Compound (92)
Article Title (6)
Article Author (88)
Assay (5)
CABOZANTINIB US12304898, Example Cabozantinib Cometriq US10227329, Compound Cabozantinib US20240174674, Compound Cabozantinib Cabometyx US10202365, Compound Cabozantinib CHEBI:72317 US12338253, Compound Cabozantinib US10464902, Cabozantinib BDBM50021574 BMS-907351 US11279688, Compound Cabozantinib cabozantinib s-malate US10183928, Cabozantinib XL-184 US10273211, Compound Cabozantinib US10774070, Compound Cabozantinib
US10287267, Compound 707 US10556885, Compound 707 US11174244, Compound 707 BDBM385240 US10508099, Compound 707 US11673881, Compound 707
US10881652, Example 707 BDBM305689 US11648243, Example 707 US10144734, Example 707 US10172845, Example 707 US10441581, Example 707
BDBM87372 US10709712, Example 707 US10245267, Example 707 US9694016, 707
US9745328, Compound 707 US9884878, Compound 707 BDBM169302 US9079866, 707
BDBM431840 US11014913, Example 707 US10870641, Example 707 US10550105, Example 707
US10478424, Example 707 US10071079, Example 707 BDBM273921
US10711020, Example 707 BDBM382996 US10273259, Example 707
US11046698, Compound I-707 BDBM424252 US10508120, Compound I-707 US10577373, Compound I-707
BDBM566139 US12221453, Compound I-707 US11414431, Compound I-707
BDBM116980 US8637532, 707
BDBM122267 US8722692, 707
BDBM177341 US9120749, 707
BDBM179054 US9126931, 707
BDBM216662 US9302989, 707
BDBM217992 US9212182, 707
BDBM88276 US9695118, 707
US8871934, 707 BDBM138114
US9034866, 707 BDBM159230
US9085555, 707 BDBM171349
US9283222, 707 BDBM214583
US9328096, 707 BDBM227019
US9434711, 707 BDBM248754
US9675593, 707 BDBM173093
BDBM170323 US9079913, MI-707
BDBM444118 US10660877, Example 707
BDBM583815 US11524959, Compound 707.
BDBM584958 US11524968, Example 707
BDBM623688 US11780845, Example 707
BDBM632437 US20230348426, Example 707
BDBM650601 US20240043427, Example 707
BDBM687686 US20240246964, Compound 707
BDBM762018 US12378224, Example 707
CHEMBL1159714 Ko 707 BDBM50421719
US10988445, Example 707 BDBM493718
US11286268, Compound 707 BDBM545221
US11292791, Example 707 BDBM547434
US11814367, Compound 707 BDBM635257
US11845723, Example 707 BDBM641805
US12384753, Example 707 BDBM763662
US20160046618, Example 707 BDBM705581
US20240116946, Example 707 BDBM666673
US20240316047, Example 707 BDBM697926
US20250145633, Example 707 BDBM739374
BDBM727845 US20250090540, Example I-707
US10150728, Example I-707 BDBM307470
US10202379, Reference Example 707 BDBM346972
US20250163057, Compound I-707 BDBM742410
US9034866, 707 BDBM159229 US9034866, 706
US11130759, Cpd. No. 707 1-(2-chlorophenyl)-4-(thiazol-4- ylamino)-7-(trifluoromethyl) pyrido[2,3-d]-pyrimidin-2(1H)-one US11084798, Cpd No 707 US11046691, Compound 707 BDBM508396
US11053244, Example 710 BDBM517285 US11053244, Example 707
US20230348426, Example 706 US20230348426, Example 707 BDBM632436
acs.jmedchem.1c00409_ST.707 BDBM429332 jm5b01461, Compound 149
NN-DIPROP-5-CT BDBM81789 5-CT,DP DP-5-CT CAS_156314 NSC_156314
BDBM120583 Roche-Dataset for PDE10A, Compound 707 US8703768, 183
BDBM29555 [3H]-5-CT
CT-20026 BDBM50487411 CHEMBL427882
US10106501, Example CT BDBM293221
BDBM293222 US10106501, Example CT-1
BDBM293223 US10106501, Example CT-2
BDBM293224 US10106501, Example CT-3
BDBM293225 US10106501, Example CT-4
BDBM293226 US10106501, Example CT-5
BDBM293231 US10106501, Example CT-10
BDBM293232 US10106501, Example CT-11
BDBM681166 US20240199555, Reference 5-CT
US10106501, Example CT-6 BDBM293227
US10106501, Example CT-7 BDBM293228
US10106501, Example CT-8 BDBM293229
US10106501, Example CT-9 BDBM293230
BDBM50478476 CHEMBL454065 CT-2108A CHEBI:65678
BDBM50478477 CHEMBL454066 CT-2108B CHEBI:65679
BDBM468045 N-((1RS,2RS)-2-Aminocyclopentyl)-5-(*S)-(4-methyl-6- phenoxypyridin-3-yl)-4-oxo-4,5-dihydro-3H-1-thia-3,5,8- triazaacenaphthylene-2-carboxamide; US10800792, Example 707 US10822348, Example 707
US10822352, Comp No. 707 US10287301, Compound 707 (2S,4R)-1-(2-(3- acetyl-5-(1H- pyrazol-4-yl)-1H- indazol-1- yl)acetyl)-N-(6- bromopyridin-2- yl)-4- fluoropyrrolidine- 2-carboxamide BDBM386752
5-CT CHEMBL18840 5-CT,DP [3H]-5-carboxamidotryptamine [3H]-5-Carboxamide tryptamine 3-(2-aminoethyl)-1H-indole-5-carboxamide [3H]-5-Carboxyamidotryptamine [3H]-5-CT BDBM21392 CHEMBL1256863 5-carboxamidotryptamine
BDBM262854 4'-(2-aminoethyl)-2-(1H- tetrazol-5-yl)-4- (trifluoromethyl)biphenyl-3- sulfonamide US9708336, 707
(R)-6-(1-(3-hydroxy-2- methylpropyl)-1H- pyrazol-4-yl)-4-(6-(4- ((6-methoxypyridin-3- yl)methyl)piperazin-1- yl)pyridin-3- yl)pyrazolo[1,5- a]pyridine-3- carbonitrile BDBM284672 US10023570, Example 707 US10174027, Example 707
BDBM418022 US11001575, Example 707 US10457669, Example 707 (2R)-2-[6-(5-chloro-2-{[(2S)-1- hydroxypropan-2-yl]amino}pyrimidin- 4-yl)-1-oxo-2,3-dihydro-1H-isoindol-2- yl]-3-hydroxy-N-[1-(3- methylphenyl)cyclopropyl]propanamide
BDBM50141287 CT 32228 5TT4A4MBLR HE066284 CT-32228 N-(4-Bromo-phenyl)-6-(5-chloro-2-methyl-phenyl)-[1,3,5]triazine-2,4-diamine CHEMBL36501
US10266526, Compound 707 1-cyclopropyl-N-[1-(3-hydroxypropyl)azetidin-3-yl]-1H-1,2,3-triazole-4-carboxamide BDBM378569
5-CT,DP CAS_74885-72-6 BDBM81784 5-carboxyamidotryptamine maleate
US9796708, Example 707 BDBM353475 4-(2,4-dimethoxyphenyl)-2-[1-(methylsulfonyl)-1,2,3,6-tetrahydropyridin-4-yl]-1H-pyrrolo[2,3-b]pyridine
US11078201, Compound I-707 US11548890, Compound I-707 (S)-7-((6- ((dimethylamino)- methyl)-5- (tetrahydrofuran- 3-yl)pyridin- 2-yl)amino)-4- (1-methyl-1H- indol-4-yl)- 2,3-dihydro- 1H-pyrrolo[3,4- c]pyridin-1-one BDBM500876 US11021481, Compound I-540
US10544143, Example 710 US10544143, Example 721 BDBM517285 US10730877, Example 727 US10544143, Example 707 US11053244, Example 727 BDBM428271 US10544143, Example 727
BDBM50526797 Ct-7001 ICEC0942 US11857552, Compound REF-001 ICEC-0942 Samuraciclib Ct7001
US12065436, Compound 708 (S)-N-(6-(5-(difluoromethyl)-1,2,4- oxadiazol-3-yl)-2,3- dihydrobenzofuran-3-yl)-4- (hydroxymethyl)picolinamide US12065436, Compound 707 BDBM691318
(2S,4aS,6aS,6bR,8aR,9S,10S,12aS,12bR,14bR)-10-(acetyloxy)-2,4a,6a,6b,9,12a-hexamethyl-13-oxo-9-{[(2-oxo-5-phenyl-2H-1,3-dioxol-4-yl)methoxy]carbonyl}-1,2,3,4,4a,5,6,6a,6b,7,8,8a,9,10,11,12,12a,12b,13,14b-icosahydropicene-2-carboxylic acid US11858959, Compound 707-1 US20240209019, Compound 707-1 BDBM642892
US10065972, Example 707 (R)-N-benzyl-1-(3-methyl-4-oxo-2-trifluoromethyl-3,4-dihydropyrido[3,2-d]pyrimidin-6-yl)pyrrolidine-2-carboxamide BDBM273196
(3R,4S)-4-(4-fluorophenyl)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-N-{[4-(trifluoromethyl)cyclohexyl]methyl}pyrrolidin-3-amine US9656955, Example 707 BDBM309185
BDBM355616 US9815796, Example 707 (R)- or (S)-N-((3-fluoro-4- ((trifluoromethyl)thio)phenyl)(1- methylcyclopropyl)methyl)-6-oxo-2- phenyl-1,6-dihydropyrimidine-4- carboxamide
BDBM407763 US10336762, Compound 707 (R)-6-(3-cyanopyrrolo[1,2- b]pyridazin-7-yl)-N-(2- fluoro-3-hydroxy-3- methylbutyl)-4-((4- fluorophenethyl)amino) nicotinamide
BDBM433004 US10577363, Compound 707 N-((2S,4S)-2-benzyl-1-(((1-(3- hydroxypropyl)piperidin-4- yl)methyl)sulfonyl)piperidin-4-yl)-5- cyclopropylisoxazole-3-carboxamide
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