Affinity DataKi: 0.300nMAssay Description:Binding affinity to human Androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.450nMAssay Description:Displacement of [3H]DHT from Androgen receptor expressed in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.550nMAssay Description:Displacement of [3H]mibolerone from Androgen receptor (unknown origin) measured by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Binding affinity to Androgen receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Binding affinity to human Androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity to human Androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]DHT from Androgen receptor expressed in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Agonist activity at Androgen receptor expressed in mouse C2C12 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]DHT from Androgen receptor expressed in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Displacement of [3H]DHT from Androgen receptor expressed in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]mibolerone from Androgen receptor (unknown origin) measured by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Binding affinity to human Androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Binding affinity to human Androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Binding affinity to bicalutamide-resistant Androgen receptor T878A mutant (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 6.20nMAssay Description:Binding affinity to rat Androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.5nMAssay Description:Binding affinity to human Androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Binding affinity to human Androgen receptor measured by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Displacement of [3H]DHT from Androgen receptor expressed in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8.70nMAssay Description:Binding affinity to human Androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity to Androgen receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Displacement of [3H]DHT from Androgen receptor expressed in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Binding affinity to human Androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Displacement of [3H]DHT from Androgen receptor expressed in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 62nMAssay Description:Binding affinity to human Androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 73nMAssay Description:Displacement of [3H]DHT from Androgen receptor expressed in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Binding affinity to wild-type Androgen receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 365nMAssay Description:Binding affinity to Androgen receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to rat Androgen receptor ligand binding domain measured by competitive ligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to rat Androgen receptor ligand binding domain measured by competitive ligand binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Antagonist activity at Androgen receptor in human MDA-kb2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Binding affinity to human Androgen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Partial agonist activity at human Androgen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Binding affinity to human Androgen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Binding affinity to human Androgen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Binding affinity to rat Androgen receptor in African green monkey COS-7 cells measured by whole-cell binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Binding affinity to Androgen receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Binding affinity to human Androgen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 3.60nMAssay Description:Binding affinity to Androgen receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 6.60nMAssay Description:Displacement of [3H]methyltrienolone from Androgen receptor expressed in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Agonist activity at Androgen receptor in human 22Rv1 cells cotransfected with pARE-LUC measured by luciferase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Antagonist activity at Androgen receptor in human MDA-kb2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Partial agonist activity at human Androgen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Binding affinity to Androgen receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Binding affinity to rat Androgen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Antagonist activity at Androgen receptor in human MDA-MB-453 cells measured by SEAP reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Antagonist activity at Androgen receptor in human MDA-MB-453 cells measured by SEAP reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Binding affinity to human Androgen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Antagonist activity at wild-type Androgen receptor (unknown origin) expressed in African green monkey COS-7 cells measured as gene transcription leve...More data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Binding affinity to rat Androgen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Binding affinity to human Androgen receptorMore data for this Ligand-Target Pair