin D using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50362533(CHEMBL1941010)
Affinity DataIC50:  3.19E+4nMAssay Description:Inhibition of human cathepsin D using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50362538(CHEMBL1941015)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin-2 using DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS as substrate by FRET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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