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Found 105 with Last Name = 'lyons' and Initial = 'dm'
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445263(CHEMBL3103651)
Affinity DataIC50:  400nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445286(CHEMBL3103907)
Affinity DataIC50:  510nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445279(CHEMBL3103914)
Affinity DataIC50:  530nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445276(CHEMBL3103917)
Affinity DataIC50:  550nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445285(CHEMBL3103908)
Affinity DataIC50:  600nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445259(CHEMBL3103655)
Affinity DataIC50:  630nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445267(CHEMBL3103647)
Affinity DataIC50:  640nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445280(CHEMBL3103913)
Affinity DataIC50:  780nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445303(CHEMBL3102870)
Affinity DataIC50:  790nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445277(CHEMBL3103916)
Affinity DataIC50:  930nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275059((Z)-1-(Benzo[b]thiophen-3-ylmethylene)-6-methyl-4-...)
Affinity DataIC50:  970nMAssay Description:Inhibition of recombinant perforin mediated lysis of human Jurkat cells pre-incubated for 30 mins with perforin followed by incubation with Jurkat ce...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50347203(CHEMBL1795754)
Affinity DataIC50:  1.04E+3nMAssay Description:Inhibition of recombinant perforin mediated lysis of human Jurkat cells pre-incubated for 30 mins with perforin followed by incubation with Jurkat ce...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445268(CHEMBL3103646)
Affinity DataIC50:  1.14E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445307(CHEMBL3104019)
Affinity DataIC50:  1.15E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445281(CHEMBL3103912)
Affinity DataIC50:  1.17E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445283(CHEMBL3103910)
Affinity DataIC50:  1.18E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445278(CHEMBL3103915)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445270(CHEMBL3103644)
Affinity DataIC50:  1.38E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445255(CHEMBL3103900)
Affinity DataIC50:  1.45E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445284(CHEMBL3103909)
Affinity DataIC50:  1.52E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445302(CHEMBL3104023)
Affinity DataIC50:  1.56E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445258(CHEMBL3103897)
Affinity DataIC50:  1.58E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445304(CHEMBL3104022)
Affinity DataIC50:  1.62E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445256(CHEMBL3103899)
Affinity DataIC50:  1.66E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445306(CHEMBL3104020)
Affinity DataIC50:  1.67E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445308(CHEMBL3104018)
Affinity DataIC50:  1.69E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445269(CHEMBL3103645)
Affinity DataIC50:  1.89E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445266(CHEMBL3103648)
Affinity DataIC50:  2.33E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445288(CHEMBL3103905)
Affinity DataIC50:  2.44E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445257(CHEMBL3103898)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445287(CHEMBL3103906)
Affinity DataIC50:  2.55E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445254(CHEMBL3103641)
Affinity DataIC50:  2.55E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50347206(CHEMBL1795762)
Affinity DataIC50:  2.87E+3nMAssay Description:Inhibition of recombinant perforin mediated lysis of human Jurkat cells pre-incubated for 30 mins with perforin followed by incubation with Jurkat ce...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445262(CHEMBL3103652)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50347209(CHEMBL1795769)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of recombinant perforin mediated lysis of human Jurkat cells pre-incubated for 30 mins with perforin followed by incubation with Jurkat ce...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445301(CHEMBL3104024)
Affinity DataIC50:  3.03E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445305(CHEMBL3104021)
Affinity DataIC50:  3.04E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50347212(CHEMBL1795772)
Affinity DataIC50:  3.08E+3nMAssay Description:Inhibition of recombinant perforin mediated lysis of human Jurkat cells pre-incubated for 30 mins with perforin followed by incubation with Jurkat ce...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445309(CHEMBL3104017)
Affinity DataIC50:  3.09E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50347202(CHEMBL1795771)
Affinity DataIC50:  3.16E+3nMAssay Description:Inhibition of recombinant perforin mediated lysis of human Jurkat cells pre-incubated for 30 mins with perforin followed by incubation with Jurkat ce...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445271(CHEMBL3103643)
Affinity DataIC50:  3.21E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50347214(CHEMBL1795775)
Affinity DataIC50:  3.24E+3nMAssay Description:Inhibition of recombinant perforin mediated lysis of human Jurkat cells pre-incubated for 30 mins with perforin followed by incubation with Jurkat ce...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445260(CHEMBL3103654)
Affinity DataIC50:  3.44E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50347204(CHEMBL1795784)
Affinity DataIC50:  3.53E+3nMAssay Description:Inhibition of recombinant perforin mediated lysis of human Jurkat cells pre-incubated for 30 mins with perforin followed by incubation with Jurkat ce...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445291(CHEMBL3103902)
Affinity DataIC50:  3.64E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50347207(CHEMBL1795773)
Affinity DataIC50:  4.18E+3nMAssay Description:Inhibition of recombinant perforin mediated lysis of human Jurkat cells pre-incubated for 30 mins with perforin followed by incubation with Jurkat ce...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445290(CHEMBL3103903)
Affinity DataIC50:  4.35E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445282(CHEMBL3103911)
Affinity DataIC50:  4.42E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50445296(CHEMBL3104231)
Affinity DataIC50:  4.53E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human [51Cr]-labelled Jurkat cells assessed as release of [51Cr] preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50347216(CHEMBL1795350)
Affinity DataIC50:  4.56E+3nMAssay Description:Inhibition of recombinant perforin mediated lysis of human Jurkat cells pre-incubated for 30 mins with perforin followed by incubation with Jurkat ce...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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