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Found 74 with Last Name = 'okonogi' and Initial = 't'
TargetEstrogen receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by PDSP Ki Database
LigandPNGBDBM50005414((estradiol)13-Methyl-7,8,9,11,12,13,14,15,16,17-de...)
Affinity DataKi:  0.830nMMore data for this Ligand-Target Pair
TargetAndrogen receptor(Rattus norvegicus (Rat))
Meiji Seika Kaisha

Curated by PDSP Ki Database
LigandPNGBDBM50025452((testosterone)17-Hydroxy-10,13-dimethyl-1,2,6,7,8,...)
Affinity DataKi:  6.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetGlucocorticoid receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by PDSP Ki Database
LigandPNGBDBM18207((1R,2S,10S,11S,13R,14R,15S,17S)-1-fluoro-14,17-dih...)
Affinity DataKi:  6.80nMMore data for this Ligand-Target Pair
TargetProgesterone receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by PDSP Ki Database
LigandPNGBDBM86680(CAS_4042 | Mpa | NSC_4042)
Affinity DataKi:  13nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Meiji Seika Kaisha

Curated by PDSP Ki Database
LigandPNGBDBM86680(CAS_4042 | Mpa | NSC_4042)
Affinity DataKi:  19nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by PDSP Ki Database
LigandPNGBDBM86678(CP8816)
Affinity DataKi:  25nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by PDSP Ki Database
LigandPNGBDBM86679(CP8863)
Affinity DataKi:  40nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by PDSP Ki Database
LigandPNGBDBM86680(CAS_4042 | Mpa | NSC_4042)
Affinity DataKi:  43nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by PDSP Ki Database
LigandPNGBDBM86678(CP8816)
Affinity DataKi:  5.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Meiji Seika Kaisha

