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Found 267 with Last Name = 'gresh' and Initial = 'n'
TargetMannose-6-phosphate isomerase(Saccharomyces cerevisiae)
Univ Paris-Sud

Curated by ChEMBL
LigandPNGBDBM50481224(CHEMBL611642)
Affinity DataKi:  1.05E+4nMAssay Description:Inhibition of Saccharomyces cerevisiae type I phosphomannose isomerase assessed as D-mannose 6-phosphate to D-fructose 6-phosphate isomerization at p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMannose-6-phosphate isomerase(Escherichia coli (strain K12))
Univ Paris-Sud

Curated by ChEMBL
LigandPNGBDBM50481224(CHEMBL611642)
Affinity DataKi:  1.15E+5nMAssay Description:Inhibition of Escherichia coli type I phosphomannose isomerase assessed as D-mannose 6-phosphate to D-fructose 6-phosphate isomerization at pH 7.1 by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM19126((1R,3R,6R,7S,8R,10S,11S,14R,15R,20S)-18-[(2S)-buta...)
Affinity DataIC50:  2nMAssay Description:Inhibition of AChE activity was determined by the spectroscopic method of Ellman using acetylthiocholine iodide as substrate, in 96-well microtiter p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM19125((1R,3R,6R,7S,8R,10S,11S,14R,15R,20S)-7-[(1S)-1-(di...)
Affinity DataIC50:  2nMAssay Description:Inhibition of AChE activity was determined by the spectroscopic method of Ellman using acetylthiocholine iodide as substrate, in 96-well microtiter p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Cnrs Umr 176

Curated by ChEMBL
LigandPNGBDBM50300042(4-[(2S)-2-{[(1S)-1-{[(1S)-1,2-dicarbamoylethyl]car...)
Affinity DataIC50:  11nMAssay Description:Inhibition of Grb2 by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Cnrs Umr 176

Curated by ChEMBL
LigandPNGBDBM50080832(CHEMBL334099 | [1-[1-(1,2-Dicarbamoyl-ethylcarbamo...)
Affinity DataIC50:  11nMAssay Description:The compound was evaluated for its potency to inhibit the interaction between Growth factor receptor bound protein 2 and phosphotyrosine-containing p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Cnrs

LigandPNGBDBM19110((3R,6R,7S,8R,10S,11R,14R,15S,20S)-18-[(2S)-butan-2...)
Affinity DataIC50:  13nMpH: 8.0 T: 2°CAssay Description:Inhibition of AChE activity was determined by the spectroscopic method of Ellman using acetylthiocholine iodide as substrate, in 96-well microtiter p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Cnrs

LigandPNGBDBM19126((1R,3R,6R,7S,8R,10S,11S,14R,15R,20S)-18-[(2S)-buta...)
Affinity DataIC50:  14nMAssay Description:Inhibition of AChE activity was determined by the spectroscopic method of Ellman using acetylthiocholine iodide as substrate, in 96-well microtiter p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50424266(CHEMBL2314466)
Affinity DataIC50:  17nMAssay Description:Inhibition of recombinant human CDK5/p25 after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Cnrs

LigandPNGBDBM19125((1R,3R,6R,7S,8R,10S,11S,14R,15R,20S)-7-[(1S)-1-(di...)
Affinity DataIC50:  18nMAssay Description:Inhibition of AChE activity was determined by the spectroscopic method of Ellman using acetylthiocholine iodide as substrate, in 96-well microtiter p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50424264(CHEMBL2314464)
Affinity DataIC50:  21nMAssay Description:Inhibition of recombinant human CDK5/p25 after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50424270(CHEMBL2314471)
Affinity DataIC50:  22nMAssay Description:Inhibition of recombinant human CDK5/p25 after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50424272(CHEMBL2314473)
Affinity DataIC50:  25nMAssay Description:Inhibition of recombinant human CDK5/p25 after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Cnrs

LigandPNGBDBM19111((3R,6R,7S,8R,10S,11R,14R,15S,20S)-18-(butan-2-yl)-...)
Affinity DataIC50:  27nMpH: 8.0 T: 2°CAssay Description:Inhibition of AChE activity was determined by the spectroscopic method of Ellman using acetylthiocholine iodide as substrate, in 96-well microtiter p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Cnrs

LigandPNGBDBM19129((3R,6R,7S,8R,10S,11R,14R,15R,20S)-18-[(2S)-butan-2...)
Affinity DataIC50:  28nMAssay Description:Inhibition of AChE activity was determined by the spectroscopic method of Ellman using acetylthiocholine iodide as substrate, in 96-well microtiter p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Cnrs

LigandPNGBDBM19101((3R,6R,7S,8R,10S,11R,14R,15S,20S)-7-[(1S)-1-(dimet...)
Affinity DataIC50:  31nMpH: 8.0 T: 2°CAssay Description:Inhibition of AChE activity was determined by the spectroscopic method of Ellman using acetylthiocholine iodide as substrate, in 96-well microtiter p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50424294(CHEMBL2314447)
Affinity DataIC50:  38nMAssay Description:Inhibition of recombinant human CDK5/p25 after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50424282(CHEMBL2314436)
Affinity DataIC50:  41nMAssay Description:Inhibition of recombinant human CDK5/p25 after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50424296(CHEMBL2314449)
Affinity DataIC50:  42nMAssay Description:Inhibition of recombinant human CDK5/p25 after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50424283(CHEMBL2314435)
Affinity DataIC50:  42nMAssay Description:Inhibition of recombinant human CDK5/p25 after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50424265(CHEMBL2314467)
Affinity DataIC50:  50nMAssay Description:Inhibition of recombinant human CDK5/p25 after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Cnrs

LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  58nMAssay Description:Inhibition of BuChE activity was determined by the spectroscopic method of Ellman using butyrylthiocholine iodide as substrate, in 96-well microtiter...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50424284(CHEMBL2314437)
Affinity DataIC50:  60nMAssay Description:Inhibition of recombinant human CDK5/p25 after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50267086(Adociaquinone B | CHEMBL476648)
Affinity DataIC50:  70nMAssay Description:Inhibition of human recombinant CDC25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Cnrs

LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  74nMAssay Description:Inhibition of AChE activity was determined by the spectroscopic method of Ellman using acetylthiocholine iodide as substrate, in 96-well microtiter p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50424295(CHEMBL2314448)
Affinity DataIC50:  76nMAssay Description:Inhibition of recombinant human CDK5/p25 after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50244787((R)-2-(1-Hydroxybut-2-ylamino)-6-[3-(2-pyridyl)phe...)
Affinity DataIC50:  80nMAssay Description:Inhibition of recombinant human CDK5/p25 after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50424271(CHEMBL2314472)
Affinity DataIC50:  90nMAssay Description:Inhibition of recombinant human CDK5/p25 after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50424279(CHEMBL2314434)
Affinity DataIC50:  100nMAssay Description:Inhibition of recombinant human CDK5/p25 after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Cnrs

LigandPNGBDBM19112((3R,6R,7S,8R,10S,11R,14R,15S,20S)-7-[(1S)-1-(dimet...)
Affinity DataIC50:  102nMpH: 8.0 T: 2°CAssay Description:Inhibition of AChE activity was determined by the spectroscopic method of Ellman using acetylthiocholine iodide as substrate, in 96-well microtiter p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Cnrs

LigandPNGBDBM19104((2S)-N-[(1R,6S,7S,8R,11R,12S,14R,15S,16R)-15-[(1S)...)
Affinity DataIC50:  105nMpH: 8.0 T: 2°CAssay Description:Inhibition of AChE activity was determined by the spectroscopic method of Ellman using acetylthiocholine iodide as substrate, in 96-well microtiter p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Cnrs

LigandPNGBDBM19122((3R,6R,7S,8R,10S,11R,14R,15S,20S)-8-hydroxy-6,10,1...)
Affinity DataIC50:  106nMAssay Description:Inhibition of AChE activity was determined by the spectroscopic method of Ellman using acetylthiocholine iodide as substrate, in 96-well microtiter p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Cnrs

LigandPNGBDBM19120((3R,6R,7S,8R,10S,11R,14R,15S,20S)-7-[(1S)-1-(dimet...)
Affinity DataIC50:  110nMAssay Description:Inhibition of AChE activity was determined by the spectroscopic method of Ellman using acetylthiocholine iodide as substrate, in 96-well microtiter p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Cnrs

LigandPNGBDBM19121(N-[(6S,7S,8R,11S,12S,14R,15S,16R)-14-hydroxy-7-(hy...)
Affinity DataIC50:  110nMAssay Description:Inhibition of AChE activity was determined by the spectroscopic method of Ellman using acetylthiocholine iodide as substrate, in 96-well microtiter p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Cnrs

LigandPNGBDBM19118((1S,6R,7S,8R,10S,11S,14R,15S,20S)-7-[(1S)-1-(dimet...)
Affinity DataIC50:  110nMAssay Description:Inhibition of AChE activity was determined by the spectroscopic method of Ellman using acetylthiocholine iodide as substrate, in 96-well microtiter p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Cnrs Umr 176

Curated by ChEMBL
LigandPNGBDBM50080831(CHEMBL434413 | [1-[1-(1,2-Dicarbamoyl-ethylcarbamo...)
Affinity DataIC50:  120nMAssay Description:The compound was evaluated for its potency to inhibit the interaction between Growth factor receptor bound protein 2 and phosphotyrosine-containing p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Cnrs

LigandPNGBDBM19105(N-[(1R,6S,7S,8R,11R,12S,14R,15S,16R)-15-[(1S)-1-(d...)
Affinity DataIC50:  120nMpH: 8.0 T: 2°CAssay Description:Inhibition of AChE activity was determined by the spectroscopic method of Ellman using acetylthiocholine iodide as substrate, in 96-well microtiter p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50420297(CHEMBL2089032)
Affinity DataIC50:  150nMAssay Description:Inhibition of human recombinant CDK9/cyclin T expressed in baculovirus-infected insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50420301(CHEMBL2089036)
Affinity DataIC50:  150nMAssay Description:Inhibition of CK1 after 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Cnrs Umr 176

Curated by ChEMBL
LigandPNGBDBM50080836(4-[2-[2-(3-Amino-benzyloxycarbonylamino)-3-(4-phos...)
Affinity DataIC50:  153nMAssay Description:The compound was evaluated for its potency to inhibit the interaction between Growth factor receptor bound protein 2 and phosphotyrosine-containing p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  157nMAssay Description:Inhibition of AChE activity was determined by the spectroscopic method of Ellman using acetylthiocholine iodide as substrate, in 96-well microtiter p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50420301(CHEMBL2089036)
Affinity DataIC50:  180nMAssay Description:Inhibition of human recombinant CDK9/cyclin T expressed in baculovirus-infected insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50420297(CHEMBL2089032)
Affinity DataIC50:  180nMAssay Description:Inhibition of CK1 after 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50424292(CHEMBL2314445)
Affinity DataIC50:  180nMAssay Description:Inhibition of recombinant human CDK5/p25 after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50420301(CHEMBL2089036)
Affinity DataIC50:  180nMAssay Description:Inhibition of human recombinant CDK5/p25 expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50420297(CHEMBL2089032)
Affinity DataIC50:  190nMAssay Description:Inhibition of human recombinant CDK5/p25 expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Cnrs Umr 176

Curated by ChEMBL
LigandPNGBDBM50080834(CHEMBL409455 | {4-[2-[2-(3-Amino-benzyloxycarbonyl...)
Affinity DataIC50:  198nMAssay Description:The compound was evaluated for its potency to inhibit the interaction between Growth factor receptor bound protein 2 and phosphotyrosine-containing p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50424263(CHEMBL2314465)
Affinity DataIC50:  200nMAssay Description:Inhibition of recombinant human CDK5/p25 after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM7533((2R)-2-[[6-(benzylamino)-9-isopropyl-purin-2-yl]am...)
Affinity DataIC50:  200nMAssay Description:Inhibition of recombinant human CDK5/p25 after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50424280(CHEMBL2311568)
Affinity DataIC50:  200nMAssay Description:Inhibition of recombinant human CDK5/p25 after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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