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Found 36 Enz. Inhib. hit(s) with all data for entry = 50034910
TargetDelta-type opioid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50290872((-)-rel-3-((4aR,12aS)-2-methyl-1,2,3,4,4a,5,12,12a...)
Affinity DataKi:  0.230nMAssay Description:inhibition of [3H]DADLE binding to delta-opioid receptor of mouse brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50450528(CHEMBL2051964)
Affinity DataKi:  0.460nMAssay Description:inhibition of [3H]DADLE binding to delta-opioid receptor of mouse brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50061061((4aR,8aS)-6-Ethyl-8a-(3-hydroxy-phenyl)-3-methyl-4...)
Affinity DataKi:  0.950nMAssay Description:inhibition of [3H]DADLE binding to delta-opioid receptor of mouse brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50290869((4aR,8aR)-7-Ethyl-4a-(3-hydroxy-phenyl)-3-methyl-4...)
Affinity DataKi:  1.5nMAssay Description:inhibition of [3H]DADLE binding to delta-opioid receptor of mouse brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50061061((4aR,8aS)-6-Ethyl-8a-(3-hydroxy-phenyl)-3-methyl-4...)
Affinity DataKi:  1.90nMAssay Description:inhibition of [3H]DADLE binding to delta-opioid receptor of mouse brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50061061((4aR,8aS)-6-Ethyl-8a-(3-hydroxy-phenyl)-3-methyl-4...)
Affinity DataKi:  1.90nMAssay Description:inhibition of [3H]DADLE binding to delta-opioid receptor of mouse brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50061063((4aR,8aS)-8a-(3-Hydroxy-phenyl)-3,6-dimethyl-4,4a,...)
Affinity DataKi:  2.10nMAssay Description:inhibition of [3H]DADLE binding to delta-opioid receptor of mouse brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50290866((4aR,8aR)-7-Ethyl-4a-(3-hydroxy-phenyl)-3-methyl-4...)
Affinity DataKi:  2.40nMAssay Description:inhibition of [3H]DADLE binding to delta-opioid receptor of mouse brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50290868((4aR,8aS)-6-Ethyl-8a-(3-hydroxy-phenyl)-3-methyl-4...)
Affinity DataKi:  2.60nMAssay Description:inhibition of [3H]DADLE binding to delta-opioid receptor of mouse brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50290870((4aR,8aR)-4a-(3-Hydroxy-phenyl)-3,7-dimethyl-4,4a,...)
Affinity DataKi:  3nMAssay Description:inhibition of [3H]DADLE binding to delta-opioid receptor of mouse brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50290871((4aR,8aS)-6-Ethyl-8a-(3-hydroxy-phenyl)-3-methyl-4...)
Affinity DataKi:  6.80nMAssay Description:inhibition of [3H]DADLE binding to delta-opioid receptor of mouse brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Mus musculus (Mouse))
TBA

Curated by ChEMBL
LigandPNGBDBM50450528(CHEMBL2051964)
Affinity DataKi:  9.5nMAssay Description:Binding affinity against Kappa opioid receptor using [3H]U-69593 radioligand in mouse brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50290867((4aR,8aS)-6-Ethyl-8a-(3-hydroxy-phenyl)-3-methyl-4...)
Affinity DataKi:  15nMAssay Description:inhibition of [3H]DADLE binding to delta-opioid receptor of mouse brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50450528(CHEMBL2051964)
Affinity DataKi:  16nMAssay Description:Inhibition of [3H]DAMGO from mouse brain homogenate Mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50290869((4aR,8aR)-7-Ethyl-4a-(3-hydroxy-phenyl)-3-methyl-4...)
Affinity DataKi:  42nMAssay Description:Inhibition of [3H]DAMGO from mouse brain homogenate Mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50290868((4aR,8aS)-6-Ethyl-8a-(3-hydroxy-phenyl)-3-methyl-4...)
Affinity DataKi:  58nMAssay Description:Inhibition of [3H]DAMGO from mouse brain homogenate Mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50290872((-)-rel-3-((4aR,12aS)-2-methyl-1,2,3,4,4a,5,12,12a...)
Affinity DataKi:  60nMAssay Description:Inhibition of [3H]DAMGO from mouse brain homogenate Mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Mus musculus (Mouse))
TBA

Curated by ChEMBL
LigandPNGBDBM50290867((4aR,8aS)-6-Ethyl-8a-(3-hydroxy-phenyl)-3-methyl-4...)
Affinity DataKi:  70nMAssay Description:Binding affinity against Kappa opioid receptor using [3H]U-69593 radioligand in mouse brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50290870((4aR,8aR)-4a-(3-Hydroxy-phenyl)-3,7-dimethyl-4,4a,...)
Affinity DataKi:  89nMAssay Description:Inhibition of [3H]DAMGO from mouse brain homogenate Mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50061063((4aR,8aS)-8a-(3-Hydroxy-phenyl)-3,6-dimethyl-4,4a,...)
Affinity DataKi:  93nMAssay Description:Inhibition of [3H]DAMGO from mouse brain homogenate Mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50290867((4aR,8aS)-6-Ethyl-8a-(3-hydroxy-phenyl)-3-methyl-4...)
Affinity DataKi:  139nMAssay Description:Inhibition of [3H]DAMGO from mouse brain homogenate Mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50290866((4aR,8aR)-7-Ethyl-4a-(3-hydroxy-phenyl)-3-methyl-4...)
Affinity DataKi:  141nMAssay Description:Inhibition of [3H]DAMGO from mouse brain homogenate Mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Mus musculus (Mouse))
TBA

Curated by ChEMBL
LigandPNGBDBM50290866((4aR,8aR)-7-Ethyl-4a-(3-hydroxy-phenyl)-3-methyl-4...)
Affinity DataKi:  169nMAssay Description:Binding affinity against Kappa opioid receptor using [3H]U-69593 radioligand in mouse brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Mus musculus (Mouse))
TBA

Curated by ChEMBL
LigandPNGBDBM50290872((-)-rel-3-((4aR,12aS)-2-methyl-1,2,3,4,4a,5,12,12a...)
Affinity DataKi:  312nMAssay Description:Binding affinity against Kappa opioid receptor using [3H]U-69593 radioligand in mouse brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50061061((4aR,8aS)-6-Ethyl-8a-(3-hydroxy-phenyl)-3-methyl-4...)
Affinity DataKi:  407nMAssay Description:Inhibition of [3H]DAMGO from mouse brain homogenate Mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50061061((4aR,8aS)-6-Ethyl-8a-(3-hydroxy-phenyl)-3-methyl-4...)
Affinity DataKi:  407nMAssay Description:Inhibition of [3H]DAMGO from mouse brain homogenate Mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Mus musculus (Mouse))
TBA

Curated by ChEMBL
LigandPNGBDBM50290869((4aR,8aR)-7-Ethyl-4a-(3-hydroxy-phenyl)-3-methyl-4...)
Affinity DataKi:  449nMAssay Description:Binding affinity against Kappa opioid receptor using [3H]U-69593 radioligand in mouse brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Mus musculus (Mouse))
TBA

Curated by ChEMBL
LigandPNGBDBM50061063((4aR,8aS)-8a-(3-Hydroxy-phenyl)-3,6-dimethyl-4,4a,...)
Affinity DataKi:  500nMAssay Description:Binding affinity against Kappa opioid receptor using [3H]U-69593 radioligand in mouse brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50290871((4aR,8aS)-6-Ethyl-8a-(3-hydroxy-phenyl)-3-methyl-4...)
Affinity DataKi:  580nMAssay Description:Inhibition of [3H]DAMGO from mouse brain homogenate Mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Mus musculus (Mouse))
TBA

Curated by ChEMBL
LigandPNGBDBM50290871((4aR,8aS)-6-Ethyl-8a-(3-hydroxy-phenyl)-3-methyl-4...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against Kappa opioid receptor using [3H]U-69593 radioligand in mouse brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Mus musculus (Mouse))
TBA

Curated by ChEMBL
LigandPNGBDBM50290870((4aR,8aR)-4a-(3-Hydroxy-phenyl)-3,7-dimethyl-4,4a,...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against Kappa opioid receptor using [3H]U-69593 radioligand in mouse brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Mus musculus (Mouse))
TBA

Curated by ChEMBL
LigandPNGBDBM50290868((4aR,8aS)-6-Ethyl-8a-(3-hydroxy-phenyl)-3-methyl-4...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against Kappa opioid receptor using [3H]U-69593 radioligand in mouse brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Mus musculus (Mouse))
TBA

Curated by ChEMBL
LigandPNGBDBM50061061((4aR,8aS)-6-Ethyl-8a-(3-hydroxy-phenyl)-3-methyl-4...)
Affinity DataKi:  1.30E+3nMAssay Description:Inhibition of [3H]DAMGO from mouse brain homogenate Mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Mus musculus (Mouse))
TBA

Curated by ChEMBL
LigandPNGBDBM50061061((4aR,8aS)-6-Ethyl-8a-(3-hydroxy-phenyl)-3-methyl-4...)
Affinity DataKi:  1.34E+3nMAssay Description:Binding affinity against Kappa opioid receptor using [3H]U-69593 radioligand in mouse brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Mus musculus (Mouse))
TBA

Curated by ChEMBL
LigandPNGBDBM50061061((4aR,8aS)-6-Ethyl-8a-(3-hydroxy-phenyl)-3-methyl-4...)
Affinity DataKi:  1.34E+3nMAssay Description:Binding affinity against Kappa opioid receptor using [3H]U-69593 radioligand in mouse brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50061061((4aR,8aS)-6-Ethyl-8a-(3-hydroxy-phenyl)-3-methyl-4...)
Affinity DataKi: >5.00E+3nMAssay Description:inhibition of [3H]DADLE binding to delta-opioid receptor of mouse brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article