Curated by PDSP Ki Database
LigandPNGBDBM86679(CP8863)
Affinity DataKi:  9.70E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by PDSP Ki Database
LigandPNGBDBM86679(CP8863)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by PDSP Ki Database
LigandPNGBDBM86680(CAS_4042 | Mpa | NSC_4042)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by PDSP Ki Database
LigandPNGBDBM86679(CP8863)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by PDSP Ki Database
LigandPNGBDBM86678(CP8816)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291167(1-((S)-Oxo-3-(R)-2-amino-1-phenyl-propyl)-pyrrolid...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50291175(((R)-1-Benzyl-2-{(S)-2-[(R)-4-guanidino-1-(thiazol...)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291175(((R)-1-Benzyl-2-{(S)-2-[(R)-4-guanidino-1-(thiazol...)
Affinity DataIC50:  2nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291173(1-((S)-2-Amino-3-(R)-phenyl-propionyl)-azetidine-2...)
Affinity DataIC50:  3nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProlyl endopeptidase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50284127(4-Phenyl-1-{(S)-2-[(S)-2-(thiazole-2-carbonyl)-pyr...)
Affinity DataIC50:  3.10nMAssay Description:Compound was evaluated for the inhibition of Prolyl endopeptidase (PEP) from pig kidney using Z-Gly-Pro-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProlyl endopeptidase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50037610(1-{(S)-2-[(S)-2-(4,5-Dihydro-thiazole-2-carbonyl)-...)
Affinity DataIC50:  3.80nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50037612(1-{(S)-2-[(S)-2-(Benzothiazole-2-carbonyl)-pyrroli...)
Affinity DataIC50:  4nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50291167(1-((S)-Oxo-3-(R)-2-amino-1-phenyl-propyl)-pyrrolid...)
Affinity DataIC50:  4.20nMAssay Description:Inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProlyl endopeptidase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50291163(4-Phenyl-1-{(S)-2-[(R)-2-(thiazole-2-carbonyl)-pyr...)
Affinity DataIC50:  4.40nMAssay Description:The compound was tested for the inhibitory activity against prolyl endo peptidase(PEP) enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProlyl endopeptidase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50037605((S)-2-[(S)-2-(Benzothiazole-2-carbonyl)-pyrrolidin...)
Affinity DataIC50:  5nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50284127(4-Phenyl-1-{(S)-2-[(S)-2-(thiazole-2-carbonyl)-pyr...)
Affinity DataIC50:  5nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50291168((S)-1-(4-Phenyl-butyryl)-pyrrolidine-2-carboxylic ...)
Affinity DataIC50:  5nMAssay Description:The compound was tested for the inhibitory activity against prolyl endo peptidase(PEP) enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProlyl endopeptidase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50037611(1-{(S)-2-[(S)-2-(Oxazolo[4,5-b]pyridine-2-carbonyl...)
Affinity DataIC50:  5.5nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50037606(1-{(S)-2-[(S)-2-(Benzooxazole-2-carbonyl)-pyrrolid...)
Affinity DataIC50:  5.60nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50037597(4-Phenyl-1-{(S)-2-[(S)-2-(thiazole-4-carbonyl)-pyr...)
Affinity DataIC50:  5.90nMAssay Description:Compound was evaluated for the inhibition of Prolyl endopeptidase (PEP) from pig kidney using Z-Gly-Pro-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProlyl endopeptidase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50037597(4-Phenyl-1-{(S)-2-[(S)-2-(thiazole-4-carbonyl)-pyr...)
Affinity DataIC50:  6.20nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50037600(4-Phenyl-1-{(S)-2-[(S)-2-(pyridine-2-carbonyl)-pyr...)
Affinity DataIC50:  6.90nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50037609(2-[2-(Thiazole-2-carbonyl)-pyrrolidine-1-carbonyl]...)
Affinity DataIC50:  8.5nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291166((R)-2-((R)-2-Amino-3-phenyl-propionylamino)-N-[(S)...)
Affinity DataIC50:  8.60nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProlyl endopeptidase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50284126((S)-1-((S)-1-(4-phenylbutanoyl)pyrrolidine-2-carbo...)
Affinity DataIC50:  8.70nMAssay Description:Compound was evaluated for the inhibition of Prolyl endopeptidase (PEP) from pig kidney using Z-Gly-Pro-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProlyl endopeptidase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50037602(1-[(S)-1-(4-Phenyl-butyryl)-pyrrolidine-2-carbonyl...)
Affinity DataIC50:  8.70nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50037604(1-{(S)-2-[(S)-2-(1H-Imidazole-2-carbonyl)-pyrrolid...)
Affinity DataIC50:  9nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50291173(1-((S)-2-Amino-3-(R)-phenyl-propionyl)-azetidine-2...)
Affinity DataIC50:  9nMAssay Description:Inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProlyl endopeptidase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50088247(CHEMBL303966 | Oxo-{(S)-1-[(S)-1-(4-phenyl-butyryl...)
Affinity DataIC50:  9.60nMAssay Description:Compound was evaluated for the inhibition of Prolyl endopeptidase (PEP) from pig kidney using Z-Gly-Pro-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProlyl endopeptidase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50037607(CHEMBL333638 | Oxo-{1-[(S)-1-(4-phenyl-butyryl)-py...)
Affinity DataIC50:  10.3nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50037603(4-Phenyl-1-{(S)-2-[(S)-2-(pyrimidine-5-carbonyl)-p...)
Affinity DataIC50:  61nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50291166((R)-2-((R)-2-Amino-3-phenyl-propionylamino)-N-[(S)...)
Affinity DataIC50:  180nMAssay Description:Inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50291172((S)-1-(3-Phenyl-propionyl)-pyrrolidine-2-carboxyli...)
Affinity DataIC50:  230nMAssay Description:Inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50291171((S)-1-(4-Phenyl-butyryl)-pyrrolidine-2-carboxylic ...)
Affinity DataIC50:  230nMAssay Description:Inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50291170((S)-1-((R)-2-Acetylamino-3-phenyl-propionyl)-pyrro...)
Affinity DataIC50:  230nMAssay Description:Inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50118724((S)-1-((R)-2-Amino-3-phenyl-propionyl)-pyrrolidine...)
Affinity DataIC50:  260nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50038001((2R,4R)-1-((S)-5-(diaminomethyleneamino)-2-(3-meth...)
Affinity DataIC50:  600nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProlyl endopeptidase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50037599(4-Phenyl-1-{(S)-2-[(S)-2-(thiazole-5-carbonyl)-pyr...)
Affinity DataIC50:  646nMAssay Description:Compound was evaluated for the inhibition of Prolyl endopeptidase (PEP) from pig kidney using Z-Gly-Pro-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291174((S)-1-((R)-2-Amino-3-phenyl-propionyl)-piperidine-...)
Affinity DataIC50:  730nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291172((S)-1-(3-Phenyl-propionyl)-pyrrolidine-2-carboxyli...)
Affinity DataIC50:  820nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProlyl endopeptidase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50037599(4-Phenyl-1-{(S)-2-[(S)-2-(thiazole-5-carbonyl)-pyr...)
Affinity DataIC50:  1.09E+3nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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