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Found 113 with Last Name = 'van aerschot' and Initial = 'a'
TargetAspartate--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50339907(((S)-2-amino-3-carboxypropanoyl)(((2R,3S,4R,5R)-5-...)
Affinity DataKi:  0.0520nMAssay Description:Inhibition of Escherichia coli BL21(DE3) Aspartyl-tRNA synthetase assessed as reduction in tRNA aminoacylation preincubated for 10 mins with Escheric...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50458119(Leusa)
Affinity DataKi:  0.139nMAssay Description:Inhibition of Escherichia coli BL21(DE3) Leucyl-tRNA synthetase assessed as reduction in tRNA aminoacylation preincubated for 10 mins with Escherichi...More data for this Ligand-Target Pair
TargetSerine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50339906(((2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-dihyd...)
Affinity DataKi:  0.180nMAssay Description:Inhibition of Escherichia coli BL21(DE3) Seryl-tRNA synthetase assessed as reduction in tRNA aminoacylation preincubated for 10 mins with Escherichia...More data for this Ligand-Target Pair
TargetLeucine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50458122(CHEMBL4204314)
Affinity DataKi:  0.654nMAssay Description:Inhibition of Escherichia coli BL21(DE3) Leucyl-tRNA synthetase assessed as reduction in tRNA aminoacylation preincubated for 10 mins with Escherichi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50524451(CHEMBL4553017)
Affinity DataKi:  1.20nMAssay Description:Inhibition of recombinant Escherichia coli BL21(DE3) isoleucyl-tRNA synthetase expressed in Escherichia coli Rosetta 2 (DE3) assessed as reduction in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50222902(CHEMBL1163069)
Affinity DataKi:  1.90nMAssay Description:Inhibition of Escherichia coli BL21(DE3) Isoleucyl-tRNA synthetase assessed as reduction in tRNA aminoacylation preincubated for 10 mins with Escheri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50569962(CHEMBL4864835)
Affinity DataKi:  2.5nMAssay Description:Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50290686(9-((E)-4-((2S,3R,4R,5S)-3,4-dihydroxy-5-(((2S,3S)-...)
Affinity DataKi:  2.5nMAssay Description:Competitive inhibition of Escherichia coli Isoleucyl-tRNA synthetaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50458121(CHEMBL1163085)
Affinity DataKi:  2.90nMAssay Description:Inhibition of Escherichia coli BL21(DE3) Tyrosyl-tRNA synthetase assessed as reduction in tRNA aminoacylation preincubated for 10 mins with Escherich...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetLeucine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50569952(CHEMBL4869028)
Affinity DataKi:  5.5nMAssay Description:Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50524359(CHEMBL4465674)
Affinity DataKi:  9.80nMAssay Description:Inhibition of purified Escherichia coli BL21 (DE3) leuRS incubated for 10 mins in presence of 14C-labeled leucine by radiolabel transfer assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Ghent

Curated by ChEMBL
LigandPNGBDBM50112193(CHEMBL52648 | N-[5-(6-Cyclopentylamino-purin-9-yl)...)
Affinity DataKi:  17nMAssay Description:Affinity for adenosine A1 receptor was determined, in the presence of GTP in rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50524360(CHEMBL3265242)
Affinity DataKi:  17nMAssay Description:Inhibition of purified Escherichia coli BL21 (DE3) ileRS incubated for 10 mins in presence of 14C-labeled isoleucine by radiolabel transfer assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50569957(CHEMBL4864965)
Affinity DataKi:  18nMAssay Description:Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50524355(CHEMBL4467328)
Affinity DataKi:  21nMAssay Description:Inhibition of purified Escherichia coli BL21 (DE3) leuRS incubated for 10 mins in presence of 14C-labeled leucine by radiolabel transfer assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Ghent

Curated by ChEMBL
LigandPNGBDBM50454674(CHEMBL2112630)
Affinity DataKi:  24nMAssay Description:Affinity for adenosine A1 receptor was determined, in the presence of GTP in rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Ghent

Curated by ChEMBL
LigandPNGBDBM50112193(CHEMBL52648 | N-[5-(6-Cyclopentylamino-purin-9-yl)...)
Affinity DataKi:  24nMAssay Description:Affinity for adenosine A1 receptor was determined, in the absence of GTP in rat cortical membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAspartate--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50458117(CHEMBL4203761)
Affinity DataKi:  25nMAssay Description:Inhibition of Escherichia coli BL21(DE3) Aspartyl-tRNA synthetase assessed as reduction in tRNA aminoacylation preincubated for 10 mins with Escheric...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50458118(CHEMBL4208126)
Affinity DataKi:  30nMAssay Description:Inhibition of Escherichia coli BL21(DE3) Tyrosyl-tRNA synthetase assessed as reduction in tRNA aminoacylation preincubated for 10 mins with Escherich...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50524361(CHEMBL4451258)
Affinity DataKi:  30nMAssay Description:Inhibition of purified Escherichia coli BL21 (DE3) leuRS incubated for 10 mins in presence of 14C-labeled leucine by radiolabel transfer assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50569960(CHEMBL4852287)
Affinity DataKi:  31nMAssay Description:Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50569963(CHEMBL4855635)
Affinity DataKi:  31nMAssay Description:Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50569958(CHEMBL4864716)
Affinity DataKi:  32nMAssay Description:Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Ghent

Curated by ChEMBL
LigandPNGBDBM50454674(CHEMBL2112630)
Affinity DataKi:  33nMAssay Description:Affinity for adenosine A1 receptor was determined, in the absence of GTP in rat cortical membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50524357(CHEMBL4558119)
Affinity DataKi:  43nMAssay Description:Inhibition of purified Escherichia coli BL21 (DE3) tyrRS incubated for 10 mins in presence of 14C-labeled tyrosine by radiolabel transfer assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetLeucine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50569954(CHEMBL4867227)
Affinity DataKi:  52nMAssay Description:Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50524354(CHEMBL3265243)
Affinity DataKi:  55nMAssay Description:Inhibition of purified Escherichia coli BL21 (DE3) ileRS incubated for 10 mins in presence of 14C-labeled isoleucine by radiolabel transfer assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Ghent

Curated by ChEMBL
LigandPNGBDBM50454666(CHEMBL2112627)
Affinity DataKi:  81nMAssay Description:Affinity for adenosine A1 receptor was determined, in the presence of GTP in rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Ghent

Curated by ChEMBL
LigandPNGBDBM50060845(CHEMBL122746 | N-[(R)-5-(6-Cyclopentylamino-purin-...)
Affinity DataKi:  83nMAssay Description:Affinity for adenosine A1 receptor was determined, in the absence of GTP in rat cortical membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Ghent

Curated by ChEMBL
LigandPNGBDBM50060845(CHEMBL122746 | N-[(R)-5-(6-Cyclopentylamino-purin-...)
Affinity DataKi:  83nMAssay Description:Affinity for adenosine A1 receptor was determined, in the absence of GTP in rat cortical membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50544145(CHEMBL4636583)
Affinity DataKi:  88nMAssay Description:Inhibition of Escherichia coli BL21(DE3) ileRS overexpressed in Escherichia coli Rosetta2(DE3) assessed as reduction in tRNA aminoacylation preincuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Ghent

Curated by ChEMBL
LigandPNGBDBM50454665(CHEMBL2112626)
Affinity DataKi:  100nMAssay Description:Affinity for adenosine A1 receptor was determined, in the presence of GTP in rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50569955(CHEMBL4876966)
Affinity DataKi:  108nMAssay Description:Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Ghent

Curated by ChEMBL
LigandPNGBDBM50453913(CHEMBL2112619)
Affinity DataKi:  110nMAssay Description:Affinity for adenosine A1 receptor was determined, in the absence of GTP in rat cortical membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Ghent

Curated by ChEMBL
LigandPNGBDBM50454666(CHEMBL2112627)
Affinity DataKi:  110nMAssay Description:Affinity for adenosine A1 receptor was determined, in the absence of GTP in rat cortical membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50544146(CHEMBL4648043)
Affinity DataKi:  114nMAssay Description:Inhibition of Escherichia coli BL21(DE3) ileRS overexpressed in Escherichia coli Rosetta2(DE3) assessed as reduction in tRNA aminoacylation preincuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Ghent

Curated by ChEMBL
LigandPNGBDBM50454665(CHEMBL2112626)
Affinity DataKi:  130nMAssay Description:Affinity for adenosine A1 receptor was determined, in the absence of GTP in rat cortical membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Ghent

Curated by ChEMBL
LigandPNGBDBM50060840(CHEMBL340299 | N-[(R)-5-(6-Cyclopentylamino-purin-...)
Affinity DataKi:  130nMAssay Description:Affinity for adenosine A1 receptor was determined, in the presence of GTP in rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50524353(CHEMBL4518549)
Affinity DataKi:  149nMAssay Description:Inhibition of purified Escherichia coli BL21 (DE3) tyrRS incubated for 10 mins in presence of 14C-labeled tyrosine by radiolabel transfer assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Ghent

Curated by ChEMBL
LigandPNGBDBM50060847(4-Cyclohexyl-N-[(R)-5-(6-cyclopentylamino-purin-9-...)
Affinity DataKi:  150nMAssay Description:Affinity for adenosine A1 receptor was determined, in the presence of GTP in rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50569961(CHEMBL4861722)
Affinity DataKi:  182nMAssay Description:Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Ghent

Curated by ChEMBL
LigandPNGBDBM50060847(4-Cyclohexyl-N-[(R)-5-(6-cyclopentylamino-purin-9-...)
Affinity DataKi:  190nMAssay Description:Affinity for adenosine A1 receptor was determined, in the absence of GTP in rat cortical membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Ghent

Curated by ChEMBL
LigandPNGBDBM50454669(CHEMBL2112632)
Affinity DataKi:  200nMAssay Description:Affinity for adenosine A1 receptor was determined, in the presence of GTP in rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Ghent

Curated by ChEMBL
LigandPNGBDBM50060840(CHEMBL340299 | N-[(R)-5-(6-Cyclopentylamino-purin-...)
Affinity DataKi:  200nMAssay Description:Affinity for adenosine A1 receptor was determined, in the absence of GTP in rat cortical membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50458120(CHEMBL4215986)
Affinity DataKi:  213nMAssay Description:Inhibition of Escherichia coli BL21(DE3) Isoleucyl-tRNA synthetase assessed as reduction in tRNA aminoacylation preincubated for 10 mins with Escheri...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Ghent

Curated by ChEMBL
LigandPNGBDBM50454669(CHEMBL2112632)
Affinity DataKi:  240nMAssay Description:Affinity for adenosine A1 receptor was determined, in the absence of GTP in rat cortical membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Ghent

Curated by ChEMBL
LigandPNGBDBM50454673(CHEMBL2112620)
Affinity DataKi:  310nMAssay Description:Affinity for adenosine A1 receptor was determined, in the presence of GTP in rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Ghent

Curated by ChEMBL
LigandPNGBDBM50454667(CHEMBL2112625)
Affinity DataKi:  350nMAssay Description:Affinity for adenosine A1 receptor was determined, in the presence of GTP in rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Ghent

Curated by ChEMBL
LigandPNGBDBM50454667(CHEMBL2112625)
Affinity DataKi:  370nMAssay Description:Affinity for adenosine A1 receptor was determined, in the absence of GTP in rat cortical membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase(Escherichia coli (strain K12))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50569956(CHEMBL4850408)
Affinity DataKi:  388nMAssay Description:Inhibition of recombinant Escherichia coli LeuRS assessed as inhibition of 14C-radiolabelled leucine transfer to tRNA leucine preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
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