Compile Data Set for Download or QSAR
maximum 50k data
Found 39 Enz. Inhib. hit(s) with all data for entry = 50025504
TargetNeutrophil collagenase(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50031795((N-(2-HYDROXAMATEMETHYLENE-4-METHYL-PENTOYL)PHENYL...)
Affinity DataIC50:  0.0460nMAssay Description:Inhibition of human recombinant MMP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50031795((N-(2-HYDROXAMATEMETHYLENE-4-METHYL-PENTOYL)PHENYL...)
Affinity DataIC50:  0.380nMAssay Description:Inhibition of human recombinant MMP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50031795((N-(2-HYDROXAMATEMETHYLENE-4-METHYL-PENTOYL)PHENYL...)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of human recombinant MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50031795((N-(2-HYDROXAMATEMETHYLENE-4-METHYL-PENTOYL)PHENYL...)
Affinity DataIC50:  8.30nMAssay Description:Inhibition of human recombinant MMP7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50031795((N-(2-HYDROXAMATEMETHYLENE-4-METHYL-PENTOYL)PHENYL...)
Affinity DataIC50:  25nMAssay Description:Inhibition of human recombinant MMP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50031795((N-(2-HYDROXAMATEMETHYLENE-4-METHYL-PENTOYL)PHENYL...)
Affinity DataIC50:  43nMAssay Description:Inhibition of human recombinant MMP3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50245248((S)-N4-hydroxy-2-isobutyl-N1-((S)-1-(methylamino)-...)
Affinity DataIC50:  48nMAssay Description:Inhibition of human recombinant MMP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50245248((S)-N4-hydroxy-2-isobutyl-N1-((S)-1-(methylamino)-...)
Affinity DataIC50:  150nMAssay Description:Inhibition of human recombinant MMP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50245248((S)-N4-hydroxy-2-isobutyl-N1-((S)-1-(methylamino)-...)
Affinity DataIC50:  170nMAssay Description:Inhibition of human recombinant MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50245248((S)-N4-hydroxy-2-isobutyl-N1-((S)-1-(methylamino)-...)
Affinity DataIC50:  640nMAssay Description:Inhibition of human recombinant MMP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50245248((S)-N4-hydroxy-2-isobutyl-N1-((S)-1-(methylamino)-...)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of human recombinant MMP7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50245248((S)-N4-hydroxy-2-isobutyl-N1-((S)-1-(methylamino)-...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of human recombinant MMP3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50272134(CHEMBL501715 | N-[(Hydroxyamino)carbonyl]-L-leucyl...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of human recombinant MMP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50272134(CHEMBL501715 | N-[(Hydroxyamino)carbonyl]-L-leucyl...)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibition of human recombinant MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50272134(CHEMBL501715 | N-[(Hydroxyamino)carbonyl]-L-leucyl...)
Affinity DataIC50:  7.00E+4nMAssay Description:Inhibition of human recombinant MMP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50245247(CHEMBL452082 | N-[(Hydroxyamino)carbonyl]-D-leucyl...)
Affinity DataIC50:  1.50E+5nMAssay Description:Inhibition of human recombinant MMP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50245247(CHEMBL452082 | N-[(Hydroxyamino)carbonyl]-D-leucyl...)
Affinity DataIC50:  2.00E+5nMAssay Description:Inhibition of human recombinant MMP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50272134(CHEMBL501715 | N-[(Hydroxyamino)carbonyl]-L-leucyl...)
Affinity DataIC50:  2.70E+5nMAssay Description:Inhibition of human recombinant MMP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50245249(CHEMBL452584 | N-(Benzyloxycarbonyl)-L-leucyl-L-ph...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human recombinant MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50245249(CHEMBL452584 | N-(Benzyloxycarbonyl)-L-leucyl-L-ph...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human recombinant MMP3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50245249(CHEMBL452584 | N-(Benzyloxycarbonyl)-L-leucyl-L-ph...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human recombinant MMP7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50245249(CHEMBL452584 | N-(Benzyloxycarbonyl)-L-leucyl-L-ph...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human recombinant MMP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50245250(CHEMBL445994 | L-Leucyl-L-phenylalanine methylamid...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human recombinant MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50245250(CHEMBL445994 | L-Leucyl-L-phenylalanine methylamid...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human recombinant MMP7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50245251(CHEMBL510082 | D-Leucyl-L-phenylalanine methylamid...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human recombinant MMP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50245251(CHEMBL510082 | D-Leucyl-L-phenylalanine methylamid...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human recombinant MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50245251(CHEMBL510082 | D-Leucyl-L-phenylalanine methylamid...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human recombinant MMP3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50245251(CHEMBL510082 | D-Leucyl-L-phenylalanine methylamid...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human recombinant MMP7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50245249(CHEMBL452584 | N-(Benzyloxycarbonyl)-L-leucyl-L-ph...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human recombinant MMP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50245251(CHEMBL510082 | D-Leucyl-L-phenylalanine methylamid...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human recombinant MMP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50245251(CHEMBL510082 | D-Leucyl-L-phenylalanine methylamid...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human recombinant MMP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50245249(CHEMBL452584 | N-(Benzyloxycarbonyl)-L-leucyl-L-ph...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human recombinant MMP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50245250(CHEMBL445994 | L-Leucyl-L-phenylalanine methylamid...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human recombinant MMP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50245247(CHEMBL452082 | N-[(Hydroxyamino)carbonyl]-D-leucyl...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human recombinant MMP7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50245247(CHEMBL452082 | N-[(Hydroxyamino)carbonyl]-D-leucyl...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human recombinant MMP3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50245247(CHEMBL452082 | N-[(Hydroxyamino)carbonyl]-D-leucyl...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human recombinant MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50245247(CHEMBL452082 | N-[(Hydroxyamino)carbonyl]-D-leucyl...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human recombinant MMP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50272134(CHEMBL501715 | N-[(Hydroxyamino)carbonyl]-L-leucyl...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human recombinant MMP7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50272134(CHEMBL501715 | N-[(Hydroxyamino)carbonyl]-L-leucyl...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human recombinant MMP3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed