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Found 236 with Last Name = 'surpateanu' and Initial = 'g'
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228427((R)-N-[(S)-1-(4-guanidino-benzylcarbamoyl)-ethyl]-...)
Affinity DataKi:  16nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50371003(CHEMBL397507)
Affinity DataKi:  2.30E+3nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228427((R)-N-[(S)-1-(4-guanidino-benzylcarbamoyl)-ethyl]-...)
Affinity DataKi: >2.50E+3nMAssay Description:Inhibition of human recombinant tPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50234567(1,4-dideoxy-1,4-imino-D-ribitol | CHEMBL261634 | I...)
Affinity DataKi:  6.10E+3nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolase expressed in Escherichia coli WK6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50260497(1,4-Dideoxy-1,4-imino-N-(4-amidinobenzyl)-D-ribito...)
Affinity DataKi:  6.70E+3nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolase expressed in Escherichia coli WK6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50260496(1,4-Dideoxy-1,4-imino-N-(4-guanidinobenzyl)-D-ribi...)
Affinity DataKi:  7.00E+3nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolase expressed in Escherichia coli WK6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228422((4-guanidino-benzyl)-carbamic acid benzyl ester | ...)
Affinity DataKi:  1.60E+4nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50260490((1S )-1,4-Dideoxy-1-(2-guanidinoethyl)-1,4-imino-D...)
Affinity DataKi:  1.80E+4nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolase expressed in Escherichia coli WK6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50370996(CHEMBL230908)
Affinity DataKi:  2.10E+4nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50370998(CHEMBL397508)
Affinity DataKi:  2.30E+4nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50371000(CHEMBL231322)
Affinity DataKi:  3.20E+4nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50260492(1,4-Dideoxy-(3-guanidinopropyl)-1,4-imino-D-ribito...)
Affinity DataKi:  4.00E+4nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolase expressed in Escherichia coli WK6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228427((R)-N-[(S)-1-(4-guanidino-benzylcarbamoyl)-ethyl]-...)
Affinity DataKi:  4.00E+4nMAssay Description:Inhibition of human plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50377915(CHEMBL1169558)
Affinity DataKi:  5.90E+4nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolase expressed in Escherichia coli WK6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50371001(CHEMBL395797)
Affinity DataKi:  6.30E+4nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50371002(CHEMBL230061)
Affinity DataKi:  8.70E+4nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50260491(1,4-Dideoxy-(2-guanidinoethyl)-1,4-imino-D-ribitol...)
Affinity DataKi:  2.86E+5nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolase expressed in Escherichia coli WK6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50260487(1-Guanidino-3,6-anhydro-1,2-dideoxy-Dallo-heptitol...)
Affinity DataKi:  3.09E+5nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolase expressed in Escherichia coli WK6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50370999(CHEMBL231025)
Affinity DataKi:  5.20E+5nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50260486(1-Guanidino-2,5-anhydro-1-deoxy-D-allitol | CHEMBL...)
Affinity DataKi:  5.45E+5nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolase expressed in Escherichia coli WK6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50260489(1-Guanidino-4,7-anhydro-1,2,3-trideoxy-Dallo-octit...)
Affinity DataKi:  6.77E+5nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolase expressed in Escherichia coli WK6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50370997(CHEMBL425996)
Affinity DataKi:  6.80E+5nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50260488(2-Guanidino-4,7-anhydro-1,2,3-trideoxy-Dallo-octit...)
Affinity DataKi:  6.85E+5nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolase expressed in Escherichia coli WK6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228422((4-guanidino-benzyl)-carbamic acid benzyl ester | ...)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of human plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228422((4-guanidino-benzyl)-carbamic acid benzyl ester | ...)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of human recombinant tPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228422((4-guanidino-benzyl)-carbamic acid benzyl ester | ...)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228422((4-guanidino-benzyl)-carbamic acid benzyl ester | ...)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50260485(2,5-Anhydro-1-deoxy-1-(trimethylammonio)-D-allitol...)
Affinity DataKi:  1.28E+6nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolase expressed in Escherichia coli WK6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50260480((2R,3S,4R,5R)-3,4-Dihydroxy-5-(hydroxymethyl)-tetr...)
Affinity DataKi:  4.50E+6nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolase expressed in Escherichia coli WK6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50206267((2S,3R,4S,5R)-2-(2-azidoethyl)-5-(hydroxymethyl)-t...)
Affinity DataKi:  5.60E+6nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50206267((2S,3R,4S,5R)-2-(2-azidoethyl)-5-(hydroxymethyl)-t...)
Affinity DataKi:  5.64E+6nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolase expressed in Escherichia coli WK6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194745(CHEMBL385900 | diphenyl 1-[(N-2-thiophenesulfonyl-...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194741(CHEMBL385158 | diphenyl 1-[(N-benzenesulfonyl-D-se...)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228418(CHEMBL393591 | methyl 1-(diphenoxyphosphoryl)-2-(4...)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228412(CHEMBL393979 | methyl 1-(bis(4-acetamidophenoxy)ph...)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194743(CHEMBL214814 | diphenyl 1-[(N-alpha-toluenesulfony...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228425(CHEMBL239118 | di-(4-acetamidophenyl) 1-(methylsul...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194743(CHEMBL214814 | diphenyl 1-[(N-alpha-toluenesulfony...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228420(CHEMBL391968 | di-(4-acetamidophenyl) 1-(benzyloxy...)
Affinity DataIC50:  4.20nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145689(CHEMBL80844 | [1-[(S)-2-((R)-2-Benzyloxycarbonylam...)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194737(CHEMBL384263 | diphenyl 1-[(N-o-methylbenzoyl-D-se...)
Affinity DataIC50:  4.40nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194742(CHEMBL263977 | diphenyl 1-[(N-benzyl-D-seryl)-L-al...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194746(CHEMBL405546 | diphenyl 1-[(N-o-methylbenzoyl-D-se...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194744(CHEMBL385897 | diphenyl 1-[(N-naphthalenesulfonyl-...)
Affinity DataIC50:  5.80nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194734(CHEMBL386275 | diphenyl 1-[(N-p-methoxybenzenesulf...)
Affinity DataIC50:  5.80nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194736(CHEMBL189823 | diphenyl 1-[(N-o,o-dimethylbenzoyl-...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194735(CHEMBL215961 | diphenyl 1-[(N-p-cyanobenzenesulfon...)
Affinity DataIC50:  6.20nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228421(CHEMBL238493 | diphenyl 1-(methylsulfonylamino)-2-...)
Affinity DataIC50:  6.60nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194738(CHEMBL386249 | diphenyl 1-[(N-p-bromobenzenesulfon...)
Affinity DataIC50:  6.60nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194732(CHEMBL214539 | di-(4-acetamidophenyl) 1-[(N-benzyl...)
Affinity DataIC50:  6.70nMAssay Description:Inhibition of [3H]-FPP incorporation into biotin-linked K-ras decapeptide (CVIM) by bovine farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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