Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50037413
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Korea Institute of Science & Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50148172BDBM50148172(KYS-05042 | N-(4-(4-fluorophenylsulfonamido)benzyl...)
Affinity DataIC50: 110nMAssay Description:Inhibition of T-type [Ca2+] channel (alpha1G) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Korea Institute of Science & Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157857BDBM50157857(2-(2-(5-aminopentylamino)-3-(biphenyl-4-yl)-3,4-di...)
Affinity DataIC50: 130nMAssay Description:Inhibition of T-type [Ca2+] channel (alpha1G) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Korea Institute of Science & Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157862BDBM50157862(2-(3-(5-aminopentyl)-2-(biphenyl-4-ylamino)-3,4-di...)
Affinity DataIC50: 140nMAssay Description:Inhibition of T-type [Ca2+] channel (alpha1G) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Korea Institute of Science & Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157864BDBM50157864(tert-butyl 5-(4-(2-(benzylamino)-2-oxoethyl)-3-(bi...)
Affinity DataIC50: 160nMAssay Description:Inhibition of T-type [Ca2+] channel (alpha1G) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Korea Institute of Science & Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157861BDBM50157861({5-[4-(Benzylcarbamoyl-methyl)-2-(biphenyl-4-ylami...)
Affinity DataIC50: 170nMAssay Description:Inhibition of T-type [Ca2+] channel (alpha1G) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Korea Institute of Science & Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50148180BDBM50148180(KYS-05041 | N-(4-(4-methylphenylsulfonamido)benzyl...)
Affinity DataIC50: 170nMAssay Description:Inhibition of T-type [Ca2+] channel (alpha1G) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Korea Institute of Science & Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157856BDBM50157856(methyl 2-(3-(5-aminopentyl)-2-(biphenyl-4-ylamino)...)
Affinity DataIC50: 300nMAssay Description:Inhibition of T-type [Ca2+] channel (alpha1G) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Korea Institute of Science & Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157860BDBM50157860(methyl 2-(2-(biphenyl-4-ylamino)-3-(5-(tert-butoxy...)
Affinity DataIC50: 370nMAssay Description:Inhibition of T-type [Ca2+] channel (alpha1G) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Korea Institute of Science & Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157859BDBM50157859(methyl 2-(2-(5-aminopentylamino)-3-(biphenyl-4-yl)...)
Affinity DataIC50: 560nMAssay Description:Inhibition of T-type [Ca2+] channel (alpha1G) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Korea Institute of Science & Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157863BDBM50157863(methyl 2-(3-(biphenyl-4-yl)-2-(5-(tert-butoxycarbo...)
Affinity DataIC50: 680nMAssay Description:Inhibition of T-type [Ca2+] channel (alpha1G) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Korea Institute of Science & Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50148175BDBM50148175(N-Benzyl-2-(3-phenyl-2-piperidin-1-yl-3,4-dihydro-...)
Affinity DataIC50: 1.16E+3nMAssay Description:Inhibition of T-type [Ca2+] channel (alpha1G) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Korea Institute of Science & Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117922BDBM50117922(CHEMBL45816 | Methoxy-acetic acid 2-(2-{[3-(1H-ben...)
Affinity DataIC50: 1.34E+3nMAssay Description:Inhibition of T-type [Ca2+] channel (alpha1G) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed