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Found 39 Enz. Inhib. hit(s) with Target = 'Baculoviral IAP repeat-containing protein 3 [238-349]'
TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM26207((2R,5S,8S)-8-[(2S)-2-(methylamino)propanamido]-7-o...)
Affinity DataKi:  4.20nM ΔG°:  -47.3kJ/molepH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader at excitation and emission wavelengths of 485 and 530 nm, respectively. The equilibri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM13212((3S,6S,9aS)-N-(diphenylmethyl)-6-[(2S)-2-(methylam...)
Affinity DataKi:  4.80nM ΔG°:  -47.0kJ/molepH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader at excitation and emission wavelengths of 485 and 530 nm, respectively. The equilibri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM26206((2R,5S,8S)-N-(diphenylmethyl)-8-[(2S)-2-(methylami...)
Affinity DataKi:  5.90nM ΔG°:  -46.5kJ/molepH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader at excitation and emission wavelengths of 485 and 530 nm, respectively. The equilibri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM26209((2R,6S,9S)-N-(diphenylmethyl)-9-[(2S)-2-(methylami...)
Affinity DataKi:  20nM ΔG°:  -43.5kJ/molepH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader at excitation and emission wavelengths of 485 and 530 nm, respectively. The equilibri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM26208((2R,5S,8S)-8-[(2S)-2-(methylamino)propanamido]-7-o...)
Affinity DataKi:  370nM ΔG°:  -36.3kJ/molepH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader at excitation and emission wavelengths of 485 and 530 nm, respectively. The equilibri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM422070(US10508103, Embodiment 23)
Affinity DataIC50: <10nMAssay Description:1) Affinity of compounds listed in table to cIAP1-BIR3, Ciap2-BIR3, XIAP-BIR3 was tested referring to Nikolovska-Colesks, Z. et.Al. (Analytical Bioch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM422074(US10508103, Embodiment 27)
Affinity DataIC50: <10nMAssay Description:1) Affinity of compounds listed in table to cIAP1-BIR3, Ciap2-BIR3, XIAP-BIR3 was tested referring to Nikolovska-Colesks, Z. et.Al. (Analytical Bioch...More data for this Ligand-Target Pair
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TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM130049(US8815927, SM-1265)
Affinity DataIC50: <10nMAssay Description:An in vitro fluorescence polarization (FP) based binding assay was used to test the binding ability of the compounds of the present invention to cert...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM422073(US10508103, Embodiment 26)
Affinity DataIC50: <10nMAssay Description:1) Affinity of compounds listed in table to cIAP1-BIR3, Ciap2-BIR3, XIAP-BIR3 was tested referring to Nikolovska-Colesks, Z. et.Al. (Analytical Bioch...More data for this Ligand-Target Pair
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TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM130048(US8815927, SM-1259)
Affinity DataIC50: <20nMAssay Description:An in vitro fluorescence polarization (FP) based binding assay was used to test the binding ability of the compounds of the present invention to cert...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM130050(US8815927, SM-1266)
Affinity DataIC50: <20nMAssay Description:An in vitro fluorescence polarization (FP) based binding assay was used to test the binding ability of the compounds of the present invention to cert...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM7006(US8815927, SM-1258)
Affinity DataIC50: <50nMAssay Description:An in vitro fluorescence polarization (FP) based binding assay was used to test the binding ability of the compounds of the present invention to cert...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM130051(US8815927, SM-1267)
Affinity DataIC50: <50nMAssay Description:An in vitro fluorescence polarization (FP) based binding assay was used to test the binding ability of the compounds of the present invention to cert...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM422075(US10508103, Embodiment 28)
Affinity DataIC50:  55nMAssay Description:1) Affinity of compounds listed in table to cIAP1-BIR3, Ciap2-BIR3, XIAP-BIR3 was tested referring to Nikolovska-Colesks, Z. et.Al. (Analytical Bioch...More data for this Ligand-Target Pair
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TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM422076(US10508103, Embodiment 29)
Affinity DataIC50:  55nMAssay Description:1) Affinity of compounds listed in table to cIAP1-BIR3, Ciap2-BIR3, XIAP-BIR3 was tested referring to Nikolovska-Colesks, Z. et.Al. (Analytical Bioch...More data for this Ligand-Target Pair
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TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM422077(US10508103, Embodiment 30)
Affinity DataIC50:  55nMAssay Description:1) Affinity of compounds listed in table to cIAP1-BIR3, Ciap2-BIR3, XIAP-BIR3 was tested referring to Nikolovska-Colesks, Z. et.Al. (Analytical Bioch...More data for this Ligand-Target Pair
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TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM422078(US10508103, Embodiment 31)
Affinity DataIC50:  55nMAssay Description:1) Affinity of compounds listed in table to cIAP1-BIR3, Ciap2-BIR3, XIAP-BIR3 was tested referring to Nikolovska-Colesks, Z. et.Al. (Analytical Bioch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM422079(US10508103, Embodiment 32)
Affinity DataIC50:  55nMAssay Description:1) Affinity of compounds listed in table to cIAP1-BIR3, Ciap2-BIR3, XIAP-BIR3 was tested referring to Nikolovska-Colesks, Z. et.Al. (Analytical Bioch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM422080(US10508103, Embodiment 36)
Affinity DataIC50:  55nMAssay Description:1) Affinity of compounds listed in table to cIAP1-BIR3, Ciap2-BIR3, XIAP-BIR3 was tested referring to Nikolovska-Colesks, Z. et.Al. (Analytical Bioch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM422081(US10508103, Embodiment 38)
Affinity DataIC50:  55nMAssay Description:1) Affinity of compounds listed in table to cIAP1-BIR3, Ciap2-BIR3, XIAP-BIR3 was tested referring to Nikolovska-Colesks, Z. et.Al. (Analytical Bioch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM422082(US10508103, Embodiment 39)
Affinity DataIC50:  55nMAssay Description:1) Affinity of compounds listed in table to cIAP1-BIR3, Ciap2-BIR3, XIAP-BIR3 was tested referring to Nikolovska-Colesks, Z. et.Al. (Analytical Bioch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM422083(US10508103, Embodiment 40)
Affinity DataIC50:  55nMAssay Description:1) Affinity of compounds listed in table to cIAP1-BIR3, Ciap2-BIR3, XIAP-BIR3 was tested referring to Nikolovska-Colesks, Z. et.Al. (Analytical Bioch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM422084(US10508103, Embodiment 42)
Affinity DataIC50:  55nMAssay Description:1) Affinity of compounds listed in table to cIAP1-BIR3, Ciap2-BIR3, XIAP-BIR3 was tested referring to Nikolovska-Colesks, Z. et.Al. (Analytical Bioch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM422085(US10508103, Embodiment 43)
Affinity DataIC50:  55nMAssay Description:1) Affinity of compounds listed in table to cIAP1-BIR3, Ciap2-BIR3, XIAP-BIR3 was tested referring to Nikolovska-Colesks, Z. et.Al. (Analytical Bioch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM422086(US10508103, Embodiment 44)
Affinity DataIC50:  55nMAssay Description:1) Affinity of compounds listed in table to cIAP1-BIR3, Ciap2-BIR3, XIAP-BIR3 was tested referring to Nikolovska-Colesks, Z. et.Al. (Analytical Bioch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM422072(US10508103, Embodiment 25)
Affinity DataIC50:  55nMAssay Description:1) Affinity of compounds listed in table to cIAP1-BIR3, Ciap2-BIR3, XIAP-BIR3 was tested referring to Nikolovska-Colesks, Z. et.Al. (Analytical Bioch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM422071(US10508103, Embodiment 24)
Affinity DataIC50:  55nMAssay Description:1) Affinity of compounds listed in table to cIAP1-BIR3, Ciap2-BIR3, XIAP-BIR3 was tested referring to Nikolovska-Colesks, Z. et.Al. (Analytical Bioch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM422069(US10508103, Embodiment 22)
Affinity DataIC50:  55nMAssay Description:1) Affinity of compounds listed in table to cIAP1-BIR3, Ciap2-BIR3, XIAP-BIR3 was tested referring to Nikolovska-Colesks, Z. et.Al. (Analytical Bioch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM422087(US10508103, Embodiment 46)
Affinity DataIC50:  55nMAssay Description:1) Affinity of compounds listed in table to cIAP1-BIR3, Ciap2-BIR3, XIAP-BIR3 was tested referring to Nikolovska-Colesks, Z. et.Al. (Analytical Bioch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM422067(US10508103, Embodiment 20)
Affinity DataIC50:  55nMAssay Description:1) Affinity of compounds listed in table to cIAP1-BIR3, Ciap2-BIR3, XIAP-BIR3 was tested referring to Nikolovska-Colesks, Z. et.Al. (Analytical Bioch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM422066(US10508103, Embodiment 19)
Affinity DataIC50:  55nMAssay Description:1) Affinity of compounds listed in table to cIAP1-BIR3, Ciap2-BIR3, XIAP-BIR3 was tested referring to Nikolovska-Colesks, Z. et.Al. (Analytical Bioch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM422065(US10508103, Embodiment 18)
Affinity DataIC50:  55nMAssay Description:1) Affinity of compounds listed in table to cIAP1-BIR3, Ciap2-BIR3, XIAP-BIR3 was tested referring to Nikolovska-Colesks, Z. et.Al. (Analytical Bioch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM422064(US10508103, Embodiment 17)
Affinity DataIC50:  55nMAssay Description:1) Affinity of compounds listed in table to cIAP1-BIR3, Ciap2-BIR3, XIAP-BIR3 was tested referring to Nikolovska-Colesks, Z. et.Al. (Analytical Bioch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM422063(US10508103, Embodiment 16)
Affinity DataIC50:  55nMAssay Description:1) Affinity of compounds listed in table to cIAP1-BIR3, Ciap2-BIR3, XIAP-BIR3 was tested referring to Nikolovska-Colesks, Z. et.Al. (Analytical Bioch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM422062(US10508103, Embodiment 14)
Affinity DataIC50:  55nMAssay Description:1) Affinity of compounds listed in table to cIAP1-BIR3, Ciap2-BIR3, XIAP-BIR3 was tested referring to Nikolovska-Colesks, Z. et.Al. (Analytical Bioch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM422061(US10508103, Embodiment 13)
Affinity DataIC50:  55nMAssay Description:1) Affinity of compounds listed in table to cIAP1-BIR3, Ciap2-BIR3, XIAP-BIR3 was tested referring to Nikolovska-Colesks, Z. et.Al. (Analytical Bioch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM422060(US10508103, Embodiment 2)
Affinity DataIC50:  55nMAssay Description:1) Affinity of compounds listed in table to cIAP1-BIR3, Ciap2-BIR3, XIAP-BIR3 was tested referring to Nikolovska-Colesks, Z. et.Al. (Analytical Bioch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM422059(US10508103, Embodiment 1)
Affinity DataIC50:  55nMAssay Description:1) Affinity of compounds listed in table to cIAP1-BIR3, Ciap2-BIR3, XIAP-BIR3 was tested referring to Nikolovska-Colesks, Z. et.Al. (Analytical Bioch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBaculoviral IAP repeat-containing protein 3 [238-349](Homo sapiens (Human))
Shanghai Institute of Organic Chemistry

LigandPNGBDBM422068(US10508103, Embodiment 21)
Affinity DataIC50:  55nMAssay Description:1) Affinity of compounds listed in table to cIAP1-BIR3, Ciap2-BIR3, XIAP-BIR3 was tested referring to Nikolovska-Colesks, Z. et.Al. (Analytical Bioch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent