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Found 428 with Last Name = 'prinz' and Initial = 'h'
TargetAndrogen receptor(Homo sapiens (Human))
Vancouver Prostate Centre (Vpc)

Curated by ChEMBL
LigandPNGBDBM50425732(ENZALUTAMIDE | US10053433, FC 4.129 | US10806720, ...)
Affinity DataIC50:  50nMAssay Description:Inhibition of full length AR transcriptional activity in human LNCAP cells harboring AR2PB-eGFP construct assessed as reduction in R1881-induced secr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAndrogen receptor(Homo sapiens (Human))
Vancouver Prostate Centre (Vpc)

Curated by ChEMBL
LigandPNGBDBM50425732(ENZALUTAMIDE | US10053433, FC 4.129 | US10806720, ...)
Affinity DataIC50:  90nMAssay Description:Inhibition of R1881-induced full length AR transcriptional activity in human LNCAP cells harboring AR2PB-eGFP construct after 72 hrs by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAndrogen receptor(Homo sapiens (Human))
Vancouver Prostate Centre (Vpc)

Curated by ChEMBL
LigandPNGBDBM50469124(CHEMBL113332)
Affinity DataIC50:  100nMAssay Description:Inhibition of full length AR transcriptional activity in human LNCAP cells harboring AR2PB-eGFP construct assessed as reduction in R1881-induced secr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50012278((2ALPHA,2''BETA,3BETA,4ALPHA,5BETA)-VINCALEUKOBLAS...)
Affinity DataIC50:  130nMAssay Description:Inhibition of pig brain tubulin polymerization after 30 mins by turbidimetric assayMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50012278((2ALPHA,2''BETA,3BETA,4ALPHA,5BETA)-VINCALEUKOBLAS...)
Affinity DataIC50:  130nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50012278((2ALPHA,2''BETA,3BETA,4ALPHA,5BETA)-VINCALEUKOBLAS...)
Affinity DataIC50:  130nMAssay Description:Inhibition of tubulin polymerization in porcine brainMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50012278((2ALPHA,2''BETA,3BETA,4ALPHA,5BETA)-VINCALEUKOBLAS...)
Affinity DataIC50:  130nMAssay Description:Inhibition of pig brain tubulin polymerization after 30 mins by turbidimetryMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50012278((2ALPHA,2''BETA,3BETA,4ALPHA,5BETA)-VINCALEUKOBLAS...)
Affinity DataIC50:  130nMAssay Description:Inhibition of pig tubulin polymerization determined after 45 mins at 37 degC by turbidimetric analysisMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50012278((2ALPHA,2''BETA,3BETA,4ALPHA,5BETA)-VINCALEUKOBLAS...)
Affinity DataIC50:  130nMAssay Description:Inhibition of porcine brain tubulin polymerizationMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50012278((2ALPHA,2''BETA,3BETA,4ALPHA,5BETA)-VINCALEUKOBLAS...)
Affinity DataIC50:  130nMAssay Description:Inhibition of pig brain tubulin polymerization after 30 mins by turbidimetry analysisMore data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
Vancouver Prostate Centre (Vpc)

Curated by ChEMBL
LigandPNGBDBM50469125(CHEMBL1210959)
Affinity DataIC50:  170nMAssay Description:Inhibition of full length AR transcriptional activity in human LNCAP cells harboring AR2PB-eGFP construct assessed as reduction in R1881-induced secr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474288(CHEMBL112192)
Affinity DataIC50:  220nMAssay Description:In vitro inhibitory concentration required to displace [3H]colchicine from its binding site on tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Vancouver Prostate Centre (Vpc)

Curated by ChEMBL
LigandPNGBDBM50469124(CHEMBL113332)
Affinity DataIC50:  232nMAssay Description:Inhibition of R1881-induced full length AR transcriptional activity in human LNCAP cells harboring AR2PB-eGFP construct after 72 hrs by fluorescence ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50477251(CHEMBL429265)
Affinity DataIC50:  290nMAssay Description:Inhibition of porcine brain tubulin polymerizationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50477242(CHEMBL240468)
Affinity DataIC50:  290nMAssay Description:Inhibition of porcine brain tubulin polymerizationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Vancouver Prostate Centre (Vpc)

Curated by ChEMBL
LigandPNGBDBM50469122(CHEMBL4278637)
Affinity DataIC50:  316nMAssay Description:Inhibition of R1881-induced full length AR transcriptional activity in human LNCAP cells harboring AR2PB-eGFP construct after 72 hrs by fluorescence ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Vancouver Prostate Centre (Vpc)

Curated by ChEMBL
LigandPNGBDBM50469121(CHEMBL1210876)
Affinity DataIC50:  340nMAssay Description:Inhibition of full length AR transcriptional activity in human LNCAP cells harboring AR2PB-eGFP construct assessed as reduction in R1881-induced secr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50035218(CHEMBL61 | PODOFILOX | Podophyllinic acid lactone ...)
Affinity DataIC50:  350nMAssay Description:Inhibition of pig tubulin polymerization determined after 45 mins at 37 degC by turbidimetric analysisMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50035218(CHEMBL61 | PODOFILOX | Podophyllinic acid lactone ...)
Affinity DataIC50:  350nMAssay Description:Inhibition of pig brain tubulin polymerization after 30 mins by turbidimetryMore data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
Vancouver Prostate Centre (Vpc)

Curated by ChEMBL
LigandPNGBDBM50469122(CHEMBL4278637)
Affinity DataIC50:  350nMAssay Description:Inhibition of full length AR transcriptional activity in human LNCAP cells harboring AR2PB-eGFP construct assessed as reduction in R1881-induced secr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50035218(CHEMBL61 | PODOFILOX | Podophyllinic acid lactone ...)
Affinity DataIC50:  350nMAssay Description:Inhibition of pig brain tubulin polymerization after 30 mins by turbidimetric assayMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50035218(CHEMBL61 | PODOFILOX | Podophyllinic acid lactone ...)
Affinity DataIC50:  350nMAssay Description:Inhibition of pig brain tubulin polymerization after 30 mins by turbidimetry analysisMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50035218(CHEMBL61 | PODOFILOX | Podophyllinic acid lactone ...)
Affinity DataIC50:  350nMAssay Description:Inhibition of porcine brain tubulin polymerizationMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50035218(CHEMBL61 | PODOFILOX | Podophyllinic acid lactone ...)
Affinity DataIC50:  350nMAssay Description:Inhibition of tubulin polymerization in porcine brainMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50035218(CHEMBL61 | PODOFILOX | Podophyllinic acid lactone ...)
Affinity DataIC50:  350nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50482385(CHEMBL1210322)
Affinity DataIC50:  360nMAssay Description:Inhibition of pig brain tubulin polymerization after 30 mins by turbidimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50469121(CHEMBL1210876)
Affinity DataIC50:  360nMAssay Description:Inhibition of pig brain tubulin polymerization after 30 mins by turbidimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50469125(CHEMBL1210959)
Affinity DataIC50:  360nMAssay Description:Inhibition of pig brain tubulin polymerization after 30 mins by turbidimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474300(CHEMBL116173)
Affinity DataIC50:  370nMAssay Description:In vitro inhibitory concentration required to displace [3H]colchicine from its binding site on TubulinMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50476049(CHEMBL219102)
Affinity DataIC50:  380nMAssay Description:Inhibition of tubulin polymerization in porcine brainMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50482387(CHEMBL1209944)
Affinity DataIC50:  380nMAssay Description:Inhibition of pig brain tubulin polymerization after 30 mins by turbidimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50477244(CHEMBL237880)
Affinity DataIC50:  390nMAssay Description:Inhibition of porcine brain tubulin polymerizationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50479547(CHEMBL455138)
Affinity DataIC50:  400nMAssay Description:Displacement of [3H]Colchicine from pig biotinylated tubulin after 2 hrs by SPAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-lipoxygenase(Bos taurus)
WestfäLische Wilhelms-UniversitäT MüNster

Curated by ChEMBL
LigandPNGBDBM50059631(6-(1,8-Dihydroxy-9-oxo-9,10-dihydro-anthracen-2-yl...)
Affinity DataIC50:  400nMAssay Description:5-LO inhibitory activity, measured by production of 5-hydroxyeicosatetraenoic acid (5-HETE) and leukotriene B4 (LTB4) in bovine polymorphonuclear leu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50482392(CHEMBL1210418)
Affinity DataIC50:  410nMAssay Description:Inhibition of pig brain tubulin polymerization after 30 mins by turbidimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50482380(CHEMBL1209943)
Affinity DataIC50:  420nMAssay Description:Inhibition of pig brain tubulin polymerization after 30 mins by turbidimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474288(CHEMBL112192)
Affinity DataIC50:  430nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50484086(CHEMBL1814612)
Affinity DataIC50:  440nMAssay Description:Inhibition of pig brain tubulin polymerization after 30 mins by turbidimetry analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50474290(CHEMBL115499)
Affinity DataIC50:  480nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-lipoxygenase(Bos taurus)
WestfäLische Wilhelms-UniversitäT MüNster

Curated by ChEMBL
LigandPNGBDBM50059608(5-(1,8-Dihydroxy-9-oxo-9,10-dihydro-anthracen-2-yl...)
Affinity DataIC50:  500nMAssay Description:5-LO inhibitory activity, measured by production of 5-hydroxyeicosatetraenoic acid (5-HETE) and leukotriene B4 (LTB4) in bovine polymorphonuclear leu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50476048(CHEMBL219439)
Affinity DataIC50:  500nMAssay Description:Inhibition of tubulin polymerization in porcine brainMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50482374(CHEMBL1210416)
Affinity DataIC50:  510nMAssay Description:Inhibition of pig brain tubulin polymerization after 30 mins by turbidimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50482379(CHEMBL1210963)
Affinity DataIC50:  520nMAssay Description:Inhibition of pig brain tubulin polymerization after 30 mins by turbidimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50479547(CHEMBL455138)
Affinity DataIC50:  520nMAssay Description:Inhibition of pig brain tubulin polymerization after 30 mins by turbidimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50483993(CHEMBL1802017)
Affinity DataIC50:  520nMAssay Description:Inhibition of pig tubulin polymerization determined after 45 mins at 37 degC by turbidimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50482372(CHEMBL1210319)
Affinity DataIC50:  530nMAssay Description:Inhibition of pig brain tubulin polymerization after 30 mins by turbidimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Westphalian Wilhelms-University

Curated by ChEMBL
LigandPNGBDBM50483990(CHEMBL1801900)
Affinity DataIC50:  570nMAssay Description:Inhibition of pig tubulin polymerization determined after 45 mins at 37 degC by turbidimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-lipoxygenase(Bos taurus)
WestfäLische Wilhelms-UniversitäT MüNster

Curated by ChEMBL
LigandPNGBDBM50059616(3-(1,8-Dihydroxy-9-oxo-9,10-dihydro-anthracen-2-yl...)
Affinity DataIC50:  600nMAssay Description:5-LO inhibitory activity, measured by production of 5-hydroxyeicosatetraenoic acid (5-HETE) and leukotriene B4 (LTB4) in bovine polymorphonuclear leu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-lipoxygenase(Bos taurus)
WestfäLische Wilhelms-UniversitäT MüNster

Curated by ChEMBL
LigandPNGBDBM50059604(4-(1,8-Dihydroxy-9-oxo-9,10-dihydro-anthracen-2-yl...)
Affinity DataIC50:  600nMAssay Description:5-LO inhibitory activity, measured by production of 5-hydroxyeicosatetraenoic acid (5-HETE) and leukotriene B4 (LTB4) in bovine polymorphonuclear leu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
Vancouver Prostate Centre (Vpc)

Curated by ChEMBL
LigandPNGBDBM50469122(CHEMBL4278637)
Affinity DataIC50:  625nMAssay Description:Displacement of Fluormone-DHT from rat GST-tagged rat AR LBD expressed in insect cells after 4 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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