Compile Data Set for Download or QSAR
Report error Found 110 Enz. Inhib. hit(s) with all data for entry = 50013506
TargetAlpha-2C adrenergic receptor(Human)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131353BDBM50131353(7,8-Dimethoxy-3-[4-((E)-2-methyl-3-phenyl-allyl)-p...)
Affinity DataKi:  0.200nMAssay Description:In vitro binding affinity towards human adrenergic alpha-2C adrenergic receptor using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131348BDBM50131348(7-Methoxy-3-[4-((E)-3-phenyl-allyl)-piperazin-1-yl...)
Affinity DataKi:  0.5nMAssay Description:In vitro binding affinity towards human alpha-2A adrenergic receptor using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131359BDBM50131359((3R,3aS)-7,8-Dimethoxy-3-[4-((E)-3-phenyl-allyl)-p...)
Affinity DataKi:  0.5nMAssay Description:In vitro binding affinity towards human adrenergic alpha-2C adrenergic receptor using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131359BDBM50131359((3R,3aS)-7,8-Dimethoxy-3-[4-((E)-3-phenyl-allyl)-p...)
Affinity DataKi:  0.5nMAssay Description:In vitro binding affinity towards human adrenergic alpha-2C adrenergic receptor using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131365BDBM50131365(7,8-Dimethoxy-3-[4-((E)-3-phenyl-but-2-enyl)-piper...)
Affinity DataKi:  0.600nMAssay Description:In vitro binding affinity towards human adrenergic alpha-2C adrenergic receptor using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131350BDBM50131350(8-Methoxy-3-[4-((E)-3-phenyl-allyl)-piperazin-1-yl...)
Affinity DataKi:  0.800nMAssay Description:In vitro binding affinity towards human alpha-2A adrenergic receptor using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131353BDBM50131353(7,8-Dimethoxy-3-[4-((E)-2-methyl-3-phenyl-allyl)-p...)
Affinity DataKi:  0.800nMAssay Description:In vitro binding affinity towards human alpha-2A adrenergic receptor using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131360BDBM50131360(3-[4-((E)-3-Phenyl-allyl)-piperazin-1-ylmethyl]-3a...)
Affinity DataKi:  0.900nMAssay Description:In vitro binding affinity towards human alpha-2A adrenergic receptor using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131359BDBM50131359((3R,3aS)-7,8-Dimethoxy-3-[4-((E)-3-phenyl-allyl)-p...)
Affinity DataKi:  1.20nMAssay Description:In vitro binding affinity towards rat serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131359BDBM50131359((3R,3aS)-7,8-Dimethoxy-3-[4-((E)-3-phenyl-allyl)-p...)
Affinity DataKi:  1.20nMAssay Description:In vitro binding affinity towards rat serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131351BDBM50131351((3R,3aS)-7,8-Dimethoxy-3-(4-naphthalen-2-ylmethyl-...)
Affinity DataKi:  1.30nMAssay Description:In vitro binding affinity towards rat serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131351BDBM50131351((3R,3aS)-7,8-Dimethoxy-3-(4-naphthalen-2-ylmethyl-...)
Affinity DataKi:  1.30nMAssay Description:In vitro binding affinity towards rat serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131346BDBM50131346((3R,3aS)-7,8-Dimethoxy-3-[4-((E)-2-methyl-3-phenyl...)
Affinity DataKi:  1.40nMAssay Description:In vitro binding affinity towards human adrenergic alpha-2C adrenergic receptor using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131346BDBM50131346((3R,3aS)-7,8-Dimethoxy-3-[4-((E)-2-methyl-3-phenyl...)
Affinity DataKi:  1.40nMAssay Description:In vitro binding affinity towards human adrenergic alpha-2C adrenergic receptor using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131365BDBM50131365(7,8-Dimethoxy-3-[4-((E)-3-phenyl-but-2-enyl)-piper...)
Affinity DataKi:  1.40nMAssay Description:In vitro binding affinity towards human alpha-2A adrenergic receptor using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131354BDBM50131354(7,8-Dimethoxy-3-(4-naphthalen-2-ylmethyl-piperazin...)
Affinity DataKi:  1.70nMAssay Description:In vitro binding affinity towards rat serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131360BDBM50131360(3-[4-((E)-3-Phenyl-allyl)-piperazin-1-ylmethyl]-3a...)
Affinity DataKi:  1.70nMAssay Description:In vitro binding affinity towards human adrenergic alpha-2C adrenergic receptor using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131366BDBM50131366(7,8-Dimethoxy-3-[4-(3-phenyl-propyl)-piperazin-1-y...)
Affinity DataKi:  1.90nMAssay Description:In vitro binding affinity towards human adrenergic alpha-2C adrenergic receptor using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131348BDBM50131348(7-Methoxy-3-[4-((E)-3-phenyl-allyl)-piperazin-1-yl...)
Affinity DataKi:  1.90nMAssay Description:In vitro binding affinity towards human adrenergic alpha-2C adrenergic receptor using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131360BDBM50131360(3-[4-((E)-3-Phenyl-allyl)-piperazin-1-ylmethyl]-3a...)
Affinity DataKi:  2nMAssay Description:In vitro binding affinity towards human alpha-2B adrenergic receptor using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50057128BDBM50057128(A-80426 | (2-Benzofuran-6-yl-ethyl)-((R)-5-methoxy...)
Affinity DataKi:  2.10nMAssay Description:In vitro binding affinity towards human adrenergic alpha-2C adrenergic receptor using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131353BDBM50131353(7,8-Dimethoxy-3-[4-((E)-2-methyl-3-phenyl-allyl)-p...)
Affinity DataKi:  2.30nMAssay Description:In vitro binding affinity towards rat serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131350BDBM50131350(8-Methoxy-3-[4-((E)-3-phenyl-allyl)-piperazin-1-yl...)
Affinity DataKi:  2.30nMAssay Description:In vitro binding affinity towards human adrenergic alpha-2C adrenergic receptor using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50057128BDBM50057128(A-80426 | (2-Benzofuran-6-yl-ethyl)-((R)-5-methoxy...)
Affinity DataKi:  2.40nMAssay Description:In vitro binding affinity towards human alpha-2A adrenergic receptor using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131359BDBM50131359((3R,3aS)-7,8-Dimethoxy-3-[4-((E)-3-phenyl-allyl)-p...)
Affinity DataKi:  2.60nMAssay Description:In vitro binding affinity towards human alpha-2A adrenergic receptor using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131359BDBM50131359((3R,3aS)-7,8-Dimethoxy-3-[4-((E)-3-phenyl-allyl)-p...)
Affinity DataKi:  2.60nMAssay Description:In vitro binding affinity towards human alpha-2A adrenergic receptor using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131346BDBM50131346((3R,3aS)-7,8-Dimethoxy-3-[4-((E)-2-methyl-3-phenyl...)
Affinity DataKi:  2.80nMAssay Description:In vitro binding affinity towards rat serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131346BDBM50131346((3R,3aS)-7,8-Dimethoxy-3-[4-((E)-2-methyl-3-phenyl...)
Affinity DataKi:  2.80nMAssay Description:In vitro binding affinity towards rat serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131354BDBM50131354(7,8-Dimethoxy-3-(4-naphthalen-2-ylmethyl-piperazin...)
Affinity DataKi:  3.10nMAssay Description:In vitro binding affinity towards human adrenergic alpha-2C adrenergic receptor using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131364BDBM50131364(7,8-Dimethoxy-3-(4-naphthalen-1-ylmethyl-piperazin...)
Affinity DataKi:  3.90nMAssay Description:In vitro binding affinity towards rat serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50057128BDBM50057128(A-80426 | (2-Benzofuran-6-yl-ethyl)-((R)-5-methoxy...)
Affinity DataKi:  4nMAssay Description:In vitro binding affinity towards rat serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131356BDBM50131356(3-[4-(1H-Inden-2-ylmethyl)-piperazin-1-ylmethyl]-7...)
Affinity DataKi:  4.10nMAssay Description:In vitro binding affinity towards rat serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131356BDBM50131356(3-[4-(1H-Inden-2-ylmethyl)-piperazin-1-ylmethyl]-7...)
Affinity DataKi:  4.70nMAssay Description:In vitro binding affinity towards human adrenergic alpha-2C adrenergic receptor using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131354BDBM50131354(7,8-Dimethoxy-3-(4-naphthalen-2-ylmethyl-piperazin...)
Affinity DataKi:  5nMAssay Description:In vitro binding affinity towards human alpha-2A adrenergic receptor using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131368BDBM50131368(3-(4-Benzo[b]thiophen-2-ylmethyl-piperazin-1-ylmet...)
Affinity DataKi:  5nMAssay Description:In vitro binding affinity towards rat serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131358BDBM50131358(3-[4-(7,8-Dimethoxy-3a,4-dihydro-3H-chromeno[4,3-c...)
Affinity DataKi:  5.30nMAssay Description:In vitro binding affinity towards human adrenergic alpha-2C adrenergic receptor using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131357BDBM50131357(4-(5-Fluoro-indan-2-ylmethyl)-4,5-dihydro-1H-imida...)
Affinity DataKi:  5.90nMAssay Description:In vitro binding affinity towards human alpha-2A adrenergic receptor using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131355BDBM50131355(7,8-Dimethoxy-3-[4-((E)-3-phenyl-allyl)-piperazin-...)
Affinity DataKi:  6.20nMAssay Description:In vitro binding affinity towards human adrenergic alpha-2C adrenergic receptor using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131352BDBM50131352(3-(4-Benzo[b]thiophen-3-ylmethyl-piperazin-1-ylmet...)
Affinity DataKi:  7.20nMAssay Description:In vitro binding affinity towards rat serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131353BDBM50131353(7,8-Dimethoxy-3-[4-((E)-2-methyl-3-phenyl-allyl)-p...)
Affinity DataKi:  7.5nMAssay Description:In vitro binding affinity towards human alpha-2B adrenergic receptor using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131367BDBM50131367(7,8-Dimethoxy-3-(4-quinolin-6-ylmethyl-piperazin-1...)
Affinity DataKi:  8.10nMAssay Description:In vitro binding affinity towards rat serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131355BDBM50131355(7,8-Dimethoxy-3-[4-((E)-3-phenyl-allyl)-piperazin-...)
Affinity DataKi:  8.30nMAssay Description:In vitro binding affinity towards rat serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131355BDBM50131355(7,8-Dimethoxy-3-[4-((E)-3-phenyl-allyl)-piperazin-...)
Affinity DataKi:  8.80nMAssay Description:In vitro binding affinity towards human alpha-2A adrenergic receptor using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131351BDBM50131351((3R,3aS)-7,8-Dimethoxy-3-(4-naphthalen-2-ylmethyl-...)
Affinity DataKi:  9.5nMAssay Description:In vitro binding affinity towards human adrenergic alpha-2C adrenergic receptor using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131351BDBM50131351((3R,3aS)-7,8-Dimethoxy-3-(4-naphthalen-2-ylmethyl-...)
Affinity DataKi:  9.5nMAssay Description:In vitro binding affinity towards human adrenergic alpha-2C adrenergic receptor using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131365BDBM50131365(7,8-Dimethoxy-3-[4-((E)-3-phenyl-but-2-enyl)-piper...)
Affinity DataKi:  10nMAssay Description:In vitro binding affinity towards rat serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131366BDBM50131366(7,8-Dimethoxy-3-[4-(3-phenyl-propyl)-piperazin-1-y...)
Affinity DataKi:  10nMAssay Description:In vitro binding affinity towards rat serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131347BDBM50131347((3R,3aS)-7,8-Dimethoxy-3-[4-((E)-3-phenyl-but-2-en...)
Affinity DataKi:  10nMAssay Description:In vitro binding affinity towards rat serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131347BDBM50131347((3R,3aS)-7,8-Dimethoxy-3-[4-((E)-3-phenyl-but-2-en...)
Affinity DataKi:  10nMAssay Description:In vitro binding affinity towards human adrenergic alpha-2C adrenergic receptor using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131347BDBM50131347((3R,3aS)-7,8-Dimethoxy-3-[4-((E)-3-phenyl-but-2-en...)
Affinity DataKi:  10nMAssay Description:In vitro binding affinity towards rat serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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