TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 0.0730nMAssay Description:Displacement of [3H]CGP12177 from human beta2 adrenoceptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 0.160nMAssay Description:Displacement of [3H]CGP12177 from human beta2 adrenoceptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 0.320nMAssay Description:Displacement of [3H]CGP12177 from human beta2 adrenoceptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 0.490nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.720nMAssay Description:Displacement of [3H]spiperone from human dopamine D4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.960nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]CGP12177 from human beta2 adrenoceptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]CGP12177 from human beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]CGP12177 from human beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR expressed in human recombinant SH-SY5Y cell membranes after 120 minsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR expressed in human recombinant SH-SY5Y cell membranes after 120 minsMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 2.60nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 3.40nMAssay Description:Displacement of [3H]CGP12177 from human beta2 adrenoceptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 4.90nMAssay Description:Displacement of [3H]N-methyl-scopolamine bromide from human recombinant muscarinic M2 receptor expressed in HEK293T cell membranes after 1 hr by liqu...More data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 5.30nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 6.80nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Displacement of [3H]spiperone from human dopamine D4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Displacement of [3H]CGP12177 from human beta2 adrenoceptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 23nMAssay Description:Displacement of [3H]N-methyl-scopolamine bromide from human recombinant muscarinic M1 receptor expressed in HEK293T cell membranes after 1 hr by liqu...More data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 29nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 41nMAssay Description:Displacement of [3H]N-methyl-scopolamine bromide from human recombinant muscarinic M3 receptor expressed in HEK293T cell membranes after 1 hr by liqu...More data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 49nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 49nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 51nMAssay Description:Displacement of [3H]CGP12177 from human beta2 adrenoceptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 55nMAssay Description:Displacement of [3H]CGP12177 from human beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 57nMAssay Description:Displacement of [3H]CGP12177 from human beta2 adrenoceptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 63nMAssay Description:Displacement of [3H]N-methyl-scopolamine bromide from human recombinant muscarinic M1 receptor expressed in HEK293T cell membranes after 1 hr by liqu...More data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 71nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 89nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 140nMAssay Description:Displacement of [3H]N-methyl-scopolamine bromide from human recombinant muscarinic M2 receptor expressed in HEK293T cell membranes after 1 hr by liqu...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 140nMAssay Description:Displacement of [3H]N-methyl-scopolamine bromide from human recombinant muscarinic M3 receptor expressed in HEK293T cell membranes after 1 hr by liqu...More data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 150nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 170nMAssay Description:Displacement of [3H]N-methyl-scopolamine bromide from human recombinant muscarinic M1 receptor expressed in HEK293T cell membranes after 1 hr by liqu...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR expressed in human recombinant SH-SY5Y cell membranes after 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 210nMAssay Description:Displacement of [3H]N-methyl-scopolamine bromide from human recombinant muscarinic M3 receptor expressed in HEK293T cell membranes after 1 hr by liqu...More data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 220nMAssay Description:Displacement of [3H]CGP12177 from human beta2 adrenoceptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 220nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 220nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair