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Found 110 with Last Name = 'perumattam' and Initial = 'j'
TargetB2 bradykinin receptor(Homo sapiens (Human))
Scios Nova

Curated by ChEMBL
LigandPNGBDBM50052513(8-Methyl-3-(2-oxo-propyl)-1-phenethyl-1,3,8-triaza...)
Affinity DataKi:  0.150nMAssay Description:Affinity to human Bradykinin receptor B2 in CHO cell membranes determined by displacement of [3H]-NPC 17731More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
Scios Nova

Curated by ChEMBL
LigandPNGBDBM50052512(1-Cyclohexyl-8-methyl-3-(2-oxo-propyl)-1,3,8-triaz...)
Affinity DataKi:  0.570nMAssay Description:Affinity to human Bradykinin receptor B2 in CHO cell membranes determined by displacement of [3H]-NPC 17731More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
Scios Nova

Curated by ChEMBL
LigandPNGBDBM50052511(8-Methyl-3-(2-oxo-propyl)-1-p-tolyl-1,3,8-triaza-s...)
Affinity DataKi:  6.30nMAssay Description:Affinity to human Bradykinin receptor B2 in CHO cell membranes determined by displacement of [3H]-NPC 17731More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
Scios Nova

Curated by ChEMBL
LigandPNGBDBM50052509(1-Cyclohexylmethyl-8-methyl-3-(2-oxo-propyl)-1,3,8...)
Affinity DataKi:  6.80nMAssay Description:Affinity to human Bradykinin receptor B2 in CHO cell membranes determined by displacement of [3H]-NPC 17731More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
Scios Nova

Curated by ChEMBL
LigandPNGBDBM50052514(8-Methyl-3-(2-oxo-propyl)-1-phenyl-1,3,8-triaza-sp...)
Affinity DataKi:  7.70nMAssay Description:Affinity to human Bradykinin receptor B2 in CHO cell membranes determined by displacement of [3H]-NPC 17731More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
Scios Nova

Curated by ChEMBL
LigandPNGBDBM50052510(8-Methyl-3-(2-oxo-propyl)-1-propyl-1,3,8-triaza-sp...)
Affinity DataKi:  27nMAssay Description:Affinity to human Bradykinin receptor B2 in CHO cell membranes determined by displacement of [3H]-NPC 17731More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50306491(2-(6-chloro-5-((2R,5S)-4-(1-(4-fluorophenyl)ethyl)...)
Affinity DataIC50:  6nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50266947(2-(6-chloro-5-((2R,5S)-4-(4-fluorobenzyl)-2,5-dime...)
Affinity DataIC50:  9nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50306493(2-(5-((2R,5S)-4-benzhydryl-2,5-dimethylpiperazine-...)
Affinity DataIC50:  9nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375063(CHEMBL255607)
Affinity DataIC50:  10nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50309525(2-(5-(4-(4-fluorobenzyl)piperidine-1-carbonyl)-6-m...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human p38alpha after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375073(CHEMBL402340)
Affinity DataIC50:  13nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50309524(2-(6-chloro-5-(4-(4-fluorobenzyl)piperidine-1-carb...)
Affinity DataIC50:  18nMAssay Description:Inhibition of human p38alpha after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50132378(((1S,3R)-4-Benzyl-2,5-dimethyl-piperazin-1-yl)-(6-...)
Affinity DataIC50:  20nMAssay Description:Inhibition of Mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50132378(((1S,3R)-4-Benzyl-2,5-dimethyl-piperazin-1-yl)-(6-...)
Affinity DataIC50:  20nMAssay Description:Inhibition of Mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375061(CHEMBL271648)
Affinity DataIC50:  21nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50306492(2-(5-((2R,5S)-4-(bis(4-fluorophenyl)methyl)-2,5-di...)
Affinity DataIC50:  24nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50306494(2-(6-chloro-5-((2R,5S)-4-(2,3-dihydro-1H-inden-1-y...)
Affinity DataIC50:  29nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375062(CHEMBL402533)
Affinity DataIC50:  32nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374982(CHEMBL403446)
Affinity DataIC50:  34nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374982(CHEMBL403446)
Affinity DataIC50:  34nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375072(CHEMBL403337)
Affinity DataIC50:  38nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375071(CHEMBL270032)
Affinity DataIC50:  46nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50306496(2-(6-chloro-5-((2R,5S)-4-(1-cyano-1-(4-fluoropheny...)
Affinity DataIC50:  47nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50306497(2-(6-chloro-5-((2R,5S)-4-(7-chloro-1H-indazol-3-yl...)
Affinity DataIC50:  48nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50309531(2-(5-(4-(4-fluorobenzyl)piperidine-1-carbonyl)-6-m...)
Affinity DataIC50:  60nMAssay Description:Inhibition of human p38alpha after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50309529(2-(3-(4-(4-fluorobenzyl)piperidine-1-carbonyl)-2-m...)
Affinity DataIC50:  90nMAssay Description:Inhibition of human p38alpha after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 11(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50266947(2-(6-chloro-5-((2R,5S)-4-(4-fluorobenzyl)-2,5-dime...)
Affinity DataIC50:  98nMAssay Description:Inhibition of p38betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50309528(2-(6-chloro-5-(4-(4-fluorobenzyl)piperidine-1-carb...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human p38alpha after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375070(CHEMBL411724)
Affinity DataIC50:  110nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375077(CHEMBL430412)
Affinity DataIC50:  110nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375064(CHEMBL402152)
Affinity DataIC50:  150nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375069(CHEMBL271426)
Affinity DataIC50:  170nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374989(CHEMBL412302)
Affinity DataIC50:  180nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374989(CHEMBL412302)
Affinity DataIC50:  180nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Scios

Curated by ChEMBL
LigandPNGBDBM50306495(2-(6-chloro-5-((2R,5S)-4-(cyano(4-fluorophenyl)met...)
Affinity DataIC50:  183nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375080(CHEMBL270141)
Affinity DataIC50:  190nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375067(CHEMBL271043)
Affinity DataIC50:  190nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374997(CHEMBL256827)
Affinity DataIC50:  230nMAssay Description:Inhibition of CaMK2delta using 3 weeks old stock solution of compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374988(CHEMBL408434)
Affinity DataIC50:  280nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375066(CHEMBL256460)
Affinity DataIC50:  280nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375001(CHEMBL411253)
Affinity DataIC50:  290nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375054(CHEMBL409856)
Affinity DataIC50:  300nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM2695(3-[1-(3-aminopropyl)-1H-indol-3-yl]-4-(1-methyl-1H...)
Affinity DataIC50:  310nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM2695(3-[1-(3-aminopropyl)-1H-indol-3-yl]-4-(1-methyl-1H...)
Affinity DataIC50:  310nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50374997(CHEMBL256827)
Affinity DataIC50:  350nMAssay Description:Inhibition of CaMK2delta using freshly stock solution of compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375003(CHEMBL258290)
Affinity DataIC50:  360nMAssay Description:Inhibition of CaMK2delta using freshly stock solution of compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50375003(CHEMBL258290)
Affinity DataIC50:  360nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM2691(3-[1-(3-aminopropyl)-1H-indol-3-yl]-4-(1H-indol-3-...)
Affinity DataIC50:  380nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM2691(3-[1-(3-aminopropyl)-1H-indol-3-yl]-4-(1H-indol-3-...)
Affinity DataIC50:  380nMAssay Description:Inhibition of CaMK2deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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