Affinity DataKi: 0.00800nMAssay Description:Ability to inhibit [125I]ET-3 binding to the Endothelin B receptor from porcine lung membranes was evaluatedMore data for this Ligand-Target Pair
Affinity DataKi: 0.0400nMAssay Description:Ability to inhibit [125I]ET1 binding to the Endothelin A receptor from porcine lung membranes was evaluatedMore data for this Ligand-Target Pair
Affinity DataKi: 0.0770nMAssay Description:Ability to inhibit [125I]ET-3 binding to the Endothelin B receptor from porcine lung membranes was evaluatedMore data for this Ligand-Target Pair
Target15-hydroxyprostaglandin dehydrogenase [NAD(+)](Homo sapiens (Human))
Ut Southwestern Medical Center
Curated by ChEMBL
Ut Southwestern Medical Center
Curated by ChEMBL
Affinity DataKi: 0.100nMAssay Description:Binding affinity to 15-PGDH (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetEndothelin receptor type B(Homo sapiens (Human))
Takarazuka Research Institute
Curated by ChEMBL
Takarazuka Research Institute
Curated by ChEMBL
Affinity DataKi: 0.140nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
TargetEndothelin receptor type B(Homo sapiens (Human))
Takarazuka Research Institute
Curated by ChEMBL
Takarazuka Research Institute
Curated by ChEMBL
Affinity DataKi: 0.210nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
TargetEndothelin receptor type B(Homo sapiens (Human))
Takarazuka Research Institute
Curated by ChEMBL
Takarazuka Research Institute
Curated by ChEMBL
Affinity DataKi: 0.230nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
TargetEndothelin receptor type B(Homo sapiens (Human))
Takarazuka Research Institute
Curated by ChEMBL
Takarazuka Research Institute
Curated by ChEMBL
Affinity DataKi: 0.230nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
TargetEndothelin receptor type B(Homo sapiens (Human))
Takarazuka Research Institute
Curated by ChEMBL
Takarazuka Research Institute
Curated by ChEMBL
Affinity DataKi: 0.230nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
TargetEndothelin receptor type B(Homo sapiens (Human))
Takarazuka Research Institute
Curated by ChEMBL
Takarazuka Research Institute
Curated by ChEMBL
Affinity DataKi: 0.240nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
TargetEndothelin receptor type B(Homo sapiens (Human))
Takarazuka Research Institute
Curated by ChEMBL
Takarazuka Research Institute
Curated by ChEMBL
Affinity DataKi: 0.240nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.25nMAssay Description:Ability to inhibit [125I]ET-3 binding to the Endothelin B receptor from porcine lung membranes was evaluatedMore data for this Ligand-Target Pair
TargetEndothelin receptor type B(Homo sapiens (Human))
Takarazuka Research Institute
Curated by ChEMBL
Takarazuka Research Institute
Curated by ChEMBL
Affinity DataKi: 0.340nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
TargetEndothelin receptor type B(Homo sapiens (Human))
Takarazuka Research Institute
Curated by ChEMBL
Takarazuka Research Institute
Curated by ChEMBL
Affinity DataKi: 0.380nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
TargetEndothelin receptor type B(Homo sapiens (Human))
Takarazuka Research Institute
Curated by ChEMBL
Takarazuka Research Institute
Curated by ChEMBL
Affinity DataKi: 0.380nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
TargetEndothelin receptor type B(Homo sapiens (Human))
Takarazuka Research Institute
Curated by ChEMBL
Takarazuka Research Institute
Curated by ChEMBL
Affinity DataKi: 0.390nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
TargetEndothelin receptor type B(Homo sapiens (Human))
Takarazuka Research Institute
Curated by ChEMBL
Takarazuka Research Institute
Curated by ChEMBL
Affinity DataKi: 0.490nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
TargetEndothelin receptor type B(Homo sapiens (Human))
Takarazuka Research Institute
Curated by ChEMBL
Takarazuka Research Institute
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
TargetEndothelin receptor type B(Homo sapiens (Human))
Takarazuka Research Institute
Curated by ChEMBL
Takarazuka Research Institute
Curated by ChEMBL
Affinity DataKi: 0.590nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
TargetEndothelin receptor type B(Homo sapiens (Human))
Takarazuka Research Institute
Curated by ChEMBL
Takarazuka Research Institute
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
TargetEndothelin receptor type B(Homo sapiens (Human))
Takarazuka Research Institute
Curated by ChEMBL
Takarazuka Research Institute
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
TargetEndothelin receptor type B(Homo sapiens (Human))
Takarazuka Research Institute
Curated by ChEMBL
Takarazuka Research Institute
Curated by ChEMBL
Affinity DataKi: 0.760nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
TargetEndothelin receptor type B(Homo sapiens (Human))
Takarazuka Research Institute
Curated by ChEMBL
Takarazuka Research Institute
Curated by ChEMBL
Affinity DataKi: 0.790nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.890nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.910nMAssay Description:Ability to inhibit [125I]ET-3 binding to the Endothelin B receptor from porcine lung membranes was evaluatedMore data for this Ligand-Target Pair
TargetEndothelin receptor type B(Homo sapiens (Human))
Takarazuka Research Institute
Curated by ChEMBL
Takarazuka Research Institute
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Ability to inhibit [125I]ET-3 binding to the Endothelin B receptor from porcine lung membranes was evaluatedMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Ability to inhibit [125I]ET-3 binding to the Endothelin B receptor from porcine lung membranes was evaluatedMore data for this Ligand-Target Pair
TargetEndothelin receptor type B(Homo sapiens (Human))
Takarazuka Research Institute
Curated by ChEMBL
Takarazuka Research Institute
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
TargetEndothelin receptor type B(Homo sapiens (Human))
Takarazuka Research Institute
Curated by ChEMBL
Takarazuka Research Institute
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
TargetEndothelin receptor type B(Homo sapiens (Human))
Takarazuka Research Institute
Curated by ChEMBL
Takarazuka Research Institute
Curated by ChEMBL
Affinity DataKi: 3.10nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
TargetEndothelin receptor type B(Homo sapiens (Human))
Takarazuka Research Institute
Curated by ChEMBL
Takarazuka Research Institute
Curated by ChEMBL
Affinity DataKi: 3.20nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
TargetEndothelin receptor type B(Homo sapiens (Human))
Takarazuka Research Institute
Curated by ChEMBL
Takarazuka Research Institute
Curated by ChEMBL
Affinity DataKi: 3.5nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.10nM ΔG°: -47.9kJ/molepH: 7.4 T: 2°CAssay Description:CE inhibition was determined using a spectrophotometric multiwell plate assay with o-NPA as a substrate. The rate of change in absorbance at 420 nm w...More data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:CE inhibition was determined using a spectrophotometric multiwell plate assay with o-NPA as a substrate. The rate of change in absorbance at 420 nm w...More data for this Ligand-Target Pair
TargetEndothelin receptor type B(Homo sapiens (Human))
Takarazuka Research Institute
Curated by ChEMBL
Takarazuka Research Institute
Curated by ChEMBL
Affinity DataKi: 4.40nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Ability to inhibit [125I]ET-3 binding to the Endothelin B receptor from porcine lung membranes was evaluatedMore data for this Ligand-Target Pair
Affinity DataKi: 5.20nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:Ability to inhibit [125I]ET-3 binding to the Endothelin B receptor from porcine lung membranes was evaluatedMore data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.40nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Binding affinity to Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.60nMAssay Description:CE inhibition was determined using a spectrophotometric multiwell plate assay with o-NPA as a substrate. The rate of change in absorbance at 420 nm w...More data for this Ligand-Target Pair