Compile Data Set for Download or QSAR
maximum 50k data
Found 74 with Last Name = 'burger' and Initial = 'am'
TargetAdenosine deaminase(Bos taurus (bovine))
University of Maryland Baltimore County

LigandPNGBDBM21955(4-amino-1-[(2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxym...)
Affinity DataKi:  1.06E+4nM ΔG°:  -28.4kJ/molepH: 7.0 T: 2°CAssay Description:The target compounds were screened against calf intestine ADA in vitro by monitoring the rate of hydrolyzing adenosine into inosine spectrophotometri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine deaminase(Bos taurus (bovine))
University of Maryland Baltimore County

LigandPNGBDBM21953(4-amino-1-[(2R,4S,5R)-4-hydroxy-5-(hydroxymethyl)o...)
Affinity DataKi:  1.21E+4nM ΔG°:  -28.1kJ/molepH: 7.0 T: 2°CAssay Description:The target compounds were screened against calf intestine ADA in vitro by monitoring the rate of hydrolyzing adenosine into inosine spectrophotometri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine deaminase(Bos taurus (bovine))
University of Maryland Baltimore County

LigandPNGBDBM21957(4-(hydrazinocarbonyl)-1-beta-D-ribofuranosyl-1H-im...)
Affinity DataKi:  2.65E+4nM ΔG°:  -26.1kJ/molepH: 7.0 T: 2°CAssay Description:The target compounds were screened against calf intestine ADA in vitro by monitoring the rate of hydrolyzing adenosine into inosine spectrophotometri...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine deaminase(Bos taurus (bovine))
University of Maryland Baltimore County

LigandPNGBDBM21956(7-amino-1-[(2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxym...)
Affinity DataKi:  5.14E+4nM ΔG°:  -24.5kJ/molepH: 7.0 T: 2°CAssay Description:The target compounds were screened against calf intestine ADA in vitro by monitoring the rate of hydrolyzing adenosine into inosine spectrophotometri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine deaminase(Bos taurus (bovine))
University of Maryland Baltimore County

LigandPNGBDBM21954(7-amino-1-[(2R,4S,5R)-4-hydroxy-5-(hydroxymethyl)o...)
Affinity DataKi:  5.20E+4nM ΔG°:  -24.5kJ/molepH: 7.0 T: 2°CAssay Description:The target compounds were screened against calf intestine ADA in vitro by monitoring the rate of hydrolyzing adenosine into inosine spectrophotometri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50012278((2ALPHA,2''BETA,3BETA,4ALPHA,5BETA)-VINCALEUKOBLAS...)
Affinity DataIC50:  130nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474288(CHEMBL112192)
Affinity DataIC50:  220nMAssay Description:In vitro inhibitory concentration required to displace [3H]colchicine from its binding site on tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50035218(CHEMBL61 | PODOFILOX | Podophyllinic acid lactone ...)
Affinity DataIC50:  350nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474300(CHEMBL116173)
Affinity DataIC50:  370nMAssay Description:In vitro inhibitory concentration required to displace [3H]colchicine from its binding site on TubulinMore data for this Ligand-Target Pair
TargetTubulin beta-2B chain(Bos taurus)
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50107672((3-Fluoro-phenyl)-(5-methoxy-1H-indol-2-yl)-methan...)
Affinity DataIC50:  390nMAssay Description:Inhibition of tubulin polymerization.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474288(CHEMBL112192)
Affinity DataIC50:  430nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474290(CHEMBL115499)
Affinity DataIC50:  480nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta-2B chain(Bos taurus)
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50107658((5-Methoxy-1H-indol-2-yl)-phenyl-methanone | (5-me...)
Affinity DataIC50:  530nMAssay Description:Inhibition of tubulin polymerization.More data for this Ligand-Target Pair
TargetTubulin beta-2B chain(Bos taurus)
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50107678((5-Methoxy-1H-indol-2-yl)-(3-methoxy-phenyl)-metha...)
Affinity DataIC50:  530nMAssay Description:Inhibition of tubulin polymerization.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474293(CHEMBL324797)
Affinity DataIC50:  630nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474298(CHEMBL321632)
Affinity DataIC50:  630nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta-2B chain(Bos taurus)
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50107677((3-Hydroxy-phenyl)-(5-methoxy-1H-indol-2-yl)-metha...)
Affinity DataIC50:  660nMAssay Description:Inhibition of tubulin polymerization.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474300(CHEMBL116173)
Affinity DataIC50:  670nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474308(CHEMBL112385)
Affinity DataIC50:  760nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM97233(CHEMBL9514 | MLS001164242 | N-[6-(2-thenoyl)-1H-be...)
Affinity DataIC50:  760nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
TargetTubulin beta-2B chain(Bos taurus)
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50107656((3,5-Dimethoxy-phenyl)-(5-methoxy-1H-indol-2-yl)-m...)
Affinity DataIC50:  810nMAssay Description:Inhibition of tubulin polymerization.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta-2B chain(Bos taurus)
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50107676((3,4-Dimethoxy-phenyl)-(5-methoxy-1H-indol-2-yl)-m...)
Affinity DataIC50:  810nMAssay Description:Inhibition of tubulin polymerization.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta-2B chain(Bos taurus)
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50107664((5-Methoxy-1H-indol-2-yl)-(3-nitro-phenyl)-methano...)
Affinity DataIC50:  850nMAssay Description:Inhibition of tubulin polymerization.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta-2B chain(Bos taurus)
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50107674(Butyric acid 3-(5-methoxy-1H-indole-2-carbonyl)-ph...)
Affinity DataIC50:  850nMAssay Description:Inhibition of tubulin polymerization.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta-2B chain(Bos taurus)
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50107693((5-Methyl-1H-indol-2-yl)-(3,4,5-trimethoxy-phenyl)...)
Affinity DataIC50:  860nMAssay Description:Inhibition of tubulin polymerization.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474286(CHEMBL419387)
Affinity DataIC50:  910nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474287(CHEMBL115488)
Affinity DataIC50:  910nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta-2B chain(Bos taurus)
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50107651((5-Methoxy-1H-indol-2-yl)-(3,4,5-trimethoxy-phenyl...)
Affinity DataIC50:  990nMAssay Description:Inhibition of tubulin polymerization.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta-2B chain(Bos taurus)
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50107662((3-Amino-phenyl)-(5-methoxy-1H-indol-2-yl)-methano...)
Affinity DataIC50:  990nMAssay Description:Inhibition of tubulin polymerization.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta-2B chain(Bos taurus)
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50107663((2-Fluoro-phenyl)-(5-methoxy-1H-indol-2-yl)-methan...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of tubulin polymerization.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50469124(CHEMBL113332)
Affinity DataIC50:  1.20E+3nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50014846((S)-N-(5,6,7,9-tetrahydro-1,2,3,10-tetramethoxy-9-...)
Affinity DataIC50:  1.26E+3nMAssay Description:In vitro inhibitory concentration required to displace [3H]colchicine from its binding site on tubulinMore data for this Ligand-Target Pair
TargetTubulin beta-2B chain(Bos taurus)
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50107670((5-Methoxy-1H-indol-2-yl)-(2-methoxy-phenyl)-metha...)
Affinity DataIC50:  1.29E+3nMAssay Description:Inhibition of tubulin polymerization.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50014846((S)-N-(5,6,7,9-tetrahydro-1,2,3,10-tetramethoxy-9-...)
Affinity DataIC50:  1.40E+3nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
TargetTubulin beta-2B chain(Bos taurus)
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50107671((5-Methoxy-1H-indol-2-yl)-(3-trifluoromethyl-pheny...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of tubulin polymerization.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta-2B chain(Bos taurus)
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50107680((5-Methoxy-1H-indol-2-yl)-p-tolyl-methanone | CHEM...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of tubulin polymerization.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta-2B chain(Bos taurus)
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50107682((5-Methoxy-1H-indol-2-yl)-(3-trifluoromethoxy-phen...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of tubulin polymerization.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474291(CHEMBL326388)
Affinity DataIC50:  1.70E+3nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474294(CHEMBL115360)
Affinity DataIC50:  1.80E+3nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta-2B chain(Bos taurus)
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50107673((3-Difluoromethylsulfanyl-phenyl)-(5-methoxy-1H-in...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of tubulin polymerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474292(CHEMBL114642)
Affinity DataIC50:  2.30E+3nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474307(CHEMBL114651)
Affinity DataIC50:  2.50E+3nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta-2B chain(Bos taurus)
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50107661((3,4-Dichloro-phenyl)-(5-methoxy-1H-indol-2-yl)-me...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of tubulin polymerization.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474306(CHEMBL326114)
Affinity DataIC50:  2.60E+3nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta-2B chain(Bos taurus)
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50107653((2-Methoxy-phenyl)-(5-methyl-1H-indol-2-yl)-methan...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of tubulin polymerization.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta-2B chain(Bos taurus)
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50107652((4-Bromo-phenyl)-(5-methoxy-1H-indol-2-yl)-methano...)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of tubulin polymerization.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474299(CHEMBL267340)
Affinity DataIC50:  4.40E+3nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta-2B chain(Bos taurus)
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50107695((5-Methoxy-1H-indol-2-yl)-o-tolyl-methanone | CHEM...)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of tubulin polymerization.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta-2B chain(Bos taurus)
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50107654((4-Chloro-phenyl)-(5-methoxy-1H-indol-2-yl)-methan...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of tubulin polymerization.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta-2B chain(Bos taurus)
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50107667((2,5-Dimethyl-phenyl)-(5-methoxy-1H-indol-2-yl)-me...)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of tubulin polymerization.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 74 total ) | Next | Last >>
Jump to: