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Found 2410 with Last Name = 'belle' and Initial = 'r'
TargetOxytocin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412919(CHEMBL475395)
Affinity DataKi:  0.794nMAssay Description:Antagonist activity at human oxytocin receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50326715(CHEMBL456263 | N-(6-methoxypyridin-3-yl)-1,2-dimet...)
Affinity DataKi:  0.794nMAssay Description:Displacement of 3H-oxytocin from human recombinant oxytocin receptor expressed in CHO cells by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412919(CHEMBL475395)
Affinity DataKi:  1.26nMAssay Description:Displacement of [3H]oxytocin from human oxytocin receptor expressed in CHO cells by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413725(CHEMBL456254)
Affinity DataKi:  1.58nMAssay Description:Binding affinity to human recombinant oxytocin receptor expressed in CHO cells by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413714(CHEMBL458635)
Affinity DataKi:  2nMAssay Description:Antagonist activity at human recombinant oxytocin receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132686(CHEMBL326466 | Dimethyl-((2S,3S)-3-naphthalen-2-yl...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]-citalopram from Serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413716(CHEMBL456464)
Affinity DataKi:  2.51nMAssay Description:Binding affinity to human recombinant oxytocin receptor expressed in CHO cells by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132687(CHEMBL324269 | [(2S,3S)-3-(6-Fluoro-naphthalen-2-y...)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]-citalopram from Serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132685(CHEMBL109571 | Dimethyl-(3-naphthalen-2-yl-bicyclo...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]-citalopram from Serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412915(CHEMBL514975)
Affinity DataKi:  3.16nMAssay Description:Antagonist activity at human oxytocin receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412936(CHEMBL481569)
Affinity DataKi:  3.16nMAssay Description:Antagonist activity at human oxytocin receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413713(CHEMBL458634)
Affinity DataKi:  3.16nMAssay Description:Antagonist activity at human recombinant oxytocin receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132679(CHEMBL111128 | Methyl-((2S,3S)-3-naphthalen-2-yl-b...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]-citalopram from Serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413717(CHEMBL515818)
Affinity DataKi:  3.98nMAssay Description:Binding affinity to human recombinant oxytocin receptor expressed in CHO cells by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132678(CHEMBL432022 | [(2S,3S)-3-(6-Fluoro-naphthalen-2-y...)
Affinity DataKi:  4.40nMAssay Description:Displacement of [3H]-citalopram from Serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132684(CHEMBL331799 | Methyl-(3-naphthalen-2-yl-bicyclo[2...)
Affinity DataKi:  4.90nMAssay Description:Displacement of [3H]-citalopram from Serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132677(CHEMBL109517 | Dimethyl-((2R,3R)-3-naphthalen-2-yl...)
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]-citalopram from Serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132683(6-((2S,3S)-3-Dimethylaminomethyl-bicyclo[2.2.1]hep...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]-WIN-35,428 from Dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413718(CHEMBL514586)
Affinity DataKi:  6.31nMAssay Description:Binding affinity to human recombinant oxytocin receptor expressed in CHO cells by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413715(CHEMBL457544)
Affinity DataKi:  6.31nMAssay Description:Binding affinity to human recombinant oxytocin receptor expressed in CHO cells by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413712(CHEMBL515660)
Affinity DataKi:  6.31nMAssay Description:Antagonist activity at human recombinant oxytocin receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataKi:  6.80nMAssay Description:Binding affinity to oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50026952((cis) [3-(3,4-Dichloro-phenyl)-bicyclo[2.2.2]oct-2...)
Affinity DataKi:  7.20nMAssay Description:In vitro inhibition of [3H]-NE re-uptake into synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413715(CHEMBL457544)
Affinity DataKi:  7.94nMAssay Description:Antagonist activity at human recombinant oxytocin receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413714(CHEMBL458635)
Affinity DataKi:  7.94nMAssay Description:Binding affinity to human recombinant oxytocin receptor expressed in CHO cells by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412921(CHEMBL473442)
Affinity DataKi:  7.94nMAssay Description:Antagonist activity at human oxytocin receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413712(CHEMBL515660)
Affinity DataKi:  10nMAssay Description:Binding affinity to human recombinant oxytocin receptor expressed in CHO cells by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413719(CHEMBL457998)
Affinity DataKi:  10nMAssay Description:Binding affinity to human recombinant oxytocin receptor expressed in CHO cells by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132680(CHEMBL322348 | [(2S,3S)-3-(6-Methoxy-naphthalen-2-...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-citalopram from Serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413723(CHEMBL458872)
Affinity DataKi:  12.6nMAssay Description:Binding affinity to human recombinant oxytocin receptor expressed in CHO cells by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413722(CHEMBL458654)
Affinity DataKi:  12.6nMAssay Description:Binding affinity to human recombinant oxytocin receptor expressed in CHO cells by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413721(CHEMBL514123)
Affinity DataKi:  12.6nMAssay Description:Binding affinity to human recombinant oxytocin receptor expressed in CHO cells by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50326715(CHEMBL456263 | N-(6-methoxypyridin-3-yl)-1,2-dimet...)
Affinity DataKi:  12.6nMAssay Description:Binding affinity to human recombinant oxytocin receptor expressed in CHO cells by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413720(CHEMBL515975)
Affinity DataKi:  12.6nMAssay Description:Binding affinity to human recombinant oxytocin receptor expressed in CHO cells by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413713(CHEMBL458634)
Affinity DataKi:  12.6nMAssay Description:Binding affinity to human recombinant oxytocin receptor expressed in CHO cells by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412930(CHEMBL482323)
Affinity DataKi:  15.8nMAssay Description:Antagonist activity at human oxytocin receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413714(CHEMBL458635)
Affinity DataKi:  15.8nMAssay Description:Antagonist activity at human recombinant vasopressin V1a receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132685(CHEMBL109571 | Dimethyl-(3-naphthalen-2-yl-bicyclo...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]-WIN-35,428 from Dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132684(CHEMBL331799 | Methyl-(3-naphthalen-2-yl-bicyclo[2...)
Affinity DataKi:  25nMAssay Description:In vitro inhibition of DA re-uptake into synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132681(CHEMBL323678 | [(2S,3S)-3-(6-Methoxy-naphthalen-2-...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]-citalopram from Serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132682(CHEMBL113136 | [(2S,3S)-3-(3-Chloro-phenyl)-bicycl...)
Affinity DataKi:  25nMAssay Description:In vitro ability of compound to inhibit 5-HT re-uptake of radiolabelled [3H]-tritium trasmitter into synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132686(CHEMBL326466 | Dimethyl-((2S,3S)-3-naphthalen-2-yl...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]-WIN-35,428 from Dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413713(CHEMBL458634)
Affinity DataKi:  25.1nMAssay Description:Antagonist activity at human recombinant vasopressin V1a receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50326715(CHEMBL456263 | N-(6-methoxypyridin-3-yl)-1,2-dimet...)
Affinity DataKi:  31.6nMAssay Description:Binding affinity to vasopressin V1b receptor by filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132677(CHEMBL109517 | Dimethyl-((2R,3R)-3-naphthalen-2-yl...)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]-WIN-35,428 from Dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413707(CHEMBL515384)
Affinity DataKi:  39.8nMAssay Description:Binding affinity to human recombinant oxytocin receptor expressed in CHO cells by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413708(CHEMBL514287)
Affinity DataKi:  39.8nMAssay Description:Binding affinity to human recombinant oxytocin receptor expressed in CHO cells by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412929(CHEMBL474621)
Affinity DataKi:  39.8nMAssay Description:Antagonist activity at human oxytocin receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132679(CHEMBL111128 | Methyl-((2S,3S)-3-naphthalen-2-yl-b...)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]-WIN-35,428 from Dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50026952((cis) [3-(3,4-Dichloro-phenyl)-bicyclo[2.2.2]oct-2...)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]-WIN-35,428 from Dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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