Affinity DataKi: 0.0603nMAssay Description:Binding affinity in Nluc-hH3R assessed in HEK293 cells by NanoBRET binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.158nMAssay Description:Binding affinity in Nluc-hH3R assessed in HEK293 cells by NanoBRET binding assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Displacement of [3H]-Diprenorphine from human mu opioid receptor expressed in HEK293-TSA cell membranes after 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.209nMAssay Description:Displacement of [3H]UR-P1294 from human H3R receptor expressed in HEK293 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.275nMAssay Description:Displacement of [3H]UR-P1294 from human H3R receptor expressed in HEK293 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
UniversitÄT Heidelberg
Curated by PDSP Ki Database
UniversitÄT Heidelberg
Curated by PDSP Ki Database
Affinity DataKi: 0.302nMAssay Description:Displacement of [3H]UR-P1294 from human H3R receptor expressed in HEK293 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.398nMAssay Description:Displacement of [3H]UR-P1294 from human H3R receptor expressed in HEK293 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
UniversitÄT Heidelberg
Curated by PDSP Ki Database
UniversitÄT Heidelberg
Curated by PDSP Ki Database
Affinity DataKi: 0.501nMAssay Description:Binding affinity in Nluc-hH3R assessed in HEK293 cells by NanoBRET binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.631nMAssay Description:Binding affinity in Nluc-hH3R assessed in HEK293T cells by NanoBRET binding assayMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
TargetAdenosine receptor A1(Rattus norvegicus (rat))
UniversitÄT Heidelberg
Curated by PDSP Ki Database
UniversitÄT Heidelberg
Curated by PDSP Ki Database
TargetAdenosine receptor A1(Rattus norvegicus (rat))
UniversitÄT Heidelberg
Curated by PDSP Ki Database
UniversitÄT Heidelberg
Curated by PDSP Ki Database
Affinity DataKi: 0.800nMAssay Description:Binding affinity against low affinity component of adenosine A1 receptors from rat brain membranes using [3H]-DPCPXMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
UniversitÄT Heidelberg
Curated by PDSP Ki Database
UniversitÄT Heidelberg
Curated by PDSP Ki Database
Affinity DataKi: 0.800nMAssay Description:Displacement of [3H]PIA from adenosine A1 receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
Affinity DataKi: 0.912nMAssay Description:Binding affinity in Nluc-hH3R assessed in HEK293 cells by NanoBRET binding assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
UniversitÄT Heidelberg
Curated by PDSP Ki Database
UniversitÄT Heidelberg
Curated by PDSP Ki Database
Affinity DataKi: 1nMAssay Description:Binding affinity against high affinity component of adenosine A1 receptors from rat brain membranes using [3H]DPCPXMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
TargetAdenosine receptor A1(Rattus norvegicus (rat))
UniversitÄT Heidelberg
Curated by PDSP Ki Database
UniversitÄT Heidelberg
Curated by PDSP Ki Database
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]PIA from adenosine A1 receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
UniversitÄT Heidelberg
Curated by PDSP Ki Database
UniversitÄT Heidelberg
Curated by PDSP Ki Database
TargetAdenosine receptor A1(Rattus norvegicus (rat))
UniversitÄT Heidelberg
Curated by PDSP Ki Database
UniversitÄT Heidelberg
Curated by PDSP Ki Database
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]PIA from adenosine A1 receptor of rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]UR-P1294 from human H3R receptor expressed in HEK293 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
Affinity DataKi: 2.5nMAssay Description:Binding affinity in Nluc-hH3R assessed in HEK293T cells by NanoBRET binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity in Nluc-hH3R assessed in HEK293T cells by NanoBRET binding assayMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
Affinity DataKi: 2.80nMAssay Description:Inhibition of adenylate cyclase via adenosine A1 receptors in rat fat cell membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
UniversitÄT Heidelberg
Curated by PDSP Ki Database
UniversitÄT Heidelberg
Curated by PDSP Ki Database
Affinity DataKi: 3.60nMAssay Description:Binding affinity against adenosine A2 receptor from rat striatal membranes with 50 nM CPA using [3H]-NECAMore data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Binding affinity against adenosine A2 receptor from rat striatal membranes with 50 nM CPA using [3H]-NECAMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
TargetAdenosine receptor A1(Rattus norvegicus (rat))
UniversitÄT Heidelberg
Curated by PDSP Ki Database
UniversitÄT Heidelberg
Curated by PDSP Ki Database
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
UniversitÄT WÜRzburg
Curated by PDSP Ki Database