Compile Data Set for Download or QSAR
maximum 50k data
Found 40 with Last Name = 'koo' and Initial = 'ka'
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278826(4-(4-(4-hydroxy-3-methoxybenzylidene)-3,5-dioxopyr...)
Affinity DataIC50:  600nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278753(1-(3,4-dichlorophenyl)-4-(4-hydroxy-3-nitrobenzyli...)
Affinity DataIC50:  600nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278086(4-(4-hydroxy-3-methoxybenzylidene)-1-(4-methoxyphe...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50187069(1-(3,4-dichlorophenyl)-4-(4-hydroxy-3-methoxybenzy...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278211(1-(4-fluorophenyl)-4-(4-hydroxy-3-methoxybenzylide...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278598(1-(3,4-dichlorophenyl)-4-(4-hydroxybenzylidene)pyr...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosinase(Homo sapiens (Human))
Amorepacific

Curated by ChEMBL
LigandPNGBDBM50109690(3,4,5-Trihydroxy-benzoic acid 2-(4-hydroxy-phenyl)...)
Affinity DataIC50:  4.93E+3nMAssay Description:Inhibition of tyrosinase in Melan-a cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278752(1-(3,4-dichlorophenyl)-4-(3,4-difluorobenzylidene)...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM7533((2R)-2-[[6-(benzylamino)-9-isopropyl-purin-2-yl]am...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosinase(Homo sapiens (Human))
Amorepacific

Curated by ChEMBL
LigandPNGBDBM50219503(2-hydroxyphenethyl 3,4,5-trihydroxybenzoate | CHEM...)
Affinity DataIC50:  1.45E+4nMAssay Description:Inhibition of tyrosinase in Melan-a cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278684(4-(2,3-dichlorobenzylidene)-1-(3,4-dichlorophenyl)...)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosinase(Homo sapiens (Human))
Amorepacific

Curated by ChEMBL
LigandPNGBDBM50219504(3-hydroxyphenethyl 3,4,5-trihydroxybenzoate | CHEM...)
Affinity DataIC50:  1.52E+4nMAssay Description:Inhibition of tyrosinase in Melan-a cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278636(4-(2-chlorobenzylidene)-1-(3,4-dichlorophenyl)pyra...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278599(4-(4-chlorobenzylidene)-1-(3,4-dichlorophenyl)pyra...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278682(1-(3,4-dichlorophenyl)-4-(3,5-dimethoxybenzylidene...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278210(1-(4-fluorophenyl)-4-(3-hydroxy-4-methoxybenzylide...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosinase(Homo sapiens (Human))
Amorepacific

Curated by ChEMBL
LigandPNGBDBM50219502(4-hydroxyphenyl beta-D-glucopyranoside | Arbutin |...)
Affinity DataIC50:  3.03E+4nMAssay Description:Inhibition of tyrosinase in Melan-a cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278755(4-(4-(2-methoxybenzylidene)-3,5-dioxopyrazolidin-1...)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278754(1-(3,4-dichlorophenyl)-4-(4-hydroxy-3,5-dimethoxyb...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278601(1-(3,4-dichlorophenyl)-4-(3-methoxybenzylidene)pyr...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278828(4-(2-methoxybenzylidene)-1-(4-methoxyphenyl)pyrazo...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278829(4-(3-methoxybenzylidene)-1-(4-methoxyphenyl)pyrazo...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278830(4-(2-fluorobenzylidene)-1-(4-methoxyphenyl)pyrazol...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278831(4-(2,3-dichlorobenzylidene)-1-(4-methoxyphenyl)pyr...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278083(4-(3,5-dimethoxybenzylidene)-1-(4-methoxyphenyl)py...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278084(4-(3,5-dihydroxybenzylidene)-1-(4-methoxyphenyl)py...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278085(4-(3-hydroxy-4-methoxybenzylidene)-1-(4-methoxyphe...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278087(4-(4-hydroxy-3,5-dimethoxybenzylidene)-1-(4-methox...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278144(1-(4-fluorophenyl)-4-(2-methoxybenzylidene)pyrazol...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278602(1-(3,4-dichlorophenyl)-4-(2-methoxybenzylidene)pyr...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278600(1-(3,4-dichlorophenyl)-4-(4-methoxybenzylidene)pyr...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278597(4-benzylidene-1-(3,4-dichlorophenyl)pyrazolidine-3...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278685(4-(2,6-dichlorobenzylidene)-1-(3,4-dichlorophenyl)...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278683(1-(3,4-dichlorophenyl)-4-(3,5-dihydroxybenzylidene...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278681(1-(3,4-dichlorophenyl)-4-(2,4-dimethoxybenzylidene...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278639(1-(3,4-dichlorophenyl)-4-(3,4-dimethoxybenzylidene...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278638(1-(3,4-dichlorophenyl)-4-(3-hydroxy-4-methoxybenzy...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278637(1-(3,4-dichlorophenyl)-4-(2-fluorobenzylidene)pyra...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278635(1-(3,4-dichlorophenyl)-4-(2-nitrobenzylidene)pyraz...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University

Curated by ChEMBL
LigandPNGBDBM50278827(4-(4-(3-hydroxy-4-methoxybenzylidene)-3,5-dioxopyr...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed