TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Displacement of [3H]-DAMGO from mu opioid receptor (unknown origin) expressed in CHO cells at 10 uMMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Displacement of [3H]-DAMGO from mu opioid receptor (unknown origin) expressed in CHO cells at 10 uMMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Displacement of [3H]-DAMGO from mu opioid receptor (unknown origin) expressed in CHO cells at 10 uMMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Displacement of [125]IBNtxA from mouse MOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 49nMAssay Description:Displacement of [125]IBNtxA from mouse DOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 79nMAssay Description:Displacement of [125]IBNtxA from mouse MOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 125nMAssay Description:Displacement of [125]IBNtxA from mouse KOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 216nMAssay Description:Displacement of [125]IBNtxA from mouse MOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 578nMAssay Description:Displacement of [125]IBNtxA from mouse MOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 649nMAssay Description:Displacement of [125]IBNtxA from mouse KOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 666nMAssay Description:Displacement of [125]IBNtxA from mouse MOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 883nMAssay Description:Displacement of [125]IBNtxA from mouse KOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 1.15E+3nMAssay Description:Displacement of [125]IBNtxA from mouse DOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 1.18E+3nMAssay Description:Displacement of [125]IBNtxA from mouse KOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 1.27E+3nMAssay Description:Displacement of [125]IBNtxA from mouse KOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 1.68E+3nMAssay Description:Displacement of [125]IBNtxA from mouse MOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 1.88E+3nMAssay Description:Displacement of [125]IBNtxA from mouse DOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 2.20E+3nMAssay Description:Displacement of [125]IBNtxA from mouse KOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 3.24E+3nMAssay Description:Displacement of [125]IBNtxA from mouse DOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 3.40E+3nMAssay Description:Displacement of [125]IBNtxA from mouse DOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 4.14E+3nMAssay Description:Displacement of [125]IBNtxA from mouse DOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 6.90E+3nMAssay Description:Displacement of [125]IBNtxA from mouse MOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 7.18E+3nMAssay Description:Displacement of [125]IBNtxA from mouse KOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 7.95E+3nMAssay Description:Displacement of [125]IBNtxA from mouse DOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at mouse DOR expressed in CHO cell membranes assessed as inhibition of DPDPE induced [35S]-GTPgammaS binding incubated for 60 min...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at mouse DOR expressed in CHO cell membranes assessed as inhibition of DPDPE induced [35S]-GTPgammaS binding incubated for 60 min...More data for this Ligand-Target Pair
Affinity DataIC50: 1.09E+4nMAssay Description:Antagonist activity at mouse MOR expressed in CHO cell membranes assessed as inhibition of DAMGO induced [35S]-GTPgammaS binding incubated for 60 min...More data for this Ligand-Target Pair
Affinity DataIC50: 1.26E+4nMAssay Description:Antagonist activity at mouse DOR expressed in CHO cell membranes assessed as inhibition of DPDPE induced [35S]-GTPgammaS binding incubated for 60 min...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 36nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 5.30nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 7.30nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 94nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 83nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 83nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 3.76E+3nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 86nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 370nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 104nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 535nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 30nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 1.11E+3nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 186nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 71nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 1.75E+4nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 1.56E+3nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 11nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 241nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 5.90nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 0.490nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 36nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair