BDBM733127 US20250115590, Compound OC-1
BDBM733128 US20250115590, Compound OC-2
BDBM733129 US20250115590, Compound OC-3
BDBM733134 US20250115590, Compound OC-8
BDBM733135 US20250115590, Compound OC-9
BDBM733136 US20250115590, Compound OC-10
BDBM733137 US20250115590, Compound OC-11
BDBM733138 US20250115590, Compound OC-12
BDBM733139 US20250115590, Compound OC-13
BDBM733140 US20250115590, Compound OC-14
US20250115590, Compound OC-4 BDBM733130
US20250115590, Compound OC-5 BDBM733131
US20250115590, Compound OC-6 BDBM733132
US20250115590, Compound OC-7 BDBM733133
Tyr-Pro-Phe-Phe-OC(CH3)3 BDBM50271442 CHEMBL500195
BDBM50090934 CHEMBL317303 L-Arg NO2-L-Dbu-OC(CH3)3
BDBM50164079 CHEMBL181624 hexafluoridoaluminate(3-) (OC-6-11)-hexafluoroaluminate(3-) [AlF6](3-) hexafluoroaluminate(3-) AlF6(3-)
US9464092, O BDBM253923 US9527857, O
BDBM50478463 7,12-O,O''-dibenzylcoclaurine CHEMBL452762
CHEMBL332491 BDBM50131651 O-1339 O-2130
BDBM50308551 biphenyl-2-ol o-diphenylol CHEMBL108829 [1,1'-biphenyl]-2-ol o-hydroxybiphenyl o-hydroxydiphenyl o-phenylphenol
(R)-O-2,3-bis(octyloxy)propyl O,O-dihydrogen phosphorothioate CHEMBL201482 BDBM50176390
(S)-O-2,3-bis(octyloxy)propyl O,O-dihydrogen phosphorothioate CHEMBL427017 BDBM50176398
BDBM50146579 O-Benzylhydroxylamine CHEMBL443652 Benzyl-O-Hydroxylamine
- Broekema, M; van Eerd, JJ; Oyen, WJ; Corstens, FH; Liskamp, RM; Boerman, OC; Harris, TD J Med Chem 48: 6442-53 (2005)
- Howard, AD; Tan, C; Shiao, LL; Palyha, OC; McKee, KK; Weinberg, DH; Feighner, SD; Cascieri, MA; Smith, RG; Van Der Ploeg, LH; Sullivan, KA FEBS Lett 405: 285-90 (1997)
- Teixeira, TS; Freitas, RF; Abrahão, O; Devienne, KF; de Souza, LR; Blaber, SI; Blaber, M; Kondo, MY; Juliano, MA; Juliano, L; Puzer, L Bioorg Med Chem Lett 21: 6112-5 (2011)
- Nieto, MI; Balo, MC; Brea, J; Caamaño, O; Fernández, F; García-Mera, X; López, C; Loza, MI; Rodríguez-Borges, JE; Vidal, B Eur J Med Chem 45: 2884-92 (2010)
- PEVARELLO, P; SODANO, M; CUSANO, V; PISCITELLI, F; TORINO, D; VITALONE, R; YOUSIF, AM; ARTAMONOV, O US Patent US20240034737 (2024)
- Trousil, S; Carroll, L; Kalusa, A; Aberg, O; Kaliszczak, M; Aboagye, EO Medchemcomm 2013: 693-696 (2013)
- Rowbottom, MW; Tucci, FC; Connors, PJ; Gross, TD; Zhu, YF; Guo, Z; Moorjani, M; Acevedo, O; Carter, L; Sullivan, SK; Xie, Q; Fisher, A; Struthers, RS; Saunders, J; Chen, C Bioorg Med Chem Lett 14: 4967-73 (2004)
- Otto, R; Penzis, R; Gaube, F; Adolph, O; Föhr, KJ; Warncke, P; Robaa, D; Appenroth, D; Fleck, C; Enzensperger, C; Lehmann, J; Winckler, T J Med Chem 58: 6710-5 (2015)
- Ali, MR; Kumar, S; Afzal, O; Shalmali, N; Sharma, M; Bawa, S Chem Biol Drug Des 87: 508-16 (2016)
- Dockendorff, C; Aisiku, O; Verplank, L; Dilks, JR; Smith, DA; Gunnink, SF; Dowal, L; Negri, J; Palmer, M; Macpherson, L; Schreiber, SL; Flaumenhaft, R ACS Med Chem Lett 3: 232-237 (2012)
- Akgul, O; Singh, S; Andring, JT; McKenna, R; Selleri, S; Carta, F; Angeli, A; Supuran, CT Eur J Med Chem 212: (2021)
- Ahmad, S; Alam, O; Naim, MJ; Shaquiquzzaman, M; Alam, MM; Iqbal, M Eur J Med Chem 157: 527-561 (2018)
- Aktaş, DA; Akinalp, G; Sanli, F; Yucel, MA; Gambacorta, N; Nicolotti, O; Karatas, OF; Algul, O; Burmaoglu, S Bioorg Med Chem Lett 30: (2020)
- Kawamura, A; Hindi, S; Mihai, DM; James, L; Aminova, O Bioorg Med Chem 16: 8824-9 (2008)
- Fiorito, J; Vendome, J; Saeed, F; Staniszewski, A; Zhang, H; Yan, S; Deng, SX; Arancio, O; Landry, DW J Med Chem 60: 8858-8875 (2017)
- Meredith, EL; Ardayfio, O; Beattie, K; Dobler, MR; Enyedy, I; Gaul, C; Hosagrahara, V; Jewell, C; Koch, K; Lee, W; Lehmann, H; McKinsey, TA; Miranda, K; Pagratis, N; Pancost, M; Patnaik, A; Phan, D; Plato, C; Qian, M; Rajaraman, V; Rao, C; Rozhitskaya, O; Ruppen, T; Shi, J; Siska, SJ; Springer, C; van Eis, M; Vega, RB; von Matt, A; Yang, L; Yoon, T; Zhang, JH; Zhu, N; Monovich, LG J Med Chem 53: 5400-21 (2010)
- Demirci, T; Arslan, M; Bilen, ÿ; Demir, D; Gençer, N; Arslan, O J Enzyme Inhib Med Chem 29: 132-6 (2014)
- Harada, H; Asano, O; Hoshino, Y; Yoshikawa, S; Matsukura, M; Kabasawa, Y; Niijima, J; Kotake, Y; Watanabe, N; Kawata, T; Inoue, T; Horizoe, T; Yasuda, N; Minami, H; Nagata, K; Murakami, M; Nagaoka, J; Kobayashi, S; Tanaka, I; Abe, S J Med Chem 44: 170-9 (2001)
- Nguyen, MH; Atasoylu, O; Wu, L; Kapilashrami, K; Pusey, M; Gallagher, K; Lai, CT; Zhao, P; Barbosa, J; Liu, K; He, C; Zhang, C; Styduhar, ED; Witten, MR; Chen, Y; Lin, L; Yang, YO; Covington, M; Diamond, S; Yeleswaram, S; Yao, W ACS Med Chem Lett 13: 1159-1164 (2022)
- Hinze, C; Aulenbacher, O; Sundermann, B; Oberboersch, S; Friderichs, E; Englberger, W; Koegel, B; Linz, K; Schick, H; Sonnenschein, H; Henkel, B; Rose, VS; Lipkin, MJ US Patent US9120797 (2015)
- Varming, T; Christophersen, P; Møller, A; Peters, D; Axelsson, O; Nielsen, E& Bioorg Med Chem Lett 6: 245-248 (1996)
- Bürli, RW; Luckhurst, CA; Aziz, O; Matthews, KL; Yates, D; Lyons, KA; Beconi, M; McAllister, G; Breccia, P; Stott, AJ; Penrose, SD; Wall, M; Lamers, M; Leonard, P; Müller, I; Richardson, CM; Jarvis, R; Stones, L; Hughes, S; Wishart, G; Haughan, AF; O'Connell, C; Mead, T; McNeil, H; Vann, J; Mangette, J; Maillard, M; Beaumont, V; Munoz-Sanjuan, I; Dominguez, C J Med Chem 56: 9934-54 (2013)
- Mamolo, MG; Zampieri, D; Zanette, C; Florio, C; Collina, S; Urbano, M; Azzolina, O; Vio, L Eur J Med Chem 43: 2073-81 (2008)
- AUGUSTYNS, K; BENRAMDANE, S; BEYENS, O; DE LOOSE, J; DE MEESTER, I; DE WINTER, H; ESPADINHA, M; FILIPPI, N; VAN DER VEKEN, P US Patent US20250353833 (2025)
- Martucci, WE; Udier-Blagovic, M; Atreya, C; Babatunde, O; Vargo, MA; Jorgensen, WL; Anderson, KS Bioorg Med Chem Lett 19: 418-23 (2008)
- Bakare, O; Lee, CM; Brandy, Y; Khraiwesh, MH US Patent US9422231 (2016)
- Rogacki, MK; Pitta, E; Balabon, O; Huss, S; Lopez-Roman, EM; Argyrou, A; Blanco-Ruano, D; Cacho, M; Vande Velde, CML; Augustyns, K; Ballell, L; Barros, D; Bates, RH; Cunningham, F; Van der Veken, P J Med Chem 61: 11221-11249 (2018)
- Ledneczki, I; Tapolcsányi, P; Gábor, E; Éles, J; Greiner, I; Schmidt, É; Némethy, Z; Kedves, RS; Balázs, O; Román, V; Lévay, G; Mahó, S Bioorg Med Chem Lett 27: 4525-4530 (2017)
- Siegel, D; Hui, HC; Doerffler, E; Clarke, MO; Chun, K; Zhang, L; Neville, S; Carra, E; Lew, W; Ross, B; Wang, Q; Wolfe, L; Jordan, R; Soloveva, V; Knox, J; Perry, J; Perron, M; Stray, KM; Barauskas, O; Feng, JY; Xu, Y; Lee, G; Rheingold, AL; Ray, AS; Bannister, R; Strickley, R; Swaminathan, S; Lee, WA; Bavari, S; Cihlar, T; Lo, MK; Warren, TK; Mackman, RL J Med Chem 60: 1648-1661 (2017)
- Jones, LH; Allan, G; Barba, O; Burt, C; Corbau, R; Dupont, T; Knöchel, T; Irving, S; Middleton, DS; Mowbray, CE; Perros, M; Ringrose, H; Swain, NA; Webster, R; Westby, M; Phillips, C J Med Chem 52: 1219-23 (2009)
- Gerhart, SV; Kellner, WA; Thompson, C; Pappalardi, MB; Zhang, XP; Montes de Oca, R; Penebre, E; Duncan, K; Boriack-Sjodin, A; Le, B; Majer, C; McCabe, MT; Carpenter, C; Johnson, N; Kruger, RG; Barbash, O Sci Rep 8:
- Cheeseman, MD; Westwood, IM; Barbeau, O; Rowlands, M; Dobson, S; Jones, AM; Jeganathan, F; Burke, R; Kadi, N; Workman, P; Collins, I; van Montfort, RL; Jones, K J Med Chem 59: 4625-36 (2016)
- O'Dowd, CR; Helm, MD; Rountree, JSS; Flasz, JT; Arkoudis, E; Miel, H; Hewitt, PR; Jordan, L; Barker, O; Hughes, C; Rozycka, E; Cassidy, E; McClelland, K; Odrzywol, E; Page, N; Feutren-Burton, S; Dvorkin, S; Gavory, G; Harrison, T ACS Med Chem Lett 9: 238-243 (2018)
- Wu, YJ; Guernon, J; McClure, A; Luo, G; Rajamani, R; Ng, A; Easton, A; Newton, A; Bourin, C; Parker, D; Mosure, K; Barnaby, O; Soars, MG; Knox, RJ; Matchett, M; Pieschl, R; Herrington, J; Chen, P; Sivarao, DV; Bristow, LJ; Meanwell, NA; Bronson, J; Olson, R; Thompson, LA; Dzierba, C Bioorg Med Chem 25: 5490-5505 (2017)
- Hortala, L; Arnaud, J; Roux, P; Oustric, D; Boulu, L; Oury-Donat, F; Avenet, P; Rooney, T; Alagille, D; Barret, O; Tamagnan, G; Barth, F Bioorg Med Chem Lett 24: 283-7 (2014)
- Skácel, J; Djukic, S; Baszczyňski, O; Kalčic, F; Bílek, T; Chalupský, K; Kozák, J; Dvořáková, A; Tloušt'ová, E; Král'ová, Z; Šmídková, M; Voldřich, J; Rumlová, M; Pachl, P; Brynda, J; Vučková, T; Fábry, M; Snášel, J; Pichová, I; Řezáčová, P; Mertlíková-Kaiserová, H; Janeba, Z J Med Chem 66: 6652-6681 (2023)
- La Regina, G; Silvestri, R; Gatti, V; Lavecchia, A; Novellino, E; Befani, O; Turini, P; Agostinelli, E Bioorg Med Chem 16: 9729-40 (2008)
- Sund, C; Belda, O; Borkakoti, N; Lindberg, J; Derbyshire, D; Vrang, L; Hamelink, E; Åhgren, C; Woestenenk, E; Wikström, K; Eneroth, A; Lindström, E; Kalayanov, G Bioorg Med Chem Lett 22: 6721-7 (2012)
- Sharma, R; Nikas, SP; Paronis, CA; Wood, JT; Halikhedkar, A; Guo, JJ; Thakur, GA; Kulkarni, S; Benchama, O; Raghav, JG; Gifford, RS; Järbe, TU; Bergman, J; Makriyannis, A J Med Chem 56: 10142-57 (2013)
- Sobolova, K; Hrabinova, M; Hepnarova, V; Kucera, T; Kobrlova, T; Benkova, M; Janockova, J; Dolezal, R; Prchal, L; Benek, O; Mezeiova, E; Jun, D; Soukup, O; Korabecny, J Eur J Med Chem 203: (2020)
- Lesuisse, D; Gourvest, JF; Hartmann, C; Tric, B; Benslimane, O; Philibert, D; Vevert, JP J Med Chem 35: 1588-97 (1992)
- Ryckmans, T; Balançon, L; Berton, O; Genicot, C; Lamberty, Y; Lallemand, B; Pasau, P; Pirlot, N; Quéré, L; Talaga, P Bioorg Med Chem Lett 12: 261-4 (2001)
- Bezencon, O; Gatfield, J; Heidmann, B; Siegrist, R; Stamm, S US Patent US10246426 (2019)
- Remen, L; Bezençon, O; Simons, L; Gaston, R; Downing, D; Gatfield, J; Roch, C; Kessler, M; Mosbacher, J; Pfeifer, T; Grisostomi, C; Rey, M; Ertel, EA; Moon, R J Med Chem 59: 8398-411 (2016)
- Venkatraman, P; Nguyen, TT; Sainlos, M; Bilsel, O; Chitta, S; Imperiali, B; Stern, LJ Nat Chem Biol 3: 222-8 (2007)
- Bobileva, O; Bokaldere, R; Gailite, V; Kaula, I; Ikaunieks, M; Duburs, G; Petrovska, R; Mandrika, I; Klovins, J; Loza, E Bioorg Med Chem 22: 3654-69 (2014)
- Boudker, O; Ryan, RM; Yernool, D; Shimamoto, K; Gouaux, E Nature 445: 387-93 (2007)
- Garrison, AT; Orsi, DL; Capstick, RA; Whomble, D; Li, J; Carter, TR; Felts, AS; Vinson, PN; Rodriguez, AL; Han, A; Hajari, K; Cho, HP; Teal, LB; Ragland, MG; Ghamari-Langroudi, M; Bubser, M; Chang, S; Schnetz-Boutaud, NC; Boutaud, O; Blobaum, AL; Foster, DJ; Niswender, CM; Conn, PJ; Lindsley, CW; Jones, CK; Han, C J Med Chem 65: 6273-6286 (2022)
- Manetti, F; Brullo, C; Magnani, M; Mosci, F; Chelli, B; Crespan, E; Schenone, S; Naldini, A; Bruno, O; Trincavelli, ML; Maga, G; Carraro, F; Martini, C; Bondavalli, F; Botta, M J Med Chem 51: 1252-9 (2008)
- Temal-Laib, T; Peixoto, C; Desroy, N; De Lemos, E; Bonnaterre, F; Bienvenu, N; Picolet, O; Sartori, E; Bucher, D; López-Ramos, M; Roca Magadán, C; Laenen, W; Flower, T; Mollat, P; Bugaud, O; Touitou, R; Pereira Fernandes, A; Lavazais, S; Monjardet, A; Borgonovi, M; Gosmini, R; Brys, R; Amantini, D; De Vos, S; Andrews, M J Med Chem 67: 380-401 (2024)
- Sağlık, BN; Osmaniye, D; Çevik, UA; Levent, S; Çavuşoğlu, BK; Büyükemir, O; Nezir, D; Karaduman, AB; Özkay, Y; Koparal, AS; Beydemir, Ş; Kaplancıklı, ZA Eur J Med Chem 198: (2020)
- Majellaro, M; Jespers, W; Crespo, A; Núñez, MJ; Novio, S; Azuaje, J; Prieto-Díaz, R; Gioé, C; Alispahic, B; Brea, J; Loza, MI; Freire-Garabal, M; Garcia-Santiago, C; Rodríguez-García, C; García-Mera, X; Caamaño, O; Fernandez-Masaguer, C; Sardina, JF; Stefanachi, A; El Maatougui, A; Mallo-Abreu, A; Åqvist, J; Gutiérrez-de-Terán, H; Sotelo, E J Med Chem 64: 458-480 (2021)
- Congreve, M; Aharony, D; Albert, J; Callaghan, O; Campbell, J; Carr, RA; Chessari, G; Cowan, S; Edwards, PD; Frederickson, M; McMenamin, R; Murray, CW; Patel, S; Wallis, N J Med Chem 50: 1124-32 (2007)
- Andrés, M; Buil, MA; Calbet, M; Casado, O; Castro, J; Eastwood, PR; Eichhorn, P; Ferrer, M; Forns, P; Moreno, I; Petit, S; Roberts, RS Bioorg Med Chem Lett 24: 5111-7 (2014)
- Jones, P; Altamura, S; Chakravarty, PK; Cecchetti, O; De Francesco, R; Gallinari, P; Ingenito, R; Meinke, PT; Petrocchi, A; Rowley, M; Scarpelli, R; Serafini, S; Steinkühler, C Bioorg Med Chem Lett 16: 5948-52 (2006)
- Arévalo, B; Bedoya, M; Kiper, AK; Vergara, F; Ramírez, D; Mazola, Y; Bustos, D; Zúñiga, R; Cikutovic, R; Cayo, A; Rinné, S; Ramirez-Apan, MT; Sepúlveda, FV; Cerda, O; López-Collazo, E; Decher, N; Zúñiga, L; Gutierrez, M; González, W J Med Chem 65: 15014-15027 (2022)
- Mak, LH; Knott, J; Scott, KA; Scott, C; Whyte, GF; Ye, Y; Mann, DJ; Ces, O; Stivers, J; Woscholski, R Bioorg Med Chem 20: 4371-6 (2012)
- Hoffman, CS; Ceyhan, O US Patent US9173884 (2015)
- Cristau, M; Devin, C; Oiry, C; Chaloin, O; Amblard, M; Bernad, N; Heitz, A; Fehrentz, JA; Martinez, J J Med Chem 43: 2356-61 (2000)
- Durek, T; Cromm, PM; White, AM; Schroeder, CI; Kaas, Q; Weidmann, J; Ahmad Fuaad, A; Cheneval, O; Harvey, PJ; Daly, NL; Zhou, Y; Dellsén, A; Österlund, T; Larsson, N; Knerr, L; Bauer, U; Kessler, H; Cai, M; Hruby, VJ; Plowright, AT; Craik, DJ J Med Chem 61: 3674-3684 (2018)
- Ceccarelli, SM; Chomienne, O; Gubler, M; Arduini, A J Med Chem 54: 3109-52 (2011)
- Ouvry, G; Bihl, F; Bouix-Peter, C; Christin, O; Defoin-Platel, C; Deret, S; Feret, C; Froude, D; Hacini-Rachinel, F; Harris, CS; Hervouet, C; Lafitte, G; Luzy, AP; Musicki, B; Orfila, D; Parnet, V; Pascau, C; Pascau, J; Pierre, R; Raffin, C; Rossio, P; Spiesse, D; Taquet, N; Thoreau, E; Vatinel, R; Vial, E; Hennequin, LF Bioorg Med Chem Lett 28: 1269-1273 (2018)
- Giorgioni, G; Ambrosini, D; Vesprini, C; Hudson, A; Nasuti, C; Di Stefano, A; Sozio, P; Ciampi, O; Costa, B; Martini, C; Carrieri, A; Carbonara, G; Enzensperger, C; Pigini, M Bioorg Med Chem 18: 7085-91 (2010)
- Son, JH; Zhu, JS; Phuan, PW; Cil, O; Teuthorn, AP; Ku, CK; Lee, S; Verkman, AS; Kurth, MJ J Med Chem 60: 2401-2410 (2017)
- Biernacki, K; Ciupak, O; Daśko, M; Rachon, J; Kozak, W; Rak, J; Kubiński, K; Masłyk, M; Martyna, A; Śliwka-Kaszyńska, M; Wietrzyk, J; Świtalska, M; Nocentini, A; Supuran, CT; Demkowicz, S J Med Chem 65: 5044-5056 (2022)
- Urbano, M; Guerrero, M; Zhao, J; Velaparthi, S; Saldanha, SA; Chase, P; Wang, Z; Civelli, O; Hodder, P; Schaeffer, MT; Brown, S; Rosen, H; Roberts, E Bioorg Med Chem Lett 22: 7135-41 (2012)
- McCoull, W; Boyd, S; Brown, MR; Coen, M; Collingwood, O; Davies, NL; Doherty, A; Fairley, G; Goldberg, K; Hardaker, E; He, G; Hennessy, EJ; Hopcroft, P; Hodgson, G; Jackson, A; Jiang, X; Karmokar, A; Lainé, AL; Lindsay, N; Mao, Y; Markandu, R; McMurray, L; McLean, N; Mooney, L; Musgrove, H; Nissink, JWM; Pflug, A; Reddy, VP; Rawlins, PB; Rivers, E; Schimpl, M; Smith, GF; Tentarelli, S; Travers, J; Troup, RI; Walton, J; Wang, C; Wilkinson, S; Williamson, B; Winter-Holt, J; Yang, D; Zheng, Y; Zhu, Q; Smith, PD J Med Chem 64: 13524-13539 (2021)
- Siegrist, R; Pozzi, D; Jacob, G; Torrisi, C; Colas, K; Braibant, B; Mawet, J; Pfeifer, T; de Kanter, R; Roch, C; Kessler, M; Corminboeuf, O; Bezençon, O J Med Chem 59: 10661-10675 (2016)
- Mougenot, P; Namane, C; Fett, E; Goumy, F; Dadji-Faïhun, R; Langot, G; Monseau, C; Onofri, B; Pacquet, F; Pascal, C; Crespin, O; Ben-Hassine, M; Ragot, JL; Van-Pham, T; Philippo, C; Chatelain-Egger, F; Péron, P; Le Bail, JC; Guillot, E; Chamiot-Clerc, P; Chabanaud, MA; Pruniaux, MP; Ménegotto, J; Schmidt, F; Venier, O; Viviani, F; Nicolai, E Bioorg Med Chem Lett 26: 25-32 (2016)
- Micheli, F; Bonanomi, G; Blaney, FE; Braggio, S; Capelli, AM; Checchia, A; Curcuruto, O; Damiani, F; Fabio, RD; Donati, D; Gentile, G; Gribble, A; Hamprecht, D; Tedesco, G; Terreni, S; Tarsi, L; Lightfoot, A; Stemp, G; Macdonald, G; Smith, A; Pecoraro, M; Petrone, M; Perini, O; Piner, J; Rossi, T; Worby, A; Pilla, M; Valerio, E; Griffante, C; Mugnaini, M; Wood, M; Scott, C; Andreoli, M; Lacroix, L; Schwarz, A; Gozzi, A; Bifone, A; Ashby, CR; Hagan, JJ; Heidbreder, C J Med Chem 50: 5076-89 (2007)
- Meltzer, D; Ethan, O; Arguin, G; Nadel, Y; Danino, O; Lecka, J; Sévigny, J; Gendron, FP; Fischer, B Bioorg Med Chem 23: 5764-73 (2015)
- Darlami, O; Pun, R; Ahn, SH; Kim, SH; Shin, D Eur J Med Chem 272:
- Josef, TT; David, O; Pascal, F; Klaus, W; Achim, S WIPO WO2022091056 (2022)
- Boland, S; Bourin, A; Alen, J; Geraets, J; Schroeders, P; Castermans, K; Kindt, N; Boumans, N; Panitti, L; Vanormelingen, J; Fransen, S; Van de Velde, S; Defert, O Bioorg Med Chem Lett 25: 4005-10 (2015)
- Fichez, J; Soulie, C; Le Corre, L; Sayon, S; Priet, S; Alvarez, K; Delelis, O; Gizzi, P; Prestat, G; Gravier-Pelletier, C; Marcelin, AG; Calvez, V; Busca, P RSC Med Chem 11: 577-582 (2020)
- Maibaum, J; Liao, SM; Vulpetti, A; Ostermann, N; Randl, S; Rüdisser, S; Lorthiois, E; Erbel, P; Kinzel, B; Kolb, FA; Barbieri, S; Wagner, J; Durand, C; Fettis, K; Dussauge, S; Hughes, N; Delgado, O; Hommel, U; Gould, T; Mac Sweeney, A; Gerhartz, B; Cumin, F; Flohr, S; Schubart, A; Jaffee, B; Harrison, R; Risitano, AM; Eder, J; Anderson, K Nat Chem Biol 12: 1105-1110 (2016)
- Rossi, AM; Riley, AM; Tovey, SC; Rahman, T; Dellis, O; Taylor, EJ; Veresov, VG; Potter, BV; Taylor, CW Nat Chem Biol 5: 631-9 (2009)
- Jagtap, PK; Garg, D; Kapp, TG; Will, CL; Demmer, O; Lührmann, R; Kessler, H; Sattler, M J Med Chem 59: 10190-10197 (2016)
- Deo, O; Alvi, S; Pham, V; Christopoulos, A; Thal, DM; Jörg, M; Capuano, B; Valant, C; Scammells, PJ J Med Chem 65: 12367-12385 (2022)
- Kozikowski, AP; Johnson, KM; Deschaux, O; Bandyopadhyay, BC; Araldi, GL; Carmona, G; Munzar, P; Smith, MP; Balster, RL; Beardsley, PM; Tella, SR J Pharmacol Exp Ther 305: 143-50 (2003)
- Hayek, S; Pietrancosta, N; Hovhannisyan, AA; Alves de Sousa, R; Bekaddour, N; Ermellino, L; Tramontano, E; Arnould, S; Sardet, C; Dairou, J; Diaz, O; Lotteau, V; Nisole, S; Melikyan, G; Herbeuval, JP; Vidalain, PO Eur J Med Chem 186: (2020)
- Horsfall, LE; Garau, G; Liénard, BM; Dideberg, O; Schofield, CJ; Frère, JM; Galleni, M Antimicrob Agents Chemother 51: 2136-42 (2007)
- Blöcher, R; Lamers, C; Wittmann, SK; Merk, D; Hartmann, M; Weizel, L; Diehl, O; Brüggerhoff, A; Boß, M; Kaiser, A; Schader, T; Göbel, T; Grundmann, M; Angioni, C; Heering, J; Geisslinger, G; Wurglics, M; Kostenis, E; Brüne, B; Steinhilber, D; Schubert-Zsilavecz, M; Kahnt, AS; Proschak, E J Med Chem 59: 61-81 (2016)
- Diouf, O; Gadeau, S; Chellé, F; Gelbcke, M; Talaga, P; Christophe, B; Gillard, M; Massingham, R; Guyaux, M Bioorg Med Chem Lett 12: 2535-9 (2002)
- Elliott, JM; Carlson, EJ; Chicchi, GG; Dirat, O; Dominguez, M; Gerhard, U; Jelley, R; Jones, AB; Kurtz, MM; Tsao, K; Wheeldon, A Bioorg Med Chem Lett 16: 2929-32 (2006)
- Chrysanthopoulos, PK; Mujumdar, P; Woods, LA; Dolezal, O; Ren, B; Peat, TS; Poulsen, SA J Med Chem 60: 7333-7349 (2017)
- Li, Y; Zhao, J; Gutgesell, LM; Shen, Z; Ratia, K; Dye, K; Dubrovskyi, O; Zhao, H; Huang, F; Tonetti, DA; Thatcher, GRJ; Xiong, R J Med Chem 63: 7186-7210 (2020)
- Lu, Y; Gutgesell, LM; Xiong, R; Zhao, J; Li, Y; Rosales, CI; Hollas, M; Shen, Z; Gordon-Blake, J; Dye, K; Wang, Y; Lee, S; Chen, H; He, D; Dubrovyskyii, O; Zhao, H; Huang, F; Lasek, AW; Tonetti, DA; Thatcher, GRJ J Med Chem 62: 11301-11323 (2019)
- Alam, A; Biscarrat, S; Blanc, I; Bono, F; Duclos, O; Mccort, G US Patent US8470847 (2013)
- Paoletti, J; Assairi, L; Gelin, M; Huteau, V; Nahori, MA; Dussurget, O; Labesse, G; Pochet, S Eur J Med Chem 124: 1041-1056 (2016)
- Schulze, VK; Klar, U; Kosemund, D; Wengner, AM; Siemeister, G; Stöckigt, D; Neuhaus, R; Lienau, P; Bader, B; Prechtl, S; Holton, SJ; Briem, H; Marquardt, T; Schirok, H; Jautelat, R; Bohlmann, R; Nguyen, D; Fernández-Montalván, AE; Bömer, U; Eberspaecher, U; Brüning, M; Döhr, O; Raschke, M; Kreft, B; Mumberg, D; Ziegelbauer, K; Brands, M; von Nussbaum, F; Koppitz, M J Med Chem 63: 8025-8042 (2020)
- Dighe, SN; Ekwudu, O; Dua, K; Chellappan, DK; Katavic, PL; Collet, TA Eur J Med Chem 176: 431-455 (2019)
- Yuan, Y; Elbegdorj, O; Beletskaya, IO; Selley, DE; Zhang, Y Bioorg Med Chem Lett 23: 5045-8 (2013)
- Savateev, K; Fedotov, V; Butorin, I; Eltsov, O; Slepukhin, P; Ulomsky, E; Rusinov, V; Litvinov, R; Babkov, D; Khokhlacheva, E; Radaev, P; Vassiliev, P; Spasov, A Eur J Med Chem 185: (2020)
- Bornot, A; Bauer, U; Brown, A; Firth, M; Hellawell, C; Engkvist, O J Med Chem 56: 1197-210 (2013)
- Engström, O; Belda, O; Kullman-Magnusson, M; Rapp, M; Böhm, K; Paul, R; Henderson, I; Derbyshire, D; Karlström, S; Parkes, KEB; Zhao, H Bioorg Med Chem Lett 30: (2020)
- Brand, S; Ko, EJ; Viayna, E; Thompson, S; Spinks, D; Thomas, M; Sandberg, L; Francisco, AF; Jayawardhana, S; Smith, VC; Jansen, C; De Rycker, M; Thomas, J; MacLean, L; Osuna-Cabello, M; Riley, J; Scullion, P; Stojanovski, L; Simeons, FRC; Epemolu, O; Shishikura, Y; Crouch, SD; Bakshi, TS; Nixon, CJ; Reid, IH; Hill, AP; Underwood, TZ; Hindley, SJ; Robinson, SA; Kelly, JM; Fiandor, JM; Wyatt, PG; Marco, M; Miles, TJ; Read, KD; Gilbert, IH J Med Chem 60: 7284-7299 (2017)
- Huang, H; Acquaviva, L; Berry, V; Bregman, H; Chakka, N; DiMauro, EF; Dovey, J; Epstein, O; Grubinska, B; Goldstein, J; Gunaydin, H; Hua, Z; Huang, X; Huang, L; Human, J; Long, A; Newcomb, J; Patel, VF; Saffran, D; Serafino, R; Schneider, S; Strathdee, C; Tang, J; Turci, S; White, R; Yu, V; Zhao, H; Wilson, C; Martin, MW ACS Med Chem Lett 3: 1059-1064 (2012)
- Nakache, P; Erez, O; Botti, S; Goutopoulos, A; Finch, H US Patent US12441689 (2025)
- Olsson, H; Sjö, P; Ersoy, O; Kristoffersson, A; Larsson, J; Nordén, B Bioorg Med Chem Lett 20: 4738-40 (2010)
- Galiano, S; Erviti, O; Pérez, S; Moreno, A; Juanenea, L; Aldana, I; Monge, A Bioorg Med Chem Lett 14: 597-9 (2004)
- Meltzer, D; Ethan, O; Arguin, G; Nadel, Y; Danino, O; Lecka, J; Sévigny, J; Gendron, FP; Fischer, B Bioorg Med Chem 23: 5764-73 (2015)
- Gopalsamy, A; Narayanan, A; Liu, S; Parikh, MD; Kyne, RE; Fadeyi, O; Tones, MA; Cherry, JJ; Nabhan, JF; LaRosa, G; Petersen, DN; Menard, C; Foley, TL; Noell, S; Ren, Y; Loria, PM; Maglich-Goodwin, J; Rong, H; Jones, LH J Med Chem 60: 3094-3108 (2017)
- Zhang, Z; Barros-Álvarez, X; Gillespie, JR; Ranade, RM; Huang, W; Shibata, S; Molasky, NMR; Faghih, O; Mushtaq, A; Choy, RKM; de Hostos, E; Hol, WGJ; Verlinde, CLMJ; Buckner, FS; Fan, E RSC Med Chem 11: 885-895 (2020)
- Fish, PV; Filippakopoulos, P; Bish, G; Brennan, PE; Bunnage, ME; Cook, AS; Federov, O; Gerstenberger, BS; Jones, H; Knapp, S; Marsden, B; Nocka, K; Owen, DR; Philpott, M; Picaud, S; Primiano, MJ; Ralph, MJ; Sciammetta, N; Trzupek, JD J Med Chem 55: 9831-7 (2012)
- Henderson, SH; Sorrell, FJ; Bennett, JM; Fedorov, O; Hanley, MT; Godoi, PH; Ruela de Sousa, R; Robinson, S; Navratilova, IH; Elkins, JM; Ward, SE Eur J Med Chem 269:
- Ravez, S; Corbet, C; Spillier, Q; Dutu, A; Robin, AD; Mullarky, E; Cantley, LC; Feron, O; Frédérick, R J Med Chem 60: 1591-1597 (2017)
- Hynes, JB; Singh, SK; Fetzer, O; Shane, B J Med Chem 35: 4078-85 (1992)
- Hortala, L; Rinaldi-Carmona, M; Congy, C; Boulu, L; Sadoun, F; Fabre, G; Finance, O; Barth, F Bioorg Med Chem Lett 20: 4573-7 (2010)
- Razzaghi-Asl, N; Firuzi, O; Hemmateenejad, B; Javidnia, K; Edraki, N; Miri, R Bioorg Med Chem 21: 6893-909 (2013)
- Davidsson, Ö; Nilsson, K; Brånalt, J; Andersson, T; Berggren, K; Chen, Y; Fjellström, O; Gradén, H; Gustafsson, L; Hermansson, NO; Jansen, F; Johannesson, P; Ohlsson, B; Tyrchan, C; Wellner, A; Wellner, E; Ölwegård-Halvarsson, M Bioorg Med Chem Lett 30: (2020)
- Hu, S; Huang, Y; Deshpande, M; Luo, G; Bruce, MA; Chen, L; Mattson, G; Iben, LG; Zhang, J; Russell, JW; Clarke, WJ; Hogan, JB; Ortiz, A; Flint, O; Henwood, A; Gao, Q; Antal-Zimanyi, I; Poindexter, GS ACS Med Chem Lett 3: 222-226 (2012)
- Fragai, M; Comito, G; Di Cesare Mannelli, L; Gualdani, R; Calderone, V; Louka, A; Richichi, B; Francesconi, O; Angeli, A; Nocentini, A; Gratteri, P; Chiarugi, P; Ghelardini, C; Tadini-Buoninsegni, F; Supuran, CT; Nativi, C J Med Chem 60: 9003-9011 (2017)
- Jacobs, MD; Black, J; Futer, O; Swenson, L; Hare, B; Fleming, M; Saxena, K J Biol Chem 280: 13728-34 (2005)
- Gautschi, O; Mack, PC; Davies, AM; Lara, PN; Gandara, DR Clin Lung Cancer 8: 93-8
- Gavelle, O; Grether, U; Kimbara, A; Nettekoven, M; Stephan, R; Rogers-Evans, M; Rombach, D; Schulz-Gasch, T US Patent US10308659 (2019)
- Oliva, P; Suresh, RR; Pasquini, S; Salmaso, V; Will, EJ; Tosh, DK; Gao, ZG; Liu, N; Gavrilova, O; Vincenzi, F; Varani, K; Jacobson, KA ACS Med Chem Lett 14: 1640-1646 (2023)
- Le Tiran, A; Le Diguarher, T; Starck, J; Henlin, J; Guillouzic, A; De Nanteuil, G; Geneste, O; Fejes, I; Tatai, J; Nyerges, M; Davidson, JE; Murray, JB; Chen, I; Durand, D US Patent US9108983 (2015)
- Singh, SB; Goetz, MA; Smith, SK; Zink, DL; Polishook, J; Onishi, R; Salowe, S; Wiltsie, J; Allocco, J; Sigmund, J; Dorso, K; de la Cruz, M; Martín, J; Vicente, F; Genilloud, O; Donald, RG; Phillips, JW Bioorg Med Chem Lett 22: 7127-30 (2012)
- Campiani, G; Butini, S; Fattorusso, C; Trotta, F; Gemma, S; Catalanotti, B; Nacci, V; Fiorini, I; Cagnotto, A; Mereghetti, I; Mennini, T; Minetti, P; Di Cesare, MA; Stasi, MA; Di Serio, S; Ghirardi, O; Tinti, O; Carminati, P J Med Chem 48: 1705-8 (2005)
- Rosenthal, AS; Dexheimer, TS; Gileadi, O; Nguyen, GH; Chu, WK; Hickson, ID; Jadhav, A; Simeonov, A; Maloney, DJ Bioorg Med Chem Lett 23: 5660-6 (2013)
- Kesteleyn, B; Bardiot, D; Bonfanti, JF; De Boeck, B; Goethals, O; Kaptein, SJF; Stoops, B; Coesemans, E; Fortin, J; Muller, P; Doublet, F; Carlens, G; Koukni, M; Smets, W; Raboisson, P; Chaltin, P; Simmen, K; Van Loock, M; Neyts, J; Marchand, A; Jonckers, THM J Med Chem 66: 8808-8821 (2023)
- Golonzhka, O; Jarpe, MB US Patent US10858323 (2020)
- von Kleist, L; Michaelis, S; Bartho, K; Graebner, O; Schlief, M; Dreger, M; Schrey, AK; Sefkow, M; Kroll, F; Koester, H; Luo, Y J Med Chem 59: 4664-75 (2016)
- Basarab, GS; Hill, PJ; Garner, CE; Hull, K; Green, O; Sherer, BA; Dangel, PB; Manchester, JI; Bist, S; Hauck, S; Zhou, F; Uria-Nickelsen, M; Illingworth, R; Alm, R; Rooney, M; Eakin, AE J Med Chem 57: 6060-82 (2014)
- Grütter, C; Simard, JR; Mayer-Wrangowski, SC; Schreier, PH; Pérez-Martín, J; Richters, A; Getlik, M; Gutbrod, O; Braun, CA; Beck, ME; Rauh, D ACS Chem Biol 7: 1257-67 (2012)
- Novotná, B; Vaneková, L; Zavřel, M; Buděšínský, M; Dejmek, M; Smola, M; Gutten, O; Tehrani, ZA; Pimková Polidarová, M; Brázdová, A; Liboska, R; Štěpánek, I; Vavřina, Z; Jandušík, T; Nencka, R; Rulíšek, L; Bouřa, E; Brynda, J; Páv, O; Birkuš, G J Med Chem 62: 10676-10690 (2019)
- Mohamed, FAM; Alakilli, SYM; El Azab, EF; Baawad, FAM; Shaaban, EIA; Alrub, HA; Hendawy, O; Gomaa, HAM; Bakr, AG; Abdelrahman, MH; Trembleau, L; Mohammed, AF; Youssif, BGM RSC Med Chem 14: 734-744 (2023)
- Henry, O; Lopez-Gallego, F; Agger, SA; Schmidt-Dannert, C; Sen, S; Shintani, D; Cornish, K; Distefano, MD Bioorg Med Chem 17: 4797-805 (2009)
- Narayanan, BC; Niu, W; Han, Y; Zou, J; Mariano, PS; Dunaway-Mariano, D; Herzberg, O Biochemistry 47: 167-82 (2008)
- Olsson, RI; Jacobson, I; Iliefski, T; Boström, J; Davidsson, Ö; Fjellström, O; Björe, A; Olsson, C; Sundell, J; Gran, U; Gyll, J; Malmberg, J; Hidestål, O; Emtenäs, H; Svensson, T; Yuan, ZQ; Strandlund, G; Åstrand, A; Lindhardt, E; Linhardt, G; Forsström, E; Högberg, Å; Persson, F; Andersson, B; Rönnborg, A; Löfberg, B Bioorg Med Chem Lett 24: 1269-73 (2014)
- Nordhoff, S; Cerezo-Gálvez, S; Deppe, H; Hill, O; López-Canet, M; Rummey, C; Thiemann, M; Matassa, VG; Edwards, PJ; Feurer, A Bioorg Med Chem Lett 19: 4201-3 (2009)
- Pochetti, G; Gavuzzo, E; Campestre, C; Agamennone, M; Tortorella, P; Consalvi, V; Gallina, C; Hiller, O ; Tschesche, H; Tucker, PA; Mazza, F J Med Chem 49: 923-31 (2006)
- Musilek, K; Komloova, M; Zavadova, V; Holas, O; Hrabinova, M; Pohanka, M; Dohnal, V; Nachon, F; Dolezal, M; Kuca, K; Jung, YS Bioorg Med Chem Lett 20: 1763-6 (2010)
- Pergola, C; Gaboriaud-Kolar, N; Jestädt, N; König, S; Kritsanida, M; Schaible, AM; Li, H; Garscha, U; Weinigel, C; Barz, D; Albring, KF; Huber, O; Skaltsounis, AL; Werz, O J Med Chem 57: 3715-23 (2014)
- Lemke, CT; Goudreau, N; Zhao, S; Hucke, O; Thibeault, D; Llinás-Brunet, M; White, PW J Biol Chem 286: 11434-43 (2011)
- León, R; de los Ríos, C; Marco-Contelles, J; Huertas, O; Barril, X; Luque, FJ; López, MG; García, AG; Villarroya, M Bioorg Med Chem 16: 7759-69 (2008)
- Saraswati, AP; Relitti, N; Brindisi, M; Osko, JD; Chemi, G; Federico, S; Grillo, A; Brogi, S; McCabe, NH; Turkington, RC; Ibrahim, O; O'Sullivan, J; Lamponi, S; Ghanim, M; Kelly, VP; Zisterer, D; Amet, R; Hannon Barroeta, P; Vanni, F; Ulivieri, C; Herp, D; Sarno, F; Di Costanzo, A; Saccoccia, F; Ruberti, G; Jung, M; Altucci, L; Gemma, S; Butini, S; Christianson, DW; Campiani, G ACS Med Chem Lett 11: 2268-2276 (2020)
- Courtney, S; Yarnold, C; Flanagan, S; Brace, G; Barker, J; Ichihara, O; Gadouleau, E; Richardson, A; Kondo, T; Imagawa, A; Nakatani, S; Suzuki, R; Kouyama, S US Patent US9732085 (2017)
- Konishi, A; Tokumasu, M; Suzuki, T; Koshiba, T; Ohsumi, K; Ikehara, O; Kodama, Y US Patent US8609715 (2013)
- Hilton-Proctor, JP; Ilyichova, O; Zheng, Z; Jennings, IG; Johnstone, RW; Shortt, J; Mountford, SJ; Scanlon, MJ; Thompson, PE Bioorg Med Chem 27: (2019)
- Meiering, S; Inhoff, O; Mies, J; Vincek, A; Garcia, G; Kramer, B; Dormeyer, M; Krauth-Siegel, RL J Med Chem 48: 4793-802 (2005)
- Yokokawa, F; Ehara, T; Kawakami, S; Irie, O; Suzuki, M; Hitomi, Y; Toyao, A US Patent US8497286 (2013)
- Jacobson, O; Weiss, ID; Szajek, L; Farber, JM; Kiesewetter, DO Bioorg Med Chem 17: 1486-93 (2009)
- Balavoine, F; Malabre, P; Alleaume, T; Rey, A; Cherfils, V; Jeanneton, O; Seigneurin-Venin, S; Revah, F Bioorg Med Chem Lett 17: 3754-9 (2007)
- ATKINSON, S; DE BRUIN, G; IZZO, F; JANSEN, C; KINZEL, O; PACKER, M; VERKAIK, S; VOETS, R US Patent US20240335431 (2024)
- Ginsburg-Shmuel, T; Haas, M; Schumann, M; Reiser, G; Kalid, O; Stern, N; Fischer, B J Med Chem 53: 1673-85 (2010)
- Kuriyama, C; Kamiyama, O; Ikeda, K; Sanae, F; Kato, A; Adachi, I; Imahori, T; Takahata, H; Okamoto, T; Asano, N Bioorg Med Chem 16: 7330-6 (2008)
- Hamaguchi, W; Kinoyama, I; Koganemaru, Y; Miyazaki, T; Kaneko, O; Sekioka, R; Washio, T US Patent US8962612 (2015)
- Honma, D; Kanno, O; Watanabe, J; Kinoshita, J; Hirasawa, M; Nosaka, E; Shiroishi, M; Takizawa, T; Yasumatsu, I; Horiuchi, T; Nakao, A; Suzuki, K; Yamasaki, T; Nakajima, K; Hayakawa, M; Yamazaki, T; Yadav, AS; Adachi, N Cancer Sci 108: 2069-2078
- Giordanetto, F; Barlaam, B; Berglund, S; Edman, K; Karlsson, O; Lindberg, J; Nylander, S; Inghardt, T Bioorg Med Chem Lett 24: 3936-43 (2014)
- Gazal, S; Gelerman, G; Ziv, O; Karpov, O; Litman, P; Bracha, M; Afargan, M; Gilon, C J Med Chem 45: 1665-71 (2002)
- Miyamoto, Y; Banno, Y; Yamashita, T; Fujimoto, T; Oi, S; Moritoh, Y; Asakawa, T; Kataoka, O; Yashiro, H; Takeuchi, K; Suzuki, N; Ikedo, K; Kosaka, T; Tsubotani, S; Tani, A; Sasaki, M; Funami, M; Amano, M; Yamamoto, Y; Aertgeerts, K; Yano, J; Maezaki, H J Med Chem 54: 831-50 (2012)
- De Pascale, M; Bissegger, L; Tarantelli, C; Beaufils, F; Prescimone, A; Mohamed Seid Hedad, H; Kayali, O; Orbegozo, C; Raguž, L; Schaefer, T; Hebeisen, P; Bertoni, F; Wymann, MP; Borsari, C Eur J Med Chem 248: (2023)
- Mesiti, F; Gaspar, A; Chavarria, D; Maruca, A; Rocca, R; Gil Martins, E; Barreiro, S; Silva, R; Fernandes, C; Gul, S; Keminer, O; Alcaro, S; Borges, F J Med Chem 64: 11169-11182 (2021)
- Lerchen, H; Cancho Grande, Y; Stelte-Ludwig, B; Sommer, A; Mahlert, C; Rebstock, A; Greven, S; Griebenow, N; Tebbe, J; Kensch, O US Patent US11806404 (2023)
- Huet, T; Kerbarh, O; Schols, D; Clayette, P; Gauchet, C; Dubreucq, G; Vincent, L; Bompais, H; Mazinghien, R; Querolle, O; Salvador, A; Lemoine, J; Lucidi, B; Balzarini, J; Petitou, M Antimicrob Agents Chemother 54: 134-42 (2009)
- Andrews, DM; Cartic, S; Cosulich, S; Divecha, N; Faulder, P; Flemington, V; Kern, O; Kettle, JG; MacDonald, E; McKelvie, J; Pike, KG; Roberts, B; Rowlinson, R; Smith, JM; Stockley, M; Swarbrick, ME; Treinies, I; Waring, MJ Bioorg Med Chem 54: (2022)
- Krenitsky, VP; Delgado, M; Nadolny, L; Sahasrabudhe, K; Ayala, L; Clareen, SS; Hilgraf, R; Albers, R; Kois, A; Hughes, K; Wright, J; Nowakowski, J; Sudbeck, E; Ghosh, S; Bahmanyar, S; Chamberlain, P; Muir, J; Cathers, BE; Giegel, D; Xu, L; Celeridad, M; Moghaddam, M; Khatsenko, O; Omholt, P; Katz, J; Pai, S; Fan, R; Tang, Y; Shirley, MA; Benish, B; Blease, K; Raymon, H; Bhagwat, S; Henderson, I; Cole, AG; Bennett, B; Satoh, Y Bioorg Med Chem Lett 22: 1427-32 (2012)
- Hecht, S; Khdour, O; Lu, J; Arce, P US Patent US8952025 (2015)
- Stokmaier, D; Khorev, O; Cutting, B; Born, R; Ricklin, D; Ernst, TO; Böni, F; Schwingruber, K; Gentner, M; Wittwer, M; Spreafico, M; Vedani, A; Rabbani, S; Schwardt, O; Ernst, B Bioorg Med Chem 17: 7254-64 (2009)
- Walker, MA; Johnson, T; Ma, Z; Banville, J; Remillard, R; Kim, O; Zhang, Y; Staab, A; Wong, H; Torri, A; Samanta, H; Lin, Z; Deminie, C; Terry, B; Krystal, M; Meanwell, N Bioorg Med Chem Lett 16: 2920-4 (2006)
- Kinzel, O; Steeneck, C; Schlüter, T; Schulz, A; Gege, C; Hahn, U; Hambruch, E; Hornberger, M; Spalwisz, A; Frick, K; Perovic-Ottstadt, S; Deuschle, U; Burnet, M; Kremoser, C Bioorg Med Chem Lett 26: 3746-53 (2016)
- Sergeev, A; Vorobyov, A; Yakubovskaya, M; Kirsanova, O; Gromova, E Bioorg Med Chem Lett 30: (2020)
- Sato, H; Kitagawa, O; Aida, Y; Chikazawa, J; Kurimoto, T; Takei, M; Fukuta, Y; Yoshida, K Bioorg Med Chem Lett 9: 1553-8 (1999)
- Polishchuk, PG; Samoylenko, GV; Khristova, TM; Krysko, OL; Kabanova, TA; Kabanov, VM; Kornylov, AY; Klimchuk, O; Langer, T; Andronati, SA; Kuz'min, VE; Krysko, AA; Varnek, A J Med Chem 58: 7681-94 (2015)
- Nazaré, M; Matter, H; Klingler, O; Al-Obeidi, F; Schreuder, H; Zoller, G; Czech, J; Lorenz, M; Dudda, A; Peyman, A; Nestler, HP; Urmann, M; Bauer, A; Laux, V; Wehner, V; Will, DW Bioorg Med Chem Lett 14: 2801-5 (2004)
- Pokhodylo, N; Finiuk, N; Klyuchivska, O; Тupychak, MA; Matiychuk, V; Goreshnik, E; Stoika, R Eur J Med Chem 241: (2022)
- Patberg, M; Isaak, A; Füsser, F; Ortiz Zacarías, NV; Vinnenberg, L; Schulte, J; Michetti, L; Grey, L; van der Horst, C; Hundehege, P; Koch, O; Heitman, LH; Budde, T; Junker, A Eur J Med Chem 226: (2021)
- Chen, P; Cheng, PT; Alam, M; Beyer, BD; Bisacchi, GS; Dejneka, T; Evans, AJ; Greytok, JA; Hermsmeier, MA; Humphreys, WG; Jacobs, GA; Kocy, O; Lin, PF; Lis, KA; Marella, MA; Ryono, DE; Sheaffer, AK; Spergel, SH; Sun, CQ; Tino, JA; Vite, G; Colonno, RJ; Zahler, R; Barrish, JC J Med Chem 39: 1991-2007 (1996)
- Peifer, C; Krasowski, A; Hämmerle, N; Kohlbacher, O; Dannhardt, G; Totzke, F; Schächtele, C; Laufer, S J Med Chem 49: 7549-53 (2006)
- Asoh, K; Kohchi, M; Hyoudoh, I; Ohtsuka, T; Masubuchi, M; Kawasaki, K; Ebiike, H; Shiratori, Y; Fukami, TA; Kondoh, O; Tsukaguchi, T; Ishii, N; Aoki, Y; Shimma, N; Sakaitani, M Bioorg Med Chem Lett 19: 1753-7 (2009)
- Degterev, A; Hitomi, J; Germscheid, M; Ch'en, IL; Korkina, O; Teng, X; Abbott, D; Cuny, GD; Yuan, C; Wagner, G; Hedrick, SM; Gerber, SA; Lugovskoy, A; Yuan, J Nat Chem Biol 4: 313-21 (2008)
- Mimura, H; Ikemura, T; Kotera, O; Sawada, M; Tashiro, S; Fuse, E; Ueno, K; Manabe, H; Ohshima, E; Karasawa, A; Miyaji, H J Pharmacol Exp Ther 314: 244-51 (2005)
- Buta, A; Maximyuk, O; Kovalskyy, D; Sukach, V; Vovk, M; Ievglevskyi, O; Isaeva, E; Isaev, D; Savotchenko, A; Krishtal, O J Med Chem 58: 4449-61 (2015)
- Khirsariya, P; Pospíšil, P; Maier, L; Boudný, M; Babáš, M; Kroutil, O; Mráz, M; Vácha, R; Paruch, K J Med Chem 65: 5701-5723 (2022)
- Surmiak, E; Ząber, J; Plewka, J; Wojtanowicz, G; Kocik-Krol, J; Kruc, O; Muszak, D; Rodríguez, I; Musielak, B; Viviano, M; Castellano, S; Skalniak, L; Magiera-Mularz, K; Holak, TA; Kalinowska-Tłuścik, J ACS Med Chem Lett 15: 36-44 (2024)
- Provencher, BA; Eshleman, AJ; Johnson, RA; Shi, X; Kryatova, O; Nelson, J; Tian, J; Gonzalez, M; Meltzer, PC; Janowsky, A J Med Chem 61: 9121-9131 (2018)
- Bröker, J; Waterson, AG; Smethurst, C; Kessler, D; Böttcher, J; Mayer, M; Gmaschitz, G; Phan, J; Little, A; Abbott, JR; Sun, Q; Gmachl, M; Rudolph, D; Arnhof, H; Rumpel, K; Savarese, F; Gerstberger, T; Mischerikow, N; Treu, M; Herdeis, L; Wunberg, T; Gollner, A; Weinstabl, H; Mantoulidis, A; Krämer, O; McConnell, DB; W Fesik, S J Med Chem 65: 14614-14629 (2022)
- Sato, K; Takahagi, H; Kubo, O; Hidaka, K; Yoshikawa, T; Kamaura, M; Nakakariya, M; Amano, N; Adachi, R; Maki, T; Take, K; Takekawa, S; Kitazaki, T; Maekawa, T Bioorg Med Chem 23: 4544-4560
- Resetar, M; Liu, X; Herdlinger, S; Kunert, O; Pferschy-Wenzig, EM; Latkolik, S; Steinacher, T; Schuster, D; Bauer, R; Dirsch, VM J Nat Prod 83: 918-926 (2020)
- Kojima, T; Asano, Y; Kurasawa, O; Hirata, Y; Iwamura, N; Wong, TT; Saito, B; Tanaka, Y; Arai, R; Yonemori, K; Miyamoto, Y; Sagiya, Y; Yaguchi, M; Shibata, S; Mizutani, A; Sano, O; Adachi, R; Satomi, Y; Hirayama, M; Aoyama, K; Hiura, Y; Kiba, A; Kitamura, S; Imamura, S Bioorg Med Chem 26: 2452-2465 (2018)
- Labeeuw, O; Levoin, N; Poupardin-Olivier, O; Calmels, T; Ligneau, X; Berrebi-Bertrand, I; Robert, P; Lecomte, JM; Schwartz, JC; Capet, M Bioorg Med Chem Lett 23: 2548-54 (2013)
- Contour-Galcéra, MO; Lavergne, O; Brezak, MC; Ducommun, B; Prévost, G Bioorg Med Chem Lett 14: 5809-12 (2004)
- Kovaleva, K; Oleshko, O; Mamontova, E; Yarovaya, O; Zakharova, O; Zakharenko, A; Kononova, A; Dyrkheeva, N; Cheresiz, S; Pokrovsky, A; Lavrik, O; Salakhutdinov, N J Nat Prod 82: 2443-2450 (2019)
- Macabuag, N; Esmieu, W; Breccia, P; Jarvis, R; Blackaby, W; Lazari, O; Urbonas, L; Eznarriaga, M; Williams, R; Strijbosch, A; Van de Bospoort, R; Matthews, K; Clissold, C; Ladduwahetty, T; Vater, H; Heaphy, P; Stafford, DG; Wang, HJ; Mangette, JE; McAllister, G; Beaumont, V; Vogt, TF; Wilkinson, HA; Doherty, EM; Dominguez, C J Med Chem 65: 12445-12459 (2022)
- Chen, CH; Lee, O; Yao, CN; Chuang, MY; Chang, YL; Chang, MH; Wen, YF; Yang, WH; Ko, CH; Chou, NT; Lin, MW; Lai, CP; Sun, CY; Wang, LM; Chen, YC; Hseu, TH; Chang, CN; Hsu, HC; Lin, HC; Chang, YL; Shih, YC; Chou, SH; Hsu, YL; Tseng, HW; Liu, CP; Tu, CM; Hu, TL; Tsai, YJ; Chen, TS; Lin, CL; Chiou, SJ; Liu, CC; Hwang, CS Bioorg Med Chem Lett 20: 6129-32 (2010)
- Chaudhary, S; Pecic, S; Legendre, O; Navarro, HA; Harding, WW Bioorg Med Chem Lett 19: 2530-2 (2009)
- Certal, V; Carry, JC; Halley, F; Virone-Oddos, A; Thompson, F; Filoche-Rommé, B; El-Ahmad, Y; Karlsson, A; Charrier, V; Delorme, C; Rak, A; Abecassis, PY; Amara, C; Vincent, L; Bonnevaux, H; Nicolas, JP; Mathieu, M; Bertrand, T; Marquette, JP; Michot, N; Benard, T; Perrin, MA; Lemaitre, O; Guerif, S; Perron, S; Monget, S; Gruss-Leleu, F; Doerflinger, G; Guizani, H; Brollo, M; Delbarre, L; Bertin, L; Richepin, P; Loyau, V; Garcia-Echeverria, C; Lengauer, C; Schio, L J Med Chem 57: 903-20 (2014)
- Lin, TI; Lenz, O; Fanning, G; Verbinnen, T; Delouvroy, F; Scholliers, A; Vermeiren, K; Rosenquist, A; Edlund, M; Samuelsson, B; Vrang, L; de Kock, H; Wigerinck, P; Raboisson, P; Simmen, K Antimicrob Agents Chemother 53: 1377-85 (2009)
- Colotta, V; Lenzi, O; Catarzi, D; Varano, F; Filacchioni, G; Martini, C; Trincavelli, L; Ciampi, O; Pugliese, AM; Traini, C; Pedata, F; Morizzo, E; Moro, S J Med Chem 52: 2407-19 (2009)
- Denèfle, T; Pramil, E; Gómez-Morales, L; Levasseur, MD; Lardé, E; Newton, C; Herry, K; Herbi, L; Lamotte, Y; Odile, E; Ancellin, N; Grondin, P; Martinez-Torres, AC; Viviani, F; Merle-Beral, H; Lequin, O; Susin, SA; Karoyan, P J Med Chem 62: 7656-7668 (2019)
- Trân, K; Murza, A; Sainsily, X; Delile, E; Couvineau, P; Côté, J; Coquerel, D; Peloquin, M; Auger-Messier, M; Bouvier, M; Lesur, O; Sarret, P; Marsault, É J Med Chem 64: 602-615 (2021)
- Stasi, LP; Artusi, R; Bovino, C; Buzzi, B; Canciani, L; Caselli, G; Colace, F; Garofalo, P; Giambuzzi, S; Larger, P; Letari, O; Mandelli, S; Perugini, L; Pucci, S; Salvi, M; Toro, P Bioorg Med Chem Lett 23: 2653-8 (2013)
- Harrison, D; Boutard, N; Brzozka, K; Bugaj, M; Chmielewski, S; Cierpich, A; Doedens, JR; Fabritius, CRY; Gabel, CA; Galezowski, M; Kowalczyk, P; Levenets, O; Mroczkowska, M; Palica, K; Porter, RA; Schultz, D; Sowinska, M; Topolnicki, G; Urbanski, P; Woyciechowski, J; Watt, AP Bioorg Med Chem Lett 30: (2020)
- Arasappan, A; Njoroge, FG; Chan, TY; Bennett, F; Bogen, SL; Chen, K; Gu, H; Hong, L; Jao, E; Liu, YT; Lovey, RG; Parekh, T; Pike, RE; Pinto, P; Santhanam, B; Venkatraman, S; Vaccaro, H; Wang, H; Yang, X; Zhu, Z; Mckittrick, B; Saksena, AK; Girijavallabhan, V; Pichardo, J; Butkiewicz, N; Ingram, R; Malcolm, B; Prongay, A; Yao, N; Marten, B; Madison, V; Kemp, S; Levy, O; Lim-Wilby, M; Tamura, S; Ganguly, AK Bioorg Med Chem Lett 15: 4180-4 (2005)
- Jain, N; Allan, G; Linton, O; Tannenbaum, P; Chen, X; Xu, J; Zhu, P; Gunnet, J; Demarest, K; Lundeen, S; Murray, W; Sui, Z Bioorg Med Chem Lett 19: 3977-80 (2009)
- Biagi, G; Costantini, A; Costantino, L; Giorgi, I; Livi, O; Pecorari, P; Rinaldi, M; Scartoni, V J Med Chem 39: 2529-35 (1996)
- Palomer, A; Pérez, JJ; Navea, S; Llorens, O; Pascual, J; García, L; Mauleón, D J Med Chem 43: 2280-4 (2000)
- Hersperger, R; Buchheit, KH; Cammisuli, S; Enz, A; Lohse, O; Ponelle, M; Schuler, W; Schweitzer, A; Walker, C; Zehender, H; Zenke, G; Zimmerlin, AG; Zollinger, M; Mazzoni, L; Fozard, JR J Med Chem 47: 4950-7 (2004)
- McKeown, SC; Hall, A; Giblin, GM; Lorthioir, O; Blunt, R; Lewell, XQ; Wilson, RJ; Brown, SH; Chowdhury, A; Coleman, T; Watson, SP; Chessell, IP; Pipe, A; Clayton, N; Goldsmith, P Bioorg Med Chem Lett 16: 4767-71 (2006)
- Llona-Minguez, S; Höglund, A; Jacques, SA; Johansson, L; Calderón-Montaño, JM; Claesson, M; Loseva, O; Valerie, NC; Lundbäck, T; Piedrafita, J; Maga, G; Crespan, E; Meijer, L; Burgos Morón, E; Baranczewski, P; Hagbjörk, AL; Svensson, R; Wiita, E; Almlöf, I; Visnes, T; Jeppsson, F; Sigmundsson, K; Jensen, AJ; Artursson, P; Jemth, AS; Stenmark, P; Warpman Berglund, U; Scobie, M; Helleday, T J Med Chem 59: 1140-8 (2016)
- Chioua, M; Samadi, A; Soriano, E; Lozach, O; Meijer, L; Marco-Contelles, J Bioorg Med Chem Lett 19: 4566-9 (2009)
- Zakharova, O; Luzina, O; Zakharenko, A; Sokolov, D; Filimonov, A; Dyrkheeva, N; Chepanova, A; Ilina, E; Ilyina, A; Klabenkova, K; Chelobanov, B; Stetsenko, D; Zafar, A; Eurtivong, C; Reynisson, J; Volcho, K; Salakhutdinov, N; Lavrik, O Bioorg Med Chem 26: 4470-4480 (2018)
- Van der Plas, SE; Kelgtermans, H; Mammoliti, O; Menet, C; Tricarico, G; De Blieck, A; Joannesse, C; De Munck, T; Lambin, D; Cowart, M; Dropsit, S; Martina, SLX; Gees, M; Wesse, AS; Conrath, K; Andrews, M J Med Chem 64: 343-353 (2021)
- Scheiner, M; Dolles, D; Gunesch, S; Hoffmann, M; Nabissi, M; Marinelli, O; Naldi, M; Bartolini, M; Petralla, S; Poeta, E; Monti, B; Falkeis, C; Vieth, M; Hübner, H; Gmeiner, P; Maitra, R; Maurice, T; Decker, M J Med Chem 62: 9078-9102 (2019)
- Labaudinière, R; Dereu, N; Cavy, F; Guillet, MC; Marquis, O; Terlain, B J Med Chem 35: 4315-24 (1992)
- Yu, L; Ikeda, K; Kato, A; Adachi, I; Godin, G; Compain, P; Martin, O; Asano, N Bioorg Med Chem 14: 7736-44 (2006)
- Diurno, MV; Mazzoni, O; Piscopo, E; Calignano, A; Giordano, F; Bolognese, A J Med Chem 35: 2910-2 (1992)
- Hajirahimkhan, A; Mbachu, O; Simmler, C; Ellis, SG; Dong, H; Nikolic, D; Lankin, DC; van Breemen, RB; Chen, SN; Pauli, GF; Dietz, BM; Bolton, JL J Nat Prod 81: 966-975 (2018)
- McCarthy, O; Musso-Buendia, A; Kaiser, M; Brun, R; Ruiz-Perez, LM; Johansson, NG; Pacanowska, DG; Gilbert, IH Eur J Med Chem 44: 678-88 (2009)
- Bumpers, QA; Pipal, RW; Benz-Weeden, AM; Brewster, JT; Cook, A; Crooks, AL; Cruz, C; Dwulet, NC; Gaudino, JJ; Golec, D; Harrison, JA; Hartley, DP; Hassanien, SH; Hicken, EJ; Kahn, D; Laird, ER; Lemieux, C; Lewandowski, N; McCown, J; McDonald, MG; McNulty, O; Mou, TC; Nguyen, P; Oko, L; Opie, LP; Otten, J; Peck, SC; Polites, VC; Randall, SD; Rosen, RZ; Savechenkov, P; Simpson, H; Singh, A; Sparks, D; Wickersham, K; Wollenberg, L; Wong, CE; Wong, J; Wu, WI; Elsayed, MSA; Hinklin, RJ; Tang, TP J Med Chem 67: 14466-14477
- Guibbal, F; Bénard, S; Patché, J; Meneyrol, V; Couprie, J; Yong-Sang, J; Meilhac, O; Jestin, E Bioorg Med Chem Lett 28: 787-792 (2018)
- Monaco, A; Zoete, V; Alghisi, GC; Rüegg, C; Michelin, O; Prior, J; Scapozza, L; Seimbille, Y Bioorg Med Chem Lett 23: 6068-72 (2013)
- Röhrig, UF; Majjigapu, SR; Caldelari, D; Dilek, N; Reichenbach, P; Ascencao, K; Irving, M; Coukos, G; Vogel, P; Zoete, V; Michielin, O Bioorg Med Chem Lett 26: 4330-3 (2016)
- Kiyeleko, S; Hocine, S; Mautino, G; Kuenemann, M; Nawrotek, A; Miallau, L; Vuillard, LM; Mirguet, O; Kotschy, A; Hanessian, S Bioorg Med Chem Lett 75: (2022)
- Ivachtchenko, A; Golovina, E; Kadieva, M; Mitkin, O; Tkachenko, S; Okun, I Bioorg Med Chem 21: 4614-27 (2013)
- Kettle, JG; Anjum, R; Barry, E; Bhavsar, D; Brown, C; Boyd, S; Campbell, A; Goldberg, K; Grondine, M; Guichard, S; Hardy, CJ; Hunt, T; Jones, RDO; Li, X; Moleva, O; Ogg, D; Overman, RC; Packer, MJ; Pearson, S; Schimpl, M; Shao, W; Smith, A; Smith, JM; Stead, D; Stokes, S; Tucker, M; Ye, Y J Med Chem 61: 8797-8810 (2018)
- Di Sarno, V; Lauro, G; Musella, S; Ciaglia, T; Vestuto, V; Sala, M; Scala, MC; Smaldone, G; Di Matteo, F; Novi, S; Tecce, MF; Moltedo, O; Bifulco, G; Campiglia, P; Gomez-Monterrey, IM; Snoeck, R; Andrei, G; Ostacolo, C; Bertamino, A Eur J Med Chem 226: (2021)
- Mravljak, J; Monasson, O; Al-Dabbagh, B; Crouvoisier, M; Bouhss, A; Gravier-Pelletier, C; Le Merrer, Y Eur J Med Chem 46: 1582-92 (2011)
- Erichsen, MN; Huynh, TH; Abrahamsen, B; Bastlund, JF; Bundgaard, C; Monrad, O; Bekker-Jensen, A; Nielsen, CW; Frydenvang, K; Jensen, AA; Bunch, L J Med Chem 53: 7180-91 (2010)
- Bennett, J; Fedorov, O; Tallant, C; Monteiro, O; Meier, J; Gamble, V; Savitsky, P; Nunez-Alonso, GA; Haendler, B; Rogers, C; Brennan, PE; Müller, S; Knapp, S J Med Chem 59: 1642-7 (2016)
- Ishiuchi, K; Hirose, D; Suzuki, T; Nakayama, W; Jiang, WP; Monthakantirat, O; Wu, JB; Kitanaka, S; Makino, T J Nat Prod 81: 1143-1147 (2018)
- Vaisburg, A; Paquin, I; Bernstein, N; Frechette, S; Gaudette, F; Leit, S; Moradei, O; Raeppel, S; Zhou, N; Bouchain, G; Woo, SH; Jin, Z; Gillespie, J; Wang, J; Fournel, M; Yan, PT; Trachy-Bourget, MC; Robert, MF; Lu, A; Yuk, J; Rahil, J; Macleod, AR; Besterman, JM; Li, Z; Delorme, D Bioorg Med Chem Lett 17: 6729-33 (2007)
- McDermott, LA; Higgins, B; Simcox, M; Luk, KC; Nevins, T; Kolinsky, K; Smith, M; Yang, H; Li, JK; Chen, Y; Ke, J; Mallalieu, N; Egan, T; Kolis, S; Railkar, A; Gerber, L; Liu, JJ; Konzelmann, F; Zhang, Z; Flynn, T; Morales, O; Chen, Y Bioorg Med Chem Lett 16: 1950-3 (2006)
- Selvakumar, K; Paidi, VR; Thangathirupathy, S; Kumar Cm, V; Alajangi, TR; Sura, MR; Mahadevu, K; Sistla, RK; Agarwal, P; Subbiah Karuppiah, AM; Nair, JS; Morampudi, O; Panda, M; Tino, JA; Cherney, RJ; Duncia, JV; Gardner, DS; Dhar, TG; Ross, AG; Gormisky, PE; Zhu, X; Seletsky, BM; Antropow, AH; Niu, D; Zhu, Z; Miao, G; Cuervo, JH US Patent US12473304 (2025)
- Filippakopoulos, P; Picaud, S; Fedorov, O; Keller, M; Wrobel, M; Morgenstern, O; Bracher, F; Knapp, S Bioorg Med Chem 20: 1878-86 (2012)
- Marugan, JJ; Huang, W; Motabar, O; Zheng, W; Xiao, J; Patnaik, S; Southall, N; Westbroek, W; Lea, WA; Simeonov, A; Goldin, E; Debernardi, MA; Sidransky, E Medchemcomm 3: 56-60 (2012)
- Nishi, T; Fukazawa, T; Ishibashi, K; Nakajima, K; Sugioka, Y; Iio, Y; Kurata, H; Itoh, K; Mukaiyama, O; Satoh, Y; Yamaguchi, T Bioorg Med Chem Lett 9: 875-80 (1999)
- Morikawa, T; Hachiman, I; Matsuo, K; Nishida, E; Ninomiya, K; Hayakawa, T; Yoshie, O; Muraoka, O; Nakayama, T J Nat Prod 79: 2005-13 (2016)
- Van Quaquebeke, E; Simon, G; André, A; Dewelle, J; El Yazidi, M; Bruyneel, F; Tuti, J; Nacoulma, O; Guissou, P; Decaestecker, C; Braekman, JC; Kiss, R; Darro, F J Med Chem 48: 849-56 (2005)
- Sato, T; Ashizawa, N; Iwanaga, T; Nakamura, H; Matsumoto, K; Inoue, T; Nagata, O Bioorg Med Chem Lett 19: 184-7 (2008)
- Kobayashi, JI; Hirasawa, H; Ozawa, T; Ozawa, T; Takeda, H; Fujimori, Y; Nakanishi, O; Kamada, N; Ikeda, T Bioorg Med Chem 25: 727-742 (2017)
- Bolli, MH; Abele, S; Birker, M; Bravo, R; Bur, D; de Kanter, R; Kohl, C; Grimont, J; Hess, P; Lescop, C; Mathys, B; Müller, C; Nayler, O; Rey, M; Scherz, M; Schmidt, G; Seifert, J; Steiner, B; Velker, J; Weller, T J Med Chem 57: 110-30 (2014)
- Schnute, ME; O'Brien, PM; Nahra, J; Morris, M; Howard Roark, W; Hanau, CE; Ruminski, PG; Scholten, JA; Fletcher, TR; Hamper, BC; Carroll, JN; Patt, WC; Shieh, HS; Collins, B; Pavlovsky, AG; Palmquist, KE; Aston, KW; Hitchcock, J; Rogers, MD; McDonald, J; Johnson, AR; Munie, GE; Wittwer, AJ; Man, CF; Settle, SL; Nemirovskiy, O; Vickery, LE; Agawal, A; Dyer, RD; Sunyer, T Bioorg Med Chem Lett 20: 576-80 (2010)
- Khatib, S; Nerya, O; Musa, R; Tamir, S; Peter, T; Vaya, J J Med Chem 50: 2676-81 (2007)
- Chesworth, R; Wessel, MD; Heyden, L; Mangano, FM; Zawistoski, M; Gegnas, L; Galluzzo, D; Lefker, B; Cameron, KO; Tickner, J; Lu, B; Castleberry, TA; Petersen, DN; Brault, A; Perry, P; Ng, O; Owen, TA; Pan, L; Ke, HZ; Brown, TA; Thompson, DD; DaSilva-Jardine, P Bioorg Med Chem Lett 15: 5562-6 (2005)
- Henderson, JA; Bilimoria, D; Bubenik, M; Cadilhac, C; Cottrell, KM; Dietrich, E; Denis, F; Ewing, N; Falardeau, G; Giroux, S; Grey, R; L'Heureux, L; Liu, B; Mani, N; Morris, M; Nicolas, O; Pereira, OZ; Poisson, C; Govinda Rao, B; Reddy, TJ; Selliah, S; Shawgo, RS; Vaillancourt, L; Wang, J; Yannopoulos, CG; Chauret, N; Berlioz-Seux, F; Chan, LC; Das, SK; Grillot, AL; Bennani, YL; Maxwell, JP Bioorg Med Chem Lett 25: 944-7 (2015)
- Labas, R; Gilbert, G; Nicole, O; Dhilly, M; Abbas, A; Tirel, O; Buisson, A; Henry, J; Barré, L; Debruyne, D; Sobrio, F Eur J Med Chem 46: 2295-309 (2011)
- Tardia, P; Stefanachi, A; Niso, M; Stolfa, DA; Mangiatordi, GF; Alberga, D; Nicolotti, O; Lattanzi, G; Carotti, A; Leonetti, F; Perrone, R; Berardi, F; Azzariti, A; Colabufo, NA; Cellamare, S J Med Chem 57: 6403-18 (2014)
- Bootorabi, F; Jänis, J; Hytönen, VP; Valjakka, J; Kuuslahti, M; Vullo, D; Niemelä, O; Supuran, CT; Parkkila, S J Enzyme Inhib Med Chem 26: 862-70 (2011)
- Pérez, RA; Fernández-Alvarez, E; Nieto, O; Piedrafita, FJ J Med Chem 35: 4584-8 (1993)
- Nain-Perez, A; Nilsson, O; Lulla, A; Håversen, L; Brear, P; Liljenberg, S; Hyvönen, M; Borén, J; Grøtli, M Eur J Med Chem 250: (2023)
- Ratcliffe, P; Abernethy, L; Ansari, N; Cameron, K; Clarkson, T; Dempster, M; Dunn, D; Easson, AM; Edwards, D; Everett, K; Feilden, H; Ho, KK; Kultgen, S; Littlewood, P; Maclean, J; McArthur, D; McGregor, D; McLuskey, H; Neagu, I; Nimz, O; Nisbet, LA; Ohlmeyer, M; Palin, R; Pham, Q; Rong, Y; Roughton, A; Sammons, M; Swanson, R; Tracey, H; Walker, G Bioorg Med Chem Lett 21: 4652-7 (2011)
- Shiraishi, M; Aramaki, Y; Seto, M; Imoto, H; Nishikawa, Y; Kanzaki, N; Okamoto, M; Sawada, H; Nishimura, O; Baba, M; Fujino, M J Med Chem 43: 2049-63 (2000)
- Murakami, T; Yoshioka, K; Sato, Y; Tanaka, M; Niwa, O; Yabuki, S Bioorg Med Chem Lett 21: 1265-9 (2011)
- Jeanty, M; Suzenet, F; Delagrange, P; Nosjean, O; Boutin, JA; Caignard, DH; Guillaumet, G Bioorg Med Chem Lett 21: 2316-9 (2011)
- Kawaguchi, M; Okabe, T; Okudaira, S; Nishimasu, H; Ishitani, R; Kojima, H; Nureki, O; Aoki, J; Nagano, T ACS Chem Biol 8: 1713-21 (2013)
- Raboisson, PJ; Hu, L; Vendeville, SM; Nyanguile, O; Tahri, A US Patent US8524716 (2013)
- Rejman, D; Rabatinová, A; Pombinho, AR; Kovačková, S; Pohl, R; Zborníková, E; Kolář, M; Bogdanová, K; Nyč, O; Sanderová, H; Látal, T; Bartůněk, P; Krásný, L J Med Chem 54: 7884-98 (2011)
- Qi, Q; Obianyo, O; Du, Y; Fu, H; Li, S; Ye, K J Med Chem 60: 7244-7255 (2017)
- Teno, N; Miyake, T; Ehara, T; Irie, O; Sakaki, J; Ohmori, O; Gunji, H; Matsuura, N; Masuya, K; Hitomi, Y; Nonomura, K; Horiuchi, M; Gohda, K; Iwasaki, A; Umemura, I; Tada, S; Kometani, M; Iwasaki, G; Cowan-Jacob, SW; Missbach, M; Lattmann, R; Betschart, C Bioorg Med Chem Lett 17: 6096-100 (2007)
- Fukuda, M; Sasaki, T; Hashimoto, T; Miyachi, H; Waki, M; Asai, A; Takikawa, O; Ohno, O; Matsuno, K Bioorg Med Chem Lett 28: 2846-2849 (2018)
- Hagihara, S; Ishizawa, K; Soga, K; Honjo, T; Takai, S; Kawano, Y; Kikuchi, M; Nishidate, A; Matsumoto, F; Murase, M; Hashimoto, N; Sasaki, C; Miyaguchi, I; Okada, O; Akashi, T; Nakayama, S; Ogasawara, Y; Endo, J Bioorg Med Chem Lett 109:
- Satoh, A; Sagara, T; Sakoh, H; Hashimoto, M; Nakashima, H; Kato, T; Goto, Y; Mizutani, S; Azuma-Kanoh, T; Tani, T; Okuda, S; Okamoto, O; Ozaki, S; Iwasawa, Y; Ohta, H; Kawamoto, H J Med Chem 52: 4091-4 (2009)
- Tanaka, A; Hattori, K; Taniguchi, K; Okitsu, O; Tabuchi, S; Nishio, M; Nagakura, Y; Maeda, N; Murai, H; Seki, J Bioorg Med Chem Lett 16: 4861-4 (2006)
- Kovaleva, K; Oleshko, O; Mamontova, E; Yarovaya, O; Zakharova, O; Zakharenko, A; Kononova, A; Dyrkheeva, N; Cheresiz, S; Pokrovsky, A; Lavrik, O; Salakhutdinov, N J Nat Prod 82: 2443-2450 (2019)
- Marriott, KS; Morrison, AZ; Moore, M; Olubajo, O; Stewart, LE Bioorg Med Chem 20: 6856-61 (2012)
- Ommi, O; Naiyaz Ahmad, M; Gajula, SNR; Wanjari, P; Sau, S; Agnivesh, PK; Sahoo, SK; Kalia, NP; Sonti, R; Nanduri, S; Dasgupta, A; Chopra, S; Yaddanapudi, VM RSC Med Chem 14: 1296-1308 (2023)
- Kempson, J; Pitts, WJ; Barbosa, J; Guo, J; Omotoso, O; Watson, A; Stebbins, K; Starling, GC; Dodd, JH; Barrish, JC; Felix, R; Fischer, K Bioorg Med Chem Lett 15: 1829-33 (2005)
- Kato, A; Okaki, T; Ifuku, S; Sato, K; Hirokami, Y; Iwaki, R; Kamori, A; Nakagawa, S; Adachi, I; Kiria, PG; Onomura, O; Minato, D; Sugimoto, K; Matsuya, Y; Toyooka, N Bioorg Med Chem 21: 6565-73 (2013)
- Whitehead, A; Ornoski, O; Raghavan, S; Berger, R; Garfunkle, J; Yang, Z; Ji, G; Jiang, F; Fu, J US Patent US10780092 (2020)
- Taylor, AM; Williams, BR; Giordanetto, F; Kelley, EH; Lescarbeau, A; Shortsleeves, K; Tang, Y; Walters, WP; Arrazate, A; Bowman, C; Brophy, E; Chan, EW; Deshmukh, G; Greisman, JB; Hunsaker, TL; Kipp, DR; Saenz Lopez-Larrocha, P; Maddalo, D; Martin, IJ; Maragakis, P; Merchant, M; Murcko, M; Nisonoff, H; Nguyen, V; Nguyen, V; Orozco, O; Owen, C; Pierce, L; Schmidt, M; Shaw, DE; Smith, S; Therrien, E; Tran, JC; Watters, J; Waters, NJ; Wilbur, J; Willmore, L J Med Chem 66: 13384-13399 (2023)
- Esteves, MA; Ortet, O; Capelo, A; Supuran, CT; Marques, SM; Santos, MA Bioorg Med Chem Lett 20: 3623-7 (2010)
- Lu, SF; Herbert, B; Haufe, G; Laue, KW; Padgett, WL; Oshunleti, O; Daly, JW; Kirk, KL J Med Chem 43: 1611-9 (2000)
- Chatterjee, J; Ovadia, O; Zahn, G; Marinelli, L; Hoffman, A; Gilon, C; Kessler, H J Med Chem 50: 5878-81 (2007)
- Turkoglu, S; Maresca, A; Alper, M; Kockar, F; Isik, S; Sinan, S; Ozensoy, O; Arslan, O; Supuran, CT Bioorg Med Chem 20: 2208-13 (2012)
- Gökhan-Kelekçi, N; Koyunoqlu, S; Yabanoqlu, S; Yesilada, K; Ozgen, O; Uçar, G; Erol, K; Kendi, E; Yesilada, A Bioorg Med Chem 17: 675-89 (2009)
- Sebhat, IK; Franklin, C; Lo, MM; Chen, D; Jewell, JP; Miller, R; Pang, J; Palyha, O; Kan, Y; Kelly, TM; Guan, XM; Marsh, DJ; Kosinski, JA; Metzger, JM; Lyons, K; Dragovic, J; Guzzo, PR; Henderson, AJ; Reitman, ML; Nargund, RP; Wyvratt, MJ ACS Med Chem Lett 2: 43-47 (2011)
- Lamaa, D; Lin, HP; Zig, L; Bauvais, C; Bollot, G; Bignon, J; Levaique, H; Pamlard, O; Dubois, J; Ouaissi, M; Souce, M; Kasselouri, A; Saller, F; Borgel, D; Jayat-Vignoles, C; Al-Mouhammad, H; Feuillard, J; Benihoud, K; Alami, M; Hamze, A J Med Chem 61: 6574-6591 (2018)
- Mowat, JS; Buchmann, B; Aiguabella Font, N; Leder, G; Carretero, R; Panknin, O; Neuhaus, R; Meier, RM; Berndt, S; Petersen, K; Offringa, R US Patent US11427578 (2022)
- Kyriakis, E; Karra, AG; Papaioannou, O; Solovou, T; Skamnaki, VT; Liggri, PGV; Zographos, SE; Szennyes, E; Bokor, É; Kun, S; Psarra, AG; Somsák, L; Leonidas, DD Bioorg Med Chem 28: (2020)
- Rojas, S; Parravicini, O; Vettorazzi, M; Tosso, R; Garro, A; Gutiérrez, L; Andújar, S; Enriz, R Eur J Med Chem 208: (2020)
- Mallart, S; Ingenito, R; Bianchi, E; Bresciani, A; Esposito, S; Gallo, M; Magotti, P; Monteagudo, E; Orsatti, L; Roversi, D; Santoprete, A; Tucci, F; Veneziano, M; Bartsch, R; Boehm, C; Brasseur, D; Bruneau, P; Corbier, A; Froissant, J; Gauzy-Lazo, L; Gervat, V; Marguet, F; Menguy, I; Minoletti, C; Nicolas, MF; Pasquier, O; Poirier, B; Raux, A; Riva, L; Janiak, P; Strobel, H; Duclos, O; Illiano, S J Med Chem 64: 2139-2150 (2021)
- Pav, O; Protivinska, E; Pressova, M; Collinsova, M; Jiracek, J; Snasel, J; Masojidkova, M; Budesinsky, M; Rosenberg, I J Med Chem 49: 3955-62 (2006)
- Lin, Z; Antemano, RR; Hughen, RW; Tianero, MD; Peraud, O; Haygood, MG; Concepcion, GP; Olivera, BM; Light, A; Schmidt, EW J Nat Prod 73: 1922-6 (2010)
- Micheli, F; Bonanomi, G; Blaney, FE; Braggio, S; Capelli, AM; Checchia, A; Curcuruto, O; Damiani, F; Fabio, RD; Donati, D; Gentile, G; Gribble, A; Hamprecht, D; Tedesco, G; Terreni, S; Tarsi, L; Lightfoot, A; Stemp, G; Macdonald, G; Smith, A; Pecoraro, M; Petrone, M; Perini, O; Piner, J; Rossi, T; Worby, A; Pilla, M; Valerio, E; Griffante, C; Mugnaini, M; Wood, M; Scott, C; Andreoli, M; Lacroix, L; Schwarz, A; Gozzi, A; Bifone, A; Ashby, CR; Hagan, JJ; Heidbreder, C J Med Chem 50: 5076-89 (2007)
- Walker, EH; Pacold, ME; Perisic, O; Stephens, L; Hawkins, PT; Wymann, MP; Williams, RL Mol Cell 6: 909-19 (2000)
- Ganellin, CR; Bishop, PB; Bambal, RB; Chan, SM; Law, JK; Marabout, B; Luthra, PM; Moore, AN; Peschard, O; Bourgeat, P; Rose, C; Vargas, F; Schwartz, JC J Med Chem 43: 664-74 (2000)
- Pothier, J; Riederer, MA; Peter, O; Leroy, X; Valdenaire, A; Gnerre, C; Fretz, H Bioorg Med Chem Lett 22: 4660-4 (2012)
- Wasilewicz, A; Kirchweger, B; Bojkova, D; Abi Saad, MJ; Langeder, J; Bütikofer, M; Adelsberger, S; Grienke, U; Cinatl, J; Petermann, O; Scapozza, L; Orts, J; Kirchmair, J; Rabenau, HF; Rollinger, JM J Nat Prod 86: 264-275 (2023)
- Reigada, C; Phanstiel, O; Miranda, MR; Pereira, CA Eur J Med Chem 147: 1-6 (2018)
- Phuangsawai, O; Beswick, P; Ratanabunyong, S; Tabtimmai, L; Suphakun, P; Obounchoey, P; Srisook, P; Horata, N; Chuckowree, I; Hannongbua, S; Ward, SE; Choowongkomon, K; Gleeson, MP Eur J Med Chem 124: 896-905 (2016)
- Desroy, N; Housseman, C; Bock, X; Joncour, A; Bienvenu, N; Cherel, L; Labeguere, V; Rondet, E; Peixoto, C; Grassot, JM; Picolet, O; Annoot, D; Triballeau, N; Monjardet, A; Wakselman, E; Roncoroni, V; Le Tallec, S; Blanque, R; Cottereaux, C; Vandervoort, N; Christophe, T; Mollat, P; Lamers, M; Auberval, M; Hrvacic, B; Ralic, J; Oste, L; van der Aar, E; Brys, R; Heckmann, B J Med Chem 60: 3580-3590 (2017)
- Steinmetzer, T; Pilgram, O; Wenzel, BM; Wiedemeyer, SJA J Med Chem 63: 1445-1472 (2020)
- Parrino, B; Carbone, A; Ciancimino, C; Spanò, V; Montalbano, A; Barraja, P; Cirrincione, G; Diana, P; Sissi, C; Palumbo, M; Pinato, O; Pennati, M; Beretta, G; Folini, M; Matyus, P; Balogh, B; Zaffaroni, N Eur J Med Chem 94: 149-62 (2015)
- Lamotte, Y; Faucher, N; Sançon, J; Pineau, O; Sautet, S; Fouchet, MH; Beneton, V; Tousaint, JJ; Saintillan, Y; Ancellin, N; Nicodeme, E; Grillot, D; Martres, P Bioorg Med Chem Lett 24: 1098-103 (2014)
- Malleron, JL; Comte, MT; Gueremy, C; Peyronel, JF; Truchon, A; Blanchard, JC; Doble, A; Piot, O; Zundel, JL; Huon, C J Med Chem 34: 2477-83 (1991)
- Adelt, S; Plettenburg, O; Stricker, R; Reiser, G; Altenbach, HJ; Vogel, G J Med Chem 42: 1262-73 (1999)
- Hall, J; Brault, A; Vincent, F; Weng, S; Wang, H; Dumlao, D; Aulabaugh, A; Aivazian, D; Castro, D; Chen, M; Culp, J; Dower, K; Gardner, J; Hawrylik, S; Golenbock, D; Hepworth, D; Horn, M; Jones, L; Jones, P; Latz, E; Li, J; Lin, LL; Lin, W; Lin, D; Lovering, F; Niljanskul, N; Nistler, R; Pierce, B; Plotnikova, O; Schmitt, D; Shanker, S; Smith, J; Snyder, W; Subashi, T; Trujillo, J; Tyminski, E; Wang, G; Wong, J; Lefker, B; Dakin, L; Leach, K PLoS ONE 12: 1-16 (2017)
- Mallinger, A; Crumpler, S; Pichowicz, M; Waalboer, D; Stubbs, M; Adeniji-Popoola, O; Wood, B; Smith, E; Thai, C; Henley, AT; Georgi, K; Court, W; Hobbs, S; Box, G; Ortiz-Ruiz, MJ; Valenti, M; De Haven Brandon, A; TePoele, R; Leuthner, B; Workman, P; Aherne, W; Poeschke, O; Dale, T; Wienke, D; Esdar, C; Rohdich, F; Raynaud, F; Clarke, PA; Eccles, SA; Stieber, F; Schiemann, K; Blagg, J J Med Chem 58: 1717-35 (2015)
- Rehwinkel, H; Hägebarth, A; Politz, O; Neuhaus, R; Bömer, U US Patent US8987286 (2015)
- White, GV; Edgar, EV; Holmes, DS; Lewell, XQ; Liddle, J; Polyakova, O; Smith, KJ; Thorpe, JH; Walker, AL; Wang, Y; Young, RJ; Hovnanian, A Bioorg Med Chem Lett 29: 821-825 (2019)
- Van Zandt, MC; Jagdmann, GE; Whitehouse, DL; Ji, M; Savoy, J; Potapova, O; Cousido-Siah, A; Mitschler, A; Howard, EI; Pyle, AM; Podjarny, AD J Med Chem 62: 8164-8177 (2019)
- Amaudrut, J; Argiriadi, MA; Barth, M; Breinlinger, EC; Bressac, D; Broqua, P; Calderwood, DJ; Chatar, M; Cusack, KP; Gauld, SB; Jacquet, S; Kamath, RV; Kort, ME; Lepais, V; Luccarini, JM; Masson, P; Montalbetti, C; Mounier, L; Potin, D; Poupardin, O; Rouaud, S; Spitzer, L; Wallace, CD Bioorg Med Chem Lett 29: 1799-1806 (2019)
- Poyraz, O; Jeankumar, VU; Saxena, S; Schnell, R; Haraldsson, M; Yogeeswari, P; Sriram, D; Schneider, G J Med Chem 56: 6457-66 (2013)
- Lang, C; Maschauer, S; Hübner, H; Gmeiner, P; Prante, O J Med Chem 56: 9361-5 (2013)
- Collina, S; Loddo, G; Urbano, M; Linati, L; Callegari, A; Ortuso, F; Alcaro, S; Laggner, C; Langer, T; Prezzavento, O; Ronsisvalle, G; Azzolina, O Bioorg Med Chem 15: 771-83 (2006)
- Panknin, O; Wagenfeld, A; Bone, W; Bender, E; Nowak-Reppel, K; Fernández-Montalván, AE; Nubbemeyer, R; Bäurle, S; Ring, S; Schmees, N; Prien, O; Schäfer, M; Friedrich, C; Zollner, TM; Steinmeyer, A; Mueller, T; Langer, G J Med Chem 63: 11854-11881 (2020)
- Tars, K; Leitans, J; Kazaks, A; Zelencova, D; Liepinsh, E; Kuka, J; Makrecka, M; Lola, D; Andrianovs, V; Gustina, D; Grinberga, S; Liepinsh, E; Kalvinsh, I; Dambrova, M; Loza, E; Pugovics, O J Med Chem 57: 2213-36 (2014)
- Pimková Polidarová, M; Břehová, P; Kaiser, MM; Smola, M; Dračínský, M; Smith, J; Marek, A; Dejmek, M; Šála, M; Gutten, O; Rulíšek, L; Novotná, B; Brázdová, A; Janeba, Z; Nencka, R; Boura, E; Páv, O; Birkuš, G J Med Chem 64: 7596-7616 (2021)
- Czodrowski, P; Mallinger, A; Wienke, D; Esdar, C; Pöschke, O; Busch, M; Rohdich, F; Eccles, SA; Ortiz-Ruiz, MJ; Schneider, R; Raynaud, FI; Clarke, PA; Musil, D; Schwarz, D; Dale, T; Urbahns, K; Blagg, J; Schiemann, K J Med Chem 59: 9337-9349 (2016)
- Léger, R; Thibaudeau, K; Robitaille, M; Quraishi, O; van Wyk, P; Bousquet-Gagnon, N; Carette, J; Castaigne, JP; Bridon, DP Bioorg Med Chem Lett 14: 4395-8 (2004)
- Martínez González, S; Hernández, AI; Varela, C; Rodríguez-Arístegui, S; Lorenzo, M; Rodríguez, A; Rivero, V; Martín, JI; Saluste, CG; Ramos-Lima, F; Cendón, E; Cebrián, D; Aguirre, E; Gomez-Casero, E; Albarrán, M; Alfonso, P; García-Serelde, B; Oyarzabal, J; Rabal, O; Mulero, F; Gonzalez-Granda, T; Link, W; Fominaya, J; Barbacid, M; Bischoff, JR; Pizcueta, P; Pastor, J Bioorg Med Chem Lett 22: 3460-6 (2012)
- Leahy, JW; Buhr, CA; Johnson, HW; Kim, BG; Baik, T; Cannoy, J; Forsyth, TP; Jeong, JW; Lee, MS; Ma, S; Noson, K; Wang, L; Williams, M; Nuss, JM; Brooks, E; Foster, P; Goon, L; Heald, N; Holst, C; Jaeger, C; Lam, S; Lougheed, J; Nguyen, L; Plonowski, A; Song, J; Stout, T; Wu, X; Yakes, MF; Yu, P; Zhang, W; Lamb, P; Raeber, O J Med Chem 55: 5467-82 (2012)
- Das, N; Bandopadhyay, P; Roy, S; Sinha, BP; Dastidar, UG; Rahaman, O; Pal, S; Ganguly, D; Talukdar, A J Med Chem 65: 11607-11632 (2022)
- Talapatra, SK; Rath, O; Clayton, E; Tomasi, S; Kozielski, F J Nat Prod 79: 1576-85 (2016)
- Sander, K; von Coburg, Y; Camelin, JC; Ligneau, X; Rau, O; Schubert-Zsilavecz, M; Schwartz, JC; Stark, H Bioorg Med Chem Lett 20: 1581-4 (2010)
- Cansfield, AD; Ladduwahetty, T; Sunose, M; Ellard, K; Lynch, R; Newton, AL; Lewis, A; Bennett, G; Zinn, N; Thomson, DW; Rüger, AJ; Feutrill, JT; Rausch, O; Watt, AP; Bergamini, G ACS Med Chem Lett 7: 768-73 (2016)
- Plut, E; Calderón, JC; Stanojlović, V; Gattor, AO; Höring, C; Humphrys, LJ; Konieczny, A; Kerres, S; Schubert, M; Keller, M; Cabrele, C; Clark, T; Reiser, O J Med Chem 66: 9642-9657 (2023)
- Meyers, KM; Kim, N; Méndez-Andino, JL; Hu, XE; Mumin, RN; Klopfenstein, SR; Wos, JA; Mitchell, MC; Paris, JL; Ackley, DC; Holbert, JK; Mittelstadt, SW; Reizes, O Bioorg Med Chem Lett 17: 814-8 (2007)
- Roussel, E; Moréno, A; Altounian, N; Philouze, C; Pérès, B; Thomas, A; Renaudet, O; Falson, P; Boumendjel, A Eur J Med Chem 202: (2020)
- Fauber, B; Rene, O; Bodil van Niel, M; Ward, S US Patent US9302985 (2016)
- van Niel, MB; Fauber, BP; Cartwright, M; Gaines, S; Killen, JC; René, O; Ward, SI; de Leon Boenig, G; Deng, Y; Eidenschenk, C; Everett, C; Gancia, E; Ganguli, A; Gobbi, A; Hawkins, J; Johnson, AR; Kiefer, JR; La, H; Lockey, P; Norman, M; Ouyang, W; Qin, A; Wakes, N; Waszkowycz, B; Wong, H Bioorg Med Chem Lett 24: 5769-76 (2014)
- Lane, T; Makarov, V; Nelson, JAE; Meeker, RB; Sanna, G; Riabova, O; Kazakova, E; Monakhova, N; Tsedilin, A; Urbina, F; Jones, T; Suchy, A; Ekins, S J Med Chem 66: 6193-6217 (2023)
- Ulven, T; Little, PB; Receveur, JM; Frimurer, TM; Rist, O; Nørregaard, PK; Högberg, T Bioorg Med Chem Lett 16: 1070-5 (2006)
- Czechtizky, W; Weston, J; Rackelmann, N; Podeschwa, M; Arndt, P; Wirth, K; Goegelein, H; Ritzeler, O; Kraft, V; Bellevergue, P; McCort, G US Patent US8912224 (2014)
- Jackson, JJ; Shibuya, GM; Ravishankar, B; Adusumilli, L; Bradford, D; Brockstedt, DG; Bucher, C; Bui, M; Cho, C; Colas, C; Cutler, G; Dukes, A; Han, X; Hu, DX; Jacobson, S; Kassner, PD; Katibah, GE; Ko, MYM; Kolhatkar, U; Leger, PR; Ma, A; Marshall, L; Maung, J; Ng, AA; Okano, A; Pookot, D; Poon, D; Ramana, C; Reilly, MK; Robles, O; Schwarz, JB; Shakhmin, AA; Shunatona, HP; Sreenivasan, R; Tivitmahaisoon, P; Xu, M; Zaw, T; Wustrow, DJ; Zibinsky, M J Med Chem 65: 12895-12924 (2022)
- Roche, O; Nettekoven, M; Vifian, W; Sarmiento, RM Bioorg Med Chem Lett 18: 4377-9 (2008)
- Altmann, E; Hommel, U; Lorthiois, EL; Maibaum, JK; Ostermann, N; Quancard, J; Randl, SA; Rogel, O; Vulpetti, A; Flohr, S US Patent US9487483 (2016)
- Rosati, O; Messina, F; Pelosi, A; Curini, M; Petrucci, V; Gertsch, J; Chicca, A Eur J Med Chem 85: 77-86 (2014)
- Meredith, EL; Ardayfio, O; Beattie, K; Dobler, MR; Enyedy, I; Gaul, C; Hosagrahara, V; Jewell, C; Koch, K; Lee, W; Lehmann, H; McKinsey, TA; Miranda, K; Pagratis, N; Pancost, M; Patnaik, A; Phan, D; Plato, C; Qian, M; Rajaraman, V; Rao, C; Rozhitskaya, O; Ruppen, T; Shi, J; Siska, SJ; Springer, C; van Eis, M; Vega, RB; von Matt, A; Yang, L; Yoon, T; Zhang, JH; Zhu, N; Monovich, LG J Med Chem 53: 5400-21 (2010)
- Moyano, N; Frydman, J; Buldain, G; Ruiz, O; Frydman, RB J Med Chem 33: 1969-74 (1990)
- ADAMS, CM; CZABANIUK, LC; FLOHR, S; GESSIER, F; HEDIGER, MC; HURTH, K; LABBE-GIGUERE, N; LIMA, F; PATEL, T; SIMIC, O; SENDZIK, M; VITREY, A; VULPETTI, A US Patent US20250115572 (2025)
- Claridge, S; Raeppel, F; Granger, MC; Bernstein, N; Saavedra, O; Zhan, L; Llewellyn, D; Wahhab, A; Deziel, R; Rahil, J; Beaulieu, N; Nguyen, H; Dupont, I; Barsalou, A; Beaulieu, C; Chute, I; Gravel, S; Robert, MF; Lefebvre, S; Dubay, M; Pascal, R; Gillespie, J; Jin, Z; Wang, J; Besterman, JM; MacLeod, AR; Vaisburg, A Bioorg Med Chem Lett 18: 2793-8 (2008)
- Wenzel, B; Li, Y; Kraus, W; Sorger, D; Sabri, O; Brust, P; Steinbach, J Bioorg Med Chem Lett 22: 2163-6 (2012)
- Eghtedari, M; Sarrafi, Y; Nadri, H; Mahdavi, M; Moradi, A; Homayouni Moghadam, F; Emami, S; Firoozpour, L; Asadipour, A; Sabzevari, O; Foroumadi, A Eur J Med Chem 128: 237-246 (2017)
- Wilson, AA; Hicks, JW; Sadovski, O; Parkes, J; Tong, J; Houle, S; Fowler, CJ; Vasdev, N J Med Chem 56: 201-9 (2013)
- Shirasaki, Y; Nakamura, M; Yamaguchi, M; Miyashita, H; Sakai, O; Inoue, J J Med Chem 49: 3926-32 (2006)
- Miyazaki, H; Ikeda, Y; Sakurai, O; Miyake, T; Tsubota, R; Okabe, J; Kuroda, M; Hisada, Y; Yanagida, T; Yoneda, H; Tsukumo, Y; Tokunaga, S; Kawata, T; Ohashi, R; Fukuda, H; Kojima, K; Kannami, A; Kifuji, T; Sato, N; Idei, A; Iguchi, T; Sakairi, T; Moritani, Y Bioorg Med Chem Lett 28: 2055-2060 (2018)
- Holenz, J; Mercè, R; Díaz, JL; Guitart, X; Codony, X; Dordal, A; Romero, G; Torrens, A; Mas, J; Andaluz, B; Hernández, S; Monroy, X; Sánchez, E; Hernández, E; Pérez, R; Cubí, R; Sanfeliu, O; Buschmann, H J Med Chem 48: 1781-95 (2005)
- Shibata, N; Nagai, K; Morita, Y; Ujikawa, O; Ohoka, N; Hattori, T; Koyama, R; Sano, O; Imaeda, Y; Nara, H; Cho, N; Naito, M J Med Chem 61: 543-575 (2018)
- Migliore, M; Habrant, D; Sasso, O; Albani, C; Bertozzi, SM; Armirotti, A; Piomelli, D; Scarpelli, R Eur J Med Chem 109: 216-37 (2016)
- Kuttruff, CA; Fleck, M; Carotta, S; Arnhof, H; Bretschneider, T; Dahmann, G; Gremel, G; Grube, A; Handschuh, S; Heimann, A; Hofmann, MH; Impagnatiello, MA; Nar, H; Rast, G; Schaaf, O; Schmidt, E; Oost, T J Med Chem 66: 9376-9400 (2023)
- Klein, M; Busch, M; Friese-Hamim, M; Crosignani, S; Fuchss, T; Musil, D; Rohdich, F; Sanderson, MP; Seenisamy, J; Walter-Bausch, G; Zanelli, U; Hewitt, P; Esdar, C; Schadt, O J Med Chem 64: 10230-10245 (2021)
- Ishiguro, N; Shimizu, H; Kishimoto, W; Ebner, T; Schaefer, O Drug Metab Dispos 41: 149-58 (2012)
- Draoui, N; Schicke, O; Fernandes, A; Drozak, X; Nahra, F; Dumont, A; Douxfils, J; Hermans, E; Dogné, JM; Corbau, R; Marchand, A; Chaltin, P; Sonveaux, P; Feron, O; Riant, O Bioorg Med Chem 21: 7107-17 (2013)
- Gonschorek, P; Zorzi, A; Maric, T; Le Jeune, M; Schüttel, M; Montagnon, M; Gómez-Ojea, R; Vollmar, DP; Whitfield, C; Reymond, L; Carle, V; Verma, H; Schilling, O; Hovnanian, A; Heinis, C J Med Chem 65: 9735-9749 (2022)
- Kopka, K; Faust, A; Keul, P; Wagner, S; Breyholz, HJ; Höltke, C; Schober, O; Schäfers, M; Levkau, B J Med Chem 49: 6704-15 (2006)
- Crosignani, S; Bombrun, A; Covini, D; Maio, M; Marin, D; Quattropani, A; Swinnen, D; Simpson, D; Sauer, W; Françon, B; Martin, T; Cambet, Y; Nichols, A; Martinou, I; Burgat-Charvillon, F; Rivron, D; Donini, C; Schott, O; Eligert, V; Novo-Perez, L; Vitte, PA; Arrighi, JF Bioorg Med Chem Lett 20: 1516-9 (2010)
- Steinmetzer, T; Schweinitz, A; Stürzebecher, A; Dönnecke, D; Uhland, K; Schuster, O; Steinmetzer, P; Müller, F; Friedrich, R; Than, ME; Bode, W; Stürzebecher, J J Med Chem 49: 4116-26 (2006)
- Wagner, B; Smieško, M; Jakob, RP; Mühlethaler, T; Cramer, J; Maier, T; Rabbani, S; Schwardt, O; Ernst, B Eur J Med Chem 272:
- Gordon, DE; Jang, GM; Bouhaddou, M; Xu, J; Obernier, K; White, KM; O'Meara, MJ; Rezelj, VV; Guo, JZ; Swaney, DL; Tummino, TA; Hüttenhain, R; Kaake, RM; Richards, AL; Tutuncuoglu, B; Foussard, H; Batra, J; Haas, K; Modak, M; Kim, M; Haas, P; Polacco, BJ; Braberg, H; Fabius, JM; Eckhardt, M; Soucheray, M; Bennett, MJ; Cakir, M; McGregor, MJ; Li, Q; Meyer, B; Roesch, F; Vallet, T; Mac Kain, A; Miorin, L; Moreno, E; Naing, ZZC; Zhou, Y; Peng, S; Shi, Y; Zhang, Z; Shen, W; Kirby, IT; Melnyk, JE; Chorba, JS; Lou, K; Dai, SA; Barrio-Hernandez, I; Memon, D; Hernandez-Armenta, C; Lyu, J; Mathy, CJP; Perica, T; Pilla, KB; Ganesan, SJ; Saltzberg, DJ; Rakesh, R; Liu, X; Rosenthal, SB; Calviello, L; Venkataramanan, S; Liboy-Lugo, J; Lin, Y; Huang, XP; Liu, Y; Wankowicz, SA; Bohn, M; Safari, M; Ugur, FS; Koh, C; Savar, NS; Tran, QD; Shengjuler, D; Fletcher, SJ; O'Neal, MC; Cai, Y; Chang, JCJ; Broadhurst, DJ; Klippsten, S; Sharp, PP; Wenzell, NA; Kuzuoglu-Ozturk, D; Wang, HY; Trenker, R; Young, JM; Cavero, DA; Hiatt, J; Roth, TL; Rathore, U; Subramanian, A; Noack, J; Hubert, M; Stroud, RM; Frankel, AD; Rosenberg, OS; Verba, KA; Agard, DA; Ott, M; Emerman, M; Jura, N; von Zastrow, M; Verdin, E; Ashworth, A; Schwartz, O; d'Enfert, C; Mukherjee, S; Jacobson, M; Malik, HS; Fujimori, DG; Ideker, T; Craik, CS; Floor, SN; Fraser, JS; Gross, JD; Sali, A; Roth, BL; Ruggero, D; Taunton, J; Kortemme, T; Beltrao, P; Vignuzzi, M; García-Sastre, A; Shokat, KM; Shoichet, BK; Krogan, NJ Nature 583: 459-468 (2020)
- Steri, R; Rupp, M; Proschak, E; Schroeter, T; Zettl, H; Hansen, K; Schwarz, O; Müller-Kuhrt, L; Müller, KR; Schneider, G; Schubert-Zsilavecz, M Bioorg Med Chem Lett 20: 2920-3 (2010)
- Eustache, J; Grob, A; Lam, C; Sellier, O; Schulz, G Bioorg Med Chem Lett 8: 2961-6 (1999)
- Zeng, Q; Nair, AG; Rosenblum, SB; Huang, HC; Lesburg, CA; Jiang, Y; Selyutin, O; Chan, TY; Bennett, F; Chen, KX; Venkatraman, S; Sannigrahi, M; Velazquez, F; Duca, JS; Gavalas, S; Huang, Y; Pu, H; Wang, L; Pinto, P; Vibulbhan, B; Agrawal, S; Ferrari, E; Jiang, CK; Li, C; Hesk, D; Gesell, J; Sorota, S; Shih, NY; Njoroge, FG; Kozlowski, JA Bioorg Med Chem Lett 23: 6585-7 (2013)
- Schormann, N; Velu, SE; Murugesan, S; Senkovich, O; Walker, K; Chenna, BC; Shinkre, B; Desai, A; Chattopadhyay, D Bioorg Med Chem 18: 4056-66 (2010)
- Choudhary, S; Singh, PK; Verma, H; Singh, H; Silakari, O Eur J Med Chem 151: 62-97 (2018)
- Puleo, DE; Kucera, K; Hammarén, HM; Ungureanu, D; Newton, AS; Silvennoinen, O; Jorgensen, WL; Schlessinger, J ACS Med Chem Lett 8: 618-621 (2017)
- Brandl, T; Raman, P; Rigollier, P; Seepersaud, M; Simic, O US Patent US8613914 (2013)
- Jiao, GS; Simo, O; Nagata, M; Oamppound39Malley, S; Hemscheidt, T; Cregar, L; Millis, SZ; Goldman, ME; Tang, C Bioorg Med Chem Lett 16: 5183-9 (2006)
- Taft, BR; Yokokawa, F; Kirrane, T; Mata, AC; Huang, R; Blaquiere, N; Waldron, G; Zou, B; Simon, O; Vankadara, S; Chan, WL; Ding, M; Sim, S; Straimer, J; Guiguemde, A; Lakshminarayana, SB; Jain, JP; Bodenreider, C; Thompson, C; Lanshoeft, C; Shu, W; Fang, E; Qumber, J; Chan, K; Pei, L; Chen, YL; Schulz, H; Lim, J; Abas, SN; Ang, X; Liu, Y; Angulo-Barturen, I; Jiménez-Díaz, MB; Gamo, FJ; Crespo-Fernandez, B; Rosenthal, PJ; Cooper, RA; Tumwebaze, P; Aguiar, ACC; Campo, B; Campbell, S; Wagner, J; Diagana, TT; Sarko, C J Med Chem 65: 3798-3813 (2022)
- Westaway, SM; Preston, AG; Barker, MD; Brown, F; Brown, JA; Campbell, M; Chung, CW; Drewes, G; Eagle, R; Garton, N; Gordon, L; Haslam, C; Hayhow, TG; Humphreys, PG; Joberty, G; Katso, R; Kruidenier, L; Leveridge, M; Pemberton, M; Rioja, I; Seal, GA; Shipley, T; Singh, O; Suckling, CJ; Taylor, J; Thomas, P; Wilson, DM; Lee, K; Prinjha, RK J Med Chem 59: 1370-87 (2016)
- Schulze, M; Siol, O; Decker, M; Lehmann, J Bioorg Med Chem Lett 20: 2946-9 (2010)
- McComas, C; Cohen, J; Huselton, C; Marella, M; Melenski, E; Mugford, C; Slayden, O; Winneker, R; Wrobel, J; Yudt, MR; Fensome, A Bioorg Med Chem Lett 22: 7119-22 (2012)
- Scholz, M; Ulbrich, HK; Soehnlein, O; Lindbom, L; Mattern, A; Dannhardt, G Bioorg Med Chem 17: 558-68 (2009)
- Finger, V; Kufa, M; Soukup, O; Castagnolo, D; Roh, J; Korabecny, J Eur J Med Chem 246: (2023)
- Teodori, E; Contino, M; Riganti, C; Bartolucci, G; Braconi, L; Manetti, D; Romanelli, MN; Trezza, A; Athanasios, A; Spiga, O; Perrone, MG; Giampietro, R; Gazzano, E; Salerno, M; Colabufo, NA; Dei, S Eur J Med Chem 182: (2019)
- Eaton, JB; Peng, JH; Schroeder, KM; George, AA; Fryer, JD; Krishnan, C; Buhlman, L; Kuo, YP; Steinlein, O; Lukas, RJ Mol Pharmacol 64: 1283-94 (2003)
- Rothweiler, U; Czarna, A; Weber, L; Popowicz, GM; Brongel, K; Kowalska, K; Orth, M; Stemmann, O; Holak, TA J Med Chem 51: 5035-42 (2008)
- Peterson, K; Kumar, R; Stenström, O; Verma, P; Verma, PR; Håkansson, M; Kahl-Knutsson, B; Zetterberg, F; Leffler, H; Akke, M; Logan, DT; Nilsson, UJ J Med Chem 61: 1164-1175 (2018)
- Correa, EA; Högestätt, ED; Sterner, O; Echeverri, F; Zygmunt, PM Bioorg Med Chem 18: 3299-306 (2010)
- Thomson, CG; Le Grand, D; Dowling, M; Beattie, D; Elphick, L; Faller, M; Freeman, M; Hardaker, E; Head, V; Hemmig, R; Hill, J; Lister, A; Pascoe, D; Rieffel, S; Shrestha, B; Steward, O; Zink, F Bioorg Med Chem Lett 31: (2021)
- Furukawa, A; Arita, T; Fukuzaki, T; Mori, M; Honda, T; Satoh, S; Matsui, Y; Wakabayashi, K; Hayashi, S; Nakamura, K; Araki, K; Kuroha, M; Tanaka, J; Wakimoto, S; Suzuki, O; Ohsumi, J Eur J Med Chem 54: 522-33 (2012)
- Cannalire, R; Tarantino, D; Astolfi, A; Barreca, ML; Sabatini, S; Massari, S; Tabarrini, O; Milani, M; Querat, G; Mastrangelo, E; Manfroni, G; Cecchetti, V Eur J Med Chem 143: 1667-1676 (2018)
- Okamoto, M; Takayama, K; Shimizu, T; Ishida, K; Takahashi, O; Furuya, T J Med Chem 52: 7323-7 (2009)
- Yoshida, Y; Terauchi, T; Naoe, Y; Kazuta, Y; Ozaki, F; Beuckmann, CT; Nakagawa, M; Suzuki, M; Kushida, I; Takenaka, O; Ueno, T; Yonaga, M Bioorg Med Chem 22: 6071-88 (2014)
- Kosugi, T; Mitchell, DR; Fujino, A; Imai, M; Kambe, M; Kobayashi, S; Makino, H; Matsueda, Y; Oue, Y; Komatsu, K; Imaizumi, K; Sakai, Y; Sugiura, S; Takenouchi, O; Unoki, G; Yamakoshi, Y; Cunliffe, V; Frearson, J; Gordon, R; Harris, CJ; Kalloo-Hosein, H; Le, J; Patel, G; Simpson, DJ; Sherborne, B; Thomas, PS; Suzuki, N; Takimoto-Kamimura, M; Kataoka, K J Med Chem 55: 6700-15 (2012)
- Kumazawa, M; Tejima, M; Fukuda, M; Takeda, S; Suzuki, K; Mizumoto, Y; Sato, K; Waki, M; Miyachi, H; Asai, A; Takikawa, O; Hashimoto, T; Ohno, O; Matsuno, K ACS Med Chem Lett 12: 211-216 (2021)
- Cavdar, H; Ekinci, D; Talaz, O; Saraçoglu, N; Sentürk, M; Supuran, CT J Enzyme Inhib Med Chem 27: 148-54 (2012)
- Shibue, T; Okamoto, I; Morita, N; Morita, H; Hirasawa, Y; Hosoya, T; Tamura, O Bioorg Med Chem Lett 21: 431-4 (2011)
- Yamasaki, K; Tani, O; Tateishi, Y; Tanabe, E; Namatame, I; Niimi, T; Furukawa, K; Sakashita, H J Med Chem 59: 2261-6 (2016)
- Tanwar, O; Tanwar, L; Shaquiquzzaman, M; Alam, MM; Akhter, M Bioorg Med Chem Lett 24: 3447-51 (2014)
- Ho, W; Tutwiler, GF; Cottrell, SC; Morgans, DJ; Tarhan, O; Mohrbacher, RJ J Med Chem 29: 2184-90 (1986)
- Müller, J; Klein, R; Tarkhanova, O; Gryniukova, A; Borysko, P; Merkl, S; Ruf, M; Neumann, A; Gastreich, M; Moroz, YS; Klebe, G; Glinca, S J Med Chem 65: 15663-15678 (2022)
- Schirrmacher, E; Schirrmacher, R; Thews, O; Dillenburg, W; Helisch, A; Wessler, I; Buhl, R; Höhnemann, S; Buchholz, HG; Bartenstein, P; Machulla, HJ; Rösch, F Bioorg Med Chem Lett 13: 2687-92 (2003)
- Campiani, G; Butini, S; Fattorusso, C; Trotta, F; Gemma, S; Catalanotti, B; Nacci, V; Fiorini, I; Cagnotto, A; Mereghetti, I; Mennini, T; Minetti, P; Di Cesare, MA; Stasi, MA; Di Serio, S; Ghirardi, O; Tinti, O; Carminati, P J Med Chem 48: 1705-8 (2005)
- Labas, R; Gilbert, G; Nicole, O; Dhilly, M; Abbas, A; Tirel, O; Buisson, A; Henry, J; Barré, L; Debruyne, D; Sobrio, F Eur J Med Chem 46: 2295-309 (2011)
- Vaccarin, C; Veit, G; Hegedus, T; Torres, O; Chilin, A; Lukacs, GL; Marzaro, G J Med Chem 67: 13891-13908
- Nagao, S; Yamane, Y; Funasaka, S; Tanaka, K; Miyazaki, K; Kotake, Y; Kamata, J; Watanabe-Miyano, S; Toyama, O; Ozawa, Y; Mizui, Y; Okamoto, K; Ito, D Bioorg Med Chem 22: 5513-29 (2014)
- Macor, JE; Gurley, D; Lanthorn, T; Loch, J; Mack, RA; Mullen, G; Tran, O; Wright, N; Gordon, JC Bioorg Med Chem Lett 11: 319-21 (2001)
- Tsuruta, O; Yuasa, H; Hashimoto, H Bioorg Med Chem Lett 6: 1989-1992 (1996)
- Smith, JM; Barlaam, B; Beattie, D; Bradshaw, L; Chan, HM; Chiarparin, E; Collingwood, O; Cooke, SL; Cronin, A; Cumming, I; Dean, E; Debreczeni, JÉ; Del Barco Barrantes, I; Diene, C; Gianni, D; Guerot, C; Guo, X; Guven, S; Hayhow, TG; Hong, T; Kemmitt, PD; Lamont, GM; Lamont, S; Lynch, JT; McWilliams, L; Moore, S; Raubo, P; Robb, GR; Robinson, J; Scott, JS; Srinivasan, B; Steward, O; Stubbs, CJ; Syson, K; Tan, L; Turner, O; Underwood, E; Urosevic, J; Vazquez-Chantada, M; Whittaker, AL; Wilson, DM; Winter-Holt, JJ J Med Chem 67: 13604-13638
- Nalli, M; Armijos Rivera, JI; Masci, D; Coluccia, A; Badia, R; Riveira-Muñoz, E; Brambilla, A; Cinquina, E; Turriziani, O; Falasca, F; Catalano, M; Limatola, C; Esté, JA; Maga, G; Silvestri, R; Crespan, E; La Regina, G Eur J Med Chem 208: (2020)
- Goswami, R; Wohlfahrt, G; Törmäkangas, O; Moilanen, A; Lakshminarasimhan, A; Nagaraj, J; Arumugam, KN; Mukherjee, S; Chacko, AR; Krishnamurthy, NR; Jaleel, M; Palakurthy, RK; Samiulla, DS; Ramachandra, M Bioorg Med Chem Lett 25: 5309-14 (2015)
- Fukatsu, K; Uchikawa, O; Kawada, M; Yamano, T; Yamashita, M; Kato, K; Hirai, K; Hinuma, S; Miyamoto, M; Ohkawa, S J Med Chem 45: 4212-21 (2002)
- Shimokawa, K; Shibata, N; Sameshima, T; Miyamoto, N; Ujikawa, O; Nara, H; Ohoka, N; Hattori, T; Cho, N; Naito, M ACS Med Chem Lett 8: 1042-1047 (2017)
- Němec, V; Remeš, M; Beňovský, P; Böck, MC; Šranková, E; Wong, JF; Cros, J; Williams, E; Tse, LH; Smil, D; Ensan, D; Isaac, MB; Al-Awar, R; Gomolková, R; Ursachi, VC; Fafílek, B; Kahounová, Z; Víchová, R; Vacek, O; Berger, BT; Wells, CI; Corona, CR; Vasta, JD; Robers, MB; Krejci, P; Souček, K; Bullock, AN; Knapp, S; Paruch, K J Med Chem 67: 12632-12659
- Sarasamkan, J; Scheunemann, M; Apaijai, N; Palee, S; Parichatikanond, W; Arunrungvichian, K; Fischer, S; Chattipakorn, S; Deuther-Conrad, W; Schüürmann, G; Brust, P; Vajragupta, O ACS Med Chem Lett 7: 890-895 (2016)
- Sibille, P; Lopez, S; Brabet, I; Valenti, O; Oueslati, N; Gaven, F; Goudet, C; Bertrand, HO; Neyton, J; Marino, MJ; Amalric, M; Pin, JP; Acher, FC J Med Chem 50: 3585-95 (2007)
- Vechorkin, O; Liu, K; Pan, J; Sokolsky, A; Ye, HF; Ye, Q; Yao, W; Hummel, J US Patent US11542265 (2023)
- Crespin, O; Nicolai, E; Venier, O US Patent US8536173 (2013)
- Law, JM; Stark, SC; Liu, K; Liang, NE; Hussain, MM; Leiendecker, M; Ito, D; Verho, O; Stern, AM; Johnston, SE; Zhang, YL; Dunn, GP; Shamji, AF; Schreiber, SL ACS Med Chem Lett 7: 944-949 (2016)
- Shippy, RR; Lin, X; Agabiti, SS; Li, J; Zangari, BM; Foust, BJ; Poe, MM; Hsiao, CC; Vinogradova, O; Wiemer, DF; Wiemer, AJ J Med Chem 60: 2373-2382 (2017)
- Traxler, PM; Wacker, O; Bach, HL; Geissler, JF; Kump, W; Meyer, T; Regenass, U; Roesel, JL; Lydon, N J Med Chem 34: 2328-37 (1991)
- Brown, A; Brown, L; Ellis, D; Puhalo, N; Smith, CR; Wallace, O; Watson, L Bioorg Med Chem Lett 18: 4278-81 (2008)
- Cázares-Körner, A; Helleday, T; Visnes, T; Wallner, O; Koolmeister, T US Patent US11970474 (2024)
- Graulich, A; Dilly, S; Farce, A; Scuvée-Moreau, J; Waroux, O; Lamy, C; Chavatte, P; Seutin, V; Liégeois, JF J Med Chem 50: 5070-5 (2007)
- Schmeck, C; Gielen-Haertwig, H; Vakalopoulos, A; Bischoff, H; Li, V; Wirtz, G; Weber, O Bioorg Med Chem Lett 20: 1740-3 (2010)
- Bruno, F; Errico, S; Pace, S; Nawrozkij, MB; Mkrtchyan, AS; Guida, F; Maisto, R; Olgaç, A; D'Amico, M; Maione, S; De Rosa, M; Banoglu, E; Werz, O; Fiorentino, A; Filosa, R Eur J Med Chem 155: 946-960 (2018)
- Boye, SV; Ortega-Caballero, F; Sinning, S; Wiborg, O; Jensen, HH; Bols, M Bioorg Med Chem Lett 17: 6019-25 (2007)
- Estiu, G; Greenberg, E; Harrison, CB; Kwiatkowski, NP; Mazitschek, R; Bradner, JE; Wiest, O J Med Chem 51: 2898-906 (2008)
- Berndt, A; Miller, S; Williams, O; Le, DD; Houseman, BT; Pacold, JI; Gorrec, F; Hon, WC; Liu, Y; Rommel, C; Gaillard, P; Rückle, T; Schwarz, MK; Shokat, KM; Shaw, JP; Williams, RL Nat Chem Biol 6: 117-24 (2010)
- McCombie, SW; Bishop, RW; Carr, D; Dobek, E; Kirkup, MP; Kirschmeier, P; Lin, S; Petrin, J; Rosinski, K; Shankar, BB; Wilson, O Bioorg Med Chem Lett 3: 1537-1542 (1993)
- Kovaleva, K; Oleshko, O; Mamontova, E; Yarovaya, O; Zakharova, O; Zakharenko, A; Kononova, A; Dyrkheeva, N; Cheresiz, S; Pokrovsky, A; Lavrik, O; Salakhutdinov, N J Nat Prod 82: 2443-2450 (2019)
- Tsuno, N; Yukimasa, A; Yoshida, O; Suzuki, S; Nakai, H; Ogawa, T; Fujiu, M; Takaya, K; Nozu, A; Yamaguchi, H; Matsuda, H; Funaki, S; Nishimura, Y; Ito, T; Nagamatsu, D; Asaki, T; Horita, N; Yamamoto, M; Hinata, M; Soga, M; Imai, M; Morioka, Y; Kanemasa, T; Sakaguchi, G; Iso, Y Bioorg Med Chem Lett 26: 4936-4941 (2016)
- Morikawa, T; Hachiman, I; Matsuo, K; Nishida, E; Ninomiya, K; Hayakawa, T; Yoshie, O; Muraoka, O; Nakayama, T J Nat Prod 79: 2005-13 (2016)
- Drabczynska, A; Müller, CE; Schiedel, A; Schumacher, B; Karolak-Wojciechowska, J; Fruzinski, A; Zobnina, W; Yuzlenko, O; Kiec-Kononowicz, K Bioorg Med Chem 15: 6956-74 (2007)
- CASTRO, AC; BURKE, MJ; WYNN, TA; RUPPEL, SK; SANTILLANA SOTO, SL; HAINES, E; XU, L; ZAVIDIJ, O US Patent US20230382863 (2023)
- Zakharova, O; Luzina, O; Zakharenko, A; Sokolov, D; Filimonov, A; Dyrkheeva, N; Chepanova, A; Ilina, E; Ilyina, A; Klabenkova, K; Chelobanov, B; Stetsenko, D; Zafar, A; Eurtivong, C; Reynisson, J; Volcho, K; Salakhutdinov, N; Lavrik, O Bioorg Med Chem 26: 4470-4480 (2018)
- Cabrele, C; Langer, M; Bader, R; Wieland, HA; Doods, HN; Zerbe, O; Beck-Sickinger, AG J Biol Chem 275: 36043-8 (2000)
- Gazal, S; Gelerman, G; Ziv, O; Karpov, O; Litman, P; Bracha, M; Afargan, M; Gilon, C J Med Chem 45: 1665-71 (2002)
- Wijtmans, M; de Graaf, C; de Kloe, G; Istyastono, EP; Smit, J; Lim, H; Boonnak, R; Nijmeijer, S; Smits, RA; Jongejan, A; Zuiderveld, O; de Esch, IJ; Leurs, R J Med Chem 54: 1693-703 (2011)
- Soares da Costa, TP; Tieu, W; Yap, MY; Zvarec, O; Bell, JM; Turnidge, JD; Wallace, JC; Booker, GW; Wilce, MC; Abell, AD; Polyak, SW ACS Med Chem Lett 3: 509-514 (2012)
- Szabó, G; Éliás, O; Erdélyi, P; Potor, A; Túrós, GI; Károlyi, BI; Varró, G; Vaskó, ÁG; Bata, I; Kapus, GL; Dohányos, Z; Bobok, AÁ; Fodor, L; Thán, M; Vastag, M; Komlódi, Z; Soukupné Kedves, RÉ; Makó, É; Süveges, B; Greiner, I J Med Chem 65: 7876-7895 (2022)
- Rupar, J; Dobričić, V; Grahovac, J; Radulović, S; Skok, Ž; Ilaš, J; Aleksić, M; Brborić, J; Čudina, O RSC Med Chem 11: 378-386 (2020)
- Kožíšek, M; Štěpánek, O; Parkan, K; Berenguer Albiñana, C; Pávová, M; Weber, J; Krӓusslich, HG; Konvalinka, J; Machara, A Bioorg Med Chem Lett 26: 3487-90 (2016)